Page last updated: 2024-09-03

ezogabine and oxotremorine

ezogabine has been researched along with oxotremorine in 2 studies

Compound Research Comparison

Studies
(ezogabine)
Trials
(ezogabine)
Recent Studies (post-2010)
(ezogabine)
Studies
(oxotremorine)
Trials
(oxotremorine)
Recent Studies (post-2010) (oxotremorine)
383262411,930699

Protein Interaction Comparison

ProteinTaxonomyezogabine (IC50)oxotremorine (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.4
Muscarinic acetylcholine receptor M4Homo sapiens (human)5
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)2.321
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M5Homo sapiens (human)8
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.7261
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.5012

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boehm, S; Lechner, SG; Mayer, M1
Boehm, S; Drobny, H; Kosenburger, K; Kubista, H; Mahlknecht, P1

Other Studies

2 other study(ies) available for ezogabine and oxotremorine

ArticleYear
Activation of M1 muscarinic receptors triggers transmitter release from rat sympathetic neurons through an inhibition of M-type K+ channels.
    The Journal of physiology, 2003, Dec-15, Volume: 553, Issue:Pt 3

    Topics: Animals; Animals, Newborn; Carbamates; Cells, Cultured; Evoked Potentials; Mecamylamine; Membrane Potentials; Muscarinic Agonists; Neurons; Norepinephrine; Oxotremorine; Pertussis Toxin; Phenylenediamines; Potassium Channels, Voltage-Gated; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Superior Cervical Ganglion; Tetrodotoxin

2003
Inhibition of transmitter release from rat sympathetic neurons via presynaptic M(1) muscarinic acetylcholine receptors.
    British journal of pharmacology, 2009, Volume: 156, Issue:8

    Topics: Acetylcholine; Action Potentials; Adrenergic Fibers; Animals; Animals, Newborn; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Carbamates; Cells, Cultured; Diamines; Dose-Response Relationship, Drug; Electric Stimulation; KCNQ Potassium Channels; Muscarinic Agonists; Muscarinic Antagonists; Neural Inhibition; Norepinephrine; omega-Conotoxin GVIA; Oxotremorine; Pertussis Toxin; Phenylenediamines; Pirenzepine; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptors, Presynaptic; Superior Cervical Ganglion; Synaptic Transmission; Time Factors; Type C Phospholipases

2009