etorphine has been researched along with 18,19-dihydroetorphine in 59 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (13.56) | 18.7374 |
1990's | 37 (62.71) | 18.2507 |
2000's | 12 (20.34) | 29.6817 |
2010's | 2 (3.39) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
He, BL; Jin, B; Li, H | 1 |
Bian, CF; Xing, SH; Xu, PC | 1 |
Bian, CF; Chen, Y; Duan, SM; Jin, GZ; Qin, W; Xing, SH; Yu, YM | 1 |
Bian, CF; Qin, W; Xing, SH | 1 |
Huang, RH; Xu, X | 1 |
Huang, M; Qin, BY; Wang, MY; Yuan, SL | 1 |
Huang, M; Qin, BY | 2 |
Li, E; Weng, L | 1 |
Miao, H; Qin, BY | 1 |
Feng, JL; Hu, XY; Liu, F; Luo, Y | 2 |
al-Essa, LY; Iwamura, T; Kataoka, T; Kohno, K; Niwa, M; Nozaki, M; Ohta, S; Tsurumi, K | 1 |
Kamei, J; Kasuya, Y; Misawa, M; Nagase, H; Suzuki, T | 1 |
Kaneto, H; Nakamura, F; Takahashi, M; Tokuyama, S | 2 |
Cai, ZJ; Ge, Y; Li, M; Sun, WL | 1 |
Iwamoto, Y; Kamei, J; Kasuya, Y; Misawa, M; Nagase, H; Suzuki, T | 1 |
Crain, SM; Shen, KF | 1 |
Kaneto, H; Takahashi, M; Tokuyama, S | 1 |
Lu, XQ; Qin, BY; Wang, DX | 1 |
Iwamura, T; Katsumata, S; Minami, M; Nakagawa, T; Satoh, M | 1 |
Kaneto, H; Nakamura, F; Nakao, K; Takahashi, M; Tokuyama, S | 1 |
Kamei, J; Nagase, H; Suzuki, T | 1 |
Feng, J; Hu, X; Liu, F; Luo, Y | 1 |
Harris, LS; Kim, SA; Martin, TJ; Smith, JE | 1 |
Huang, C; Wang, A; Zhang, Q | 1 |
Chen, DH; Miao, H; Qin, BY; Yang, Y | 1 |
Beardsley, PM; Harris, LS | 1 |
Jin, Y; Wu, L; Xia, Y | 1 |
Aceto, MD; Bowman, ER; Harris, LS | 1 |
Ling, K; Pei, G; Pu, L; Ren, XH; Yin, DL; Zhao, J | 1 |
Bai, HQ; Li, FY; Li, Y; Wu, WR; Zhang, KR; Zheng, JW | 1 |
Cai, Z; Chen, J; Ha, Y; Ren, Y; Wang, G; Wang, W; Xie, L; Zhang, K; Zheng, J | 1 |
Hairston, CT; Harris, LS; Lutz, PO; Martin, TJ; Porreca, F | 1 |
Cheng, LX; Sha, LJ; Zhang, ZX | 1 |
Qin, BY; Wang, DX | 1 |
Chen, XP; Guo, QD; Shi, TS | 1 |
Bai, HQ; Li, N; Li, Y; Wu, WR; Zhang, KR; Zheng, JW | 1 |
Chen, MH; Li, QS; Ma, HJ; Shen, Y; Zuo, XJ | 1 |
Li, FY; Li, Y; Wu, WR; Zheng, JW | 1 |
Liu, ZH; Zhang, KG | 1 |
Akil, H; Lee, KO; Traynor, JR; Woods, JH | 1 |
Aceto, MD; Harris, LS; Ji, Z; Scates, SM | 1 |
Gong, ZH; Liu, JG; Qin, BY | 2 |
Hayashi, T; Kawase, M; Morimoto, Y; Ohmori, S; Saito, S | 2 |
Hayashi, T; Kawase, M; Morimoto, Y; Ohmori, S; Saito, S; Sugibayashi, K | 1 |
Morimoto, Y; Ohmori, S; Sugiyama, Y | 1 |
Fang, L; Kawase, M; Morimoto, Y; Ohmori, S; Saito, S | 1 |
Benyhe, S; Biyashev, D; Borsodi, A; Garadnay, S; Makleit, S; Marton, J | 1 |
Morimoto, Y; Ohmori, S | 1 |
Husbands, SM; Lewis, JW | 1 |
France, CR; Gauthier, CR; Gerak, LR | 1 |
Chen, XJ; Chi, ZQ; He, Y; Jin, WQ; Liu, ZH; Shen, QX; Zhang, HP | 1 |
Han, JS; Luo, F; Ming, XY; Wang, W | 1 |
Chi, ZQ; Liu, JG; Sun, JF; Tao, YM; Wang, YH; Xu, XJ | 1 |
Baily, P; Boom, M; Dahan, A; Niesters, M; Oksche, A; Olofsen, E; Sarton, E; Smith, KJ; van Velzen, M | 1 |
2 review(s) available for etorphine and 18,19-dihydroetorphine
Article | Year |
---|---|
Dihydroetorphine: a potent analgesic: pharmacology, toxicology, pharmacokinetics, and clinical effects.
Topics: Administration, Cutaneous; Analgesics, Opioid; Animals; Clinical Trials as Topic; Drug Tolerance; Etorphine; Humans; In Vitro Techniques; Opioid-Related Disorders; Pain, Intractable; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 2002 |
Opioid ligands having delayed long-term antagonist activity: potential pharmacotherapies for opioid abuse.
Topics: Analgesics, Opioid; Animals; Buprenorphine; Drug Evaluation, Preclinical; Etorphine; Humans; Hydromorphone; Ligands; Morphinans; Narcotic Antagonists; Receptors, Opioid, mu; Structure-Activity Relationship; Substance-Related Disorders | 2003 |
3 trial(s) available for etorphine and 18,19-dihydroetorphine
Article | Year |
---|---|
[Influence of dihydroetorphine hydrochloride and tramadol on labor pain and umbilical blood gas].
Topics: Analgesia, Obstetrical; Analgesics, Opioid; Blood Gas Analysis; Etorphine; Female; Humans; Tramadol; Umbilical Arteries; Umbilical Veins; Uterine Contraction | 1995 |
[Colonic dialysis therapy of Chinese herbal medicine in abstinance of heroin addicts--report of 75 cases].
Topics: Adolescent; Adult; Analgesics, Opioid; Colon; Dialysis; Drugs, Chinese Herbal; Etorphine; Female; Follow-Up Studies; Heroin Dependence; Humans; Male; Methadone | 1997 |
Analgesic and Respiratory Depressant Effects of R-dihydroetorphine: A Pharmacokinetic-Pharmacodynamic Analysis in Healthy Male Volunteers.
Topics: Adolescent; Adult; Analgesia; Analgesics, Opioid; Dose-Response Relationship, Drug; Double-Blind Method; Etorphine; Healthy Volunteers; Humans; Infusions, Intravenous; Male; Middle Aged; Pain Measurement; Respiratory Insufficiency; Young Adult | 2019 |
54 other study(ies) available for etorphine and 18,19-dihydroetorphine
Article | Year |
---|---|
[Narcotics combined with low-flow nitrous oxide in open-heart surgery].
Topics: Adolescent; Analgesics, Opioid; Anesthesia; Cardiac Surgical Procedures; Child; Etorphine; Female; Fentanyl; Heart Septal Defects, Ventricular; Humans; Male; Morphinans; Nitrous Oxide | 1986 |
[The interactions between dihydroetorphine, L-tetrahydropalmatine, B-7601 and diazepam].
Topics: Alkaloids; Anesthesia, General; Anesthesia, Intravenous; Animals; Antipsychotic Agents; Benzilates; Berberine Alkaloids; Diazepam; Dogs; Drug Interactions; Etorphine; Female; Male; Mice; Morphinans; Piperidines; Rabbits | 1986 |
[Interaction of analgesics and l-stepholidine].
Topics: Analgesics; Animals; Berberine; Berberine Alkaloids; Dogs; Drug Synergism; Electroencephalography; Etorphine; Female; Heart Rate; Male; Meperidine; Mice; Pain; Rabbits; Respiration; Sensory Thresholds | 1986 |
Relationship between dihydroetorphine and cholinergic system in the inhibition of respiration and heart rate.
Topics: Animals; Atropine; Cerebral Ventricles; Etorphine; Heart Rate; Injections, Intraventricular; Morphinans; Pilocarpine; Rabbits; Respiration | 1986 |
[Phosphorimetric method for the determination of dihydroetorphine and its application].
Topics: Animals; Brain Chemistry; Etorphine; Mice; Morphinans; Rabbits | 1988 |
[Pharmacodynamics and pharmacokinetics of dihydroetorphine hydrochloride administered sublingually in mice and rats].
Topics: Administration, Sublingual; Analgesics; Animals; Biological Availability; Etorphine; Female; Male; Mice; Morphinans | 1988 |
[Analgesic and other CNS depressive effects of dihydroetorphine (author's transl)].
Topics: Analgesics; Animals; Dogs; Etorphine; Female; Immobilization; Male; Mice; Morphinans; Motor Activity; Nalorphine; Rabbits; Respiration | 1982 |
[Physical dependence of dihydroetorphine in mice and monkeys (author's transl)].
Topics: Analgesics; Animals; Etorphine; Female; Humans; Macaca mulatta; Male; Mice; Morphinans; Morphine Dependence; Opioid-Related Disorders; Substance Withdrawal Syndrome | 1982 |
Influences of locus coeruleus lesions and reserpine treatment on opioid physical dependence in rats.
Topics: Animals; Body Weight; Etorphine; Female; Locus Coeruleus; Male; Morphine Dependence; Neurons; Opioid-Related Disorders; Rats; Rats, Wistar; Reserpine; Substance Withdrawal Syndrome | 1995 |
Identification of dihydroetorphine in biological fluids by gas chromatography-mass spectrometry.
Topics: Etorphine; Gas Chromatography-Mass Spectrometry; Humans; Imidazoles; Methylene Chloride; Sensitivity and Specificity; Substance-Related Disorders | 1995 |
Opioid receptor interaction and adenylyl cyclase inhibition of dihydroetorphine: direct comparison with etorphine.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Brain; Etorphine; Gerbillinae; Guinea Pigs; Humans; Male; Placenta; Rats; Rats, Wistar; Receptors, Opioid | 1995 |
Antinociceptive effect of dihydroetorphine in diabetic mice.
Topics: Analgesia; Analgesics, Opioid; Animals; Binding, Competitive; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Etorphine; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Male; Mice; Mice, Inbred ICR; Naloxone; Naltrexone; Narcotic Antagonists; Pain Measurement; Receptors, Opioid, delta; Receptors, Opioid, mu | 1995 |
Physical dependence produced by dihydroetorphine in mice.
Topics: Analgesics; Animals; Etorphine; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Morphine Dependence; Naloxone; Opioid-Related Disorders; Substance Withdrawal Syndrome | 1994 |
[Monitoring of dihydroetorphine hydrochloride in biological fluid].
Topics: Etorphine; Gas Chromatography-Mass Spectrometry; Humans; Substance Abuse Detection | 1994 |
[Clinical assessment of physical dependence potential of dihydroetorphine hydrochloride (DHE)].
Topics: Administration, Sublingual; Adolescent; Adult; Analgesics, Opioid; Etorphine; Female; Heroin; Heroin Dependence; Humans; Male; Methadone; Substance Withdrawal Syndrome; Substance-Related Disorders | 1994 |
Antitussive effect of dihydroetorphine in mice.
Topics: Alkylating Agents; Animals; Antitussive Agents; Cough; Dose-Response Relationship, Drug; Etorphine; Injections, Intraperitoneal; Male; Mice; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1994 |
Antagonists at excitatory opioid receptors on sensory neurons in culture increase potency and specificity of opiate analgesics and attenuate development of tolerance/dependence.
Topics: Analgesics; Animals; Cells, Cultured; Diprenorphine; Drug Tolerance; Electrophysiology; Enkephalin, Leucine-2-Alanine; Etorphine; Ganglia, Spinal; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Neurons, Afferent; Opioid-Related Disorders | 1994 |
Antinociceptive effect of dihydroetorphine and its tolerance/dependence liability in mice.
Topics: Analgesics; Animals; Body Weight; Drug Tolerance; Etorphine; Male; Mice; Mice, Inbred Strains; Morphine; Motor Activity; Naloxone; Naltrexone; Narcotic Antagonists; Pain Measurement; Substance-Related Disorders | 1993 |
Dihydroetorphine is a mu-receptor-selective ligand.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Etorphine; Injections, Intraventricular; Mice; Radioligand Assay; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1995 |
Pharmacological study of dihydroetorphine in cloned mu-, delta- and kappa-opioid receptors.
Topics: Animals; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Etorphine; Narcotic Antagonists; Narcotics; Pertussis Toxin; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Proteins; Virulence Factors, Bordetella | 1995 |
A potent mu-opioid receptor agonist, dihydroetorphine, fails to produce the conditioned place preference in mice.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Choice Behavior; Conditioning, Operant; Conditioning, Psychological; Dose-Response Relationship, Drug; Etorphine; Male; Mice; Morphine; Morphine Dependence | 1996 |
Agonist and antagonist properties of dihydroetorphine for mu-opioid receptors in mice.
Topics: Analgesics, Opioid; Animals; Buprenorphine; Etorphine; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphine; Nociceptors; Pain Measurement; Receptors, Opioid, mu | 1996 |
Antinociceptive effect of dihydroetorphine following various routes of administration: a comparative study with morphine.
Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Etorphine; Male; Mice; Mice, Inbred Strains; Morphine; Pain Measurement | 1996 |
Determination of dihydroetorphine in biological fluids by gas chromatography-mass spectrometry using selected-ion monitoring.
Topics: Analgesics, Opioid; Calibration; Etorphine; Gas Chromatography-Mass Spectrometry; Humans; Hydrogen-Ion Concentration; Opioid-Related Disorders; Reference Standards; Reproducibility of Results; Solvents | 1996 |
Potent reinforcing effects of dihydroetorphine in rats.
Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Etorphine; Fentanyl; Heroin; Male; Morphine; Morphine Derivatives; Rats; Rats, Inbred F344; Substance Withdrawal Syndrome; Substance-Related Disorders | 1997 |
[Effect of dihydroetorphini hydrochloride on mice parturition].
Topics: Abdominal Pain; Analgesics, Opioid; Anesthetics, Local; Animals; Etorphine; Female; Labor, Obstetric; Mice; Morphine; Pregnancy; Procaine | 1996 |
Ultrastructural changes in rat locus coeruleus induced by chronic opioids.
Topics: Analgesics; Animals; Endoplasmic Reticulum, Rough; Etorphine; Locus Coeruleus; Male; Morphine; Myelin Sheath; Naloxone; Narcotic Antagonists; Narcotics; Neurons; Polyribosomes; Rats; Rats, Wistar; Synaptic Vesicles | 1997 |
Evaluation of the discriminative stimulus and reinforcing effects of dihydroetorphine.
Topics: Analgesics, Opioid; Animals; Discrimination Learning; Dose-Response Relationship, Drug; Etorphine; Heroin; Macaca mulatta; Male; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration; Substance-Related Disorders | 1997 |
[Clinical study on painless labor under drugs combined with acupuncture analgesia].
Topics: Acupressure; Acupuncture Analgesia; Adult; Analgesics, Opioid; Ear, External; Etorphine; Evoked Potentials, Somatosensory; Female; Humans; Labor, Obstetric; Magnetics; Pain Threshold; Pregnancy; Transcutaneous Electric Nerve Stimulation; Uterine Contraction | 1996 |
Etorphines: mu-opioid receptor-selective antinociception and low physical dependence capacity.
Topics: Analgesics, Opioid; Animals; Etorphine; Female; Macaca mulatta; Male; Mice; Mice, Inbred ICR; Pain Threshold; Receptors, Opioid, mu; Substance-Related Disorders | 1997 |
Differential neurotoxicity of etorphine-like opiates: lack of correlation with their ability to activate opiate receptors.
Topics: Animals; Cell Survival; Etorphine; Guanosine 5'-O-(3-Thiotriphosphate); Heroin; Humans; Narcotics; Neuroblastoma; Neurotoxins; PC12 Cells; Rats; Receptors, Opioid; Structure-Activity Relationship; Thebaine; Tumor Cells, Cultured | 1998 |
Involvement of mu-opioid receptors and alpha-adrenoceptors in the immunomodulatory effects of dihydroetorphine.
Topics: Adjuvants, Immunologic; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Analgesics, Opioid; Animals; Cell Division; Etorphine; Female; Immunosuppressive Agents; Interleukin-2; Lymphocytes; Mice; Mice, Inbred BALB C; Naloxone; Narcotic Antagonists; Phentolamine; Propranolol; Receptors, Adrenergic, alpha; Receptors, Opioid, mu | 1998 |
Psychic dependent potential of dihydroetorphine.
Topics: Analgesics, Opioid; Animals; Etorphine; Haplorhini; Mice; Opioid-Related Disorders; Rats | 1998 |
Anti-allodynic actions of intravenous opioids in the nerve injured rat: potential utility of heroin and dihydroetorphine against neuropathic pain.
Topics: Analgesics, Opioid; Animals; Drug Evaluation; Etorphine; Fentanyl; Heroin; Infusions, Intravenous; Ligation; Male; Morphine; Nerve Compression Syndromes; Pain; Rats; Rats, Inbred F344; Spinal Nerves | 1998 |
[Binding of [3H] dihydroetorphine to opioid receptors in rat brain membrane].
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Cell Membrane; Etorphine; Female; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, Opioid | 1996 |
[Studies on transdermal delivery system of dihydroetorphine hydrochloride].
Topics: Administration, Cutaneous; Analgesics, Opioid; Animals; Drug Delivery Systems; Etorphine; Rabbits; Rats; Rats, Wistar; Skin | 1996 |
Immunosuppressive effects of dihydroetorphine, a potent narcotic analgesic, in dihydroetorphine-dependent mice.
Topics: Analgesics, Opioid; Animals; Antibody-Producing Cells; Body Weight; Cell Division; Dose-Response Relationship, Drug; Etorphine; Female; Hypersensitivity, Delayed; Immunosuppressive Agents; Lymphocyte Count; Lymphocyte Subsets; Lymphocytes; Lymphokines; Mice; Mice, Inbred C57BL; Naloxone; Opioid-Related Disorders; Organ Size; Spleen; Substance Withdrawal Syndrome; Thymus Gland | 1999 |
[Decrease of cAMP and increase of amino acids contents in mouse brain after dihydroetorphine tolerance].
Topics: Amino Acids; Analgesics, Opioid; Animals; Aspartic Acid; Brain; Cyclic AMP; Drug Tolerance; Etorphine; gamma-Aminobutyric Acid; Glutamic Acid; Mice | 1998 |
Immunosuppressive effects of intravenous self administration of dihydroetorphine on lymphocyte functions in rats.
Topics: Animals; Cell Division; Etorphine; Immunosuppressive Agents; Injections, Intravenous; Interleukin-2; Lymphocytes; Male; Rats; Rats, Wistar; Self Administration; Spleen; Substance-Related Disorders | 1998 |
Dihydroetorphine-induced place preference was mediated by dopamine D1 receptors in rats.
Topics: Animals; Behavior, Animal; Benzazepines; Dopamine Agonists; Etorphine; Haloperidol; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Sulpiride | 1999 |
Differential binding properties of oripavines at cloned mu- and delta-opioid receptors.
Topics: Analgesics, Opioid; Animals; Benzamides; Binding, Competitive; Buprenorphine; Cloning, Molecular; Diprenorphine; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Naloxone; Piperazines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Sulfur Radioisotopes; Thebaine; Tritium; Tumor Cells, Cultured | 1999 |
Dihydroetorphine: physical dependence and stereotypy after continuous infusion in the rat.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Body Weight; Dose-Response Relationship, Drug; Etorphine; Infusions, Parenteral; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 2000 |
Effects of opioid receptor agonists on cAMP second messenger system.
Topics: Adenylyl Cyclases; Analgesics, Opioid; Buprenorphine; Cyclic AMP; Etorphine; Glioma; Humans; Hybrid Cells; Methadone; Morphine; Neuroblastoma; Opioid-Related Disorders; Receptors, Opioid; Receptors, Opioid, delta; Tumor Cells, Cultured | 1999 |
Effects of low-pH treatment on cAMP second messenger system regulated by different opioid agonists.
Topics: Adenylyl Cyclases; Analgesics, Opioid; Buprenorphine; Cyclic AMP; Etorphine; Glioma; Humans; Hybrid Cells; Hydrogen-Ion Concentration; Methadone; Morphine; Neuroblastoma; Opioid-Related Disorders; Receptors, Opioid, delta; Tumor Cells, Cultured | 1999 |
Quantitative determination of dihydroetorphine in rat plasma and brain by liquid chromatography-tandem mass spectrometry.
Topics: Analgesics, Opioid; Animals; Brain Chemistry; Buprenorphine; Calibration; Chromatography, High Pressure Liquid; Etorphine; Male; Mass Spectrometry; Quality Control; Rats; Reference Standards; Reproducibility of Results; Solutions | 2000 |
Pharmacokinetic and pharmacodynamic evaluations of a potent analgesic, dihydroetorphine, in hairless rat.
Topics: Algorithms; Analgesics, Opioid; Animals; Bile; Biological Availability; Biotransformation; Blood Proteins; Central Nervous System; Etorphine; Glucuronides; Injections, Intraventricular; Pain Measurement; Protein Binding; Rats; Rats, Inbred Strains | 2001 |
Transdermal delivery of the potent analgesic dihydroetorphine: kinetic analysis of skin permeation and analgesic effect in the hairless rat.
Topics: Administration, Cutaneous; Analgesics, Opioid; Animals; Bandages; Brain; Etorphine; In Vitro Techniques; Infusion Pumps; Kinetics; Male; Models, Biological; Rats; Rats, Mutant Strains; Skin; Skin Absorption; Solutions; Time Factors | 2000 |
A protective effect against undesirable increase of dihydroetorphine permeation through damaged skin by using pressure-sensitive adhesive tape with an ethylene-vinyl acetate co-polymer membrane.
Topics: Adhesives; Analgesics, Opioid; Animals; Etorphine; Permeability; Polyvinyls; Rats; Skin | 2001 |
Tolerance to analgesia and dependence liability by topical application of dihydroetorphine to hairless rats.
Topics: Administration, Cutaneous; Analgesics, Opioid; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Drug Tolerance; Etorphine; Formaldehyde; Inflammation; Infusions, Intravenous; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotic Antagonists; Rats; Rats, Nude; Substance-Related Disorders; Time Factors; Weight Loss | 2001 |
Biochemical characterisation of newly developed beta-etorphine and beta-dihydroetorphine derivatives.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Etorphine; Guanosine 5'-O-(3-Thiotriphosphate); Naloxone; Radioligand Assay; Rats; Rats, Wistar; Structure-Activity Relationship; Sulfur Radioisotopes; Tritium | 2002 |
Discriminative stimulus and antinociceptive effects of dihydroetorphine in rhesus monkeys.
Topics: Analgesics, Opioid; Animals; Discrimination Learning; Etorphine; Female; Macaca mulatta; Male; Morphine; Naltrexone | 2003 |
Binding affinity to and dependence on some opioids in Sf9 insect cells expressing human mu-opioid receptor.
Topics: Analgesics, Opioid; Animals; Baculoviridae; Binding, Competitive; Cells, Cultured; Cyclic AMP; Etorphine; Female; Fentanyl; Heroin; Male; Mice; Opioid-Related Disorders; Receptors, Opioid, mu; Spodoptera; Transfection | 2003 |
Tramadol and dihydroetorphine produce synergistic analgesic effect and postpones acute opiate tolerance in rats.
Topics: Analgesics, Opioid; Animals; Drug Synergism; Drug Tolerance; Etorphine; Female; Male; Pain; Rats; Rats, Wistar; Tramadol | 2005 |
Paradoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.
Topics: Analgesics, Opioid; Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Endocytosis; Etorphine; Fentanyl; Guanosine 5'-O-(3-Thiotriphosphate); Morphine; Opioid-Related Disorders; Receptors, Opioid, mu | 2010 |