Page last updated: 2024-09-05

ezlopitant and naloxone

ezlopitant has been researched along with naloxone in 1 studies

Compound Research Comparison

Studies
(ezlopitant)
Trials
(ezlopitant)
Recent Studies (post-2010)
(ezlopitant)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
222120,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomyezlopitant (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Honda, M; Ono, H; Tanabe, M; Yamamoto, S1

Other Studies

1 other study(ies) available for ezlopitant and naloxone

ArticleYear
Spinal ventral root after-discharges as a pain index: involvement of NK-1 and NMDA receptors.
    Brain research, 2006, Apr-12, Volume: 1082, Issue:1

    Topics: Action Potentials; Analysis of Variance; Animals; Benzylamines; Bridged Bicyclo Compounds, Heterocyclic; Diterpenes; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Excitatory Amino Acid Antagonists; Ketamine; Male; Mephenesin; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Neurotoxins; Pain; Pain Measurement; Physical Stimulation; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Receptors, Neurokinin-1; Spinal Nerve Roots; Time Factors

2006