ezogabine has been researched along with oxotremorine in 2 studies
Studies (ezogabine) | Trials (ezogabine) | Recent Studies (post-2010) (ezogabine) | Studies (oxotremorine) | Trials (oxotremorine) | Recent Studies (post-2010) (oxotremorine) |
---|---|---|---|---|---|
383 | 26 | 241 | 1,930 | 6 | 99 |
Protein | Taxonomy | ezogabine (IC50) | oxotremorine (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 0.4 | |
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 5 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 2.321 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 2.7261 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 2.7261 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 2.7261 | |
Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | 8 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 2.7261 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 4.5012 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Boehm, S; Lechner, SG; Mayer, M | 1 |
Boehm, S; Drobny, H; Kosenburger, K; Kubista, H; Mahlknecht, P | 1 |
2 other study(ies) available for ezogabine and oxotremorine
Article | Year |
---|---|
Activation of M1 muscarinic receptors triggers transmitter release from rat sympathetic neurons through an inhibition of M-type K+ channels.
Topics: Animals; Animals, Newborn; Carbamates; Cells, Cultured; Evoked Potentials; Mecamylamine; Membrane Potentials; Muscarinic Agonists; Neurons; Norepinephrine; Oxotremorine; Pertussis Toxin; Phenylenediamines; Potassium Channels, Voltage-Gated; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Superior Cervical Ganglion; Tetrodotoxin | 2003 |
Inhibition of transmitter release from rat sympathetic neurons via presynaptic M(1) muscarinic acetylcholine receptors.
Topics: Acetylcholine; Action Potentials; Adrenergic Fibers; Animals; Animals, Newborn; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Carbamates; Cells, Cultured; Diamines; Dose-Response Relationship, Drug; Electric Stimulation; KCNQ Potassium Channels; Muscarinic Agonists; Muscarinic Antagonists; Neural Inhibition; Norepinephrine; omega-Conotoxin GVIA; Oxotremorine; Pertussis Toxin; Phenylenediamines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptors, Presynaptic; Superior Cervical Ganglion; Synaptic Transmission; Time Factors; Type C Phospholipases | 2009 |