etorphine has been researched along with diprenorphine in 96 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 64 (66.67) | 18.7374 |
| 1990's | 24 (25.00) | 18.2507 |
| 2000's | 7 (7.29) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 1 (1.04) | 2.80 |
| Authors | Studies |
|---|---|
| Klein, P; Nelson, WL | 1 |
| Portoghese, PS; Takemori, AE | 1 |
| Bernard, D; Coop, A; MacKerell, AD | 1 |
| Casella, G; Clouet, DH; Mulé, SJ | 1 |
| Atweh, SF; Kuhar, MJ | 3 |
| Braestrup, C; Squires, RF | 1 |
| Herz, A; Höllt, V | 1 |
| Bongso, TA; Perera, BM | 1 |
| Nowrouzian, I; Schels, HF | 1 |
| Denis, JP; Grange, M | 1 |
| Hillidge, CJ | 1 |
| Magonigle, RA; Stauber, EH; Vaughn, HW | 1 |
| Bush, M; Ensley, PK; Mehren, K; Rapley, W | 1 |
| Farnsworth, RJ; Stowe, CM | 1 |
| Hillidge, CJ; Lees, P | 2 |
| Rafferty, GC | 1 |
| Edwards, RH; Evans, CJ; Keith, DE; Magendzo, K; Morrison, H | 1 |
| Meunier, JC; Mollereau, C; Puget, A; Roussin-Pascaud, A | 1 |
| Attali, B; Vogel, Z | 1 |
| Frances, B; Meunier, JC; Moisand, C; Puget, A | 1 |
| Levy, R; Simantov, R | 1 |
| von Hegel, G; Wiesner, H | 1 |
| Baillat, G; Mazarguil, H; Meunier, JC; Mollereau, C; Pascaud, A; Puget, A | 2 |
| Law, PY; Loh, HH; Louie, AK; Zhan, JN | 1 |
| Cros, J; Francés, B; Meunier, JC; Porthé, G; Verrier, B | 1 |
| Frances, B; Meunier, JC; Moisand, C | 1 |
| Livett, BG; Marley, PD | 1 |
| Hom, DS; Law, PY; Loh, HH; Ungar, HG | 1 |
| Curell, J; Hitzemann, R; Murphy, M | 1 |
| Cho, TM; Nozaki, M | 1 |
| Costa, T; Gramsch, C; Herz, A; Wüster, M | 1 |
| Richards, ML; Sadée, W | 1 |
| Richards, ML; Sadée, W; Yu, VC | 1 |
| Charness, ME; Diamond, I; Querimit, LA | 1 |
| Klein, C; Levy, R; Simantov, R | 1 |
| Frances, B; Jauzac, P; Meunier, JC; Moisand, C; Puget, A | 1 |
| Brown, SR; Cox, BM; Puttfarcken, P; Werling, LL | 1 |
| Bunn, SJ; Livett, BG; Marley, PD | 1 |
| Bunn, SJ; Marley, PD | 1 |
| Asa, CS; Eagle, TC; Plotka, ED; Seal, US; Siniff, DB; Tester, JR | 1 |
| Dorr, L; Kock, R; Pearce, PC | 1 |
| Barron, BA; Hexum, TD | 1 |
| Appia, F; Chariot, J; Rozé, C; Vaille, C | 1 |
| Cho, TM; Yamato, C | 1 |
| Law, PY; Tao, PL | 1 |
| Frances, B; Jauzac, P; Meunier, JC; Puget, A | 1 |
| Grevel, J; Richards, ML; Rosenbaum, JS; Sadée, W | 1 |
| Klee, WA; Koski, G; Simonds, WF | 1 |
| Cho, JS; Cho, TM; Loh, HH; Yamato, C | 1 |
| Brase, DA | 1 |
| Cuénoud, S; Fulpius, BW; Rüegg, UT; Simon, EJ | 1 |
| Herz, A; Rosenbaum, JS; Sadée, W | 1 |
| Kurowski, M; Perry, DC; Rosenbaum, JS; Sadée, W | 1 |
| Tolkovsky, AM | 1 |
| Brown, DR; Holtzman, SG; Locke, KW | 1 |
| Meunier, JC; Puget, A | 1 |
| Cho, TM; Ge, BL; Loh, HH; Smith, AP; Yamato, C | 1 |
| Jauzac, P; Meunier, JC; Puget, A | 2 |
| Gioannini, TL; Hiller, JM; Itzhak, Y; Simon, EJ | 1 |
| Holford, NH; Rosenbaum, JS; Sadée, W | 1 |
| Aman, RA; Holford, NH; Richards, ML; Rosenbaum, JS; Sadée, W | 1 |
| DeRossett, SE; Holtzman, SG | 1 |
| Costa, E; Guidotti, A; Hanbauer, I; Saiani, L | 1 |
| Fisker, AV; Philipsen, HP; Stage, I | 1 |
| Becker, M; Beglinger, R | 1 |
| Hattingh, J; Knox, CM; Raath, JP | 1 |
| Jauzac, P; Polastron, J | 1 |
| Crain, SM; Shen, KF | 1 |
| Jauzac, P; Mazarguil, H; Meunier, JC; Mur, M; Polastron, J; Puget, A | 1 |
| Chin, H; Kim, DS; Klee, WA | 1 |
| Feigenbaum, JJ; Simantov, R | 1 |
| Butour, JL; Meunier, JC; Moisand, C; Mollereau, C; Parmentier, M | 1 |
| Blake, AD; Bot, G; Freeman, JC; Reisine, T | 1 |
| Osofsky, SA | 1 |
| Ralph, HK; Vogelnest, L | 1 |
| Grandy, DK; Hirota, K; Hirst, RA; Lambert, DG | 1 |
| Bertin, B; Capeyrou, R; Corbani, M; Emorine, LJ; Lepage, JF; Riond, J | 1 |
| Boardman, WS; Geiser, D; Jensen, J; Loomis, MR; Mehren, KG; Ramsay, EC | 1 |
| Calvo, F; Castanas, E; Hatzoglou, A; Martin, PM; Panagiotou, S | 1 |
| Burd, AL; El-Kouhen, R; Erickson, LJ; Law, PY; Loh, HH | 1 |
| Emorine, LJ; Exner, T; Gaibelet, G; Liaubet, L; Masson, JM; Meilhoc, E; Nürnberg, B; Riond, J; Saves, I | 1 |
| Chen, J; Chi, ZQ; Li, CL; Pei, G; Shen, QX; Wang, CH; Wei, Q; Zhou, DH | 1 |
| Akil, H; Lee, KO; Traynor, JR; Woods, JH | 1 |
| Russell, M | 1 |
| Ambuehl, M; Giacometti, M; Janovsky, M; Tataruch, F | 1 |
| Gafni, M; Keren, O; Sarne, Y; Shapira, M | 1 |
| Buss, PE; Meltzer, DG | 1 |
| Gafni, M; Sarne, Y; Shapira, M | 1 |
| Chen, C; Chong, PL; Huang, P; Liu-Chen, LY; Xu, W; Yoon, SI | 1 |
| Chen, C; Chong, PL; Huang, P; Liu-Chen, LY; Unterwald, EM; Xu, W; Yoon, SI | 1 |
| Beytell, P; du Preez, JH; du Preez, P; Felippe, J; Gleed, RD; Jago, M; Kotting, B; Manuel, B; Miller, MA; Morkel, E; Morkel, PV; Parry, SA; Radcliffe, RW | 1 |
1 review(s) available for etorphine and diprenorphine
| Article | Year |
|---|---|
In vivo receptor occupation by opiates and correlation to the pharmacological effect.
Topics: Animals; Binding Sites; Brain; Cerebellum; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Mice; Naltrexone; Narcotics; Rats; Receptors, Opioid; Stereoisomerism | 1978 |
1 trial(s) available for etorphine and diprenorphine
| Article | Year |
|---|---|
THE PULMONARY AND METABOLIC EFFECTS OF SUSPENSION BY THE FEET COMPARED WITH LATERAL RECUMBENCY IN IMMOBILIZED BLACK RHINOCEROSES (DICEROS BICORNIS) CAPTURED BY AERIAL DARTING.
Topics: Animals; Animals, Wild; Diprenorphine; Energy Metabolism; Etorphine; Female; Hypnotics and Sedatives; Immobilization; Male; Naltrexone; Narcotic Antagonists; Perissodactyla; Posture; Respiratory Physiological Phenomena | 2021 |
94 other study(ies) available for etorphine and diprenorphine
| Article | Year |
|---|---|
O3-(2-carbomethoxyallyl) ethers of opioid ligands derived from oxymorphone, naltrexone, etorphine, diprenorphine, norbinaltorphimine, and naltrindole. Unexpected O3-dealkylation in the opioid radioligand displacement assay.
Topics: Alkylation; Animals; Brain; Diprenorphine; Drug Stability; Ethers; Etorphine; Guinea Pigs; Indoles; Methacrylates; Molecular Structure; Morphinans; Naltrexone; Narcotic Antagonists; Narcotics; Oxymorphone; Phenols; Radioligand Assay; Receptors, Opioid; Tritium | 1992 |
Different receptor sites mediate opioid agonism and antagonism.
Topics: Animals; Binding Sites; Kinetics; Naltrexone; Narcotic Antagonists; Narcotics; Receptors, Opioid; Structure-Activity Relationship | 1983 |
Quantitative conformationally sampled pharmacophore for delta opioid ligands: reevaluation of hydrophobic moieties essential for biological activity.
Topics: Animals; Cell Line, Tumor; Enkephalin, Leucine; Hydrophobic and Hydrophilic Interactions; Ligands; Models, Molecular; Molecular Conformation; Phenylalanine; Quantitative Structure-Activity Relationship; Rats; Receptors, Opioid, delta | 2007 |
The specificity of binding of the narcotic agonist etorphine in synaptic membranes of rat brain in vivo.
Topics: Animals; Brain; Diprenorphine; Etorphine; Male; Morphinans; Naloxone; Rats; Receptors, Neurotransmitter; Stereoisomerism; Synaptic Membranes | 1975 |
Autoradiographic localization of opiate receptors in rat brain. I. Spinal cord and lower medulla.
Topics: Afferent Pathways; Animals; Binding Sites; Diprenorphine; Etorphine; Glossopharyngeal Nerve; Male; Medulla Oblongata; Rats; Receptors, Opioid; Spinal Cord; Trigeminal Nerve; Vagus Nerve | 1977 |
Autoradiographic localization of opiate receptors in rat brain. II. The brain stem.
Topics: Animals; Autoradiography; Binding Sites; Brain Mapping; Brain Stem; Diencephalon; Diprenorphine; Etorphine; Histocytochemistry; Male; Medulla Oblongata; Mesencephalon; Optic Lobe, Nonmammalian; Pons; Rats; Receptors, Opioid | 1977 |
Autoradiographic localization of opiate receptors in rat brain. III. The telencephalon.
Topics: Amygdala; Animals; Autoradiography; Basal Ganglia; Cerebral Cortex; Diprenorphine; Etorphine; Hippocampus; Rats; Receptors, Opioid; Stereoisomerism; Telencephalon | 1977 |
Characteristics and regional distributions of two distinct [3H]naloxone binding sites in the rat brain.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cyclazocine; Diprenorphine; Etorphine; In Vitro Techniques; Male; Morphine; Nalorphine; Naloxone; Organ Specificity; Rats; Receptors, Opioid; Temperature | 1978 |
Observations on the use of etorphine alone and in combination with acepromazine maleate for immobilisation of aggressive Asian elephants (Elephas maximus).
Topics: Acepromazine; Aggression; Animals; Diprenorphine; Elephants; Etorphine; Humans; Immobilization; Male; Morphinans | 1978 |
The effects of reversible narcotic immobilisation in the Iranian camel.
Topics: Acepromazine; Animals; Camelus; Diprenorphine; Etorphine; Female; Immobilization; Iran; Male; Morphinans; Neuroleptanalgesia | 1977 |
[Various late complications observed after anesthesia of the zebu (Bos indicus) with the compound Immuobilon-Revivon ND].
Topics: Animals; Body Temperature Regulation; Cattle; Diprenorphine; Etorphine; Male; Morphinans; Neuroleptanalgesia; Pulmonary Edema | 1977 |
The influence of neuroleptanalgesia on the serum activity of muscle enzymes in ponies.
Topics: Acepromazine; Animals; Creatine Kinase; Diprenorphine; Etorphine; Female; Fructose-Bisphosphate Aldolase; Horses; Hydroxybutyrate Dehydrogenase; Male; Morphinans; Muscles; Myocardium; Neuroleptanalgesia | 1978 |
The immobilization of wapiti with etorphine hydrochloride.
Topics: Acepromazine; Animals; Artiodactyla; Diprenorphine; Etorphine; Female; Immobilization; Male; Morphinans; Time Factors | 1977 |
Immobilization of giraffes with xylazine and etorphine hydrochloride.
Topics: Animals; Animals, Zoo; Artiodactyla; Ataxia; Diprenorphine; Doxapram; Etorphine; Female; Hoof and Claw; Immobilization; Male; Mandibular Fractures; Morphinans; Salivation; Thiazines; Tooth Extraction; Xylazine | 1976 |
Depression of a newborn elk calf associated with the prepartum use of etorphine hydrochloride in the dam.
Topics: Animals; Animals, Newborn; Artiodactyla; Diprenorphine; Etorphine; Female; Immobilization; Labor Presentation; Maternal-Fetal Exchange; Morphinans; Pregnancy; Respiration | 1976 |
Proceedings: Influence of etorphine acepromazine and diprenorphine on respiratory function in ponies.
Topics: Acepromazine; Animals; Carbon Dioxide; Depression, Chemical; Diprenorphine; Drug Combinations; Etorphine; Horses; Morphinans; Oxygen; Respiration | 1975 |
Letter: Immobilon/Revivon in the bull.
Topics: Acepromazine; Animals; Cattle; Cattle Diseases; Diprenorphine; Drug Combinations; Etorphine; Male; Morphinans; Respiratory Insufficiency | 1976 |
Proceedings: Influence of etorphine, acepromazine and diprenorphine on cardiovascular function in ponies.
Topics: Acepromazine; Animals; Diprenorphine; Etorphine; Hemodynamics; Horses; Morphinans; Stimulation, Chemical; Time Factors | 1976 |
Cloning of a delta opioid receptor by functional expression.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Blotting, Northern; Blotting, Southern; Cell Line; Cyclic AMP; Diprenorphine; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; Gene Expression; Humans; Kinetics; Models, Structural; Molecular Sequence Data; Naloxone; Narcotics; Protein Structure, Secondary; Receptors, Opioid, delta; Sequence Homology, Amino Acid; Transfection; Tumor Cells, Cultured | 1992 |
Regulation by Na+ ions and GppNHp of the interaction between a G protein and the amphibian type of opioid receptor.
Topics: Animals; Digitonin; Diprenorphine; Etorphine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Membranes; Rana ridibunda; Receptors, Opioid; Sodium; Temperature | 1990 |
Characterization of kappa opiate receptors in rat spinal cord-dorsal root ganglion cocultures and their regulation by chronic opiate treatment.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cell Differentiation; Cells, Cultured; Diprenorphine; Etorphine; Ganglia, Spinal; Morphinans; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord | 1990 |
Apparent precoupling of kappa- but not mu-opioid receptors with a G protein in the absence of agonist.
Topics: Animals; Centrifugation, Density Gradient; Cerebellum; Digitonin; Diprenorphine; Etorphine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Kinetics; Membranes; Narcotic Antagonists; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium; Tritium | 1990 |
Neuronal activation regulates the expression of opioid receptors: possible role of glial-derived factors and voltage-dependent ion channels.
Topics: Animals; Brain; Calcium Channels; Cell Aggregation; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Neurons; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Channels; Tetrodotoxin; Veratridine | 1989 |
[The immobilization of giraffes].
Topics: Animals; Artiodactyla; Diprenorphine; Etorphine; Female; Hyaluronoglucosaminidase; Immobilization; Male; Xylazine | 1989 |
Characterization, solubilization and purification of an opioid receptor from the brain of the frog Rana ridibunda.
Topics: Animals; Brain; Diprenorphine; Etorphine; Kinetics; Rana ridibunda; Receptors, Opioid; Solubility | 1986 |
Modification of opioid receptor activity by acid phosphatase in neuroblastoma x glioma NG108-15 hybrid cells.
Topics: Acid Phosphatase; Animals; Chromatography, High Pressure Liquid; Cyclic AMP; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Glioma; Guanfacine; Guanidines; Hybrid Cells; Neuroblastoma; Phenylacetates; Receptors, Opioid | 1988 |
The kappa-opioid receptor from human placenta: hydrodynamic characteristics and evidence for its association with a G protein.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Binding, Competitive; Centrifugation, Density Gradient; Chromatography, Gel; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Female; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Microvilli; Oligopeptides; Placenta; Pregnancy; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride | 1988 |
5'-Guanylylimidodiphosphate decreases affinity for agonists and apparent molecular size of a frog brain opioid receptor in digitonin solution.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Digitonin; Diprenorphine; Etorphine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Molecular Weight; Rana ridibunda; Receptors, Opioid | 1988 |
Na+ ions and Gpp(NH)p selectively inhibit agonist interactions at mu- and kappa-opioid receptor sites in rabbit and guinea-pig cerebellum membranes.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzomorphans; Binding, Competitive; Cerebellum; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Guinea Pigs; Hydrogen-Ion Concentration; In Vitro Techniques; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium | 1985 |
Effects of opioid compounds on desensitization of the nicotinic response of isolated bovine adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Diprenorphine; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Methionine; Epinephrine; Etorphine; Morphine; Naloxone; Nicotine; Norepinephrine; Peptide Fragments; Potassium | 1987 |
Effects of cycloheximide and tunicamycin on opiate receptor activities in neuroblastoma X glioma NG108-15 hybrid cells.
Topics: Adenylyl Cyclase Inhibitors; Cyclic AMP; Cycloheximide; Diprenorphine; Etorphine; Glioma; Glucosamine; Humans; Hybrid Cells; Neuroblastoma; Proteins; Receptors, Opioid; Tritium; Tunicamycin | 1985 |
Opiate receptor thermodynamics: agonist and antagonist binding.
Topics: Animals; Brain; Diprenorphine; Etorphine; In Vitro Techniques; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium; Temperature; Thermodynamics | 1985 |
Effects of 5,5'-dithiobis-(2-nitrobenzoic acid) on opiate binding to both the membrane-bound receptor and the partially purified opiate receptor.
Topics: Animals; Butorphanol; Cell Membrane; Dihydromorphine; Diprenorphine; Dithionitrobenzoic Acid; Dithiothreitol; Etorphine; Morphine; Nalorphine; Naloxone; Naltrexone; Nitrobenzoates; Oxymorphone; Rats; Receptors, Opioid | 1985 |
Multiple states of opioid receptors may modulate adenylate cyclase in intact neuroblastoma X glioma hybrid cells.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cyclic AMP; Diprenorphine; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Glioma; Hybrid Cells; Kinetics; Ligands; Morphine; Naloxone; Neuroblastoma; Neurons; Receptors, Opioid; Receptors, Opioid, delta | 1985 |
In vivo opiate receptor binding of oripavines to mu, delta and kappa sites in rat brain as determined by an ex vivo labeling method.
Topics: Animals; Brain; Buprenorphine; Diprenorphine; Etorphine; Kinetics; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thebaine | 1985 |
A human neuroblastoma cell line expresses mu and delta opioid receptor sites.
Topics: Bone Neoplasms; Cell Line; Child, Preschool; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Etorphine; Female; Guanylyl Imidodiphosphate; Humans; Kinetics; Naloxone; Neuroblastoma; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Sodium Chloride | 1986 |
Ethanol increases the expression of functional delta-opioid receptors in neuroblastoma x glioma NG108-15 hybrid cells.
Topics: Cell Line; Cyclic AMP; Cycloheximide; Dactinomycin; Diprenorphine; DNA; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethanol; Etorphine; Glioma; Hybridomas; Naloxone; Neuroblastoma; Phenylisopropyladenosine; Receptors, Opioid; Receptors, Opioid, delta; Sodium; Transcription, Genetic | 1986 |
Subcellular compartmentation of opioid receptors: modulation by enkephalin and alkaloids.
Topics: Animals; Cell Line; Cell Membrane; Centrifugation, Density Gradient; Chloroquine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Glioma; Golgi Apparatus; Kinetics; Lysosomes; Microsomes; Neuroblastoma; Receptors, Opioid | 1986 |
Differential regulation of two molecular forms of a mu-opioid receptor type by sodium ions, manganese ions and by guanyl-5'-yl imidodiphosphate.
Topics: Adenylyl Cyclases; Allosteric Regulation; Animals; Cell Membrane; Cerebellum; Diprenorphine; Drug Antagonism; Etorphine; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Manganese; Molecular Weight; Protein Binding; Rabbits; Receptors, Opioid; Receptors, Opioid, mu; Sodium | 1986 |
Sodium regulation of agonist binding at opioid receptors. II. Effects of sodium replacement on opioid binding in guinea pig cortical membranes.
Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Guinea Pigs; Male; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium | 1986 |
Prostanoid responses of bovine adrenal medullary cells: lack of effect of opioids.
Topics: Adrenal Medulla; Animals; Catecholamines; Cattle; Cells, Cultured; Dinoprostone; Diprenorphine; Etorphine; Inositol Phosphates; Morphinans; Phosphatidylinositols; Prostaglandins E | 1988 |
Lack of effect of opioid compounds on angiotensin II responses of bovine adrenal medullary cells.
Topics: Adrenal Medulla; Angiotensin II; Animals; Catecholamines; Cattle; Cells, Cultured; Diprenorphine; Etorphine; Inositol Phosphates; Morphinans; Sugar Phosphates | 1988 |
Rapid reversible immobilization of feral stallions using etorphine hydrochloride, xylazine hydrochloride and atropine sulfate.
Topics: Acepromazine; Animals; Animals, Wild; Atropine; Diprenorphine; Etorphine; Horses; Immobilization; Male; Morphinans; Thiazines; Xylazine; Yohimbine | 1987 |
'Anaesthetic death' in a black fallow deer.
Topics: Acepromazine; Animals; Blood Pressure; Deer; Diprenorphine; Electrocardiography; Etorphine; Female; Heart Arrest; Immobilization; Oxygen Inhalation Therapy; Positive-Pressure Respiration; Xylazine | 1985 |
Modulation of bovine adrenal gland secretion by etorphine and diprenorphine.
Topics: Acetylcholine; Adrenal Glands; Animals; Catecholamines; Cattle; Dimethylphenylpiperazinium Iodide; Diprenorphine; Enkephalin, Methionine; Etorphine; Morphinans | 1986 |
Etorphine inhibition of pancreatic exocrine secretion in rats: comparison with methadone.
Topics: Anesthesia; Animals; Deoxyglucose; Diprenorphine; Electric Stimulation; Etorphine; Male; Methadone; Morphinans; Naloxone; Pancreas; Rats; Rats, Inbred Strains; Time Factors; Vagus Nerve | 1986 |
Possible involvements of negative cooperativity in opiate agonist receptor interactions.
Topics: Allosteric Regulation; Animals; Brain; Diprenorphine; Etorphine; In Vitro Techniques; Kinetics; Rats; Receptors, Opioid | 1984 |
Down regulation of opiate receptor in rat brain after chronic etorphine treatment.
Topics: Animals; Brain; Diprenorphine; Etorphine; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Time Factors | 1984 |
Solubilization of two molecular forms of the frog brain opioid receptor.
Topics: Animals; Brain; Diprenorphine; Etorphine; Ranidae; Receptors, Opioid; Sodium; Solubility | 1984 |
In vivo characterization of four types of opioid binding sites in rat brain.
Topics: Analgesics, Opioid; Animals; Brain; Buprenorphine; Diprenorphine; Etorphine; Fentanyl; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Sufentanil; Tritium | 1983 |
Guanine nucleotides inhibit binding of agonists and antagonists to soluble opiate receptors.
Topics: Animals; Cell Line; Cell Membrane; Diprenorphine; Etorphine; Glioma; Guanine Nucleotides; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hybrid Cells; Kinetics; Mice; Morphinans; Neuroblastoma; Rats; Receptors, Opioid | 1981 |
Solubilization of membrane bound opiate receptor from rat brain.
Topics: Animals; Brain Chemistry; Dextrorphan; Diprenorphine; Etorphine; Levorphanol; Male; Rats; Receptors, Opioid; Sodium Chloride; Solubility; Sonication; Subcellular Fractions | 1981 |
Studies on brain opiate receptor stability in vitro: inhibition of opiate receptor binding by adenosine-5'-diphosphate.
Topics: Adenine Nucleotides; Adenosine Diphosphate; Animals; Binding, Competitive; Brain; Diprenorphine; Drug Stability; Etorphine; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Structure-Activity Relationship | 1981 |
Inactivation and solubilization of opiate receptors by phospholipases A2.
Topics: Animals; Brain; Cell Membrane; Detergents; Diprenorphine; Etorphine; Kinetics; Phospholipases; Phospholipases A; Phospholipases A2; Rats; Receptors, Opioid; Solubility | 1982 |
Buprenorphine: differential interaction with opiate receptor subtypes in vivo.
Topics: Allosteric Regulation; Animals; Binding, Competitive; Brain; Buprenorphine; Diprenorphine; Etorphine; In Vitro Techniques; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid | 1982 |
[3H]-etorphine and [3H]-diprenorphine receptor binding in vitro and in vivo: differential effect of Na+ and guanylyl imidodiphosphate.
Topics: Animals; Brain; Diprenorphine; Etorphine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium | 1982 |
Etorphine binds to multiple opiate receptors of the caudate nucleus with equal affinity but with different kinetics.
Topics: Animals; Binding, Competitive; Caudate Nucleus; Diprenorphine; Edetic Acid; Etorphine; In Vitro Techniques; Kinetics; Membranes; Morphinans; Morphine; Naloxone; Receptors, Opioid; Sodium Chloride | 1982 |
Effects of opiate antagonists and putative mu- and kappa-agonists on milk intake in rat and squirrel monkey.
Topics: Animals; Buprenorphine; Cyclazocine; Diazepam; Diprenorphine; Drinking; Ethylketocyclazocine; Etorphine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Taste | 1982 |
[Opiate receptor(s) of the frog brain: soluble-phase separation of the macromolecular complexes of an agonist and an antagonist].
Topics: Animals; Brain; Centrifugation, Density Gradient; Digitonin; Diprenorphine; Etorphine; Macromolecular Substances; Ranidae; Receptors, Opioid; Solubility | 1983 |
Isolation of opiate binding components by affinity chromatography and reconstitution of binding activities.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Chromatography, Affinity; Diprenorphine; Etorphine; Kinetics; Rats; Receptors, Opioid; Structure-Activity Relationship | 1983 |
Physical separation of the agonist and antagonist forms of a mu opiate receptor?
Topics: Animals; Cell Membrane; Cerebellum; Diprenorphine; Etorphine; Morphinans; Rabbits; Receptors, Opioid; Receptors, Opioid, mu; Solubility | 1983 |
Distinct molecular forms of opiate binding in the frog brain.
Topics: Animals; Brain; Cell Membrane; Digitonin; Diprenorphine; Etorphine; Morphinans; Ranidae; Receptors, Opioid; Solubility | 1983 |
Effect of digitonin on the binding of opiate agonists and antagonists to membrane-bound and soluble opioid binding sites.
Topics: Animals; Brain; Bufo marinus; Digitonin; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Etorphine; Male; Naloxone; Oxymorphone; Rats; Rats, Inbred Strains; Receptors, Opioid; Species Specificity | 1984 |
Opiate receptor binding-effect relationship: sufentanil and etorphine produce analgesia at the mu-site with low fractional receptor occupancy.
Topics: Animals; Brain; Diprenorphine; Drug Interactions; Etorphine; Fentanyl; Morphinans; Naloxone; Pain; Rats; Receptors, Opioid; Sufentanil | 1984 |
Discrimination of three types of opioid binding sites in rat brain in vivo.
Topics: Animals; Binding, Competitive; Brain; Diprenorphine; Etorphine; Fentanyl; Male; Naloxone; Rats; Receptors, Opioid; Sufentanil | 1984 |
Effects of naloxone, diprenorphine, buprenorphine and etorphine on unpunished and punished food-reinforced responding in the squirrel monkey.
Topics: Animals; Buprenorphine; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Female; Male; Morphinans; Naloxone; Punishment; Reinforcement, Psychology; Saimiri | 1984 |
Modulation of nicotinic receptor function by opiate recognition sites highly selective for Met5-enkephalin[Arg6Phe7].
Topics: Acetylcholine; Adrenal Medulla; Animals; Binding Sites; Bungarotoxins; Cattle; Cell Membrane; Cells, Cultured; Diprenorphine; Dogs; Endorphins; Enkephalin, Methionine; Epinephrine; Etorphine; Norepinephrine; Receptors, Cholinergic; Receptors, Nicotinic; Splanchnic Nerves | 1983 |
Use of etorphine-acepromazine and diprenorphine in reversible neuroleptanalgesia of rats.
Topics: Acepromazine; Animals; Behavior, Animal; Diprenorphine; Drug Evaluation; Etorphine; Female; Male; Morphinans; Neuroleptanalgesia; Rats; Rats, Inbred Strains; Respiration | 1982 |
Effects of Immobilon and Revivon on the cardiovascular system and acid base status of the Göttingen minipig.
Topics: Acepromazine; Animals; Atropine; Cardiac Output; Cardiovascular System; Diprenorphine; Etorphine; Heart Rate; Morphinans; Myocardial Contraction; Swine; Vascular Resistance | 1980 |
Arterial blood pressure of the African elephant (Loxodonta africana) under etorphine anaesthesia and after remobilisation with diprenorphine.
Topics: Anesthesia, General; Animals; Blood Pressure; Diprenorphine; Ejaculation; Electric Stimulation; Elephants; Etorphine; Male | 1994 |
Different subtypes of opioid receptors have different affinities for G-proteins.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Amino Acid Sequence; Animals; Binding, Competitive; Cerebellum; Colforsin; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Etorphine; GTP-Binding Proteins; Guinea Pigs; Humans; Hybrid Cells; Molecular Sequence Data; Morphine; Naloxone; Neoplasm Proteins; Nerve Tissue Proteins; Neuroblastoma; Oligopeptides; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Tumor Cells, Cultured | 1994 |
Antagonists at excitatory opioid receptors on sensory neurons in culture increase potency and specificity of opiate analgesics and attenuate development of tolerance/dependence.
Topics: Analgesics; Animals; Cells, Cultured; Diprenorphine; Drug Tolerance; Electrophysiology; Enkephalin, Leucine-2-Alanine; Etorphine; Ganglia, Spinal; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Neurons, Afferent; Opioid-Related Disorders | 1994 |
SK-N-BE: a human neuroblastoma cell line containing two subtypes of delta-opioid receptors.
Topics: Adenylyl Cyclases; Binding, Competitive; Centrifugation, Density Gradient; Diprenorphine; Down-Regulation; Etorphine; GTP-Binding Proteins; Humans; Ligands; Neuroblastoma; Receptors, Opioid, delta; Tumor Cells, Cultured | 1994 |
Agonist regulation of the expression of the delta opioid receptor in NG108-15 cells.
Topics: Animals; Blotting, Northern; Cell Line; Diprenorphine; Down-Regulation; Etorphine; Hybrid Cells; Membrane Proteins; Mice; Morphine; Nalorphine; Narcotic Antagonists; Narcotics; Neuroblastoma; Rats; Receptors, Opioid, delta; RNA, Messenger | 1995 |
Lack of effect of gamma-hydroxybutyrate on mu, delta and kappa opioid receptor binding.
Topics: Adjuvants, Anesthesia; Analgesics; Animals; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Glioma; Guinea Pigs; Naloxone; Narcotic Antagonists; Narcotics; Neuroblastoma; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium Oxybate; Tritium; Tumor Cells, Cultured | 1996 |
Replacement of Gln280 by His in TM6 of the human ORL1 receptor increases affinity but reduces intrinsic activity of opioids.
Topics: Adenylyl Cyclase Inhibitors; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Diprenorphine; Dynorphins; Etorphine; Fentanyl; Glutamine; Histamine; Humans; Kinetics; Ligands; Naltrexone; Narcotic Antagonists; Narcotics; Nociceptin; Nociceptin Receptor; Opioid Peptides; Receptors, Opioid | 1996 |
Differential opioid agonist regulation of the mouse mu opioid receptor.
Topics: Adenylate Cyclase Toxin; Analgesics; Animals; Buprenorphine; Colforsin; Cyclic AMP; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Levorphanol; Methadone; Mice; Morphine; Pertussis Toxin; Receptors, Opioid, mu; Virulence Factors, Bordetella | 1997 |
A practical anesthesia monitoring protocol for free-ranging adult African elephants (Loxodonta africana).
Topics: Anesthesia; Animals; Animals, Wild; Body Temperature; Diprenorphine; Elephants; Etorphine; Female; Heart Rate; Immobilization; Male; Monitoring, Physiologic; Narcotic Antagonists; Narcotics; Oximetry; Oxygen; Pulse; Respiration | 1997 |
Chemical immobilisation of giraffe to facilitate short procedures.
Topics: Acepromazine; Analgesics, Opioid; Animals; Animals, Zoo; Antipsychotic Agents; Artiodactyla; Body Temperature; Diprenorphine; Etorphine; Female; Heart Rate; Immobilization; Injections; Male; Narcotic Antagonists; New South Wales; Preoperative Care; Respiration | 1997 |
Coupling of the cloned rat kappa-opioid receptor to adenylyl cyclase is dependent on receptor expression.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylyl Cyclases; Analgesics; Animals; Benzomorphans; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Gene Expression; Narcotic Antagonists; Phosphodiesterase Inhibitors; Pyrrolidines; Rats; Receptors, Opioid, kappa; Transfection | 1997 |
Agonist-induced signaling and trafficking of the mu-opioid receptor: role of serine and threonine residues in the third cytoplasmic loop and C-terminal domain.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Enzyme Activation; Etorphine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Morphine; Mutagenesis, Site-Directed; Receptors, Opioid, mu; Serine; Signal Transduction; Threonine | 1997 |
Chemical restraint of the Nile hippopotamus (Hippopotamus amphibius) in captivity.
Topics: Acepromazine; Adjuvants, Anesthesia; Analgesics, Opioid; Anesthetics, Inhalation; Animals; Animals, Zoo; Artiodactyla; Atropine; Body Temperature; Diprenorphine; Dopamine Antagonists; Etorphine; Fasting; Female; Heart Rate; Immobilization; Injections, Intramuscular; Isoflurane; Male; Narcotic Antagonists; Oximetry; Oxygen; Respiration; Retrospective Studies; Xylazine | 1998 |
Modulation of the estrogen-regulated proteins cathepsin D and pS2 by opioid agonists in hormone-sensitive breast cancer cell lines (MCF7 and T47D): evidence for an interaction between the two systems.
Topics: Breast Neoplasms; Cathepsin D; Cell Division; Cycloheximide; Cytosol; Diprenorphine; Dose-Response Relationship, Drug; Estradiol; Ethylketocyclazocine; Etorphine; Female; Humans; Inhibitory Concentration 50; Narcotic Antagonists; Narcotics; Neoplasms, Hormone-Dependent; Protein Synthesis Inhibitors; Proteins; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins | 1998 |
Identification of serine 356 and serine 363 as the amino acids involved in etorphine-induced down-regulation of the mu-opioid receptor.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Cell Line; Colforsin; Cyclic AMP; Diprenorphine; Down-Regulation; Etorphine; Glutamic Acid; Humans; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Protein Structure, Secondary; Receptors, Opioid, mu; Recombinant Fusion Proteins; Sequence Deletion; Serine; Transfection | 1998 |
Nonselective coupling of the human mu-opioid receptor to multiple inhibitory G-protein isoforms.
Topics: Binding Sites; Binding, Competitive; Buprenorphine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Etorphine; Gene Expression; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Protein Binding; Protein Isoforms; Receptors, Opioid, mu; Recombinant Proteins; Saccharomyces cerevisiae; Spheroplasts; Transformation, Genetic | 1999 |
Human mu-opioid receptor overexpressed in baculovirus system and its pharmacological characterizations.
Topics: Animals; Baculoviridae; Cells, Cultured; Cyclic AMP; Diprenorphine; Etorphine; Fentanyl; Gene Expression; Insecta; Radioligand Assay; Receptors, Opioid, mu; Transfection | 1998 |
Differential binding properties of oripavines at cloned mu- and delta-opioid receptors.
Topics: Analgesics, Opioid; Animals; Benzamides; Binding, Competitive; Buprenorphine; Cloning, Molecular; Diprenorphine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Naloxone; Piperazines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Sulfur Radioisotopes; Thebaine; Tritium; Tumor Cells, Cultured | 1999 |
Availability of Large Animal Immobilon and Revivon.
Topics: Animals; Diprenorphine; Drug Approval; Drug Combinations; Etorphine; Methotrimeprazine; Narcotic Antagonists; United Kingdom; Veterinary Medicine | 1999 |
A Zoletil-Rompun mixture as an alternative to the use of opioids for immobilization of feral red deer.
Topics: Acepromazine; Adrenergic alpha-Agonists; Anesthetics, Dissociative; Animals; Animals, Wild; Benzodiazepines; Blood Glucose; Deer; Diprenorphine; Drug Combinations; Etorphine; Heart Rate; Hemoglobins; Imidazoles; Immobilization; Mydriatics; Narcotic Antagonists; Oximetry; Slovakia; Statistics, Nonparametric; Tiletamine; Urea; Xylazine; Yohimbine; Zolazepam | 2000 |
Divers pathways mediate delta-opioid receptor down regulation within the same cell.
Topics: Acetylcysteine; Analgesics, Opioid; Animals; Antirheumatic Agents; Chloroquine; Cysteine Proteinase Inhibitors; Diprenorphine; Down-Regulation; Etorphine; Flavonoids; Genistein; GTP-Binding Proteins; Humans; Kidney; MAP Kinase Signaling System; Narcotic Antagonists; Neuroblastoma; Phosphorylation; Radioligand Assay; Receptors, Opioid, delta; Staurosporine; Teprotide; Transfection; Tritium; Tumor Cells, Cultured | 2001 |
Changes in respiratory function following the intramuscular administration of etorphine to boer goats (Capra hircus).
Topics: Animals; Blood Gas Analysis; Carbon Dioxide; Diprenorphine; Etorphine; Female; Goats; Immobilization; Injections, Intramuscular; Narcotic Antagonists; Narcotics; Oxygen Consumption; Partial Pressure; Respiration; Respiratory Dead Space; Respiratory Function Tests; Tidal Volume; Time Factors | 2001 |
Long-term interactions between opioid and cannabinoid agonists at the cellular level: cross-desensitization and downregulation.
Topics: Animals; Cell Line; Cell Membrane; Chlorocebus aethiops; COS Cells; Cyclic AMP; Cyclohexanols; Diprenorphine; Down-Regulation; Drug Interactions; Etorphine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Mice; Narcotic Antagonists; Rats; Receptors, Cannabinoid; Receptors, Drug; Receptors, Opioid; Receptors, Opioid, delta; Signal Transduction; Transfection | 2003 |
Cholesterol reduction by methyl-beta-cyclodextrin attenuates the delta opioid receptor-mediated signaling in neuronal cells but enhances it in non-neuronal cells.
Topics: Animals; Anticholesteremic Agents; beta-Cyclodextrins; Brain; Caveolin 1; Cell Line, Tumor; CHO Cells; Cholesterol; Cricetinae; Cricetulus; Diprenorphine; Enkephalin, D-Penicillamine (2,5)-; Etorphine; G(M1) Ganglioside; Hybrid Cells; Levorphanol; Membrane Microdomains; Membrane Proteins; Naloxone; Neurons; Oligopeptides; Receptors, Opioid, delta; Signal Transduction | 2007 |
Agonist treatment did not affect association of mu opioid receptors with lipid rafts and cholesterol reduction had opposite effects on the receptor-mediated signaling in rat brain and CHO cells.
Topics: Animals; Binding, Competitive; Brain; Caveolin 1; CHO Cells; Cholesterol; Cricetinae; Cricetulus; Diprenorphine; Dose-Response Relationship, Drug; Etorphine; Male; Membrane Microdomains; Morphine; Naloxone; Narcotic Antagonists; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Signal Transduction; Transfection | 2007 |