etravirine has been researched along with nelfinavir in 4 studies
Studies (etravirine) | Trials (etravirine) | Recent Studies (post-2010) (etravirine) | Studies (nelfinavir) | Trials (nelfinavir) | Recent Studies (post-2010) (nelfinavir) |
---|---|---|---|---|---|
572 | 90 | 321 | 1,240 | 230 | 240 |
Protein | Taxonomy | etravirine (IC50) | nelfinavir (IC50) |
---|---|---|---|
Tyrosine-protein kinase Fyn | Homo sapiens (human) | 7.971 | |
Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | 8.852 | |
ATP-dependent translocase ABCB1 | Homo sapiens (human) | 3.3938 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 1.275 | |
ATP-dependent translocase ABCB1 | Mus musculus (house mouse) | 2.3 | |
Sodium-dependent noradrenaline transporter | Homo sapiens (human) | 8.852 | |
Protease | Human immunodeficiency virus 1 | 0.53 | |
Protease | Human immunodeficiency virus 1 | 0.0054 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 3 (75.00) | 24.3611 |
2020's | 1 (25.00) | 2.80 |
Authors | Studies |
---|---|
Doak, AK; Prusiner, SB; Shoichet, BK; Wille, H | 1 |
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M | 1 |
Cruz, JP; Machado, M; Mendes, AM; PrudĂȘncio, M; Sanches-Vaz, M | 1 |
1 review(s) available for etravirine and nelfinavir
Article | Year |
---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
3 other study(ies) available for etravirine and nelfinavir
Article | Year |
---|---|
Colloid formation by drugs in simulated intestinal fluid.
Topics: Buffers; Chemical Precipitation; Colloids; Intestine, Small; Light; Microscopy, Electron, Transmission; Pharmaceutical Preparations; Scattering, Radiation; Solubility | 2010 |
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries | 2023 |
Inhibition of
Topics: Alkynes; Animals; Anti-Retroviral Agents; Antimalarials; Benzoxazines; Cell Line; Cyclopropanes; Disease Models, Animal; Hepatocytes; Humans; Malaria; Male; Mice, Inbred C57BL; Nelfinavir; Nitriles; Plasmodium berghei; Pyridazines; Pyrimidines | 2017 |