etravirine has been researched along with r-82913 in 1 studies
Studies (etravirine) | Trials (etravirine) | Recent Studies (post-2010) (etravirine) | Studies (r-82913) | Trials (r-82913) | Recent Studies (post-2010) (r-82913) |
---|---|---|---|---|---|
572 | 90 | 321 | 65 | 1 | 0 |
Protein | Taxonomy | etravirine (IC50) | r-82913 (IC50) |
---|---|---|---|
Chain A, Reverse Transcriptase | Human immunodeficiency virus type 1 (CLONE 12) | 0.033 | |
Chain A, Reverse Transcriptase | Human immunodeficiency virus 1 | 0.033 | |
Chain B, Reverse Transcriptase | Human immunodeficiency virus 1 | 0.033 | |
Gag-Pol polyprotein | HIV-1 M:B_HXB2R | 2.0078 | |
Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | 0.45 | |
Protease | Human immunodeficiency virus 1 | 3.8155 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
De Corte, BL | 1 |
1 review(s) available for etravirine and r-82913
Article | Year |
---|---|
From 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk](1,4)benzodiazepin-2(1H)-one (TIBO) to etravirine (TMC125): fifteen years of research on non-nucleoside inhibitors of HIV-1 reverse transcriptase.
Topics: Anti-HIV Agents; Benzodiazepines; Drug Design; Drug Resistance, Viral; HIV Reverse Transcriptase; Imidazoles; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors | 2005 |