Page last updated: 2024-09-05

etravirine and methadone

etravirine has been researched along with methadone in 3 studies

Compound Research Comparison

Studies
(etravirine)
Trials
(etravirine)
Recent Studies (post-2010)
(etravirine)
Studies
(methadone)
Trials
(methadone)
Recent Studies (post-2010) (methadone)
5729032113,6301,4633,957

Protein Interaction Comparison

ProteinTaxonomyetravirine (IC50)methadone (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)7.5
Mu-type opioid receptorHomo sapiens (human)0.0041
Delta-type opioid receptorHomo sapiens (human)1.09
Kappa-type opioid receptorHomo sapiens (human)0.512
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)9.7724

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
De Smedt, G; Hoetelmans, RM; Kakuda, TN; Peeters, M; Schöller-Gyüre, M; Stevens, T; van den Brink, W; Vanaken, H; Vandermeulen, K; Woodfall, B1
Garcés, PA; Tena, EV1

Reviews

2 review(s) available for etravirine and methadone

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
[Etravirine in first-line therapy].
    Enfermedades infecciosas y microbiologia clinica, 2009, Volume: 27 Suppl 2

    Topics: Anti-HIV Agents; Chemical and Drug Induced Liver Injury; Drug Eruptions; Drug Interactions; Drug Resistance, Multiple, Viral; Genes, pol; Hepatitis, Viral, Human; Heroin Dependence; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Mental Disorders; Methadone; Multicenter Studies as Topic; Nitriles; Patient Compliance; Pyridazines; Pyrimidines; Randomized Controlled Trials as Topic; Reverse Transcriptase Inhibitors; Substance Abuse, Intravenous

2009

Trials

1 trial(s) available for etravirine and methadone

ArticleYear
Pharmacokinetic and pharmacodynamic study of the concomitant administration of methadone and TMC125 in HIV-negative volunteers.
    Journal of clinical pharmacology, 2008, Volume: 48, Issue:3

    Topics: Adult; Area Under Curve; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Exanthema; Headache; HIV Seronegativity; Humans; Male; Metabolic Clearance Rate; Methadone; Middle Aged; Nausea; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors; Stereoisomerism; Tablets

2008