Page last updated: 2024-08-23

etorphine and methadone

etorphine has been researched along with methadone in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-199015 (60.00)18.7374
1990's7 (28.00)18.2507
2000's3 (12.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Govoni, S; Kumakura, K; Spano, PF; Tonon, GC; Trabucchi, M1
Kapitsopoulos, G; Makhay, MM; Young, AM1
Culpepper-Morgan, J; Holt, PR; Kreek, MJ; LaRoche, D; O'Bryan, L; Zhang, J1
Carino, MA; Horita, A; Yamawaki, S1
Gibson, A; Vernadakis, A1
Hynes, MD; Leander, JD; Reel, JK; Zimmerman, DM1
Frank, GB; Shetty, SS1
Appia, F; Chariot, J; Rozé, C; Vaille, C1
Clouet, DH; Yonehara, N1
Paktor, J; Vaught, JL1
Cochin, J; Miller, JM; Pelikan, EW; Rosow, CE1
Goldstein, FJ; Malseed, RT; Ossipov, MH1
Gibson, DA; Vernadakis, A1
Busse, LW; Fujimoto, JM; Lange, DG; Roerig, SC1
Clouet, DH; Williams, N1
Cai, ZJ; Ge, Y; Li, M; Sun, WL1
Blake, AD; Bot, G; Freeman, JC; Reisine, T1
Blake, AD; Bot, G; Li, S; Reisine, T1
Cheng, LX; Sha, LJ; Zhang, ZX1
Gong, ZH; Liu, JG; Qin, BY2
Aibak, H; Beaudet, A; Cahill, CM; Collier, B; Esdaile, MJ; Kieffer, BL; Morinville, A1
Arttamangkul, S; Low, MJ; Pintar, J; Quillinan, N; von Zastrow, M; Williams, JT1
Dighe, SV; Madia, PA; Sirohi, S; Walker, EA; Yoburn, BC1

Reviews

1 review(s) available for etorphine and methadone

ArticleYear
Biochemical reactions between opiate receptor binding and inhibition of neurotransmission.
    NIDA research monograph, 1984, Volume: 54

    Topics: Adenylyl Cyclases; Animals; Brain Chemistry; Calcium; Calmodulin; Etorphine; Humans; Methadone; Molecular Weight; Morphine; Narcotics; Nerve Endings; Nerve Tissue Proteins; Opioid-Related Disorders; Phosphodiesterase Inhibitors; Phosphorylation; Protein Binding; Protein Kinases; Receptors, Opioid; Synaptic Transmission

1984

Trials

1 trial(s) available for etorphine and methadone

ArticleYear
[Colonic dialysis therapy of Chinese herbal medicine in abstinance of heroin addicts--report of 75 cases].
    Zhongguo Zhong xi yi jie he za zhi Zhongguo Zhongxiyi jiehe zazhi = Chinese journal of integrated traditional and Western medicine, 1997, Volume: 17, Issue:2

    Topics: Adolescent; Adult; Analgesics, Opioid; Colon; Dialysis; Drugs, Chinese Herbal; Etorphine; Female; Follow-Up Studies; Heroin Dependence; Humans; Male; Methadone

1997

Other Studies

23 other study(ies) available for etorphine and methadone

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Interaction of narcotic analgesics with dopamine receptors in rat brain.
    Pharmacological research communications, 1975, Volume: 07, Issue:1

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Corpus Striatum; Cyclic AMP; Depression, Chemical; Dextromoramide; Dextropropoxyphene; Dopamine; Enzyme Activation; Etorphine; Fentanyl; In Vitro Techniques; Male; Methadone; Rats; Receptors, Drug

1975
Tolerance to morphine-like stimulus effects of mu opioid agonists.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 257, Issue:2

    Topics: Animals; Buprenorphine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Tolerance; Etorphine; Male; Methadone; Morphine; Rats; Rats, Inbred Strains

1991
Orally administered kappa as well as mu opiate agonists delay gastrointestinal transit time in the guinea pig.
    Life sciences, 1988, Volume: 42, Issue:21

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Administration, Oral; Animals; Etorphine; Gastrointestinal Motility; Guinea Pigs; Male; Methadone; Morphine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1988
Analeptic effect of opiate receptor agonists in rabbits.
    Neuroscience letters, 1985, Mar-22, Volume: 55, Issue:1

    Topics: Animals; Arousal; Brain; Central Nervous System Stimulants; Codeine; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Ethylketocyclazocine; Etorphine; Male; Meperidine; Methadone; Morphine; Naltrexone; Narcotics; Phenazocine; Rabbits; Receptors, Opioid; Reflex

1985
Neurotoxicity of opiates during brain development: in vivo and in vitro studies.
    Progress in clinical and biological research, 1985, Volume: 163C

    Topics: Abnormalities, Drug-Induced; Animals; Binding Sites; Brain; Cells, Cultured; Chick Embryo; Etorphine; In Vitro Techniques; Methadone; Methadyl Acetate; Neurons; Receptors, Opioid; Tritium

1985
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Biological Assay; Buprenorphine; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Etorphine; Fentanyl; Methadone; Mice; Morphine; Muscle Contraction; Nalbuphine; Nalorphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, mu

1987
Mechanism for the opioid-induced twitch potentiations of frog's skeletal muscle.
    Canadian journal of physiology and pharmacology, 1986, Volume: 64, Issue:7

    Topics: Animals; Calcium; Dextrorphan; Etorphine; In Vitro Techniques; Meperidine; Methadone; Morphine; Muscle Contraction; Muscles; Narcotics; Rana pipiens; Stimulation, Chemical

1986
Etorphine inhibition of pancreatic exocrine secretion in rats: comparison with methadone.
    European journal of pharmacology, 1986, Feb-11, Volume: 121, Issue:1

    Topics: Anesthesia; Animals; Deoxyglucose; Diprenorphine; Electric Stimulation; Etorphine; Male; Methadone; Morphinans; Naloxone; Pancreas; Rats; Rats, Inbred Strains; Time Factors; Vagus Nerve

1986
Differential analgesic cross-tolerance to morphine between lipophilic and hydrophilic narcotic agonists.
    Life sciences, 1984, Jan-02, Volume: 34, Issue:1

    Topics: Analgesics, Opioid; Animals; Blood-Brain Barrier; Dose-Response Relationship, Drug; Drug Tolerance; Etorphine; Injections, Intraventricular; Injections, Subcutaneous; Male; Methadone; Mice; Morphine; Morphine Derivatives; Narcotics; Receptors, Opioid

1984
Opiates and thermoregulation in mice. I. Agonists.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 213, Issue:2

    Topics: Animals; Benzimidazoles; Body Temperature Regulation; Codeine; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Hydromorphone; Isonipecotic Acids; Levorphanol; Male; Meperidine; Methadone; Mice; Morphine; Narcotics; Oxymorphone

1980
Feline analgesia following central administration of opioids.
    Neuropharmacology, 1984, Volume: 23, Issue:8

    Topics: Analgesia; Animals; Cats; Etorphine; Injections, Subcutaneous; Male; Methadone; Microinjections; Morphine; Narcotics; Periaqueductal Gray; Reaction Time

1984
Effects of N-LAAM on [3H]etorphine binding in neuronal-enriched cell cultures.
    Neurochemical research, 1983, Volume: 8, Issue:9

    Topics: Animals; Binding Sites; Brain; Cells, Cultured; Chick Embryo; Etorphine; Guanosine Triphosphate; Magnesium; Methadone; Methadyl Acetate; Morphinans; Narcotics; Neurons; Sodium; Tritium

1983
Withdrawal tolerance and unidirectional non-cross-tolerance in narcotic pellet-implanted mice.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Drug Implants; Drug Tolerance; Etorphine; Heroin; Humans; Male; Methadone; Mice; Morphine; Narcotics; Opioid-Related Disorders; Solubility; Substance Withdrawal Syndrome

1983
The role of calmodulin in opioid-induced changes in the phosphorylation of rat striatal synaptic membrane proteins.
    Neurochemical research, 1982, Volume: 7, Issue:9

    Topics: Animals; Calcium; Calcium-Binding Proteins; Calmodulin; Corpus Striatum; Etorphine; Kinetics; Male; Membrane Proteins; Methadone; Morphinans; Morphine; Phosphorylation; Protein Kinases; Rats; Synaptic Membranes; Synaptosomes

1982
[Clinical assessment of physical dependence potential of dihydroetorphine hydrochloride (DHE)].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1994, Volume: 29, Issue:4

    Topics: Administration, Sublingual; Adolescent; Adult; Analgesics, Opioid; Etorphine; Female; Heroin; Heroin Dependence; Humans; Male; Methadone; Substance Withdrawal Syndrome; Substance-Related Disorders

1994
Differential opioid agonist regulation of the mouse mu opioid receptor.
    The Journal of biological chemistry, 1997, Jan-10, Volume: 272, Issue:2

    Topics: Adenylate Cyclase Toxin; Analgesics; Animals; Buprenorphine; Colforsin; Cyclic AMP; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Levorphanol; Methadone; Mice; Morphine; Pertussis Toxin; Receptors, Opioid, mu; Virulence Factors, Bordetella

1997
Opioid regulation of the mouse delta-opioid receptor expressed in human embryonic kidney 293 cells.
    Molecular pharmacology, 1997, Volume: 52, Issue:2

    Topics: Adenylyl Cyclases; Animals; Antibodies, Monoclonal; Cell Line; Colforsin; Cyclic AMP; Down-Regulation; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; GTP-Binding Proteins; Humans; Methadone; Mice; Morphine; Point Mutation; Radioligand Assay; Receptors, Opioid, delta; Signal Transduction; Structure-Activity Relationship

1997
Effects of opioid receptor agonists on cAMP second messenger system.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:5

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Buprenorphine; Cyclic AMP; Etorphine; Glioma; Humans; Hybrid Cells; Methadone; Morphine; Neuroblastoma; Opioid-Related Disorders; Receptors, Opioid; Receptors, Opioid, delta; Tumor Cells, Cultured

1999
Effects of low-pH treatment on cAMP second messenger system regulated by different opioid agonists.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1999, Volume: 20, Issue:6

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Buprenorphine; Cyclic AMP; Etorphine; Glioma; Humans; Hybrid Cells; Hydrogen-Ion Concentration; Methadone; Morphine; Neuroblastoma; Opioid-Related Disorders; Receptors, Opioid, delta; Tumor Cells, Cultured

1999
Regulation of delta-opioid receptor trafficking via mu-opioid receptor stimulation: evidence from mu-opioid receptor knock-out mice.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Jun-15, Volume: 23, Issue:12

    Topics: Animals; Area Under Curve; Behavior, Animal; Cell Membrane; Dose-Response Relationship, Drug; Drug Administration Schedule; Etorphine; Female; Fentanyl; Male; Methadone; Mice; Mice, Inbred C57BL; Mice, Knockout; Morphine; Narcotics; Pain Measurement; Posterior Horn Cells; Protein Transport; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Time; Up-Regulation

2003
Differential activation and trafficking of micro-opioid receptors in brain slices.
    Molecular pharmacology, 2008, Volume: 74, Issue:4

    Topics: Analgesics, Opioid; Animals; Brain; Chelating Agents; Egtazic Acid; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fluorescent Antibody Technique, Direct; Locus Coeruleus; Methadone; Mice; Mice, Knockout; Mice, Transgenic; Morphine; Neurons; Oxycodone; Oxymorphone; Protein Transport; Radioligand Assay; Receptors, Opioid, mu; Recombinant Fusion Proteins; Time Factors

2008
Dosing protocol and analgesic efficacy determine opioid tolerance in the mouse.
    Psychopharmacology, 2009, Volume: 207, Issue:3

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Tolerance; Etorphine; Hydrocodone; Infusions, Intravenous; Male; Methadone; Mice; Oxycodone

2009