Page last updated: 2024-08-25

falipamil and cardiovascular agents

falipamil has been researched along with cardiovascular agents in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199015 (68.18)18.7374
1990's6 (27.27)18.2507
2000's1 (4.55)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Doerr, T; Trautwein, W1
Eberlein, W; Heider, J; Kobinger, W; Lillie, C; Luger, P; Müller, P; Noll, K; Psiorz, M; Reiffen, M1
Ilias, W; Lackner, F; Zimpfer, M1
Darragh, A; Hallinan, D; Koss, FW; Lambe, R; Roth, W1
Daemmgen, JW; Gross, GJ1
Brunner, F; Kukovetz, WR1
Ferry, A; Hilaire, J; Jaillon, P; Lecocq, B; Lecocq, V; Maria, JF; Naudascher, M1
Morgan, G; Siegl, PK1
Akahane, K; Chiba, S; Furukawa, Y; Haniuda, M; Ogiwara, Y1
McDonald, TF; Pelzer, D; Trautwein, W1
Brutsaert, DL; De Clerck, NM; Sys, SU1
Kobinger, W; Lillie, C2
Broustet, JP; Colle, JP; Hilaire, J; Theron, M1
Bijleveld, RE; Bom, HP; Verdouw, PD1
Kawada, M; Satoh, K; Taira, N1
Anders, G; Brachmann, J; Hamman, HD; Jauernig, R; Kübler, W; Rizos, I; Senges, J1
Antoni, H; Hohnloser, S; Homburger, H; Weirich, J1
Dämmgen, J; Diederen, W; Kadatz, R1
Boucher, M; Chapuy, E; Chassaing, C; Duchêne-Marullaz, P1
Boucher, M; Chapuy, E; Chassaing, C1
Büter, I; Gams, E; Hohlfeld, T; Schipke, JD; Schmitz-Spanke, S1

Reviews

1 review(s) available for falipamil and cardiovascular agents

ArticleYear
[Selective I(f) channel inhibition: an alternative for treating coronary artery disease?].
    Herz, 2006, Volume: 31, Issue:1

    Topics: Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Benzazepines; Cardiotonic Agents; Cardiovascular Agents; Clonidine; Coronary Artery Disease; Humans; Isoindoles; Ivabradine; Phthalimides; Practice Guidelines as Topic; Practice Patterns, Physicians'

2006

Trials

2 trial(s) available for falipamil and cardiovascular agents

ArticleYear
Effects of falipamil (AQ-A 39) on heart rate and blood pressure in resting and exercising healthy volunteers.
    Journal of cardiovascular pharmacology, 1989, Volume: 14, Issue:1

    Topics: Adult; Blood Pressure; Cardiovascular Agents; Double-Blind Method; Exercise; Heart Rate; Humans; Isoindoles; Male; Phthalimides

1989
Cardiovascular effects of AQ-A 39 in healthy volunteers.
    British journal of clinical pharmacology, 1983, Volume: 16, Issue:6

    Topics: Adult; Blood Pressure; Cardiovascular Agents; Cardiovascular System; Heart Rate; Humans; Isoindoles; Male; Phthalimides; Physical Exertion; Propranolol

1983

Other Studies

19 other study(ies) available for falipamil and cardiovascular agents

ArticleYear
On the mechanism of the "specific bradycardic action" of the verapamil derivative UL-FS 49.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:4

    Topics: Action Potentials; Animals; Benzazepines; Cardiovascular Agents; Electric Stimulation; Electrophysiology; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Ion Channels; Isoindoles; Myocardial Contraction; Myocardium; Phthalimides; Rabbits; Sinoatrial Node; Verapamil

1990
Specific bradycardic agents. 1. Chemistry, pharmacology, and structure-activity relationships of substituted benzazepinones, a-new class of compounds exerting antiischemic properties.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:5

    Topics: Animals; Anti-Arrhythmia Agents; Benzazepines; Calcium Channel Blockers; Cardiovascular Agents; Chemical Phenomena; Chemistry; Coronary Disease; Guinea Pigs; Heart Rate; Isoindoles; Molecular Conformation; Muscle, Smooth, Vascular; Myocardial Contraction; Nifedipine; Phthalimides; Rabbits; Rats; Structure-Activity Relationship; Verapamil

1990
[The intraoperative use of falipamil (AQ-A39), a new calcium antagonist with specific bradytropic properties].
    Der Anaesthesist, 1990, Volume: 39, Issue:10

    Topics: Adult; Aged; Anti-Arrhythmia Agents; Calcium Channel Blockers; Cardiovascular Agents; Female; Hemodynamics; Humans; Intraoperative Complications; Isoindoles; Male; Middle Aged; Phthalimides; Tachycardia

1990
Pharmacokinetics of falipamil after intravenous administration to humans.
    Journal of pharmaceutical sciences, 1990, Volume: 79, Issue:5

    Topics: Adult; Cardiovascular Agents; Humans; Injections, Intravenous; Isoindoles; Male; Phthalimides

1990
Effect of the new specific bradycardia agent AQ-A39 (falipamil) on coronary collateral blood flow in dogs.
    Journal of cardiovascular pharmacology, 1987, Volume: 10, Issue:1

    Topics: Animals; Bradycardia; Cardiovascular Agents; Collateral Circulation; Coronary Circulation; Dogs; Female; Hemodynamics; Isoindoles; Male; Phthalimides; Regional Blood Flow

1987
Binding of two specific bradycardic agents, alinidine and AQ-A 39, to muscarinic receptors of guinea pig atria and ventricle.
    Journal of cardiovascular pharmacology, 1988, Volume: 11, Issue:2

    Topics: Animals; Binding, Competitive; Cardiovascular Agents; Clonidine; Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Isoindoles; Myocardium; Phthalimides; Quinuclidines; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Receptors, Muscarinic

1988
Effects of a specific bradycardic agent (AQ-A39) and verapamil on beta-adrenergic responses in isolated guinea pig atria.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:2

    Topics: Animals; Cardiovascular Agents; Female; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Isoindoles; Isoproterenol; Male; Myocardial Contraction; Phthalimides; Receptors, Adrenergic, beta; Verapamil

1987
Bradycardic effects of AQ-A 39 (falipamil) in situ and in isolated, blood-perfused dog hearts. Comparison with alinidine and verapamil.
    Japanese heart journal, 1988, Volume: 29, Issue:6

    Topics: Animals; Cardiovascular Agents; Clonidine; Dogs; Dose-Response Relationship, Drug; Heart; Heart Atria; Heart Rate; Isoindoles; Myocardial Contraction; Phthalimides; Verapamil

1988
Calcium channel block and recovery from block in mammalian ventricular muscle treated with organic channel inhibitors.
    Pflugers Archiv : European journal of physiology, 1982, Volume: 394, Issue:2

    Topics: Action Potentials; Animals; Calcium; Cardiovascular Agents; Cats; Dose-Response Relationship, Drug; Gallopamil; Heart; In Vitro Techniques; Ion Channels; Isoindoles; Phthalimides; Verapamil

1982
Effects of AQA39 on contractile performance of isolated mammalian ventricular myocardium.
    European journal of pharmacology, 1984, Aug-03, Volume: 103, Issue:1-2

    Topics: Animals; Calcium Channel Blockers; Cardiovascular Agents; Cats; In Vitro Techniques; Isoindoles; Myelin Sheath; Myocardial Contraction; Myocardium; Papillary Muscles; Phthalimides

1984
Cardiovascular characterization of UL-FS 49, 1,3,4,5-tetrahydro-7,8-dimethoxy-3-[3-][2-(3,4-dimethoxyphenyl)ethyl] methylimino]propyl]-2H-3-benzazepin-2-on hydrochloride, a new "specific bradycardic agent".
    European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Benzazepines; Blood Pressure; Cardiovascular Agents; Cats; Dogs; Electric Stimulation; Electrocardiography; Female; Guinea Pigs; Heart Rate; Hemodynamics; In Vitro Techniques; Isoindoles; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Parasympatholytics; Phthalimides; Potassium; Rabbits

1984
Cardiovascular responses to increasing plasma concentrations of AQ-A 39 Cl, a new compound with negative chronotropic effects.
    Arzneimittel-Forschung, 1983, Volume: 33, Issue:5

    Topics: Anesthesia; Animals; Cardiovascular Agents; Coronary Circulation; Depression, Chemical; Electrocardiography; Heart Rate; Hemodynamics; Isoindoles; Phthalimides; Pulmonary Circulation; Swine

1983
Analyses of the cardiac action of the bradycardic agent, AQ-A 39, by use of isolated, blood-perfused dog-heart preparations.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:2

    Topics: Animals; Cardiovascular Agents; Coronary Circulation; Dogs; Heart; Heart Conduction System; Heart Rate; In Vitro Techniques; Isoindoles; Male; Myocardial Contraction; Papillary Muscles; Perfusion; Phthalimides; Vasodilation

1984
Effect of nifedipine and AQ-A 39 on the sinoatrial and atrioventricular nodes of the rabbit and their antiarrhythmic action on atrioventricular nodal reentrant tachycardia.
    Cardiovascular research, 1983, Volume: 17, Issue:3

    Topics: Action Potentials; Animals; Atrioventricular Node; Cardiovascular Agents; Heart Conduction System; Isoindoles; Nifedipine; Phthalimides; Pyridines; Rabbits; Sinoatrial Node; Tachycardia

1983
Electrophysiological studies on effects of AQ-A 39 in the isolated guinea pig heart and myocardial preparations.
    Arzneimittel-Forschung, 1982, Volume: 32, Issue:7

    Topics: Action Potentials; Animals; Barium; Cardiovascular Agents; Electric Stimulation; Electrophysiology; Guinea Pigs; Heart; In Vitro Techniques; Isoindoles; Membrane Potentials; Papillary Muscles; Phthalimides; Purkinje Fibers

1982
Cardiovascular actions of 5,6-dimethoxy-2-(3-[(alpha-(3,4-dimethoxy) phenylethyl)-methylamino] propyl) phthalimidine (AQ-A 39), a specific bradycardic agent.
    Arzneimittel-Forschung, 1981, Volume: 31, Issue:4

    Topics: Animals; Cardiovascular Agents; Cats; Coronary Circulation; Dogs; Female; Guinea Pigs; Heart Rate; Hemodynamics; Isoindoles; Male; Mice; Myocardial Contraction; Myocardium; Oxygen Consumption; Phthalimides; Rabbits; Rats; Species Specificity; Verapamil

1981
AQ-A 39 (5,6-dimethoxy-2-[3[[alpha-(3,4-dimethoxy)-phenylethyl]methylamino]propyl]phtalimidine), a specific bradycardic agent with direct action on the heart.
    European journal of pharmacology, 1981, Jun-19, Volume: 72, Issue:2-3

    Topics: Animals; Blood Pressure; Cardiovascular Agents; Cats; Coronary Vessels; Dogs; Electrocardiography; Female; Guinea Pigs; Heart; Heart Rate; In Vitro Techniques; Isoindoles; Male; Myocardial Contraction; Myocardium; Oxygen Consumption; Parasympathetic Nervous System; Phthalimides

1981
Chronotropic cardiac effects of falipamil in conscious dogs: interactions with the autonomic nervous system and various ionic conductances.
    Journal of cardiovascular pharmacology, 1994, Volume: 23, Issue:4

    Topics: Animals; Atropine; Autonomic Nervous System; Blood Pressure; Cardiovascular Agents; Dogs; Female; Heart Rate; Ion Channels; Isoindoles; Male; Phthalimides; Pindolol; Quinidine; Receptors, Adrenergic, beta; Receptors, Muscarinic; Stimulation, Chemical; Verapamil

1994
Cardiac electrophysiological effects of falipamil in the conscious dog: comparison with alinidine.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Animals; Atrioventricular Node; Blood Pressure; Bundle of His; Cardiovascular Agents; Clonidine; Dogs; Electroencephalography; Electrophysiology; Female; Heart; Heart Rate; Isoindoles; Male; Phthalimides; Sinoatrial Node

1996