Page last updated: 2024-08-24

fananserin and 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine

fananserin has been researched along with 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine in 3 studies

Research

Studies (3)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	2 (66.67)	29.6817
2010's	0 (0.00)	24.3611
2020's	1 (33.33)	2.80

Authors

Authors	Studies
Bentley, G; Blurton, P; Bristow, LJ; Burkamp, F; Castro, JL; Chapman, K; Cheng, SK; Clarkson, R; Cook, GP; Fletcher, SR; Hutson, PH; MacLeod, AM; Marwood, R; O'Connor, D; Patel, S; Shepheard, S; Spinks, D; Tudge, M; van Niel, MB	1
Giordanetto, F; Leach, AG; Zachariae, U	1
Chen, Z; Collier, T; Fu, H; Liang, SH; Rong, J; Zhou, J	1

Reviews

1 review(s) available for fananserin and 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine

Article	Year
Positron Emission Tomography (PET) Imaging Tracers for Serotonin Receptors. Journal of medicinal chemistry, 2022, 08-25, Volume: 65, Issue:16 Topics: Brain; Humans; Ligands; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin	2022

Other Studies

2 other study(ies) available for fananserin and 1-(2,4-difluorophenethyl)-4-(4-fluorophenylsulfonyl)piperidine

Article	Year
4-(Phenylsulfonyl)piperidines: novel, selective, and bioavailable 5-HT(2A) receptor antagonists. Journal of medicinal chemistry, 2002, Jan-17, Volume: 45, Issue:2 Topics: Administration, Oral; Animals; Benzamides; Biological Availability; Brain; Cation Transport Proteins; Cell Line; Cricetinae; DNA-Binding Proteins; Drug Evaluation, Preclinical; Electrocardiography; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Ferrets; Humans; In Vitro Techniques; Male; Microsomes, Liver; Nitriles; Piperidines; Potassium Channels; Potassium Channels, Voltage-Gated; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Structure-Activity Relationship; Sulfones; Trans-Activators; Transcriptional Regulator ERG	2002
Side chain flexibilities in the human ether-a-go-go related gene potassium channel (hERG) together with matched-pair binding studies suggest a new binding mode for channel blockers. Journal of medicinal chemistry, 2009, Jul-23, Volume: 52, Issue:14 Topics: Binding Sites; Ether-A-Go-Go Potassium Channels; Humans; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Potassium Channel Blockers; Protein Binding; Protein Conformation	2009

Article

Year

4-(Phenylsulfonyl)piperidines: novel, selective, and bioavailable 5-HT(2A) receptor antagonists.

Journal of medicinal chemistry, 2002, Jan-17, Volume: 45, Issue:2

Topics: Administration, Oral; Animals; Benzamides; Biological Availability; Brain; Cation Transport Proteins; Cell Line; Cricetinae; DNA-Binding Proteins; Drug Evaluation, Preclinical; Electrocardiography; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Ferrets; Humans; In Vitro Techniques; Male; Microsomes, Liver; Nitriles; Piperidines; Potassium Channels; Potassium Channels, Voltage-Gated; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Structure-Activity Relationship; Sulfones; Trans-Activators; Transcriptional Regulator ERG

2002

Side chain flexibilities in the human ether-a-go-go related gene potassium channel (hERG) together with matched-pair binding studies suggest a new binding mode for channel blockers.

Journal of medicinal chemistry, 2009, Jul-23, Volume: 52, Issue:14

Topics: Binding Sites; Ether-A-Go-Go Potassium Channels; Humans; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Potassium Channel Blockers; Protein Binding; Protein Conformation

2009