famotidine and histamine

famotidine has been researched along with histamine in 95 studies

Research

Studies (95)

TimeframeStudies, this research(%)All Research%
pre-199019 (20.00)18.7374
1990's38 (40.00)18.2507
2000's25 (26.32)29.6817
2010's8 (8.42)24.3611
2020's5 (5.26)2.80

Authors

AuthorsStudies
Berlin, R; Borow, KM; Ehler, D; Neumann, A1
Buschauer, A; Höer, A; Schwaner, I; Seifert, R1
Harada, T; Irifune, M; Matsunaga, T; Ogino, S1
Fukui, H; Inagaki, N; Kanamura, A; Kubo, A; Wada, H1
Krielaart, MJ; van Buuren, KJ; Veenstra, DM1
Inatomi, N; Nagaya, H; Satoh, H1
Aihara, H; Isobe, Y; Muramatsu, M; Otomo, S1
Fujii, K1
Fukui, H; Inagaki, N; Kanamura, A; Kondou, H; Koyama, Y; Wada, H1
Fujihara, A; Kamato, T; Miyata, K; Takeda, M1
Matsuki, T; Ohhashi, T1
Hannemann, H; Sewing, KF1
Yoshinaga, E1
Fujimoto, K; Fukagawa, K; Ookuma, K; Sakata, T; Shiraishi, T; Wada, H; Yoshimatsu, H1
Emami, S; Fagot, D; Gespach, C1
Itowi, N; Matsumura, K; Nakayama, T; Tsai, CL; Wada, H; Yamatodani, A1
Smith, JL1
Miederer, SE; Ruoff, HJ; Schepp, W; Wulfhekel, U1
Coruzzi, G; Noci, MT1
Bertaccini, G; Coruzzi, G1
Reeves, JJ; Stables, R1
Gillam, EM; Mason, SR; Reilly, PE1
Klotz, U; Kuhlmann, U; Machleidt, C; Mettang, T; Weber, J1
Chaya, M; De Heng, S; Hirooka, Y; Mitsuma, T; Nogimori, T; Ohtake, K1
Chaya, M; Mitsuma, T; Nogimori, T; Sun, DH1
Hirooka, Y; Mitsuma, T; Nogimori, T1
Kamada, T; Kawano, S; Sato, N; Takeda, M1
Maeno, H; Takagi, T; Takeda, M1
Harada, M; Maeno, H; Terai, M1
Fujiwara, T; Kohchi, M; Matsumoto, H; Miyoshi, A; Nakamura, M; Ohe, K1
Akuzawa, S; Ito, H; Kamato, T; Kobayashi-Uchida, A; Nagakura, Y; Nishida, A; Shishido, T; Takinami, Y; Yamano, M; Yuki, H1
Haruma, K; Kajiyama, G; Sumii, K; Sumii, M; Tari, A; Yamamoto, G1
Bado, A; Braquet, P; Laigneau, JP; Lewin, MJ; Moizo, L; Sobhani, I; Tarrade, T1
Kuriyama, K; Shimamoto, Y; Suga, K; Tomonaga, M; Yamaguchi, M1
Akaike, N; Munakata, M1
Fujihara, A; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H1
Haga, N; Itoh, Z; Matsunaga, Y; Mizumoto, A; Mizusawa, F; Sano, I; Ueki, S; Yamamoto, O1
Doi, T; Jayasekara, LA; Kurokawa, M; Machidori, H; Niki, N; Sakata, T; Yoshimatsu, H1
Chida, Y; Inaba, N; Ohnishi, H; Onodera, S; Shibata, M; Yamaura, T1
Bhasin, DK; Khosla, PP; Sachdev, A; Saha, N; Sankaranahyanan, A; Sharma, PL; Singh, K1
Ikarashi, Y; Kawano, O; Misaki, N; Ohba, S; Uchida, M1
Haruma, K; Kajiyama, G; Sachs, G; Sumii, K; Sumii, M; Tari, A; Walsh, JH; Wu, V; Yamamoto, G; Yonei, Y1
Haga, N; Itoh, Z; Matsunaga, Y; Mizumoto, A; Yamamoto, O1
Honda, K; Ito, H; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H1
Feng, CJ; Jahr, JS; Kang, B; Kaye, AD; Nossaman, BD; Paxtor, C1
Kaumann, AJ; Lynham, JA; Sanders, L1
Black, JW; Gerskowitch, VP; Harper, EA; Hull, RA; Roberts, SP; Shankley, NP; Watt, GF1
Akuzawa, S; Miyata, K; Nishida, A; Takemoto, Y; Uchida-Kobayashi, A1
Black, JW; Gerskowitch, VP; Hills, DM; Roberts, SP; Shankley, NP; Welsh, NJ1
Akuzawa, S; Ito, H; Miyake, A; Miyata, K; Nishida, A; Takemoto, Y; Takinami, Y; Yuki, H1
Linday, LA1
Bast, A; Bruinier, B; Hol, BE; Jansen, HM; Krouwels, FH; Lutter, R; Out, TA1
Arai, H; Inoie, M; Marubuchi, S1
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C1
Inagaki, N; Kawasaki, H; Musoh, K; Nagai, H; Nagao, M; Nakamura, N1
Ishiguro, I; Kobayashi, T; Ohta, Y1
Philippu, A; Prast, H; Tran, MH1
Attarzadeh, M; Farzin, D1
Hosoda, H; Inomata, N; Itoh, Z; Kangawa, K; Kojima, M; Masuda, Y; Ohnuma, N; Tanaka, S; Tanaka, T1
Itoh, T; Kajikuri, J; Suzuki, Y; Suzumori, K; Yamamoto, T1
Borrelli, F; Tavares, IA; Welsh, NJ1
Chi, L; Dileepan, KN; Li, Y; Stechschulte, DJ1
Hasebe, K; Horie, S; Komasaka, M; Watanabe, K; Yano, S1
Cohen, IL; DeCresce, R; Linday, LA; Shindledecker, R; Tsiouris, JA1
Hirotsu, S; Nakahara, M; Tomita, Y; Uchiwa, H; Yoshida, M1
Akerman, S; Goadsby, PJ; Kaube, H; Williamson, DJ1
Borrelli, F; Tavares, IA1
Jeong, JH; Lee, TS; Shin, CY; Sohn, UD; Song, HJ; Yun, MC1
Baroukh, B; Guez, D; Lesclous, P; Saffar, JL; Vignery, A1
Girish, K; Kole, PL; Nagappa, AN; Pandi, PV; Rahul Mishra, PK; Shanmukha, I1
Khuder, SA; Quan, WD; Walker, PR1
Eckman, JR; Wagner, MC; Wick, TM1
Baroukh, B; Gallina, S; Guez, D; Lesclous, P; Saffar, JL; Schramm, F1
Johno, Y; Miura, S; Ohno, S; Onouhi, T; Ro, S; Takayama, K; Tanaka, T; Yakabi, K1
Khan, UW; Rai, U1
Ancha, HR; Ceresa, BP; Damera, G; Harty, RF; Kurella, RR; Stewart, CA1
Kato, S; Kawashima, J; Yakabi, K1
Imatake, K; Matsui, T; Moriyama, M1
Aihara, E; Honda, M; Ito, Y; Kato, S; Mitsufuji, S; Okuda, S; Takeuchi, K; Yoshikawa, T1
Borodavkina, MV; Dolgikh, MP; Dugina, YL; Ogorodnikova, TV; Sergeeva, SA; Sorokina, IV; Tolstikova, TG; Zhukova, NA1
Asakura, M; Asanuma, H; Fujita, M; Kim, J; Kitakaze, M; Komamura, K; Minamino, T; Sanada, S; Sasaki, H; Sugimachi, M; Takahama, H; Takashima, S; Wakeno, M1
Chen, Z; He, G; Hu, J; Jia, M; Li, T; Lu, J; Luo, X; Ma, X; Meng, J; Ohtsu, H1
Kraus, MM; Philippu, A; Prast, H1
Akdis, CA; Barcik, W; Chassard, C; Ferstl, R; Frei, R; Konieczna, P; Lacroix, C; Lauener, RP; O'Mahony, L; Schiavi, E; Ziegler, M1
Chen, Z; Hou, WW; Lou, GD; Tang, YY; Wang, RR; Yu, J; Yue, JX; Zhang, SH1
Akdis, CA; Ferstl, R; Frei, R; Groeger, D; Jutel, M; Konieczna, P; OʼMahony, L; Perez, NR; Schiavi, E; Smolinska, S1
Allakonda, L; Appavoo, A; Nair, RR; Potnuri, AG; Saheera, S1
Nikfar, A; Rasouli, M1
Theoharides, TC1
Abdulai, SI; Chandra, S; Ishola, AA; Joshi, T; Pundir, H; Tijjani, H1
Amiri, S; Barikro, K; Khodakarami, S; Masoumi, K; Mohseni, M; Mohseni, MS; Raeisi, F; Raiesi, O; Raissi, V; Sharifan, Y1
Andersson, U; Brines, M; Chang, EH; Chavan, SS; George, SJ; Pavlov, VA; Silverman, HA; Thompson, DA; Tracey, KJ; Tsaava, T; Tynan, A; Yang, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Biagini, GA; Chandramohanadas, R; Darling, C; DeGrado, WF; Diamond, SL; Fisher, N; Greenbaum, DC; Jing, H; Jo, H; Lucumi, E; Napper, AD; Shone, AE; Ward, SA1

Reviews

5 review(s) available for famotidine and histamine

ArticleYear
[Physiological control mechanism of gastrointestinal motility].
    Nihon Heikatsukin Gakkai zasshi, 1990, Volume: 26, Issue:2

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Famotidine; Gastrins; Gastrointestinal Motility; Histamine; Histamine H2 Antagonists; Imidazoles; Norepinephrine; Octreotide; Tetrodotoxin

1990
Prophylaxis of symptoms of hyperhistaminemia after the treatment of acute promyelocytic leukemia with all-trans retinoic acid.
    Acta haematologica, 1994, Volume: 92, Issue:2

    Topics: Basophils; Chlorpheniramine; Drug Therapy, Combination; Famotidine; Histamine; Humans; Karyotyping; Leukemia, Promyelocytic, Acute; Leukocyte Count; Male; Middle Aged; Tretinoin

1994
Continuous infusion interleukin-2 and antihistamines in metastatic kidney cancer.
    Cancer biotherapy & radiopharmaceuticals, 2005, Volume: 20, Issue:5

    Topics: Adjuvants, Immunologic; Antineoplastic Agents; Cimetidine; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-2; Kidney Neoplasms; Neoplasm Metastasis; Ranitidine; Time Factors; Treatment Outcome

2005
Ghrelin and gastric acid secretion.
    World journal of gastroenterology, 2008, Nov-07, Volume: 14, Issue:41

    Topics: Animals; Famotidine; Gastric Acid; Gastric Mucosa; Gastrins; Ghrelin; Histamine; Histamine H2 Antagonists; Histamine Release; Histidine Decarboxylase; Humans; Stomach; Vagotomy; Vagus Nerve

2008
Therapeutic Status of Famotidine in COVID-19 Patients: A Review.
    Infectious disorders drug targets, 2022, Volume: 22, Issue:3

    Topics: COVID-19 Drug Treatment; Famotidine; Fever; Histamine; Humans; SARS-CoV-2

2022

Trials

4 trial(s) available for famotidine and histamine

ArticleYear
Influence of histamine receptors on basal left ventricular contractile tone in humans: assessment using the H2 receptor antagonist famotidine and the beta-adrenoceptor antagonist esmolol as pharmacologic probes.
    Journal of the American College of Cardiology, 1992, Volume: 19, Issue:6

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Double-Blind Method; Echocardiography, Doppler; Famotidine; Hemodynamics; Histamine; Humans; Middle Aged; Muscle Tonus; Myocardial Contraction; Propanolamines; Receptors, Histamine H2; Reference Values; Ventricular Function, Left

1992
Effect of H2-blockers, cimetidine and famotidine, on histamine nasal provocative test.
    ORL; journal for oto-rhino-laryngology and its related specialties, 1992, Volume: 54, Issue:3

    Topics: Adult; Cimetidine; Double-Blind Method; Famotidine; Histamine; Humans; Male; Middle Aged; Nasal Mucosa; Nasal Provocation Tests; Respiratory Hypersensitivity; Sneezing

1992
Clinical evaluation of the effect of omeprazole, cimetidine, famotidine and ranitidine on histamine induced cutaneous wheal and flare response.
    International journal of clinical pharmacology, therapy, and toxicology, 1993, Volume: 31, Issue:7

    Topics: Adult; Cimetidine; Drug Hypersensitivity; Dyspepsia; Famotidine; Female; Histamine; Histamine H2 Antagonists; Humans; India; Male; Middle Aged; Omeprazole; Ranitidine

1993
Famotidine treatment of children with autistic spectrum disorders: pilot research using single subject research design.
    Journal of neural transmission (Vienna, Austria : 1996), 2001, Volume: 108, Issue:5

    Topics: Autistic Disorder; Body Weight; Brain; Child; Child, Preschool; Dose-Response Relationship, Drug; Double-Blind Method; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Male; Pilot Projects; Receptors, Histamine H2; Research Design; Treatment Outcome

2001

Other Studies

86 other study(ies) available for famotidine and histamine

ArticleYear
Histamine increases cytosolic Ca2+ in HL-60 promyelocytes predominantly via H2 receptors with an unique agonist/antagonist profile and induces functional differentiation.
    Molecular pharmacology, 1992, Volume: 42, Issue:2

    Topics: Adenosine Triphosphate; Calcium; Cations; Cell Differentiation; Cyclic AMP; Cytosol; Dimaprit; Famotidine; Guanidines; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Ion Channels; Leukemia, Experimental; Leukemia, Promyelocytic, Acute; Phosphatidylinositols; Receptors, Histamine H2; Stimulation, Chemical; Thiourea; Tumor Cells, Cultured

1992
Histamine-induced cyclic AMP accumulation in type-1 and type-2 astrocytes in primary culture.
    European journal of pharmacology, 1991, Nov-13, Volume: 208, Issue:3

    Topics: Animals; Astrocytes; Cells, Cultured; Cyclic AMP; Famotidine; Histamine; Kinetics; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Stimulation, Chemical

1991
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
    Agents and actions, 1990, Volume: 31, Issue:1-2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea

1990
Differences in the antisecretory actions of the proton pump inhibitor AG-1749 (lansoprazole) and the histamine H2-receptor antagonist famotidine in rats and dogs.
    Japanese journal of pharmacology, 1991, Volume: 55, Issue:4

    Topics: 2-Pyridinylmethylsulfinylbenzimidazoles; Animals; Anti-Ulcer Agents; Bethanechol Compounds; Dogs; Famotidine; Female; Gastric Acid; Gastric Mucosa; Histamine; Hydrogen-Ion Concentration; Lansoprazole; Male; Omeprazole; Pentagastrin; Peptones; Pylorus; Rats; Rats, Inbred Strains

1991
H2-receptor antagonism by a novel compound IT-066 assessed from [14C]aminopyrine accumulation in rabbit parietal cells.
    European journal of pharmacology, 1990, Mar-27, Volume: 178, Issue:3

    Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Cimetidine; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Piperidines; Pyridines; Rabbits

1990
Histamine-induced inositol phosphate accumulation in type-2 astrocytes.
    Biochemical and biophysical research communications, 1991, Jun-14, Volume: 177, Issue:2

    Topics: Animals; Astrocytes; Cells, Cultured; Chlorpheniramine; Famotidine; Histamine; Inositol Phosphates; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine

1991
Cardiovascular and bronchial actions of famotidine in anesthetized dogs.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:11

    Topics: Airway Resistance; Anesthesia; Animals; Bronchi; Cimetidine; Dogs; Electrocardiography; Famotidine; Female; Halothane; Heart; Hemodynamics; Histamine; Male; Nitrous Oxide; Pentobarbital; Propranolol

1990
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 2

    Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation

1990
Interaction of ranitidine and famotidine with guinea pig-isolated parietal cells.
    Pharmacology, 1986, Volume: 33, Issue:5

    Topics: Animals; Famotidine; Guinea Pigs; Histamine; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Parietal Cells, Gastric; Ranitidine; Thiazoles

1986
[Mechanism of prevention of stress ulcer by vagotomy and famotidine: viewed from the transmucosal potential difference and histamine staining by a fluorescence histochemical method].
    Nihon geka hokan. Archiv fur japanische Chirurgie, 1986, Jul-01, Volume: 55, Issue:4

    Topics: Animals; Famotidine; Gastric Mucosa; Histamine; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Staining and Labeling; Stomach Ulcer; Stress, Physiological; Thiazoles; Vagotomy

1986
Neuronal histamine modulates feeding behavior through H1-receptor in rat hypothalamus.
    The American journal of physiology, 1989, Volume: 256, Issue:3 Pt 2

    Topics: Animals; Chlorpheniramine; Cimetidine; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Motor Activity; Neurons; Promethazine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Reference Values; Thiazoles

1989
Pharmacological control of the human gastric histamine H2 receptor by famotidine: comparison with H1, H2 and H3 receptor agonists and antagonists.
    European journal of clinical investigation, 1989, Volume: 19, Issue:1

    Topics: Adenylyl Cyclases; Cyclic AMP; Famotidine; Gastric Fundus; Histamine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Methylhistamines; Piperidines; Ranitidine; Receptors, Histamine; Stomach Neoplasms; Thiazoles; Triprolidine

1989
Effects of histamine on thermosensitive neurons in rat preoptic slice preparations.
    Neuroscience letters, 1989, Jul-31, Volume: 102, Issue:2-3

    Topics: Animals; Body Temperature Regulation; Dose-Response Relationship, Drug; Electrophysiology; Famotidine; Female; Histamine; Histamine H2 Antagonists; Neurons; Preoptic Area; Pyrilamine; Rats; Rats, Inbred Strains; Temperature

1989
Clinical pharmacology of famotidine.
    Digestion, 1985, Volume: 32 Suppl 1

    Topics: Animals; Cimetidine; Circadian Rhythm; Dogs; Dose-Response Relationship, Drug; Duodenal Ulcer; Famotidine; Food; Gastric Acid; Half-Life; Histamine; Histamine H2 Antagonists; Humans; Kinetics; Pentagastrin; Pepsin A; Prolactin; Rats; Tetragastrin; Thiazoles; Time Factors

1985
[Isolated human gastric mucosa cells--studies on physiologic and pharmacologic regulatory mechanisms].
    Klinische Wochenschrift, 1986, Jan-02, Volume: 64, Issue:1

    Topics: Adenylyl Cyclases; Adult; Aged; Aminopyrine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Humans; Intrinsic Factor; Microscopy, Electron; Middle Aged; Parietal Cells, Gastric; Prostaglandins; Ranitidine; Thiazoles

1986
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
    Bollettino della Societa italiana di biologia sperimentale, 1986, Sep-30, Volume: 62, Issue:9

    Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea

1986
Famotidine and ranitidine: any difference in the duration of action?
    Pharmacological research communications, 1987, Volume: 19, Issue:1

    Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors

1987
The antisecretory profile of action of the H2-receptor antagonists, famotidine, loxtidine, ranitidine and L-643,441 on the rat isolated gastric mucosa.
    Agents and actions, 1987, Volume: 20, Issue:1-2

    Topics: Animals; Bucladesine; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Methacholine Chloride; Methacholine Compounds; Ranitidine; Rats; Thiadiazoles; Thiazoles; Triazoles

1987
Differential inhibition of human liver phenacetin O-deethylation by histamine and four histamine H2-receptor antagonists.
    Xenobiotica; the fate of foreign compounds in biological systems, 1988, Volume: 18, Issue:4

    Topics: Binding Sites; Binding, Competitive; Catalysis; Chromatography, Thin Layer; Cimetidine; Cytochrome P-450 CYP1A2; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Imidazoles; Microsomes, Liver; Oxidation-Reduction; Oxidoreductases; Ranitidine; Thiazoles

1988
Cimetidine (but not ranitidine or famotidine) affects histamine determination.
    Lancet (London, England), 1988, Sep-24, Volume: 2, Issue:8613

    Topics: Cimetidine; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles

1988
Effect of histamine and its blockers on plasma beta-endorphin-like immunoreactivity in rats.
    Endocrinologia experimentalis, 1987, Volume: 21, Issue:2

    Topics: Animals; beta-Endorphin; Endorphins; Famotidine; Histamine; Hypothalamus; Male; Pituitary Gland; Pituitary Gland, Anterior; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles

1987
Effects of histamine and related compounds on thyrotropin secretion in rats.
    Hormone research, 1986, Volume: 23, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Famotidine; Histamine; Histidine; Male; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles; Thyrotropin; Thyrotropin-Releasing Hormone

1986
Effects of histamine and its blocker on thyrotropin releasing hormone release from rat adrenal gland in vitro.
    Endocrinologia experimentalis, 1987, Volume: 21, Issue:4

    Topics: Adrenal Glands; Animals; Famotidine; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles; Thyrotropin-Releasing Hormone

1987
Hemodynamics of the gastric mucosa and gastric ulceration in rats and in patients with gastric ulcer.
    Digestive diseases and sciences, 1986, Volume: 31, Issue:2 Suppl

    Topics: Animals; Blood Volume; Famotidine; Gastric Mucosa; Hemodynamics; Histamine; Humans; Microcirculation; Oxygen Consumption; Rats; Spectrophotometry; Stomach Ulcer; Stress, Physiological; Thiazoles

1986
Effect of a new potent H2-blocker, 3-]]]2-[(diaminomethylene)amino]-4-thiazolyl]methyl]-thio]-N2-sulfamoylpropionamidine (YM-11170) on gastric secretion induced by histamine and food in conscious dogs.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 256, Issue:1

    Topics: Animals; Cimetidine; Dogs; Famotidine; Food; Gastric Acid; Histamine; Histamine H2 Antagonists; Thiazoles

1982
Effect of a new potent H2-receptor antagonist 3[[[2-[(diaminomethylene)amino]-4-thiazolyl]methyl]thio]-N2- sulfamoylpropionamidine (YM-11170) on gastric mucosal histamine-sensitive adenylate cyclase from guinea pig.
    Biochemical pharmacology, 1983, May-15, Volume: 32, Issue:10

    Topics: Adenylyl Cyclases; Animals; Cimetidine; Dinoprostone; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Guinea Pigs; Hippocampus; Histamine; Histamine H2 Antagonists; Male; Prostaglandins E; Thiazoles

1983
Effect of H2-receptor antagonists, cimetidine and YM-11170, on serum gastrin levels in lumen-perfused rats.
    Digestive diseases and sciences, 1983, Volume: 28, Issue:11

    Topics: Animals; Cimetidine; Famotidine; Gastric Acid; Gastric Acidity Determination; Gastric Mucosa; Gastrins; Histamine; Infusions, Parenteral; Male; Perfusion; Rats; Rats, Inbred Strains; Thiazoles

1983
Gastrin receptor antagonist YM022 prevents hypersecretion after long-term acid suppression.
    The American journal of physiology, 1995, Volume: 269, Issue:5 Pt 1

    Topics: Animals; Benzodiazepines; Cell Count; Enterochromaffin Cells; Famotidine; Female; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Omeprazole; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Time Factors

1995
Famotidine, a histamine-2-receptor antagonist, inhibits the increase in rat gastric H+/K(+)-ATPase mRNA induced by intravenous infusion of gastrin 17 and histamine.
    Digestive diseases and sciences, 1995, Volume: 40, Issue:9

    Topics: Actins; Animals; Blotting, Northern; Famotidine; Gastrins; Gene Expression; H(+)-K(+)-Exchanging ATPase; Histamine; Histamine H2 Antagonists; Hormones; Infusions, Intravenous; Male; Parietal Cells, Gastric; Premedication; Rats; Rats, Wistar; Receptors, Histamine H2; RNA, Messenger

1995
Platelet-activating factor stimulates gastric acid secretion in isolated rabbit gastric glands.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Aminopyrine; Animals; Azepines; Biological Transport; Calcium; Carbachol; Dose-Response Relationship, Drug; Egtazic Acid; Famotidine; Fluorescent Dyes; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Kinetics; Male; Platelet Activating Factor; Rabbits; Thiazoles; Thienopyridines; Triazoles; Verapamil

1995
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
    The Journal of physiology, 1994, Oct-15, Volume: 480 ( Pt 2)

    Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine

1994
Antisecretory effects of a novel and long-lasting histamine H2-receptor antagonist, YM-14471, in rats and dogs.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:3

    Topics: Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H2 Antagonists; Infusions, Intravenous; Male; Omeprazole; Pyrimidinones; Rats; Rats, Wistar; Thiazoles

1993
Inhibition of phase III activity by acid in canine stomach.
    Regulatory peptides, 1994, Jun-16, Volume: 52, Issue:1

    Topics: Animals; Disease Models, Animal; Dogs; Duodenal Ulcer; Electrodes; Electrophysiology; Famotidine; Female; Gastric Acid; Gastrointestinal Motility; Histamine; Hydrogen-Ion Concentration; Male; Motilin; Muscle Contraction; Muscle, Smooth; Stomach Ulcer

1994
Hypothalamic neuronal histamine regulates feeding circadian rhythm in rats.
    Brain research, 1994, Apr-04, Volume: 641, Issue:2

    Topics: Animals; Cerebral Ventricles; Chlorpheniramine; Circadian Rhythm; Darkness; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histidine Decarboxylase; Hypothalamus; Infusions, Parenteral; Light; Male; Methylhistidines; Neurons; Rats; Rats, Wistar

1994
Gastric antisecretory effect of FRG-8813, a new histamine H2 receptor antagonist, in rats and dogs.
    European journal of pharmacology, 1993, Apr-28, Volume: 235, Issue:2-3

    Topics: Acetamides; Animals; Cimetidine; Dogs; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Ligation; Male; Perfusion; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley

1993
Effect of the novel histamine H2-antagonist 5,6-dimethyl-2-[4-[3-(1- piperidinomethyl)phenoxy]-(z)-2-butenylamino]-4(1H)-pyrimidine dihydrochloride on histamine-induced gastric acid secretion in Heidenhain pouch dogs.
    Arzneimittel-Forschung, 1993, Volume: 43, Issue:8

    Topics: Administration, Oral; Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Injections, Intravenous; Male; Piperidines; Pyrimidinones

1993
Effect of histamine on rat gastric H(+)-K(+)-ATPase alpha-subunit expression.
    The American journal of physiology, 1994, Volume: 266, Issue:3 Pt 1

    Topics: Animals; Famotidine; Gastric Mucosa; Gastrins; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; Male; Microscopy, Electron; Rats; Rats, Wistar; RNA, Messenger; Stomach

1994
Inhibition of phase III activity by acidifying stomach in vagally denervated and innervated dogs with gastric pouches.
    Gastroenterology, 1994, Volume: 106, Issue:6

    Topics: Acids; Animals; Denervation; Dogs; Duodenum; Famotidine; Gastrointestinal Motility; Gastroplasty; Histamine; Hydrogen-Ion Concentration; Infusions, Intravenous; Motilin; Reference Values; Stomach; Vagus Nerve

1994
Histamine H2-receptor plays only a minor role in histamine-induced wheal response in the squirrel monkey and guinea pig.
    Japanese journal of pharmacology, 1993, Volume: 63, Issue:1

    Topics: Animals; Chlorpheniramine; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Female; Guinea Pigs; Histamine; Histamine Agonists; Injections, Intradermal; Male; Pyridines; Ranitidine; Receptors, Histamine H2; Saimiri; Urticaria

1993
Analysis of responses to vancomycin in carotid blood flow in the male rat.
    Journal of medicine, 1995, Volume: 26, Issue:3-4

    Topics: Animals; Anti-Bacterial Agents; Blood Flow Velocity; Carotid Arteries; Diphenhydramine; Dose-Response Relationship, Drug; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Vancomycin; Vasodilation

1995
Chronic beta 1-adrenoceptor blockade sensitises the H1 and H2 receptor systems in human atrium: rôle of cyclic nucleotides.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:6

    Topics: Adrenergic beta-Antagonists; Arrhythmias, Cardiac; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Dose-Response Relationship, Drug; Famotidine; Female; Heart; Heart Atria; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Middle Aged; Myocardial Contraction; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Stimulation, Chemical

1996
Analysis of the variation in the action of L-365,260 at CCKB/gastrin receptors in rat, guinea-pig and mouse isolated gastric tissue assays.
    British journal of pharmacology, 1996, Volume: 118, Issue:7

    Topics: Animals; Benzodiazepinones; Binding, Competitive; Famotidine; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscle, Smooth; Pentagastrin; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Species Specificity; Stomach

1996
Comparative evaluation of the role of endogenous gastrin in basal acid secretion in conscious rats provided with chronic fistula and pylorus ligation.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:3

    Topics: Animals; Atropine; Benzodiazepines; Chronic Disease; Famotidine; Gastric Acid; Gastric Fistula; Gastrins; Histamine; Ligation; Male; Parasympathetic Nervous System; Pylorus; Rats; Rats, Sprague-Dawley

1996
Pharmacological analysis of the CCKB/gastrin receptors mediating pentagastrin-stimulated gastric acid secretion in the isolated stomach of the immature rat.
    British journal of pharmacology, 1996, Volume: 119, Issue:7

    Topics: Animals; Binding, Competitive; Enterochromaffin Cells; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Models, Biological; Pentagastrin; Rats; Rats, Wistar; Receptors, Cholecystokinin; Stimulation, Chemical

1996
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs.
    Digestive diseases and sciences, 1997, Volume: 42, Issue:4

    Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Devazepide; Dogs; Dose-Response Relationship, Drug; Eating; Famotidine; Gastric Acid; Histamine; Histamine H2 Antagonists; Hormone Antagonists; Male; Methacholine Chloride; Muscarinic Antagonists; Pentagastrin; Peptones; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Stomach

1997
Oral famotidine: a potential treatment for children with autism.
    Medical hypotheses, 1997, Volume: 48, Issue:5

    Topics: Administration, Oral; Adult; Animals; Autistic Disorder; Child; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Kidney; Models, Biological; Neurotransmitter Agents; Psychopharmacology; Safety; Schizophrenia

1997
Histamine affects interleukin-4, interleukin-5, and interferon-gamma production by human T cell clones from the airways and blood.
    American journal of respiratory cell and molecular biology, 1998, Volume: 18, Issue:5

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Asthma; Bronchoalveolar Lavage Fluid; Clone Cells; Cyclic AMP; Dinoprostone; Enzyme Activation; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Impromidine; Interferon-gamma; Interleukin-2; Interleukin-4; Interleukin-5; Lung; Methylhistamines; Piperidines; Pyridines; Ranitidine; T-Lymphocytes; Triprolidine

1998
Histamine H2-receptor antagonism of T-593, an anti-ulcer agent: studies on aminopyrine accumulation in isolated canine gastric mucosal cells.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:3

    Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Carbon Radioisotopes; Cholinergic Agonists; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Guanidines; Histamine; Histamine H2 Antagonists; Omeprazole; Pentagastrin; Pirenzepine; Ranitidine; Sulfones

1998
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles

1999
Participation of histamine H1 and H2 receptors in passive cutaneous anaphylaxis-induced scratching behavior in ICR mice.
    European journal of pharmacology, 1999, Feb-19, Volume: 367, Issue:2-3

    Topics: Animals; Anti-Allergic Agents; Behavior, Animal; Capillary Permeability; Cetirizine; Drug Interactions; Famotidine; Female; Free Radical Scavengers; Histamine; Histamine H2 Antagonists; Mice; Mice, Inbred ICR; p-Methoxy-N-methylphenethylamine; Passive Cutaneous Anaphylaxis; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Terfenadine; Time Factors

1999
Role of endogenous serotonin and histamine in the pathogenesis of gastric mucosal lesions in unanaesthetised rats with a single treatment of compound 48/80, a mast cell degranulator.
    Pharmacological research, 1999, Volume: 39, Issue:4

    Topics: Adrenergic Uptake Inhibitors; Amitriptyline; Animals; Cell Degranulation; Cimetidine; Cyproheptadine; Famotidine; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mast Cells; Methysergide; p-Methoxy-N-methylphenethylamine; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Stomach Ulcer; Tripelennamine

1999
Histaminergic H2 receptor ligands modulate acetylcholine release in the ventral striatum.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1999, Volume: 48 Suppl 1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Corpus Striatum; Dimaprit; Dopamine; Dopamine Agonists; Dopamine Antagonists; Famotidine; gamma-Aminobutyric Acid; Histamine; Histamine H2 Antagonists; Male; Neurons; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2

1999
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
    European journal of pharmacology, 2000, Sep-15, Volume: 404, Issue:1-2

    Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines

2000
Ghrelin stimulates gastric acid secretion and motility in rats.
    Biochemical and biophysical research communications, 2000, Oct-05, Volume: 276, Issue:3

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Ghrelin; Histamine; Histamine H2 Antagonists; Male; Peptide Hormones; Peptides; Peristalsis; Rats; Rats, Sprague-Dawley; Stomach; Vagotomy

2000
Modified histamine-induced NO-mediated relaxation in resistance arteries in pre-eclampsia.
    European journal of pharmacology, 2000, Dec-20, Volume: 410, Issue:1

    Topics: Adult; Arteries; Atrial Natriuretic Factor; Cyclic GMP; Down-Regulation; Endothelium, Vascular; Famotidine; Female; Histamine; Humans; Isometric Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroarginine; Pre-Eclampsia; Pregnancy; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Vascular Resistance; Vasodilation

2000
Inhibition of gastric acid secretion by nimesulide: a possible factor in its gastric tolerability.
    Clinical and experimental rheumatology, 2001, Volume: 19, Issue:1 Suppl 22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Indomethacin; Male; Mice; Mice, Inbred C57BL; Muscarine; Perfusion; Sulfonamides

2001
Histamine-induced production of interleukin-6 and interleukin-8 by human coronary artery endothelial cells is enhanced by endotoxin and tumor necrosis factor-alpha.
    Microvascular research, 2001, Volume: 61, Issue:3

    Topics: Cells, Cultured; Chemokine CCL2; Coronary Vessels; Diphenhydramine; Drug Synergism; Endothelium, Vascular; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-6; Interleukin-8; Lipopolysaccharides; NF-kappa B; Tumor Necrosis Factor-alpha

2001
Stimulatory effects of nitric oxide donors on gastric acid secretion in isolated mouse stomach.
    European journal of pharmacology, 2001, May-25, Volume: 420, Issue:2-3

    Topics: Animals; Bethanechol; Dose-Response Relationship, Drug; Electric Stimulation; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Mice; Nitric Oxide Donors; Nitroprusside; Stomach; Time Factors; Vagus Nerve; Vasodilator Agents

2001
Histamine is involved in ultraviolet B-induced pigmentation of guinea pig skin.
    The Journal of investigative dermatology, 2002, Volume: 118, Issue:2

    Topics: Animals; Cattle; Cells, Cultured; Drug Administration Schedule; Erythema; Famotidine; Guinea Pigs; Histamine; Histamine H2 Antagonists; Humans; Melanocytes; Radiation Injuries; Ranitidine; Skin Pigmentation; Ultraviolet Rays

2002
The role of histamine in dural vessel dilation.
    Brain research, 2002, Nov-22, Volume: 956, Issue:1

    Topics: Animals; Blood Pressure; Dura Mater; Electric Stimulation; Enzyme Inhibitors; Famotidine; Histamine; Histamine Antagonists; Male; Meningeal Arteries; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Time Factors; Vasodilation

2002
Effect of nimesulide on gastric acid secretion in the mouse stomach in vitro.
    Life sciences, 2003, Jan-10, Volume: 72, Issue:8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Dose-Response Relationship, Drug; Drug Combinations; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Indomethacin; Male; Mice; Mice, Inbred C57BL; Stomach; Sulfonamides

2003
Signaling via histamine receptors in cat duodenal smooth muscle cells.
    Molecules and cells, 2003, Oct-31, Volume: 16, Issue:2

    Topics: Alkaloids; Animals; Benzophenanthridines; Cats; Duodenum; Enzyme Inhibitors; Ethylmaleimide; Famotidine; Heparin; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Muscle Contraction; Myocytes, Smooth Muscle; Pertussis Toxin; Phenanthridines; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide Phospholipase C; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Signal Transduction

2003
Histamine participates in the early phase of trabecular bone loss in ovariectomized rats.
    Bone, 2004, Volume: 34, Issue:1

    Topics: Animals; Body Weight; Bone Resorption; Cimetidine; Famotidine; Female; Femur; Histamine; Immunohistochemistry; Kinetics; Mast Cells; Osteoclasts; Ovariectomy; Rats

2004
Role of surface activity in the biological actions of ranitidine and famotidine.
    Colloids and surfaces. B, Biointerfaces, 2004, Jun-01, Volume: 35, Issue:3-4

    Topics: Acetylcholine; Cholesterol; Famotidine; Histamine; Ions; Membranes, Artificial; Micelles; Molecular Structure; Permeability; Phosphatidylcholines; Ranitidine; Surface Properties

2004
Histamine increases sickle erythrocyte adherence to endothelium.
    British journal of haematology, 2006, Volume: 132, Issue:4

    Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules

2006
Histamine mediates osteoclastic resorption only during the acute phase of bone loss in ovariectomized rats.
    Experimental physiology, 2006, Volume: 91, Issue:3

    Topics: Animals; Bone Resorption; Famotidine; Female; Histamine; Histamine H2 Antagonists; Osteoclasts; Ovariectomy; Rats; Rats, Wistar; Sodium Chloride

2006
Histamine mediates the stimulatory action of ghrelin on acid secretion in rat stomach.
    Digestive diseases and sciences, 2006, Volume: 51, Issue:8

    Topics: Animals; Famotidine; Gastric Acid; Gastric Mucosa; Ghrelin; Growth Hormone; Histamine; Histamine H2 Antagonists; Histidine Decarboxylase; Male; Peptide Hormones; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stomach; Vagotomy

2006
Differential effects of histamine on Leydig cell and testicular macrophage activities in wall lizards: precise role of H1/H2 receptor subtypes.
    The Journal of endocrinology, 2007, Volume: 194, Issue:2

    Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Famotidine; Histamine; Histamine Antagonists; Leydig Cells; Lizards; Macrophages; Male; Phagocytosis; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Superoxides; Testosterone

2007
Histamine stimulation of MMP-1(collagenase-1) secretion and gene expression in gastric epithelial cells: role of EGFR transactivation and the MAP kinase pathway.
    The international journal of biochemistry & cell biology, 2007, Volume: 39, Issue:11

    Topics: Collagenases; Epithelial Cells; ErbB Receptors; Famotidine; Gene Expression Regulation, Enzymologic; Heparin-binding EGF-like Growth Factor; Histamine; Humans; Intercellular Signaling Peptides and Proteins; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Protein Kinase Inhibitors; Quinazolines; RNA, Small Interfering; Stomach; Time Factors; Transcriptional Activation; Tyrphostins

2007
The effect and mechanism of action of capsaicin on gastric acid output.
    Journal of gastroenterology, 2009, Volume: 44, Issue:5

    Topics: Animals; Benzodiazepines; Bethanechol; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastrins; Histamine; Histamine H2 Antagonists; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Agonists; Rats; Rats, Wistar; Somatostatin; Stomach; Vagus Nerve

2009
Phosphodiesterase isozymes involved in regulating acid secretion in the isolated mouse stomach.
    Journal of physiology and pharmacology : an official journal of the Polish Physiological Society, 2009, Volume: 60 Suppl 7

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; Isoenzymes; Male; Mice; Organ Specificity; Perfusion; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Rolipram; Stomach; Time Factors

2009
Antiulcer activity of preparations containing ultralow doses of antibodies in modeled chronic ulcer in rats.
    Bulletin of experimental biology and medicine, 2009, Volume: 148, Issue:3

    Topics: Acetates; Animals; Anti-Ulcer Agents; Antibodies; Famotidine; Gastrins; Histamine; Male; Rats; Rats, Wistar; Receptors, Histamine H2; Stomach Ulcer

2009
A histamine H₂ receptor blocker ameliorates development of heart failure in dogs independently of β-adrenergic receptor blockade.
    Basic research in cardiology, 2010, Volume: 105, Issue:6

    Topics: Adrenergic beta-Antagonists; Animals; Carbazoles; Cardiac Catheterization; Cardiac Pacing, Artificial; Cardiotonic Agents; Carvedilol; Cyclic AMP; Disease Models, Animal; Dogs; Echocardiography; Famotidine; Heart Failure; Histamine; Histamine H2 Antagonists; Immunohistochemistry; Mast Cells; Propanolamines; Pulmonary Wedge Pressure; Stroke Volume; Ventricular Function, Left

2010
Arrhythmogenic effect of sympathetic histamine in mouse hearts subjected to acute ischemia.
    Molecular medicine (Cambridge, Mass.), 2012, Feb-10, Volume: 18

    Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Atenolol; Famotidine; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; Histamine Release; Histidine Decarboxylase; Mice; Mice, Knockout; Myocardial Ischemia; Myocardium; Norepinephrine; Sympathetic Nervous System; Tachycardia, Ventricular; Ventricular Fibrillation

2012
Facilitation of short-term memory by histaminergic neurons in the nucleus accumbens is independent of cholinergic and glutamatergic transmission.
    British journal of pharmacology, 2013, Volume: 170, Issue:1

    Topics: Acetylcholine; Animals; Famotidine; Glutamic Acid; Histamine; Histamine Antagonists; Learning; Male; Memory, Short-Term; Neurons; Nucleus Accumbens; Piperidines; Rats; Rats, Sprague-Dawley; Time Factors

2013
Histamine receptor 2 is a key influence in immune responses to intestinal histamine-secreting microbes.
    The Journal of allergy and clinical immunology, 2014, Volume: 134, Issue:3

    Topics: Animals; Cell Line; Coculture Techniques; Cytokines; Famotidine; Histamine; Humans; Immunity; Immunomodulation; Intestines; Lactobacillus; Mice; Mice, Inbred Strains; Mice, Knockout; Microbiota; NF-kappa B; Receptors, Histamine H2

2014
Histamine upregulates Nav1.8 expression in primary afferent neurons via H2 receptors: involvement in neuropathic pain.
    CNS neuroscience & therapeutics, 2014, Volume: 20, Issue:10

    Topics: Animals; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Famotidine; Ganglia, Spinal; Histamine; Histamine Agonists; Histamine H2 Antagonists; Hyperalgesia; Male; NAV1.8 Voltage-Gated Sodium Channel; Pain Measurement; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; Sciatica; Sensory Receptor Cells; Up-Regulation

2014
Histamine Receptor 2 is Required to Suppress Innate Immune Responses to Bacterial Ligands in Patients with Inflammatory Bowel Disease.
    Inflammatory bowel diseases, 2016, Volume: 22, Issue:7

    Topics: Adult; Animals; Case-Control Studies; Cells, Cultured; Colitis, Ulcerative; Crohn Disease; Cytokines; Disease Models, Animal; Down-Regulation; Famotidine; Female; Flagellin; Gene Expression; Histamine; Histamine H2 Antagonists; Humans; Immunity, Innate; Intestinal Mucosa; Ligands; Lipopolysaccharides; Lipoproteins; Lymphocyte Count; Male; Mice; Mice, SCID; Middle Aged; Monocytes; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H4; Severity of Illness Index; Th1 Cells; Th17 Cells; Toll-Like Receptors; Weight Loss; Young Adult

2016
Association of histamine with hypertension-induced cardiac remodeling and reduction of hypertrophy with the histamine-2-receptor antagonist famotidine compared with the beta-blocker metoprolol.
    Hypertension research : official journal of the Japanese Society of Hypertension, 2018, Volume: 41, Issue:12

    Topics: Adrenergic beta-1 Receptor Antagonists; Age Factors; Animals; Blood Pressure; Cardiomegaly; Famotidine; Histamine; Histamine H2 Antagonists; Hypertension; Male; Metoprolol; Myocardium; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H2; Ventricular Remodeling

2018
Hypolipemic effects of histamine is due to inhibition of VLDL secretion from the liver: involvement of both H1 and H2-receptors.
    Archives of physiology and biochemistry, 2022, Volume: 128, Issue:6

    Topics: Animals; Cetirizine; Cholesterol; Famotidine; Histamine; Histamine Agonists; Lipids; Liver; Male; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Triglycerides

2022
Potential association of mast cells with coronavirus disease 2019.
    Annals of allergy, asthma & immunology : official publication of the American College of Allergy, Asthma, & Immunology, 2021, Volume: 126, Issue:3

    Topics: Cell Communication; Cholecalciferol; COVID-19; COVID-19 Drug Treatment; Cromolyn Sodium; Cyproheptadine; Cytokines; Famotidine; Histamine; Histamine Antagonists; Humans; Lung; Luteolin; Macrophages; Mast Cells; SARS-CoV-2; Severity of Illness Index; Substance P

2021
Molecular basis for the repurposing of histamine H2-receptor antagonist to treat COVID-19.
    Journal of biomolecular structure & dynamics, 2022, Volume: 40, Issue:13

    Topics: Cimetidine; COVID-19 Drug Treatment; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Molecular Docking Simulation

2022
Famotidine activates the vagus nerve inflammatory reflex to attenuate cytokine storm.
    Molecular medicine (Cambridge, Mass.), 2022, 05-16, Volume: 28, Issue:1

    Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Anti-Inflammatory Agents; COVID-19; Cytokine Release Syndrome; Famotidine; Histamine; Histamine H2 Antagonists; Lipopolysaccharides; Mice; Reflex; Vagus Nerve

2022
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay.
    Antimicrobial agents and chemotherapy, 2010, Volume: 54, Issue:9

    Topics: Animals; Antimalarials; Drug Resistance, Multiple; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum

2010