Page last updated: 2024-09-04

ezetimibe and propofol

ezetimibe has been researched along with propofol in 4 studies

Compound Research Comparison

Studies
(ezetimibe)
Trials
(ezetimibe)
Recent Studies (post-2010)
(ezetimibe)
Studies
(propofol)
Trials
(propofol)
Recent Studies (post-2010) (propofol)
2,4845631,46516,8275,1886,805

Protein Interaction Comparison

ProteinTaxonomyezetimibe (IC50)propofol (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)8.1667
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)9.393
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)7.596
Gamma-aminobutyric acid receptor subunit alpha-1Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit gamma-2Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)8.1667
Prostaglandin G/H synthase 1Homo sapiens (human)3.832
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)8.1667
Sodium-dependent noradrenaline transporter Homo sapiens (human)9.393
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)8.3
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-3Homo sapiens (human)8
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)8.1667
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)8.3
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)8.3
5-hydroxytryptamine receptor 2BHomo sapiens (human)5.499
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)8.3
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)8.1667
GABA theta subunitRattus norvegicus (Norway rat)8.1667
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)8.1667

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chang, TK; Ensom, MH; Kiang, TK1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Galetin, A; Gill, KL; Houston, JB1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1

Reviews

2 review(s) available for ezetimibe and propofol

ArticleYear
UDP-glucuronosyltransferases and clinical drug-drug interactions.
    Pharmacology & therapeutics, 2005, Volume: 106, Issue:1

    Topics: Clinical Trials as Topic; Drug Interactions; Enzyme Activation; Enzyme Induction; Glucuronides; Glucuronosyltransferase; Humans; Pharmaceutical Preparations; Pharmacogenetics; Polymorphism, Genetic

2005
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

2 other study(ies) available for ezetimibe and propofol

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Characterization of in vitro glucuronidation clearance of a range of drugs in human kidney microsomes: comparison with liver and intestinal glucuronidation and impact of albumin.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:4

    Topics: Adult; Aged; Female; Glucuronides; Glucuronosyltransferase; Humans; In Vitro Techniques; Intestinal Mucosa; Intestines; Kidney; Liver; Male; Metabolic Clearance Rate; Microsomes; Middle Aged; Organ Specificity; Pharmaceutical Preparations; Predictive Value of Tests; Protein Binding; Serum Albumin, Bovine; Substrate Specificity; Young Adult

2012