felodipine and dihydropyridines

felodipine has been researched along with dihydropyridines in 38 studies

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-19902 (5.26)18.7374
1990's20 (52.63)18.2507
2000's9 (23.68)29.6817
2010's7 (18.42)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adams, ME; Cohen, CJ; Ertel, EA; Leibowitz, MD; Smith, MM; Venema, VJ1
Bladen, C; Dunn, SM1
Edgar, B; Eriksson, UG; Lundahl, J; Miniscalco, A; Regårdh, CG1
Dong, H; Lu, YQ; Wang, Q; Yang, QQ; Yang, ZC1
Bäärnhielm, C; Berntsson, P; Brian, WR; Guengerich, FP; Iwasaki, M; Sari, MA1
Guengerich, FP; Kim, DH1
Breimer, DD; Roosemalen, MC; Soons, PA1
Boström, S; Nilsson, A; Westerlund, C1
Bäärnhielm, C; Hansson, G1
Lanfranchi, J1
Bülow, A; Johansson, B1
Abrahamsson, T; Akerblom, B; Nordlander, M; Thalén, P1
Atassi, G; Guilbaud, N; Kraus-Berthier, L; Leonce, S; Lombet, A; Peglion, JL; Pierre, A1
Arnold, JM; Bailey, DG; Spence, JD1
Agrotis, A; Bobik, A; Little, PJ; Saltis, J1
Block, LH; Nauck, M; Rödler, S; Roth, M; Tamm, M1
Block, LH; Eickelberg, O; Erne, P; Kohler, E; Roth, M1
Knaus, EE; Yiu, S1
Kikuchi, K; Sugawara, H; Tobise, K1
Sharma, RK; Wang, JH; Wu, Z1
Bossi, M; Tiberti, G1
Knaus, EE; Yiu, SH1
de Vries, RJ; Dunselman, PH; van Veldhuisen, DJ1
Corradi, L; Fogari, R; Malalamani, GD; Mugellini, A; Preti, P; Zoppi, A1
Mielcarek, J1
Bollo, S; Bontá, M; Caballero, E; Maya, JD; Medarde, M; Morello, A; Núñez-Vergara, LJ; Puebla, P; Repetto, Y; Rodriguez, A; San Feliciano, A; Squella, JA; Tellez, R; Zelada, U1
Bolla, G; Grassi, G; Mancia, G; Seravalle, G; Turri, C1
Mann, S1
Achard, JM; Fournier, A; Mansour, J; Modeliard, SS; Serot, JM1
Mielcarek, J; Naskrent, M1
Elhebir, ES; Hilmi, SC; Hughes, JD1
Chen, L; Jiao, Y; Jin, H; Ke, YN; Li, DY; Liu, MX; Wang, BY; Wang, L; Wang, Y; Yang, HY; Zhao, XL; Zheng, JT1
Dai, Q; Gong, J; Jin, H; Lu, X; Peng, J; Wang, B; Wang, H; Wu, Y; Xu, M; Xu, X; Yan, J; Zhang, M; Zhao, S2
Bombelli, M; Brambilla, G; Casati, A; Cuspidi, C; Grassi, G; Mancia, G; Pizzalla, DP; Riva, M; Seravalle, G1
De Luca, M; Ioele, G; Ragno, G; Spatari, C1
Cheng, KC; Cheng, KH; Cheng, KY; Lai, WT; Lee, CW; Yang, YH1

Reviews

3 review(s) available for felodipine and dihydropyridines

ArticleYear
[Calcium antagonists and treatment of chronic heart failure].
    Archives des maladies du coeur et des vaisseaux, 1995, Volume: 88, Issue:4 Suppl

    Topics: Animals; Atrial Fibrillation; Calcium Channel Blockers; Dihydropyridines; Felodipine; Heart Failure; Hemodynamics; Humans; Systole; Ventricular Function, Left

1995
Grapefruit juice and drugs. How significant is the interaction?
    Clinical pharmacokinetics, 1994, Volume: 26, Issue:2

    Topics: Beverages; Biological Availability; Citrus; Dihydropyridines; Drug Interactions; Felodipine; Flavanones; Flavonoids; Half-Life; Humans; Nifedipine; Nitrendipine

1994
Efficacy and safety of calcium channel blockers in heart failure: focus on recent trials with second-generation dihydropyridines.
    American heart journal, 2000, Volume: 139, Issue:2 Pt 1

    Topics: Amlodipine; Calcium Channel Blockers; Dihydropyridines; Exercise Test; Exercise Tolerance; Felodipine; Heart Failure; Hemodynamics; Humans; Ventricular Function, Left

2000

Trials

6 trial(s) available for felodipine and dihydropyridines

ArticleYear
Effects of different dihydropyridine calcium antagonists on plasma norepinephrine in essential hypertension.
    Journal of hypertension, 2000, Volume: 18, Issue:12

    Topics: Adult; Aged; Amlodipine; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Dihydropyridines; Double-Blind Method; Felodipine; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Nitrobenzenes; Norepinephrine; Piperazines; Sympathetic Nervous System

2000
Short-versus long-term effects of different dihydropyridines on sympathetic and baroreflex function in hypertension.
    Hypertension (Dallas, Tex. : 1979), 2003, Volume: 41, Issue:3

    Topics: Antihypertensive Agents; Baroreflex; Blood Pressure; Dihydropyridines; Double-Blind Method; Felodipine; Heart Rate; Humans; Hypertension; Male; Middle Aged; Muscle, Skeletal; Norepinephrine; Sympathetic Nervous System; Time Factors

2003
[Efficacy and safety of aranidipine in Chinese patients with mild-to-moderate essential hypertension].
    Zhonghua yi xue za zhi, 2013, Oct-22, Volume: 93, Issue:39

    Topics: Antihypertensive Agents; Dihydropyridines; Double-Blind Method; Essential Hypertension; Felodipine; Female; Humans; Hypertension; Male; Middle Aged

2013
Lercanidipine hydrochloride versus felodipine sustained-release for mild-to-moderate hypertension: a multi-center, randomized clinical trial.
    Current medical research and opinion, 2015, Volume: 31, Issue:1

    Topics: Adolescent; Adult; Aged; Antihypertensive Agents; Delayed-Action Preparations; Dihydropyridines; Felodipine; Female; Follow-Up Studies; Humans; Hypertension; Male; Middle Aged; Treatment Outcome; Young Adult

2015
Differential effects of enalapril-felodipine versus enalapril-lercanidipine combination drug treatment on sympathetic nerve traffic and metabolic profile in obesity-related hypertension.
    Journal of the American Society of Hypertension : JASH, 2016, Volume: 10, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Blood Pressure Monitoring, Ambulatory; Calcium Channel Blockers; Cross-Over Studies; Dihydropyridines; Double-Blind Method; Drug Therapy, Combination; Enalapril; Felodipine; Female; Heart Rate; Humans; Hypertension; Insulin Resistance; Male; Metabolome; Middle Aged; Norepinephrine; Obesity; Random Allocation; Sympathetic Nervous System

2016
Effects of lercanidipine hydrochloride versus felodipine sustained-release on day-to-day home blood pressure variability.
    Current medical research and opinion, 2016, Volume: 32, Issue:sup2

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Delayed-Action Preparations; Dihydropyridines; Felodipine; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Treatment Outcome

2016

Other Studies

29 other study(ies) available for felodipine and dihydropyridines

ArticleYear
High affinity block of myocardial L-type calcium channels by the spider toxin omega-Aga-toxin IIIA: advantages over 1,4-dihydropyridines.
    Molecular pharmacology, 1992, Volume: 42, Issue:6

    Topics: Agatoxins; Animals; Calcium Channel Blockers; Cells, Cultured; Dihydropyridines; Felodipine; Guinea Pigs; Heart Atria; In Vitro Techniques; Ion Channel Gating; Male; Myocardium; Spider Venoms; Substrate Specificity

1992
Low-affinity binding sites for 1,4-dihydropyridines in skeletal muscle transverse tubule membranes revealed by changes in the fluorescence of felodipine.
    Biochemistry, 1992, Apr-28, Volume: 31, Issue:16

    Topics: Animals; Binding Sites; Binding, Competitive; Calcium Channel Blockers; Cations; Cell Membrane; Dihydropyridines; Felodipine; Fluorescent Dyes; Isradipine; Kinetics; Muscles; Rabbits; Spectrometry, Fluorescence

1992
Inhibition of dihydropyridine metabolism in rat and human liver microsomes by flavonoids found in grapefruit juice.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 261, Issue:3

    Topics: Adult; Aged; Animals; Beverages; Citrus; Dihydropyridines; Felodipine; Flavanones; Flavonoids; Humans; Male; Microsomes, Liver; Middle Aged; Nifedipine; Quercetin; Rats; Rats, Inbred Strains; Stereoisomerism

1992
Antagonistic effects of dihydropyridines and verapamil on CaCl2 and 5-HT-evoked contraction in porcine coronary artery.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1991, Volume: 12, Issue:5

    Topics: Animals; Calcium Chloride; Coronary Vessels; Dihydropyridines; Felodipine; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Nicardipine; Nifedipine; Nimodipine; Serotonin Antagonists; Swine; Verapamil

1991
Oxidation of dihydropyridine calcium channel blockers and analogues by human liver cytochrome P-450 IIIA4.
    Journal of medicinal chemistry, 1991, Volume: 34, Issue:6

    Topics: Calcium Channel Blockers; Chromatography, High Pressure Liquid; Cimetidine; Cytochrome P-450 Enzyme System; Dihydropyridines; Felodipine; Humans; Kinetics; Microsomes, Liver; Nifedipine; Norpregnenes; Oxidation-Reduction

1991
In vitro inhibition of dihydropyridine oxidation and aflatoxin B1 activation in human liver microsomes by naringenin and other flavonoids.
    Carcinogenesis, 1990, Volume: 11, Issue:12

    Topics: Aflatoxins; Chamomile; Chromatography, High Pressure Liquid; Dihydropyridines; Felodipine; Flavanones; Flavins; Flavonoids; Gene Expression Regulation; Hesperidin; Humans; In Vitro Techniques; Kaempferols; Microsomes, Liver; Oils, Volatile; Plants, Medicinal; Quercetin; Transcriptional Activation

1990
Enantioselective determination of felodipine and other chiral dihydropyridine calcium entry blockers in human plasma.
    Journal of chromatography, 1990, Jun-29, Volume: 528, Issue:2

    Topics: Calcium Channel Blockers; Chromatography, Gas; Chromatography, High Pressure Liquid; Dihydropyridines; Felodipine; Humans; Male; Nitrendipine; Stereoisomerism

1990
A 62 kDa protein is photoaffinity labelled by [3H]felodipine in vascular smooth muscle, but not in cardiac and skeletal muscle.
    Biochemical pharmacology, 1989, Dec-01, Volume: 38, Issue:23

    Topics: Affinity Labels; Animals; Cytosol; Dihydropyridines; Electrophoresis, Polyacrylamide Gel; Felodipine; Female; Male; Muscle Proteins; Muscle, Smooth, Vascular; Muscles; Myocardium; Swine

1989
Oxidation of 1,4-dihydropyridines by prostaglandin synthase and the peroxidic function of cytochrome P-450. Demonstration of a free radical intermediate.
    Biochemical pharmacology, 1986, May-01, Volume: 35, Issue:9

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Cytochrome P-450 Enzyme System; Dihydropyridines; Electron Spin Resonance Spectroscopy; Felodipine; Free Radicals; Glutathione; In Vitro Techniques; Male; Microsomes; Nifedipine; Oxidation-Reduction; Oxygen Consumption; Peroxidases; Prostaglandin-Endoperoxide Synthases; Pyridines; Rats; Rats, Inbred Strains

1986
Membrane stretch evoked by cell swelling increases contractile activity in vascular smooth muscle through dihydropyridine-sensitive pathways.
    Acta physiologica Scandinavica, 1994, Volume: 152, Issue:4

    Topics: Animals; Calcium; Calcium Channel Blockers; Cell Membrane; Cell Size; Dihydropyridines; Diltiazem; Felodipine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Osmosis; Portal Vein; Rats; Rats, Sprague-Dawley; Stress, Mechanical; Verapamil

1994
Vascular versus myocardial selectivity of dihydropyridine calcium antagonists as studied in vivo and in vitro.
    Pharmacology & toxicology, 1995, Volume: 76, Issue:1

    Topics: Amlodipine; Animals; Calcium Channel Blockers; Dihydropyridines; Dose-Response Relationship, Drug; Felodipine; Heart; Heart Rate; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Nifedipine; Organ Specificity; Rats; Rats, Inbred SHR

1995
In vivo reversal of multidrug resistance by two new dihydropyridine derivatives, S16317 and S16324.
    Acta oncologica (Stockholm, Sweden), 1994, Volume: 33, Issue:6

    Topics: Adenocarcinoma; Animals; Antineoplastic Combined Chemotherapy Protocols; Calcium Channels; Colonic Neoplasms; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Drug Screening Assays, Antitumor; Drug Synergism; Felodipine; Female; Humans; Leukemia P388; Mice; Mice, Inbred DBA; Neoplasm Transplantation; Tumor Cells, Cultured; Vincristine

1994
Dihydropyridine Ca2+ channel antagonists inhibit the salvage pathway for DNA synthesis in human vascular smooth muscle cells.
    European journal of pharmacology, 1993, Feb-15, Volume: 244, Issue:3

    Topics: Calcium Channel Blockers; Cell Division; Cells, Cultured; Dihydropyridines; Diltiazem; DNA; Epidermal Growth Factor; Felodipine; Gene Expression Regulation; Genes, fos; Humans; Immunoblotting; Mammary Arteries; Muscle, Smooth, Vascular; Nisoldipine; Thymidine; Verapamil

1993
Ca(2+)-channel blockers modulate the expression of interleukin-6 and interleukin-8 genes in human vascular smooth muscle cells.
    Journal of molecular and cellular cardiology, 1995, Volume: 27, Issue:10

    Topics: Adrenergic beta-Antagonists; Amlodipine; Calcium Channel Blockers; Calcium Channels; Calcium Channels, L-Type; Cells, Cultured; Dihydropyridines; Diuretics; Felodipine; Fibroblasts; Furosemide; Gene Expression Regulation; Humans; Interleukin-6; Interleukin-8; Isradipine; Lung; Muscle Proteins; Muscle, Smooth, Vascular; Nitrobenzenes; Piperazines; Propranolol; Transcription, Genetic

1995
Ca2+ channel blockers modulate metabolism of collagens within the extracellular matrix.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, May-28, Volume: 93, Issue:11

    Topics: Amlodipine; Becaplermin; Calcium Channel Blockers; Cells, Cultured; Collagen; Collagenases; Dihydropyridines; Diltiazem; Enzyme Activation; Extracellular Matrix; Felodipine; Fibroblasts; Humans; Kinetics; Lung; Metalloendopeptidases; Muscle, Smooth, Vascular; Nitrobenzenes; Piperazines; Platelet-Derived Growth Factor; Procollagen; Proline; Proto-Oncogene Proteins c-sis; Transcription, Genetic; Verapamil

1996
Synthesis, biological evaluation, calcium channel antagonist activity, and anticonvulsant activity of felodipine coupled to a dihydropyridine-pyridinium salt redox chemical delivery system.
    Journal of medicinal chemistry, 1996, Nov-08, Volume: 39, Issue:23

    Topics: Animals; Anticonvulsants; Biotransformation; Brain; Calcium Channel Blockers; Dihydropyridines; Felodipine; Male; Mice; Oxidation-Reduction; Pyridinium Compounds; Rats; Rats, Sprague-Dawley; Sodium Chloride

1996
Antioxidant effects of calcium antagonists on rat myocardial membrane lipid peroxidation.
    Hypertension research : official journal of the Japanese Society of Hypertension, 1996, Volume: 19, Issue:4

    Topics: Adenosine Diphosphate; Animals; Antioxidants; Calcium Channel Blockers; Cell Membrane; Dihydropyridines; Diltiazem; Felodipine; Fumarates; Heart; Iron; Lipid Peroxidation; Male; Myocardium; Nicardipine; Nifedipine; Nisoldipine; Nitrendipine; Oxidation-Reduction; Rats; Rats, Sprague-Dawley; Verapamil

1996
Mechanisms of inhibition of calmodulin-stimulated cyclic nucleotide phosphodiesterase by dihydropyridine calcium antagonists.
    Journal of neurochemistry, 1997, Volume: 69, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Binding, Competitive; Brain; Calcium; Calcium Channel Blockers; Calmodulin; Cattle; Cyclic Nucleotide Phosphodiesterases, Type 1; Dihydropyridines; Felodipine; Isoenzymes; Molecular Weight; Nicardipine; Phosphodiesterase Inhibitors

1997
[Stable angina pectoris: what is the role of calcium antagonists?].
    Giornale italiano di cardiologia, 1997, Volume: 27, Issue:10

    Topics: Adrenergic beta-Antagonists; Angina Pectoris; Atenolol; Calcium Channel Blockers; Clinical Trials as Topic; Dihydropyridines; Diltiazem; Drug Therapy, Combination; Felodipine; Humans; Metoprolol; Multicenter Studies as Topic; Nifedipine; Randomized Controlled Trials as Topic; Verapamil

1997
Synthesis, calcium channel antagonist activity, and anticonvulsant activity of 3-ethyl 5-methyl 1,4-dihydro-2-[(2-hydroxyethoxy) methyl]-6-methyl-4-(2,3-dichlorophenyl)-3,5-pyridinedicarboxylate coupled to a 1-methyl-1,4-dihydropyridyl-3-carbonyl chemical
    Archiv der Pharmazie, 1999, Volume: 332, Issue:10

    Topics: Animals; Anticonvulsants; Calcium Channel Blockers; Dihydropyridines; Felodipine; Guinea Pigs; Mice; Muscle, Smooth; Nimodipine

1999
Normal-phase TLC separation of enantiomers of 1.4-dihydropyridine derivatives.
    Drug development and industrial pharmacy, 2001, Volume: 27, Issue:2

    Topics: Calcium Channel Blockers; Chromatography, Thin Layer; Dihydropyridines; Felodipine; Methanol; Nifedipine; Solvents; Stereoisomerism

2001
Effects of 3-chloro-phenyl-1,4-dihydropyridine derivatives on Trypanosome cruzi epimastigotes.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2000, Volume: 125, Issue:1

    Topics: Animals; Calcium Channel Blockers; Cell Movement; Dihydropyridines; Electrochemistry; Felodipine; Nicardipine; Oxidation-Reduction; Oxygen Consumption; Trypanocidal Agents; Trypanosoma cruzi

2000
Dihydropyridines are not substitutable without careful monitoring.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 2002, Volume: 92, Issue:8

    Topics: Adverse Drug Reaction Reporting Systems; Amlodipine; Antihypertensive Agents; Calcium Channel Blockers; Delayed-Action Preparations; Dihydropyridines; Felodipine; Humans; Nifedipine

2002
Dihydropyridines, felodipine, and PHARMAC.
    The New Zealand medical journal, 2005, Jul-15, Volume: 118, Issue:1218

    Topics: Angina Pectoris; Calcium Channel Blockers; Dihydropyridines; Drug Approval; Drug Industry; Felodipine; Humans; Hypertension; National Health Programs; New Zealand; Therapeutic Equivalency

2005
FEVER study: a trial further supporting the concept of a blood pressure-independent stroke protective effect by dihydropyridines.
    Journal of hypertension, 2006, Volume: 24, Issue:6

    Topics: Aged; Antihypertensive Agents; Blood Pressure; Dihydropyridines; Felodipine; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Stroke

2006
The effect of ionizing radiation of 1,4-dihydropyridine derivatives in the solid state.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2007, Volume: 67, Issue:1

    Topics: Calcium Channel Blockers; Dihydropyridines; Electron Spin Resonance Spectroscopy; Felodipine; Gamma Rays; Humans; Hypertension; Models, Molecular; Molecular Conformation; Myocardial Ischemia; Nifedipine; Nimodipine

2007
Calcium Antagonists Use and Its Association with Lower Urinary Tract Symptoms: A Cross-Sectional Study.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: Aged; Calcium Channel Blockers; Cross-Sectional Studies; Dihydropyridines; Felodipine; Female; Humans; Hypertension; Interviews as Topic; Logistic Models; Lower Urinary Tract Symptoms; Male; Middle Aged; Odds Ratio; Severity of Illness Index; Surveys and Questionnaires

2013
Photostabilization studies of antihypertensive 1,4-dihydropyridines using polymeric containers.
    International journal of pharmaceutics, 2016, May-30, Volume: 505, Issue:1-2

    Topics: Antihypertensive Agents; Dihydropyridines; Drug Packaging; Drug Stability; Drug Storage; Felodipine; Glass; Light; Pharmaceutical Solutions; Photolysis; Polyethylene Terephthalates; Polymers; Time Factors

2016
Long-term outcomes of lercanidipine versus other calcium channel blockers in newly diagnosed hypertension: a nationwide cohort study.
    Current medical research and opinion, 2017, Volume: 33, Issue:6

    Topics: Adolescent; Adult; Aged; Amlodipine; Blood Pressure; Calcium Channel Blockers; Cohort Studies; Dihydropyridines; Felodipine; Female; Humans; Hypertension; Male; Middle Aged; Retrospective Studies; Stroke; Taiwan; Young Adult

2017