etravirine has been researched along with loviride in 4 studies
Studies (etravirine) | Trials (etravirine) | Recent Studies (post-2010) (etravirine) | Studies (loviride) | Trials (loviride) | Recent Studies (post-2010) (loviride) |
---|---|---|---|---|---|
572 | 90 | 321 | 34 | 12 | 4 |
Protein | Taxonomy | etravirine (IC50) | loviride (IC50) |
---|---|---|---|
Protease | Human immunodeficiency virus 1 | 0.5 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (25.00) | 29.6817 |
2010's | 3 (75.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
De Corte, BL | 1 |
De Clercq, E; Li, D; Liu, X; Zhan, P | 1 |
Gu, SX; Ju, XL; Liu, GY; Lu, HH; Zhu, YY | 1 |
Annaert, P; Augustijns, P; Bevernage, J; Brouwers, J; Forier, T; Tack, J | 1 |
2 review(s) available for etravirine and loviride
Article | Year |
---|---|
From 4,5,6,7-tetrahydro-5-methylimidazo[4,5,1-jk](1,4)benzodiazepin-2(1H)-one (TIBO) to etravirine (TMC125): fifteen years of research on non-nucleoside inhibitors of HIV-1 reverse transcriptase.
Topics: Anti-HIV Agents; Benzodiazepines; Drug Design; Drug Resistance, Viral; HIV Reverse Transcriptase; Imidazoles; Nitriles; Pyridazines; Pyrimidines; Reverse Transcriptase Inhibitors | 2005 |
Advances in diarylpyrimidines and related analogues as HIV-1 nonnucleoside reverse transcriptase inhibitors.
Topics: Anti-HIV Agents; HIV Infections; HIV Reverse Transcriptase; HIV-1; Humans; Molecular Docking Simulation; Pyrimidines; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 2018 |
2 other study(ies) available for etravirine and loviride
Article | Year |
---|---|
Strategies for the design of HIV-1 non-nucleoside reverse transcriptase inhibitors: lessons from the development of seven representative paradigms.
Topics: Anti-HIV Agents; Benzodiazepines; Binding Sites; Crystallography, X-Ray; Drug Design; HIV Reverse Transcriptase; HIV-1; Hydrogen Bonding; Imidazoles; Indoles; Nitriles; Reverse Transcriptase Inhibitors; Structure-Activity Relationship | 2012 |
Excipient-mediated supersaturation stabilization in human intestinal fluids.
Topics: Acetamides; Acetophenones; Adult; Body Fluids; Danazol; Excipients; Female; Fenofibrate; Humans; Intestines; Male; Nitriles; Pharmaceutical Preparations; Polymers; Pyridazines; Pyrimidines; Ritonavir; Solubility; Young Adult | 2011 |