Page last updated: 2024-09-04

ezetimibe and dalcetrapib

ezetimibe has been researched along with dalcetrapib in 4 studies

Compound Research Comparison

Studies
(ezetimibe)
Trials
(ezetimibe)
Recent Studies (post-2010)
(ezetimibe)
Studies
(dalcetrapib)
Trials
(dalcetrapib)
Recent Studies (post-2010) (dalcetrapib)
2,4845631,46516638103

Protein Interaction Comparison

ProteinTaxonomyezetimibe (IC50)dalcetrapib (IC50)
Cholesteryl ester transfer proteinHomo sapiens (human)4.1

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Rosenson, RS1
Abt, M; Derks, M; Phelan, M1
Blum, D; Chaput, E; Derks, M; Kallend, D; Niesor, EJ; Staempfli, A1
Akinsanya, KO; Castro-Perez, J; Chen, Y; Daniels, E; Johns, DG; Previs, SF; Roddy, TP; Wang, SP; Zhou, H1

Trials

2 trial(s) available for ezetimibe and dalcetrapib

ArticleYear
Lack of clinically relevant drug-drug interactions when dalcetrapib is co-administered with ezetimibe.
    British journal of clinical pharmacology, 2010, Volume: 70, Issue:6

    Topics: Adolescent; Adult; Aged; Amides; Anticholesteremic Agents; Azetidines; Cross-Over Studies; Drug Administration Schedule; Drug Interactions; Esters; Ezetimibe; Humans; Hypertension; Lipids; Male; Middle Aged; Sulfhydryl Compounds; Young Adult

2010
Effect of dalcetrapib, a CETP modulator, on non-cholesterol sterol markers of cholesterol homeostasis in healthy subjects.
    Atherosclerosis, 2011, Volume: 219, Issue:2

    Topics: Amides; Animals; Anticholesteremic Agents; Azetidines; Biomarkers; Cholestanol; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cricetinae; Cross-Over Studies; Desmosterol; Esters; Ezetimibe; Homeostasis; Humans; Intestinal Absorption; Lipid Metabolism; Male; Mesocricetus; Models, Animal; Phytosterols; Quinolines; Sitosterols; Sulfhydryl Compounds; Switzerland

2011

Other Studies

2 other study(ies) available for ezetimibe and dalcetrapib

ArticleYear
Functional assessment of HDL: Moving beyond static measures for risk assessment.
    Cardiovascular drugs and therapy, 2010, Volume: 24, Issue:1

    Topics: Amides; Animals; Anticholesteremic Agents; Azetidines; Cardiovascular Diseases; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials as Topic; Esters; Ezetimibe; Glucose; Humans; Insulin; Lipase; Lipoproteins, HDL; Niacin; Quinolines; Risk Assessment; Risk Factors; Sulfhydryl Compounds

2010
In vivo effects of anacetrapib on preβ HDL: improvement in HDL remodeling without effects on cholesterol absorption.
    Journal of lipid research, 2013, Volume: 54, Issue:10

    Topics: Amides; Animals; Anticholesteremic Agents; Area Under Curve; Azetidines; Cholesterol; Cholesterol Ester Transfer Proteins; Cricetinae; Diet, High-Fat; Drug Evaluation, Preclinical; Dyslipidemias; Esters; Ezetimibe; High-Density Lipoproteins, Pre-beta; Humans; Intestinal Absorption; Male; Mesocricetus; Oxazolidinones; Sulfhydryl Compounds

2013