ezogabine has been researched along with himbacine in 1 studies
Studies (ezogabine) | Trials (ezogabine) | Recent Studies (post-2010) (ezogabine) | Studies (himbacine) | Trials (himbacine) | Recent Studies (post-2010) (himbacine) |
---|---|---|---|---|---|
383 | 26 | 241 | 73 | 0 | 9 |
Protein | Taxonomy | ezogabine (IC50) | himbacine (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 0.0175 | |
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 0.1144 | |
Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | 1.016 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 0.5482 | |
Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | 0.3336 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kaba, H; Takahashi, Y | 1 |
1 other study(ies) available for ezogabine and himbacine
Article | Year |
---|---|
Muscarinic receptor type 1 (M1) stimulation, probably through KCNQ/Kv7 channel closure, increases spontaneous GABA release at the dendrodendritic synapse in the mouse accessory olfactory bulb.
Topics: Alkaloids; Animals; Anticonvulsants; Calcium; Calcium Channel Blockers; Calcium Channels, R-Type; Carbachol; Carbamates; Cholinergic Agonists; Dendrites; Diclofenac; Excitatory Amino Acid Antagonists; Furans; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channel Gating; KCNQ Potassium Channels; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Naphthalenes; Nimodipine; Olfactory Bulb; Patch-Clamp Techniques; Phenylenediamines; Piperidines; Pirenzepine; Potassium Channel Blockers; Receptor, Muscarinic M1; Receptors, Glutamate; Synapses | 2010 |