Page last updated: 2024-09-04

ezetimibe and bms201038

ezetimibe has been researched along with bms201038 in 9 studies

Compound Research Comparison

Studies
(ezetimibe)
Trials
(ezetimibe)
Recent Studies (post-2010)
(ezetimibe)
Studies
(bms201038)
Trials
(bms201038)
Recent Studies (post-2010) (bms201038)
2,4845631,46512813106

Protein Interaction Comparison

ProteinTaxonomyezetimibe (IC50)bms201038 (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0008
Microsomal triglyceride transfer protein large subunitHomo sapiens (human)0.0056

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (22.22)29.6817
2010's6 (66.67)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Bloedon, LT; McKenney, J; Rader, DJ; Samaha, FF; Sasiela, WJ1
Davidson, MH1
Ballantyne, CM; Catapano, AL; Norata, GD1
Reiner, Z1
Diekmann, J; Farr, M; Horstkotte, D; Mellwig, KP; van Buuren, F1
Cai, T; Can, A; Castro, VM; Dligach, D; Du, R; Finan, S; Gainer, V; Murphy, S; Savova, G; Shadick, NA; Weiss, ST; Yu, S1
Catapano, AL; Hovingh, GK; Raal, FJ1
Hegele, RA; Tsimikas, S1
Bacalbasa, N; Bratu, OG; Crismaru, I; Diaconu, CC; Gaman, MA; Pantea Stoian, A; Stanescu, AMA1

Reviews

5 review(s) available for ezetimibe and bms201038

ArticleYear
Novel nonstatin strategies to lower low-density lipoprotein cholesterol.
    Current atherosclerosis reports, 2009, Volume: 11, Issue:1

    Topics: Animals; Anticholesteremic Agents; Azetidines; Benzimidazoles; Carrier Proteins; Cholesterol, LDL; Ezetimibe; Farnesyl-Diphosphate Farnesyltransferase; Humans; Hypercholesterolemia; Indoles; Oligonucleotides; Oxazepines; Piperidines; Proprotein Convertase 9; Proprotein Convertases; Pyridines; Serine Endopeptidases; Serine Proteinase Inhibitors

2009
New therapeutic principles in dyslipidaemia: focus on LDL and Lp(a) lowering drugs.
    European heart journal, 2013, Volume: 34, Issue:24

    Topics: Azetidines; Benzimidazoles; Benzodiazepines; Carrier Proteins; Cholesterol, LDL; Dicarboxylic Acids; Dyslipidemias; Ezetimibe; Fatty Acids; Humans; Hypolipidemic Agents; Lipoprotein(a); Oligonucleotides; Oxazolidinones; Proprotein Convertase 9; Proprotein Convertases; Serine Endopeptidases

2013
Resistance and intolerance to statins.
    Nutrition, metabolism, and cardiovascular diseases : NMCD, 2014, Volume: 24, Issue:10

    Topics: Anticholesteremic Agents; Azetidines; Benzimidazoles; Bile Acids and Salts; Cholesterol, LDL; Drug Resistance; Drug Therapy, Combination; Drug Tolerance; Ezetimibe; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypercholesterolemia; Multidrug Resistance-Associated Protein 2; Pharmacogenetics; Polymorphism, Genetic

2014
Familial hypercholesterolemia treatments: Guidelines and new therapies.
    Atherosclerosis, 2018, Volume: 277

    Topics: Anticholesteremic Agents; Benzimidazoles; Biomarkers; Blood Component Removal; Cholesterol, LDL; Down-Regulation; Drug Therapy, Combination; Ezetimibe; Genetic Predisposition to Disease; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hyperlipoproteinemia Type II; PCSK9 Inhibitors; Phenotype; Practice Guidelines as Topic; Proprotein Convertase 9; Serine Proteinase Inhibitors; Treatment Outcome

2018
Low-density lipoprotein cholesterol lowering treatment: the current approach.
    Lipids in health and disease, 2020, May-06, Volume: 19, Issue:1

    Topics: Antibodies, Monoclonal, Humanized; Anticholesteremic Agents; Atherosclerosis; Benzimidazoles; Bile Acids and Salts; Carrier Proteins; Cholesterol, LDL; Dicarboxylic Acids; Europe; Ezetimibe; Fatty Acids; Gene Expression; Guidelines as Topic; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypercholesterolemia; PCSK9 Inhibitors; Proprotein Convertase 9; RNA, Small Interfering

2020

Trials

1 trial(s) available for ezetimibe and bms201038

ArticleYear
Inhibition of microsomal triglyceride transfer protein alone or with ezetimibe in patients with moderate hypercholesterolemia.
    Nature clinical practice. Cardiovascular medicine, 2008, Volume: 5, Issue:8

    Topics: Aged; Anticholesteremic Agents; Azetidines; Benzimidazoles; Carrier Proteins; Cholesterol, LDL; Double-Blind Method; Drug Therapy, Combination; Ezetimibe; Female; Humans; Hypercholesterolemia; Male; Microsomes; Middle Aged; Severity of Illness Index; Treatment Outcome

2008

Other Studies

3 other study(ies) available for ezetimibe and bms201038

ArticleYear
[Homozygous hypercholesterolemia - new therapeutic options in cases with complete lack of LDL- receptor].
    Deutsche medizinische Wochenschrift (1946), 2016, Volume: 141, Issue:12

    Topics: Adult; Anticholesteremic Agents; Benzimidazoles; Blood Component Removal; Codon, Terminator; Combined Modality Therapy; Coronary Disease; DNA Mutational Analysis; Ezetimibe; Female; Homozygote; Humans; Hyperlipoproteinemia Type II; Myocardial Revascularization; Receptors, LDL; Simvastatin

2016
Lipid-Lowering Agents and High HDL (High-Density Lipoprotein) Are Inversely Associated With Intracranial Aneurysm Rupture.
    Stroke, 2018, Volume: 49, Issue:5

    Topics: Adult; Aged; Aneurysm, Ruptured; Benzimidazoles; Cholesterol, HDL; Cholesterol, LDL; Cholestyramine Resin; Colestipol; Ezetimibe; Female; Fibric Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Intracranial Aneurysm; Logistic Models; Male; Middle Aged; Multivariate Analysis; Odds Ratio; Oligonucleotides; PCSK9 Inhibitors; Propensity Score; Protective Factors

2018
Lipid-Lowering Agents.
    Circulation research, 2019, Volume: 124, Issue:3

    Topics: Antibodies, Monoclonal; Anticholesteremic Agents; Benzimidazoles; Caproates; Cholesterol, HDL; Cholesterol, LDL; Diacylglycerol O-Acyltransferase; Dicarboxylic Acids; Dyslipidemias; Ezetimibe; Fatty Acids; Genetic Therapy; Humans; Hypertriglyceridemia; Hypolipidemic Agents; Lipoprotein(a); Oligonucleotides; RNA, Small Interfering

2019