famotidine has been researched along with histamine in 95 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 19 (20.00) | 18.7374 |
1990's | 38 (40.00) | 18.2507 |
2000's | 25 (26.32) | 29.6817 |
2010's | 8 (8.42) | 24.3611 |
2020's | 5 (5.26) | 2.80 |
Authors | Studies |
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Berlin, R; Borow, KM; Ehler, D; Neumann, A | 1 |
Buschauer, A; Höer, A; Schwaner, I; Seifert, R | 1 |
Harada, T; Irifune, M; Matsunaga, T; Ogino, S | 1 |
Fukui, H; Inagaki, N; Kanamura, A; Kubo, A; Wada, H | 1 |
Krielaart, MJ; van Buuren, KJ; Veenstra, DM | 1 |
Inatomi, N; Nagaya, H; Satoh, H | 1 |
Aihara, H; Isobe, Y; Muramatsu, M; Otomo, S | 1 |
Fujii, K | 1 |
Fukui, H; Inagaki, N; Kanamura, A; Kondou, H; Koyama, Y; Wada, H | 1 |
Fujihara, A; Kamato, T; Miyata, K; Takeda, M | 1 |
Matsuki, T; Ohhashi, T | 1 |
Hannemann, H; Sewing, KF | 1 |
Yoshinaga, E | 1 |
Fujimoto, K; Fukagawa, K; Ookuma, K; Sakata, T; Shiraishi, T; Wada, H; Yoshimatsu, H | 1 |
Emami, S; Fagot, D; Gespach, C | 1 |
Itowi, N; Matsumura, K; Nakayama, T; Tsai, CL; Wada, H; Yamatodani, A | 1 |
Smith, JL | 1 |
Miederer, SE; Ruoff, HJ; Schepp, W; Wulfhekel, U | 1 |
Coruzzi, G; Noci, MT | 1 |
Bertaccini, G; Coruzzi, G | 1 |
Reeves, JJ; Stables, R | 1 |
Gillam, EM; Mason, SR; Reilly, PE | 1 |
Klotz, U; Kuhlmann, U; Machleidt, C; Mettang, T; Weber, J | 1 |
Chaya, M; De Heng, S; Hirooka, Y; Mitsuma, T; Nogimori, T; Ohtake, K | 1 |
Chaya, M; Mitsuma, T; Nogimori, T; Sun, DH | 1 |
Hirooka, Y; Mitsuma, T; Nogimori, T | 1 |
Kamada, T; Kawano, S; Sato, N; Takeda, M | 1 |
Maeno, H; Takagi, T; Takeda, M | 1 |
Harada, M; Maeno, H; Terai, M | 1 |
Fujiwara, T; Kohchi, M; Matsumoto, H; Miyoshi, A; Nakamura, M; Ohe, K | 1 |
Akuzawa, S; Ito, H; Kamato, T; Kobayashi-Uchida, A; Nagakura, Y; Nishida, A; Shishido, T; Takinami, Y; Yamano, M; Yuki, H | 1 |
Haruma, K; Kajiyama, G; Sumii, K; Sumii, M; Tari, A; Yamamoto, G | 1 |
Bado, A; Braquet, P; Laigneau, JP; Lewin, MJ; Moizo, L; Sobhani, I; Tarrade, T | 1 |
Kuriyama, K; Shimamoto, Y; Suga, K; Tomonaga, M; Yamaguchi, M | 1 |
Akaike, N; Munakata, M | 1 |
Fujihara, A; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H | 1 |
Haga, N; Itoh, Z; Matsunaga, Y; Mizumoto, A; Mizusawa, F; Sano, I; Ueki, S; Yamamoto, O | 1 |
Doi, T; Jayasekara, LA; Kurokawa, M; Machidori, H; Niki, N; Sakata, T; Yoshimatsu, H | 1 |
Chida, Y; Inaba, N; Ohnishi, H; Onodera, S; Shibata, M; Yamaura, T | 1 |
Bhasin, DK; Khosla, PP; Sachdev, A; Saha, N; Sankaranahyanan, A; Sharma, PL; Singh, K | 1 |
Ikarashi, Y; Kawano, O; Misaki, N; Ohba, S; Uchida, M | 1 |
Haruma, K; Kajiyama, G; Sachs, G; Sumii, K; Sumii, M; Tari, A; Walsh, JH; Wu, V; Yamamoto, G; Yonei, Y | 1 |
Haga, N; Itoh, Z; Matsunaga, Y; Mizumoto, A; Yamamoto, O | 1 |
Honda, K; Ito, H; Kamato, T; Miyata, K; Nishida, A; Takeda, M; Yuki, H | 1 |
Feng, CJ; Jahr, JS; Kang, B; Kaye, AD; Nossaman, BD; Paxtor, C | 1 |
Kaumann, AJ; Lynham, JA; Sanders, L | 1 |
Black, JW; Gerskowitch, VP; Harper, EA; Hull, RA; Roberts, SP; Shankley, NP; Watt, GF | 1 |
Akuzawa, S; Miyata, K; Nishida, A; Takemoto, Y; Uchida-Kobayashi, A | 1 |
Black, JW; Gerskowitch, VP; Hills, DM; Roberts, SP; Shankley, NP; Welsh, NJ | 1 |
Akuzawa, S; Ito, H; Miyake, A; Miyata, K; Nishida, A; Takemoto, Y; Takinami, Y; Yuki, H | 1 |
Linday, LA | 1 |
Bast, A; Bruinier, B; Hol, BE; Jansen, HM; Krouwels, FH; Lutter, R; Out, TA | 1 |
Arai, H; Inoie, M; Marubuchi, S | 1 |
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C | 1 |
Inagaki, N; Kawasaki, H; Musoh, K; Nagai, H; Nagao, M; Nakamura, N | 1 |
Ishiguro, I; Kobayashi, T; Ohta, Y | 1 |
Philippu, A; Prast, H; Tran, MH | 1 |
Attarzadeh, M; Farzin, D | 1 |
Hosoda, H; Inomata, N; Itoh, Z; Kangawa, K; Kojima, M; Masuda, Y; Ohnuma, N; Tanaka, S; Tanaka, T | 1 |
Itoh, T; Kajikuri, J; Suzuki, Y; Suzumori, K; Yamamoto, T | 1 |
Borrelli, F; Tavares, IA; Welsh, NJ | 1 |
Chi, L; Dileepan, KN; Li, Y; Stechschulte, DJ | 1 |
Hasebe, K; Horie, S; Komasaka, M; Watanabe, K; Yano, S | 1 |
Cohen, IL; DeCresce, R; Linday, LA; Shindledecker, R; Tsiouris, JA | 1 |
Hirotsu, S; Nakahara, M; Tomita, Y; Uchiwa, H; Yoshida, M | 1 |
Akerman, S; Goadsby, PJ; Kaube, H; Williamson, DJ | 1 |
Borrelli, F; Tavares, IA | 1 |
Jeong, JH; Lee, TS; Shin, CY; Sohn, UD; Song, HJ; Yun, MC | 1 |
Baroukh, B; Guez, D; Lesclous, P; Saffar, JL; Vignery, A | 1 |
Girish, K; Kole, PL; Nagappa, AN; Pandi, PV; Rahul Mishra, PK; Shanmukha, I | 1 |
Khuder, SA; Quan, WD; Walker, PR | 1 |
Eckman, JR; Wagner, MC; Wick, TM | 1 |
Baroukh, B; Gallina, S; Guez, D; Lesclous, P; Saffar, JL; Schramm, F | 1 |
Johno, Y; Miura, S; Ohno, S; Onouhi, T; Ro, S; Takayama, K; Tanaka, T; Yakabi, K | 1 |
Khan, UW; Rai, U | 1 |
Ancha, HR; Ceresa, BP; Damera, G; Harty, RF; Kurella, RR; Stewart, CA | 1 |
Kato, S; Kawashima, J; Yakabi, K | 1 |
Imatake, K; Matsui, T; Moriyama, M | 1 |
Aihara, E; Honda, M; Ito, Y; Kato, S; Mitsufuji, S; Okuda, S; Takeuchi, K; Yoshikawa, T | 1 |
Borodavkina, MV; Dolgikh, MP; Dugina, YL; Ogorodnikova, TV; Sergeeva, SA; Sorokina, IV; Tolstikova, TG; Zhukova, NA | 1 |
Asakura, M; Asanuma, H; Fujita, M; Kim, J; Kitakaze, M; Komamura, K; Minamino, T; Sanada, S; Sasaki, H; Sugimachi, M; Takahama, H; Takashima, S; Wakeno, M | 1 |
Chen, Z; He, G; Hu, J; Jia, M; Li, T; Lu, J; Luo, X; Ma, X; Meng, J; Ohtsu, H | 1 |
Kraus, MM; Philippu, A; Prast, H | 1 |
Akdis, CA; Barcik, W; Chassard, C; Ferstl, R; Frei, R; Konieczna, P; Lacroix, C; Lauener, RP; O'Mahony, L; Schiavi, E; Ziegler, M | 1 |
Chen, Z; Hou, WW; Lou, GD; Tang, YY; Wang, RR; Yu, J; Yue, JX; Zhang, SH | 1 |
Akdis, CA; Ferstl, R; Frei, R; Groeger, D; Jutel, M; Konieczna, P; OʼMahony, L; Perez, NR; Schiavi, E; Smolinska, S | 1 |
Allakonda, L; Appavoo, A; Nair, RR; Potnuri, AG; Saheera, S | 1 |
Nikfar, A; Rasouli, M | 1 |
Theoharides, TC | 1 |
Abdulai, SI; Chandra, S; Ishola, AA; Joshi, T; Pundir, H; Tijjani, H | 1 |
Amiri, S; Barikro, K; Khodakarami, S; Masoumi, K; Mohseni, M; Mohseni, MS; Raeisi, F; Raiesi, O; Raissi, V; Sharifan, Y | 1 |
Andersson, U; Brines, M; Chang, EH; Chavan, SS; George, SJ; Pavlov, VA; Silverman, HA; Thompson, DA; Tracey, KJ; Tsaava, T; Tynan, A; Yang, H | 1 |
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM | 1 |
Biagini, GA; Chandramohanadas, R; Darling, C; DeGrado, WF; Diamond, SL; Fisher, N; Greenbaum, DC; Jing, H; Jo, H; Lucumi, E; Napper, AD; Shone, AE; Ward, SA | 1 |
5 review(s) available for famotidine and histamine
Article | Year |
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[Physiological control mechanism of gastrointestinal motility].
Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Famotidine; Gastrins; Gastrointestinal Motility; Histamine; Histamine H2 Antagonists; Imidazoles; Norepinephrine; Octreotide; Tetrodotoxin | 1990 |
Prophylaxis of symptoms of hyperhistaminemia after the treatment of acute promyelocytic leukemia with all-trans retinoic acid.
Topics: Basophils; Chlorpheniramine; Drug Therapy, Combination; Famotidine; Histamine; Humans; Karyotyping; Leukemia, Promyelocytic, Acute; Leukocyte Count; Male; Middle Aged; Tretinoin | 1994 |
Continuous infusion interleukin-2 and antihistamines in metastatic kidney cancer.
Topics: Adjuvants, Immunologic; Antineoplastic Agents; Cimetidine; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-2; Kidney Neoplasms; Neoplasm Metastasis; Ranitidine; Time Factors; Treatment Outcome | 2005 |
Ghrelin and gastric acid secretion.
Topics: Animals; Famotidine; Gastric Acid; Gastric Mucosa; Gastrins; Ghrelin; Histamine; Histamine H2 Antagonists; Histamine Release; Histidine Decarboxylase; Humans; Stomach; Vagotomy; Vagus Nerve | 2008 |
Therapeutic Status of Famotidine in COVID-19 Patients: A Review.
Topics: COVID-19 Drug Treatment; Famotidine; Fever; Histamine; Humans; SARS-CoV-2 | 2022 |
4 trial(s) available for famotidine and histamine
Article | Year |
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Influence of histamine receptors on basal left ventricular contractile tone in humans: assessment using the H2 receptor antagonist famotidine and the beta-adrenoceptor antagonist esmolol as pharmacologic probes.
Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Double-Blind Method; Echocardiography, Doppler; Famotidine; Hemodynamics; Histamine; Humans; Middle Aged; Muscle Tonus; Myocardial Contraction; Propanolamines; Receptors, Histamine H2; Reference Values; Ventricular Function, Left | 1992 |
Effect of H2-blockers, cimetidine and famotidine, on histamine nasal provocative test.
Topics: Adult; Cimetidine; Double-Blind Method; Famotidine; Histamine; Humans; Male; Middle Aged; Nasal Mucosa; Nasal Provocation Tests; Respiratory Hypersensitivity; Sneezing | 1992 |
Clinical evaluation of the effect of omeprazole, cimetidine, famotidine and ranitidine on histamine induced cutaneous wheal and flare response.
Topics: Adult; Cimetidine; Drug Hypersensitivity; Dyspepsia; Famotidine; Female; Histamine; Histamine H2 Antagonists; Humans; India; Male; Middle Aged; Omeprazole; Ranitidine | 1993 |
Famotidine treatment of children with autistic spectrum disorders: pilot research using single subject research design.
Topics: Autistic Disorder; Body Weight; Brain; Child; Child, Preschool; Dose-Response Relationship, Drug; Double-Blind Method; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Male; Pilot Projects; Receptors, Histamine H2; Research Design; Treatment Outcome | 2001 |
86 other study(ies) available for famotidine and histamine
Article | Year |
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Histamine increases cytosolic Ca2+ in HL-60 promyelocytes predominantly via H2 receptors with an unique agonist/antagonist profile and induces functional differentiation.
Topics: Adenosine Triphosphate; Calcium; Cations; Cell Differentiation; Cyclic AMP; Cytosol; Dimaprit; Famotidine; Guanidines; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Ion Channels; Leukemia, Experimental; Leukemia, Promyelocytic, Acute; Phosphatidylinositols; Receptors, Histamine H2; Stimulation, Chemical; Thiourea; Tumor Cells, Cultured | 1992 |
Histamine-induced cyclic AMP accumulation in type-1 and type-2 astrocytes in primary culture.
Topics: Animals; Astrocytes; Cells, Cultured; Cyclic AMP; Famotidine; Histamine; Kinetics; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Stimulation, Chemical | 1991 |
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea | 1990 |
Differences in the antisecretory actions of the proton pump inhibitor AG-1749 (lansoprazole) and the histamine H2-receptor antagonist famotidine in rats and dogs.
Topics: 2-Pyridinylmethylsulfinylbenzimidazoles; Animals; Anti-Ulcer Agents; Bethanechol Compounds; Dogs; Famotidine; Female; Gastric Acid; Gastric Mucosa; Histamine; Hydrogen-Ion Concentration; Lansoprazole; Male; Omeprazole; Pentagastrin; Peptones; Pylorus; Rats; Rats, Inbred Strains | 1991 |
H2-receptor antagonism by a novel compound IT-066 assessed from [14C]aminopyrine accumulation in rabbit parietal cells.
Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Cimetidine; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Piperidines; Pyridines; Rabbits | 1990 |
Histamine-induced inositol phosphate accumulation in type-2 astrocytes.
Topics: Animals; Astrocytes; Cells, Cultured; Chlorpheniramine; Famotidine; Histamine; Inositol Phosphates; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine | 1991 |
Cardiovascular and bronchial actions of famotidine in anesthetized dogs.
Topics: Airway Resistance; Anesthesia; Animals; Bronchi; Cimetidine; Dogs; Electrocardiography; Famotidine; Female; Halothane; Heart; Hemodynamics; Histamine; Male; Nitrous Oxide; Pentobarbital; Propranolol | 1990 |
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation | 1990 |
Interaction of ranitidine and famotidine with guinea pig-isolated parietal cells.
Topics: Animals; Famotidine; Guinea Pigs; Histamine; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Parietal Cells, Gastric; Ranitidine; Thiazoles | 1986 |
[Mechanism of prevention of stress ulcer by vagotomy and famotidine: viewed from the transmucosal potential difference and histamine staining by a fluorescence histochemical method].
Topics: Animals; Famotidine; Gastric Mucosa; Histamine; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Staining and Labeling; Stomach Ulcer; Stress, Physiological; Thiazoles; Vagotomy | 1986 |
Neuronal histamine modulates feeding behavior through H1-receptor in rat hypothalamus.
Topics: Animals; Chlorpheniramine; Cimetidine; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Motor Activity; Neurons; Promethazine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Reference Values; Thiazoles | 1989 |
Pharmacological control of the human gastric histamine H2 receptor by famotidine: comparison with H1, H2 and H3 receptor agonists and antagonists.
Topics: Adenylyl Cyclases; Cyclic AMP; Famotidine; Gastric Fundus; Histamine; Histamine H2 Antagonists; Humans; In Vitro Techniques; Methylhistamines; Piperidines; Ranitidine; Receptors, Histamine; Stomach Neoplasms; Thiazoles; Triprolidine | 1989 |
Effects of histamine on thermosensitive neurons in rat preoptic slice preparations.
Topics: Animals; Body Temperature Regulation; Dose-Response Relationship, Drug; Electrophysiology; Famotidine; Female; Histamine; Histamine H2 Antagonists; Neurons; Preoptic Area; Pyrilamine; Rats; Rats, Inbred Strains; Temperature | 1989 |
Clinical pharmacology of famotidine.
Topics: Animals; Cimetidine; Circadian Rhythm; Dogs; Dose-Response Relationship, Drug; Duodenal Ulcer; Famotidine; Food; Gastric Acid; Half-Life; Histamine; Histamine H2 Antagonists; Humans; Kinetics; Pentagastrin; Pepsin A; Prolactin; Rats; Tetragastrin; Thiazoles; Time Factors | 1985 |
[Isolated human gastric mucosa cells--studies on physiologic and pharmacologic regulatory mechanisms].
Topics: Adenylyl Cyclases; Adult; Aged; Aminopyrine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Humans; Intrinsic Factor; Microscopy, Electron; Middle Aged; Parietal Cells, Gastric; Prostaglandins; Ranitidine; Thiazoles | 1986 |
[Effect of a new H2 receptor antagonist, famotidine, on gastric secretion].
Topics: Animals; Cats; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea | 1986 |
Famotidine and ranitidine: any difference in the duration of action?
Topics: Animals; Cats; Dimaprit; Famotidine; Gastric Acid; Gastric Juice; Histamine; Histamine H2 Antagonists; Ranitidine; Rats; Thiazoles; Thiourea; Time Factors | 1987 |
The antisecretory profile of action of the H2-receptor antagonists, famotidine, loxtidine, ranitidine and L-643,441 on the rat isolated gastric mucosa.
Topics: Animals; Bucladesine; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Methacholine Chloride; Methacholine Compounds; Ranitidine; Rats; Thiadiazoles; Thiazoles; Triazoles | 1987 |
Differential inhibition of human liver phenacetin O-deethylation by histamine and four histamine H2-receptor antagonists.
Topics: Binding Sites; Binding, Competitive; Catalysis; Chromatography, Thin Layer; Cimetidine; Cytochrome P-450 CYP1A2; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Imidazoles; Microsomes, Liver; Oxidation-Reduction; Oxidoreductases; Ranitidine; Thiazoles | 1988 |
Cimetidine (but not ranitidine or famotidine) affects histamine determination.
Topics: Cimetidine; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Ranitidine; Thiazoles | 1988 |
Effect of histamine and its blockers on plasma beta-endorphin-like immunoreactivity in rats.
Topics: Animals; beta-Endorphin; Endorphins; Famotidine; Histamine; Hypothalamus; Male; Pituitary Gland; Pituitary Gland, Anterior; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles | 1987 |
Effects of histamine and related compounds on thyrotropin secretion in rats.
Topics: Animals; Dose-Response Relationship, Drug; Famotidine; Histamine; Histidine; Male; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles; Thyrotropin; Thyrotropin-Releasing Hormone | 1986 |
Effects of histamine and its blocker on thyrotropin releasing hormone release from rat adrenal gland in vitro.
Topics: Adrenal Glands; Animals; Famotidine; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pyrilamine; Rats; Rats, Inbred Strains; Thiazoles; Thyrotropin-Releasing Hormone | 1987 |
Hemodynamics of the gastric mucosa and gastric ulceration in rats and in patients with gastric ulcer.
Topics: Animals; Blood Volume; Famotidine; Gastric Mucosa; Hemodynamics; Histamine; Humans; Microcirculation; Oxygen Consumption; Rats; Spectrophotometry; Stomach Ulcer; Stress, Physiological; Thiazoles | 1986 |
Effect of a new potent H2-blocker, 3-]]]2-[(diaminomethylene)amino]-4-thiazolyl]methyl]-thio]-N2-sulfamoylpropionamidine (YM-11170) on gastric secretion induced by histamine and food in conscious dogs.
Topics: Animals; Cimetidine; Dogs; Famotidine; Food; Gastric Acid; Histamine; Histamine H2 Antagonists; Thiazoles | 1982 |
Effect of a new potent H2-receptor antagonist 3[[[2-[(diaminomethylene)amino]-4-thiazolyl]methyl]thio]-N2- sulfamoylpropionamidine (YM-11170) on gastric mucosal histamine-sensitive adenylate cyclase from guinea pig.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Dinoprostone; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Guinea Pigs; Hippocampus; Histamine; Histamine H2 Antagonists; Male; Prostaglandins E; Thiazoles | 1983 |
Effect of H2-receptor antagonists, cimetidine and YM-11170, on serum gastrin levels in lumen-perfused rats.
Topics: Animals; Cimetidine; Famotidine; Gastric Acid; Gastric Acidity Determination; Gastric Mucosa; Gastrins; Histamine; Infusions, Parenteral; Male; Perfusion; Rats; Rats, Inbred Strains; Thiazoles | 1983 |
Gastrin receptor antagonist YM022 prevents hypersecretion after long-term acid suppression.
Topics: Animals; Benzodiazepines; Cell Count; Enterochromaffin Cells; Famotidine; Female; Gastric Acid; Gastric Mucosa; Gastrins; Histamine; Histidine Decarboxylase; Omeprazole; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Time Factors | 1995 |
Famotidine, a histamine-2-receptor antagonist, inhibits the increase in rat gastric H+/K(+)-ATPase mRNA induced by intravenous infusion of gastrin 17 and histamine.
Topics: Actins; Animals; Blotting, Northern; Famotidine; Gastrins; Gene Expression; H(+)-K(+)-Exchanging ATPase; Histamine; Histamine H2 Antagonists; Hormones; Infusions, Intravenous; Male; Parietal Cells, Gastric; Premedication; Rats; Rats, Wistar; Receptors, Histamine H2; RNA, Messenger | 1995 |
Platelet-activating factor stimulates gastric acid secretion in isolated rabbit gastric glands.
Topics: Aminopyrine; Animals; Azepines; Biological Transport; Calcium; Carbachol; Dose-Response Relationship, Drug; Egtazic Acid; Famotidine; Fluorescent Dyes; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Kinetics; Male; Platelet Activating Factor; Rabbits; Thiazoles; Thienopyridines; Triazoles; Verapamil | 1995 |
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine | 1994 |
Antisecretory effects of a novel and long-lasting histamine H2-receptor antagonist, YM-14471, in rats and dogs.
Topics: Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Histamine H2 Antagonists; Infusions, Intravenous; Male; Omeprazole; Pyrimidinones; Rats; Rats, Wistar; Thiazoles | 1993 |
Inhibition of phase III activity by acid in canine stomach.
Topics: Animals; Disease Models, Animal; Dogs; Duodenal Ulcer; Electrodes; Electrophysiology; Famotidine; Female; Gastric Acid; Gastrointestinal Motility; Histamine; Hydrogen-Ion Concentration; Male; Motilin; Muscle Contraction; Muscle, Smooth; Stomach Ulcer | 1994 |
Hypothalamic neuronal histamine regulates feeding circadian rhythm in rats.
Topics: Animals; Cerebral Ventricles; Chlorpheniramine; Circadian Rhythm; Darkness; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histidine Decarboxylase; Hypothalamus; Infusions, Parenteral; Light; Male; Methylhistidines; Neurons; Rats; Rats, Wistar | 1994 |
Gastric antisecretory effect of FRG-8813, a new histamine H2 receptor antagonist, in rats and dogs.
Topics: Acetamides; Animals; Cimetidine; Dogs; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Ligation; Male; Perfusion; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley | 1993 |
Effect of the novel histamine H2-antagonist 5,6-dimethyl-2-[4-[3-(1- piperidinomethyl)phenoxy]-(z)-2-butenylamino]-4(1H)-pyrimidine dihydrochloride on histamine-induced gastric acid secretion in Heidenhain pouch dogs.
Topics: Administration, Oral; Animals; Cimetidine; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Injections, Intravenous; Male; Piperidines; Pyrimidinones | 1993 |
Effect of histamine on rat gastric H(+)-K(+)-ATPase alpha-subunit expression.
Topics: Animals; Famotidine; Gastric Mucosa; Gastrins; H(+)-K(+)-Exchanging ATPase; Histamine; Hydrogen-Ion Concentration; Male; Microscopy, Electron; Rats; Rats, Wistar; RNA, Messenger; Stomach | 1994 |
Inhibition of phase III activity by acidifying stomach in vagally denervated and innervated dogs with gastric pouches.
Topics: Acids; Animals; Denervation; Dogs; Duodenum; Famotidine; Gastrointestinal Motility; Gastroplasty; Histamine; Hydrogen-Ion Concentration; Infusions, Intravenous; Motilin; Reference Values; Stomach; Vagus Nerve | 1994 |
Histamine H2-receptor plays only a minor role in histamine-induced wheal response in the squirrel monkey and guinea pig.
Topics: Animals; Chlorpheniramine; Dimaprit; Dose-Response Relationship, Drug; Famotidine; Female; Guinea Pigs; Histamine; Histamine Agonists; Injections, Intradermal; Male; Pyridines; Ranitidine; Receptors, Histamine H2; Saimiri; Urticaria | 1993 |
Analysis of responses to vancomycin in carotid blood flow in the male rat.
Topics: Animals; Anti-Bacterial Agents; Blood Flow Velocity; Carotid Arteries; Diphenhydramine; Dose-Response Relationship, Drug; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Vancomycin; Vasodilation | 1995 |
Chronic beta 1-adrenoceptor blockade sensitises the H1 and H2 receptor systems in human atrium: rôle of cyclic nucleotides.
Topics: Adrenergic beta-Antagonists; Arrhythmias, Cardiac; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Dose-Response Relationship, Drug; Famotidine; Female; Heart; Heart Atria; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Middle Aged; Myocardial Contraction; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Stimulation, Chemical | 1996 |
Analysis of the variation in the action of L-365,260 at CCKB/gastrin receptors in rat, guinea-pig and mouse isolated gastric tissue assays.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Famotidine; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscle, Smooth; Pentagastrin; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Species Specificity; Stomach | 1996 |
Comparative evaluation of the role of endogenous gastrin in basal acid secretion in conscious rats provided with chronic fistula and pylorus ligation.
Topics: Animals; Atropine; Benzodiazepines; Chronic Disease; Famotidine; Gastric Acid; Gastric Fistula; Gastrins; Histamine; Ligation; Male; Parasympathetic Nervous System; Pylorus; Rats; Rats, Sprague-Dawley | 1996 |
Pharmacological analysis of the CCKB/gastrin receptors mediating pentagastrin-stimulated gastric acid secretion in the isolated stomach of the immature rat.
Topics: Animals; Binding, Competitive; Enterochromaffin Cells; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Models, Biological; Pentagastrin; Rats; Rats, Wistar; Receptors, Cholecystokinin; Stimulation, Chemical | 1996 |
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs.
Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Devazepide; Dogs; Dose-Response Relationship, Drug; Eating; Famotidine; Gastric Acid; Histamine; Histamine H2 Antagonists; Hormone Antagonists; Male; Methacholine Chloride; Muscarinic Antagonists; Pentagastrin; Peptones; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Stomach | 1997 |
Oral famotidine: a potential treatment for children with autism.
Topics: Administration, Oral; Adult; Animals; Autistic Disorder; Child; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Kidney; Models, Biological; Neurotransmitter Agents; Psychopharmacology; Safety; Schizophrenia | 1997 |
Histamine affects interleukin-4, interleukin-5, and interferon-gamma production by human T cell clones from the airways and blood.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Albuterol; Asthma; Bronchoalveolar Lavage Fluid; Clone Cells; Cyclic AMP; Dinoprostone; Enzyme Activation; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Impromidine; Interferon-gamma; Interleukin-2; Interleukin-4; Interleukin-5; Lung; Methylhistamines; Piperidines; Pyridines; Ranitidine; T-Lymphocytes; Triprolidine | 1998 |
Histamine H2-receptor antagonism of T-593, an anti-ulcer agent: studies on aminopyrine accumulation in isolated canine gastric mucosal cells.
Topics: Aminopyrine; Animals; Anti-Ulcer Agents; Bucladesine; Carbachol; Carbon Radioisotopes; Cholinergic Agonists; Dogs; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Guanidines; Histamine; Histamine H2 Antagonists; Omeprazole; Pentagastrin; Pirenzepine; Ranitidine; Sulfones | 1998 |
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles | 1999 |
Participation of histamine H1 and H2 receptors in passive cutaneous anaphylaxis-induced scratching behavior in ICR mice.
Topics: Animals; Anti-Allergic Agents; Behavior, Animal; Capillary Permeability; Cetirizine; Drug Interactions; Famotidine; Female; Free Radical Scavengers; Histamine; Histamine H2 Antagonists; Mice; Mice, Inbred ICR; p-Methoxy-N-methylphenethylamine; Passive Cutaneous Anaphylaxis; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Terfenadine; Time Factors | 1999 |
Role of endogenous serotonin and histamine in the pathogenesis of gastric mucosal lesions in unanaesthetised rats with a single treatment of compound 48/80, a mast cell degranulator.
Topics: Adrenergic Uptake Inhibitors; Amitriptyline; Animals; Cell Degranulation; Cimetidine; Cyproheptadine; Famotidine; Gastric Mucosa; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mast Cells; Methysergide; p-Methoxy-N-methylphenethylamine; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Stomach Ulcer; Tripelennamine | 1999 |
Histaminergic H2 receptor ligands modulate acetylcholine release in the ventral striatum.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Corpus Striatum; Dimaprit; Dopamine; Dopamine Agonists; Dopamine Antagonists; Famotidine; gamma-Aminobutyric Acid; Histamine; Histamine H2 Antagonists; Male; Neurons; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2 | 1999 |
Influence of different histamine receptor agonists and antagonists on apomorphine-induced licking behavior in rat.
Topics: Animals; Apomorphine; Chlorpheniramine; Dimaprit; Diphenhydramine; Dopamine Agonists; Drug Interactions; Famotidine; Histamine; Histamine Agonists; Histamine Antagonists; Imidazoles; Male; Piperidines; Ranitidine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Thiourea; Toluidines | 2000 |
Ghrelin stimulates gastric acid secretion and motility in rats.
Topics: Animals; Atropine; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Ghrelin; Histamine; Histamine H2 Antagonists; Male; Peptide Hormones; Peptides; Peristalsis; Rats; Rats, Sprague-Dawley; Stomach; Vagotomy | 2000 |
Modified histamine-induced NO-mediated relaxation in resistance arteries in pre-eclampsia.
Topics: Adult; Arteries; Atrial Natriuretic Factor; Cyclic GMP; Down-Regulation; Endothelium, Vascular; Famotidine; Female; Histamine; Humans; Isometric Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroarginine; Pre-Eclampsia; Pregnancy; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Vascular Resistance; Vasodilation | 2000 |
Inhibition of gastric acid secretion by nimesulide: a possible factor in its gastric tolerability.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Indomethacin; Male; Mice; Mice, Inbred C57BL; Muscarine; Perfusion; Sulfonamides | 2001 |
Histamine-induced production of interleukin-6 and interleukin-8 by human coronary artery endothelial cells is enhanced by endotoxin and tumor necrosis factor-alpha.
Topics: Cells, Cultured; Chemokine CCL2; Coronary Vessels; Diphenhydramine; Drug Synergism; Endothelium, Vascular; Famotidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-6; Interleukin-8; Lipopolysaccharides; NF-kappa B; Tumor Necrosis Factor-alpha | 2001 |
Stimulatory effects of nitric oxide donors on gastric acid secretion in isolated mouse stomach.
Topics: Animals; Bethanechol; Dose-Response Relationship, Drug; Electric Stimulation; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Mice; Nitric Oxide Donors; Nitroprusside; Stomach; Time Factors; Vagus Nerve; Vasodilator Agents | 2001 |
Histamine is involved in ultraviolet B-induced pigmentation of guinea pig skin.
Topics: Animals; Cattle; Cells, Cultured; Drug Administration Schedule; Erythema; Famotidine; Guinea Pigs; Histamine; Histamine H2 Antagonists; Humans; Melanocytes; Radiation Injuries; Ranitidine; Skin Pigmentation; Ultraviolet Rays | 2002 |
The role of histamine in dural vessel dilation.
Topics: Animals; Blood Pressure; Dura Mater; Electric Stimulation; Enzyme Inhibitors; Famotidine; Histamine; Histamine Antagonists; Male; Meningeal Arteries; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Time Factors; Vasodilation | 2002 |
Effect of nimesulide on gastric acid secretion in the mouse stomach in vitro.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Dose-Response Relationship, Drug; Drug Combinations; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine H2 Antagonists; Hydrogen-Ion Concentration; In Vitro Techniques; Indomethacin; Male; Mice; Mice, Inbred C57BL; Stomach; Sulfonamides | 2003 |
Signaling via histamine receptors in cat duodenal smooth muscle cells.
Topics: Alkaloids; Animals; Benzophenanthridines; Cats; Duodenum; Enzyme Inhibitors; Ethylmaleimide; Famotidine; Heparin; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Muscle Contraction; Myocytes, Smooth Muscle; Pertussis Toxin; Phenanthridines; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide Phospholipase C; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Signal Transduction | 2003 |
Histamine participates in the early phase of trabecular bone loss in ovariectomized rats.
Topics: Animals; Body Weight; Bone Resorption; Cimetidine; Famotidine; Female; Femur; Histamine; Immunohistochemistry; Kinetics; Mast Cells; Osteoclasts; Ovariectomy; Rats | 2004 |
Role of surface activity in the biological actions of ranitidine and famotidine.
Topics: Acetylcholine; Cholesterol; Famotidine; Histamine; Ions; Membranes, Artificial; Micelles; Molecular Structure; Permeability; Phosphatidylcholines; Ranitidine; Surface Properties | 2004 |
Histamine increases sickle erythrocyte adherence to endothelium.
Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules | 2006 |
Histamine mediates osteoclastic resorption only during the acute phase of bone loss in ovariectomized rats.
Topics: Animals; Bone Resorption; Famotidine; Female; Histamine; Histamine H2 Antagonists; Osteoclasts; Ovariectomy; Rats; Rats, Wistar; Sodium Chloride | 2006 |
Histamine mediates the stimulatory action of ghrelin on acid secretion in rat stomach.
Topics: Animals; Famotidine; Gastric Acid; Gastric Mucosa; Ghrelin; Growth Hormone; Histamine; Histamine H2 Antagonists; Histidine Decarboxylase; Male; Peptide Hormones; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stomach; Vagotomy | 2006 |
Differential effects of histamine on Leydig cell and testicular macrophage activities in wall lizards: precise role of H1/H2 receptor subtypes.
Topics: Animals; Cells, Cultured; Dose-Response Relationship, Drug; Famotidine; Histamine; Histamine Antagonists; Leydig Cells; Lizards; Macrophages; Male; Phagocytosis; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Superoxides; Testosterone | 2007 |
Histamine stimulation of MMP-1(collagenase-1) secretion and gene expression in gastric epithelial cells: role of EGFR transactivation and the MAP kinase pathway.
Topics: Collagenases; Epithelial Cells; ErbB Receptors; Famotidine; Gene Expression Regulation, Enzymologic; Heparin-binding EGF-like Growth Factor; Histamine; Humans; Intercellular Signaling Peptides and Proteins; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Protein Kinase Inhibitors; Quinazolines; RNA, Small Interfering; Stomach; Time Factors; Transcriptional Activation; Tyrphostins | 2007 |
The effect and mechanism of action of capsaicin on gastric acid output.
Topics: Animals; Benzodiazepines; Bethanechol; Calcitonin Gene-Related Peptide; Capsaicin; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastrins; Histamine; Histamine H2 Antagonists; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Agonists; Rats; Rats, Wistar; Somatostatin; Stomach; Vagus Nerve | 2009 |
Phosphodiesterase isozymes involved in regulating acid secretion in the isolated mouse stomach.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Famotidine; Gastric Acid; Gastric Mucosa; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; Isoenzymes; Male; Mice; Organ Specificity; Perfusion; Phosphodiesterase Inhibitors; Pituitary Adenylate Cyclase-Activating Polypeptide; Rolipram; Stomach; Time Factors | 2009 |
Antiulcer activity of preparations containing ultralow doses of antibodies in modeled chronic ulcer in rats.
Topics: Acetates; Animals; Anti-Ulcer Agents; Antibodies; Famotidine; Gastrins; Histamine; Male; Rats; Rats, Wistar; Receptors, Histamine H2; Stomach Ulcer | 2009 |
A histamine H₂ receptor blocker ameliorates development of heart failure in dogs independently of β-adrenergic receptor blockade.
Topics: Adrenergic beta-Antagonists; Animals; Carbazoles; Cardiac Catheterization; Cardiac Pacing, Artificial; Cardiotonic Agents; Carvedilol; Cyclic AMP; Disease Models, Animal; Dogs; Echocardiography; Famotidine; Heart Failure; Histamine; Histamine H2 Antagonists; Immunohistochemistry; Mast Cells; Propanolamines; Pulmonary Wedge Pressure; Stroke Volume; Ventricular Function, Left | 2010 |
Arrhythmogenic effect of sympathetic histamine in mouse hearts subjected to acute ischemia.
Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Atenolol; Famotidine; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; Histamine Release; Histidine Decarboxylase; Mice; Mice, Knockout; Myocardial Ischemia; Myocardium; Norepinephrine; Sympathetic Nervous System; Tachycardia, Ventricular; Ventricular Fibrillation | 2012 |
Facilitation of short-term memory by histaminergic neurons in the nucleus accumbens is independent of cholinergic and glutamatergic transmission.
Topics: Acetylcholine; Animals; Famotidine; Glutamic Acid; Histamine; Histamine Antagonists; Learning; Male; Memory, Short-Term; Neurons; Nucleus Accumbens; Piperidines; Rats; Rats, Sprague-Dawley; Time Factors | 2013 |
Histamine receptor 2 is a key influence in immune responses to intestinal histamine-secreting microbes.
Topics: Animals; Cell Line; Coculture Techniques; Cytokines; Famotidine; Histamine; Humans; Immunity; Immunomodulation; Intestines; Lactobacillus; Mice; Mice, Inbred Strains; Mice, Knockout; Microbiota; NF-kappa B; Receptors, Histamine H2 | 2014 |
Histamine upregulates Nav1.8 expression in primary afferent neurons via H2 receptors: involvement in neuropathic pain.
Topics: Animals; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Famotidine; Ganglia, Spinal; Histamine; Histamine Agonists; Histamine H2 Antagonists; Hyperalgesia; Male; NAV1.8 Voltage-Gated Sodium Channel; Pain Measurement; Pain Threshold; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; Sciatica; Sensory Receptor Cells; Up-Regulation | 2014 |
Histamine Receptor 2 is Required to Suppress Innate Immune Responses to Bacterial Ligands in Patients with Inflammatory Bowel Disease.
Topics: Adult; Animals; Case-Control Studies; Cells, Cultured; Colitis, Ulcerative; Crohn Disease; Cytokines; Disease Models, Animal; Down-Regulation; Famotidine; Female; Flagellin; Gene Expression; Histamine; Histamine H2 Antagonists; Humans; Immunity, Innate; Intestinal Mucosa; Ligands; Lipopolysaccharides; Lipoproteins; Lymphocyte Count; Male; Mice; Mice, SCID; Middle Aged; Monocytes; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H4; Severity of Illness Index; Th1 Cells; Th17 Cells; Toll-Like Receptors; Weight Loss; Young Adult | 2016 |
Association of histamine with hypertension-induced cardiac remodeling and reduction of hypertrophy with the histamine-2-receptor antagonist famotidine compared with the beta-blocker metoprolol.
Topics: Adrenergic beta-1 Receptor Antagonists; Age Factors; Animals; Blood Pressure; Cardiomegaly; Famotidine; Histamine; Histamine H2 Antagonists; Hypertension; Male; Metoprolol; Myocardium; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Histamine H2; Ventricular Remodeling | 2018 |
Hypolipemic effects of histamine is due to inhibition of VLDL secretion from the liver: involvement of both H1 and H2-receptors.
Topics: Animals; Cetirizine; Cholesterol; Famotidine; Histamine; Histamine Agonists; Lipids; Liver; Male; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Triglycerides | 2022 |
Potential association of mast cells with coronavirus disease 2019.
Topics: Cell Communication; Cholecalciferol; COVID-19; COVID-19 Drug Treatment; Cromolyn Sodium; Cyproheptadine; Cytokines; Famotidine; Histamine; Histamine Antagonists; Humans; Lung; Luteolin; Macrophages; Mast Cells; SARS-CoV-2; Severity of Illness Index; Substance P | 2021 |
Molecular basis for the repurposing of histamine H2-receptor antagonist to treat COVID-19.
Topics: Cimetidine; COVID-19 Drug Treatment; Famotidine; Histamine; Histamine H2 Antagonists; Humans; Molecular Docking Simulation | 2022 |
Famotidine activates the vagus nerve inflammatory reflex to attenuate cytokine storm.
Topics: alpha7 Nicotinic Acetylcholine Receptor; Animals; Anti-Inflammatory Agents; COVID-19; Cytokine Release Syndrome; Famotidine; Histamine; Histamine H2 Antagonists; Lipopolysaccharides; Mice; Reflex; Vagus Nerve | 2022 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship | 2008 |
Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay.
Topics: Animals; Antimalarials; Drug Resistance, Multiple; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum | 2010 |