felodipine and bergamottin

felodipine has been researched along with bergamottin in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bailey, DG; Bend, JR; Dresser, GK; Freeman, DJ; Kreeft, JH; Munoz, C1
Bailey, DG; Malhotra, S; Paine, MF; Watkins, PB1
Bailey, DG; Bend, JR; Dresser, GK1
Bailey, DG; CilliƩ, D; Cohen, L; Dijkstra, HP; Goosen, TC; He, K; Hollenberg, PF; Rheeders, M; Williams, JA; Woster, PM; Yu, C1

Trials

4 trial(s) available for felodipine and bergamottin

ArticleYear
Grapefruit-felodipine interaction: effect of unprocessed fruit and probable active ingredients.
    Clinical pharmacology and therapeutics, 2000, Volume: 68, Issue:5

    Topics: Administration, Oral; Adult; Antioxidants; Area Under Curve; Beverages; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Delayed-Action Preparations; Drug Interactions; Felodipine; Female; Flavanones; Flavonoids; Furocoumarins; Half-Life; Humans; Male; Mixed Function Oxygenases; Radiation-Sensitizing Agents

2000
Seville orange juice-felodipine interaction: comparison with dilute grapefruit juice and involvement of furocoumarins.
    Clinical pharmacology and therapeutics, 2001, Volume: 69, Issue:1

    Topics: 5-Methoxypsoralen; Administration, Oral; Adult; Antihypertensive Agents; Beverages; Biological Availability; Caco-2 Cells; Citrus; Cross-Over Studies; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; DNA, Complementary; Enzyme Activation; Enzyme Inhibitors; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Humans; Male; Methoxsalen; Mixed Function Oxygenases

2001
Bergamottin, lime juice, and red wine as inhibitors of cytochrome P450 3A4 activity: comparison with grapefruit juice.
    Clinical pharmacology and therapeutics, 2003, Volume: 73, Issue:6

    Topics: Adult; Area Under Curve; Beverages; Biotransformation; Calcium Channel Blockers; Citrus; Citrus paradisi; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Drug Interactions; Enzyme Inhibitors; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Half-Life; Humans; Male; Middle Aged; NADP; Radiation-Sensitizing Agents; Wine

2003
Bergamottin contribution to the grapefruit juice-felodipine interaction and disposition in humans.
    Clinical pharmacology and therapeutics, 2004, Volume: 76, Issue:6

    Topics: Adult; Area Under Curve; Biological Availability; Biotransformation; Calcium Channel Blockers; Capsules; Chromatography, High Pressure Liquid; Citrus; Cross-Over Studies; Delayed-Action Preparations; Felodipine; Female; Food-Drug Interactions; Furocoumarins; Humans; Male; Spectrophotometry, Ultraviolet

2004