Page last updated: 2024-09-04

ezetimibe and avasimibe

ezetimibe has been researched along with avasimibe in 4 studies

Compound Research Comparison

Studies
(ezetimibe)
Trials
(ezetimibe)
Recent Studies (post-2010)
(ezetimibe)
Studies
(avasimibe)
Trials
(avasimibe)
Recent Studies (post-2010) (avasimibe)
2,4845631,46577630

Protein Interaction Comparison

ProteinTaxonomyezetimibe (IC50)avasimibe (IC50)
Sterol O-acyltransferase 1Rattus norvegicus (Norway rat)0.5345
Sterol O-acyltransferase 2Homo sapiens (human)9.2
Sterol O-acyltransferase 1Homo sapiens (human)1.526
Sterol O-acyltransferase 1Mus musculus (house mouse)0.47
Acyl-CoA:cholesterol acyltransferase Oryctolagus cuniculus (rabbit)7.6

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Brown, WV1
Bruckert, E1
Brust, FR; da Silva Vaz, I; Juliano, MA; Macedo, AJ; Termignoni, C; Waldman, J; Xavier, MA1

Reviews

2 review(s) available for ezetimibe and avasimibe

ArticleYear
Therapies on the horizon for cholesterol reduction.
    Clinical cardiology, 2001, Volume: 24, Issue:8 Suppl

    Topics: Acetamides; Acetates; Anticholesteremic Agents; Azetidines; Carrier Proteins; Cholestyramine Resin; Ezetimibe; Fluorobenzenes; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hydroxysteroid Dehydrogenases; Hypercholesterolemia; Membrane Glycoproteins; Pyrimidines; Rosuvastatin Calcium; Sterol O-Acyltransferase; Sulfonamides; Sulfonic Acids

2001
New advances in lipid-modifying therapies for reducing cardiovascular risk.
    Cardiology, 2002, Volume: 97, Issue:2

    Topics: Acetamides; Acetates; Azetidines; Cardiovascular Diseases; Cholesterol, LDL; Drug Therapy, Combination; Ezetimibe; Fluorobenzenes; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Niacin; Pyrimidines; Rosuvastatin Calcium; Sulfonamides; Sulfonic Acids

2002

Other Studies

2 other study(ies) available for ezetimibe and avasimibe

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Interfering with cholesterol metabolism impairs tick embryo development and turns eggs susceptible to bacterial colonization.
    Ticks and tick-borne diseases, 2021, Volume: 12, Issue:6

    Topics: Absorption, Physiological; Acetamides; Animals; Anticholesteremic Agents; Cholesterol, Dietary; Cytochrome P-450 CYP3A Inducers; Embryo, Nonmammalian; Ezetimibe; Female; Larva; Rhipicephalus; Sulfonamides; Tick Control

2021