Page last updated: 2024-09-05

etravirine and nelfinavir

etravirine has been researched along with nelfinavir in 4 studies

Compound Research Comparison

Studies
(etravirine)
Trials
(etravirine)
Recent Studies (post-2010)
(etravirine)
Studies
(nelfinavir)
Trials
(nelfinavir)
Recent Studies (post-2010) (nelfinavir)
572903211,240230240

Protein Interaction Comparison

ProteinTaxonomyetravirine (IC50)nelfinavir (IC50)
Tyrosine-protein kinase FynHomo sapiens (human)7.971
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)8.852
ATP-dependent translocase ABCB1Homo sapiens (human)3.3938
Cytochrome P450 3A4Homo sapiens (human)1.275
ATP-dependent translocase ABCB1Mus musculus (house mouse)2.3
Sodium-dependent noradrenaline transporter Homo sapiens (human)8.852
Protease Human immunodeficiency virus 10.53
Protease Human immunodeficiency virus 10.0054

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (75.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Doak, AK; Prusiner, SB; Shoichet, BK; Wille, H1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Cruz, JP; Machado, M; Mendes, AM; PrudĂȘncio, M; Sanches-Vaz, M1

Reviews

1 review(s) available for etravirine and nelfinavir

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

3 other study(ies) available for etravirine and nelfinavir

ArticleYear
Colloid formation by drugs in simulated intestinal fluid.
    Journal of medicinal chemistry, 2010, May-27, Volume: 53, Issue:10

    Topics: Buffers; Chemical Precipitation; Colloids; Intestine, Small; Light; Microscopy, Electron, Transmission; Pharmaceutical Preparations; Scattering, Radiation; Solubility

2010
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Inhibition of
    Frontiers in cellular and infection microbiology, 2017, Volume: 7

    Topics: Alkynes; Animals; Anti-Retroviral Agents; Antimalarials; Benzoxazines; Cell Line; Cyclopropanes; Disease Models, Animal; Hepatocytes; Humans; Malaria; Male; Mice, Inbred C57BL; Nelfinavir; Nitriles; Plasmodium berghei; Pyridazines; Pyrimidines

2017