Page last updated: 2024-08-23

etoposide and thiazoles

etoposide has been researched along with thiazoles in 50 studies

Research

Studies (50)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (20.00)18.2507
2000's26 (52.00)29.6817
2010's12 (24.00)24.3611
2020's2 (4.00)2.80

Authors

AuthorsStudies
Hotta, T; Kawamoto, K; Kiya, K; Kurisu, K; Mikami, T; Nakada, Y; Saito, Y; Uozumi, T; Yamada, K1
Endo, Y; Kimura, H; Kinoshita, K; Miyazaki, I; Ninomiya, I; Ohyama, S; Sasaki, T; Tanaka, M; Tugawa, K; Yonemura, Y1
Fujita, H; Ishizaki, T; Itoh, R; Okada, H; Yamamoto, T; Yasuda, J1
Gemba, K; Kiura, K; Matsumura, T; Moritaka, T; Ohnoshi, T; Segawa, Y; Shibayama, T; Tabata, M; Takigawa, N; Ueoka, H1
Asaga, T; Kawahara, S; Osawa, Y; Yanoma, S; Yoshida, A1
Fujimura, S; Kobayashi, S; Okada, S; Yoshida, H1
Häcker, G; Roloff, S; Wilhelm, S1
Borg, AG; Burgess, R; Fisher, A; Grey, M; Wood, P; Yin, JA1
Fujita, M; Higashino, K; Tsuchida, T1
Passaniti, A; Wang, W1
Aikou, T; Akiyama, S; Furukawa, T; Ikeda, R; Kitazono, M; Nagayama, S; Okumura, H; Seto, K; Sumizawa, T1
Goker, E; Karabulut, B; Omay, SB; Sanli, UA; Sezgin, C; Terzioglu, E; Uslu, R1
Chao, Y; Chen, LT; Huang, TS; Shu, CH1
Mahyar-Roemer, M; Roemer, K1
Dixon, JE; Donner, DB; Durden, DL; Mayo, LD; Tonks, NK1
Bassi, L; Carloni, M; Fonti, E; Meschini, R; Palitti, F; Palma de la Peña, N1
Akeshima, R; Iba, T; Itamochi, H; Kamazawa, S; Kanamori, Y; Kigawa, J; Sultana, H; Terakawa, N1
Deguchi, N; Murai, M; Nonaka, S; Ueno, M; Yamazaki, R1
Creutzig, U; Hählen, K; Harbott, J; Huismans, DR; Kaspers, GJ; Pieters, R; Slater, RM; Veerman, AJ; Zimmermann, M; Zwaan, CM1
Abe, A; Emi, N; Kanbe, E; Kawabe, T; Saito, H; Towatari, M1
Chan, SL; Gilman, CP; Greig, N; Guo, Z; Mattson, MP; Zhu, X1
Akaike, T; Fang, J; Greish, K; Maeda, H; Sawa, T1
Gabbert, HE; Gerharz, CD; Reinecke, P; Schmitz, M; Steckstor, M1
Bielawski, J; Dbaibo, GS; Gillanders, WE; Hannun, YA; Johnson, KR; Kozhaya, L; Obeid, LM; Osta, W; Taha, TA1
Colakogullari, M; Ulukaya, E; Wood, EJ1
Deveraux, QL; Engels, IH; Wagner, KW1
Alaoui-Jamali, MA; Chow, TY; Griller, D; Yeh, C; Yuen, L1
André, A; Braekman, JC; Bruyneel, F; Darro, F; Decaestecker, C; Dewelle, J; El Yazidi, M; Guissou, P; Kiss, R; Nacoulma, O; Simon, G; Tuti, J; Van Quaquebeke, E1
Burlet, S; Dono, R; Garino, C; Kraus, JL; Laras, Y; Maina, F; Moumen, A; Pietrancosta, N; Quéléver, G1
Faden, AI; Lea, PM; Movsesyan, VA1
Parent, AD; Tamaki, N; Yin, D; Zhang, JH1
Chang, KT; Chiu, CH; Huang, CY; Lok, YY; Tsai, CM1
Shi, YP; We, QY; Wu, QX1
Bähr, M; Dono, R; Kraus, JL; Lamballe, F; Lingor, P; Maina, F; Moumen, A; Pietrancosta, N; Planchamp, V1
Lee, HJ; Lee, HK; Park, HT; Seo, IA; Suh, DJ1
Mashima, T; Matsuura, M; Miyata, S; Okabe, S; Sato, S; Seimiya, H; Sugimoto, Y; Tsuruo, T1
Arkin, MR; Byl, JA; Conroy, A; Fox, JA; Hawtin, RE; McDowell, RS; Nguyen, T; Osheroff, N; Stockett, DE; Yang, W1
Kanomata, N; Kozuka, Y; Kurebayashi, J; Moriya, T; Sonoo, H; Watanabe, M1
Kim, JH; Lee, WH; Suk, K; Zheng, LT1
Akao, Y; Horiike, S; Kobayashi, S; Kobayashi, T; Kuroda, J; Matsumoto, Y; Nagoshi, H; Nishida, K; Sasaki, N; Shimura, Y; Taki, T; Taniwaki, M; Tsutsumi, Y; Yamamoto, M1
Bai, W; Bepler, G; Dong, H; Khochbin, S; Nicosia, SV; Wang, L; Williams, KA; Xiang, S; Zhang, X1
Evangelatov, A; Skrobanska, R; Yordanov, G1
Li, QG; Tong, Y; Xia, Q; Xing, TY; Zhang, JJ; Zhang, M1
Borchmann, P; Engert, A; Monsef, I; Rancea, M; Skoetz, N; Will, A1
Chen, X; Dai, H; Qian, Z; Wang, Y; Xu, X; Zhao, Y1
Bajrektarević, D; Filipič, M; Gajski, G; Garaj-Vrhovac, V; Gerić, M; Novak, M; Nunić, J; Žegura, B1
Burdova, K; Lindqvist, A; Macurek, L; Müllers, E; Silva Cascales, H1
Czaplinski, S; Fulda, S; Habermann, K; Hugle, M; Vogler, M1
Gopas, J; Gopinath, P; Muraleedharan, KM; Nandakumar, N1
Bakr, RB; El Azab, IH; Elkanzi, NAA1

Other Studies

50 other study(ies) available for etoposide and thiazoles

ArticleYear
Glutathione and cellular response of ACNU-resistant rat glioma sublines to drugs and radiation.
    International journal of cancer, 1991, Jul-30, Volume: 48, Issue:6

    Topics: Animals; Buthionine Sulfoximine; Cell Line; Cell Survival; Dose-Response Relationship, Radiation; Doxorubicin; Drug Resistance; Etoposide; Glioma; Glutathione; Kinetics; Methionine Sulfoximine; Nimustine; Pyrrolidonecarboxylic Acid; Rats; Thiazoles; Thiazolidines; Vinblastine

1991
[Chemosensitivity test for gastric cancer by in vitro MTT assay].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1991, Volume: 18, Issue:10

    Topics: Antineoplastic Agents; Carbazilquinone; Cisplatin; Doxorubicin; Drug Screening Assays, Antitumor; Etoposide; Fluorouracil; Humans; Mitomycin; Mitomycins; Stomach Neoplasms; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
[Estimation of medroxyprogesterone acetate (MPA) and etoposide against a human uterine endometrial cancer].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1994, Volume: 21, Issue:14

    Topics: Animals; Cell Division; Drug Synergism; Endometrial Neoplasms; Etoposide; Female; Humans; Medroxyprogesterone Acetate; Mice; Mice, Nude; Subrenal Capsule Assay; Tetrazolium Salts; Thiazoles

1994
[In vitro comparison of podophyllotoxin analogues; etoposide, teniposide and NK 611 using human lung cancer cell lines].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1993, Volume: 20, Issue:4

    Topics: Adenocarcinoma; Antineoplastic Agents; Carcinoma, Small Cell; Carcinoma, Squamous Cell; Cell Division; Drug Resistance; Drug Screening Assays, Antitumor; Etoposide; Humans; Lung Neoplasms; Podophyllotoxin; Teniposide; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1993
[In vitro chemosensitivity test for seven undifferentiated thyroid carcinoma cell lines using MTT assay].
    Gan to kagaku ryoho. Cancer & chemotherapy, 1996, Volume: 23, Issue:4

    Topics: Antineoplastic Agents; Bleomycin; Carcinoma; Cisplatin; Cyclophosphamide; Dactinomycin; Doxorubicin; Drug Screening Assays, Antitumor; Etoposide; Humans; Methotrexate; Tetrazolium Salts; Thiazoles; Thyroid Neoplasms; Tumor Cells, Cultured; Vincristine

1996
Indomethacin enhances the cytotoxicity of VCR and ADR in human pulmonary adenocarcinoma cells.
    The Tohoku journal of experimental medicine, 1997, Volume: 181, Issue:3

    Topics: Adenocarcinoma; Adjuvants, Pharmaceutic; Coloring Agents; Doxorubicin; Drug Combinations; Drug Screening Assays, Antitumor; Etoposide; Humans; Indomethacin; Lung Neoplasms; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Vincristine

1997
Inhibition of etoposide-induced apoptotic events by azide.
    Immunology letters, 1997, Volume: 59, Issue:1

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Azides; Coumarins; Etoposide; Flow Cytometry; Fluorescent Dyes; Humans; Jurkat Cells; Oligopeptides; Proto-Oncogene Proteins c-bcl-2; Tetrazolium Salts; Thiazoles; Ultraviolet Rays

1997
Effect on cell kill of addition of multidrug resistance modifiers cyclosporin A and PSC 833 to cytotoxic agents in acute myeloid leukaemia.
    Leukemia research, 1997, Volume: 21, Issue:9

    Topics: Acute Disease; Adolescent; Adult; Aged; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Coloring Agents; Cyclosporine; Cyclosporins; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Effect of vesnarinone in combination with anti-cancer drugs on lung cancer cell lines.
    Anti-cancer drugs, 1999, Volume: 10, Issue:1

    Topics: Adenocarcinoma; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Small Cell; Cell Division; Cisplatin; Coloring Agents; Deoxycytidine; DNA Fragmentation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Etoposide; Flow Cytometry; Gemcitabine; Humans; Lung Neoplasms; Pyrazines; Quinolines; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1999
Extracellular matrix inhibits apoptosis and enhances endothelial cell differentiation by a NfkappaB-dependent mechanism.
    Journal of cellular biochemistry, 1999, Jun-01, Volume: 73, Issue:3

    Topics: Apoptosis; bcl-2-Associated X Protein; Cell Cycle; Cell Differentiation; Cell Line; Cell Nucleus; Cell Survival; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Cytoplasm; DNA-Binding Proteins; Dose-Response Relationship, Drug; Endothelium, Vascular; Estradiol; Etoposide; Extracellular Matrix; Humans; I-kappa B Proteins; NF-kappa B; NF-KappaB Inhibitor alpha; Nucleic Acid Synthesis Inhibitors; Oligonucleotides, Antisense; Paclitaxel; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Receptors, Estrogen; Tetrazolium Salts; Thiazoles; Time Factors; Transfection

1999
Reversal of LRP-associated drug resistance in colon carcinoma SW-620 cells.
    International journal of cancer, 2001, Jan-01, Volume: 91, Issue:1

    Topics: Alkaloids; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Benzylisoquinolines; Butyrates; Carcinoma; Cell Nucleus; Colonic Neoplasms; Coloring Agents; Cyclic P-Oxides; Cytoplasm; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Neoplasm; Etoposide; Humans; Microscopy, Fluorescence; Neoplasm Proteins; Nicotinic Acids; RNA, Catalytic; Tetrazolium Salts; Thiazoles; Time Factors; Tumor Cells, Cultured; Vault Ribonucleoprotein Particles

2001
Arsenic trioxide-mediated cytotoxicity and apoptosis in prostate and ovarian carcinoma cell lines.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2000, Volume: 6, Issue:12

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Antioxidants; Apoptosis; Arsenic Trioxide; Arsenicals; Butylated Hydroxyanisole; Carcinogens; Cisplatin; DNA Fragmentation; Dose-Response Relationship, Drug; Doxorubicin; Enzyme-Linked Immunosorbent Assay; Etoposide; Female; Flow Cytometry; Humans; Male; Ovarian Neoplasms; Oxides; Prostatic Neoplasms; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2000
Evaluation of GL331 in combination with paclitaxel: GL331's interference with paclitaxel-induced cell cycle perturbation and apoptosis.
    Anti-cancer drugs, 2001, Volume: 12, Issue:3

    Topics: Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Blotting, Western; Calcium-Binding Proteins; Carrier Proteins; CDC2 Protein Kinase; Cell Cycle; Cell Cycle Proteins; Cell Nucleus; Cyclin B; Cyclin B1; DNA, Neoplasm; Dose-Response Relationship, Drug; Drug Antagonism; Drug Evaluation; Drug Interactions; Drug Therapy, Combination; Etoposide; Flow Cytometry; Fungal Proteins; Humans; Nasopharyngeal Neoplasms; Nuclear Proteins; Paclitaxel; Precipitin Tests; Protein Kinases; Tetrazolium Salts; Thiazoles; Toxicity Tests; Tumor Cells, Cultured

2001
p21 Waf1/Cip1 can protect human colon carcinoma cells against p53-dependent and p53-independent apoptosis induced by natural chemopreventive and therapeutic agents.
    Oncogene, 2001, Jun-07, Volume: 20, Issue:26

    Topics: Adenocarcinoma; Alleles; Amino Acid Chloromethyl Ketones; Anticarcinogenic Agents; Antineoplastic Agents; Apoptosis; Benzothiazoles; Butyrates; Cisplatin; Colonic Neoplasms; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; Cysteine Proteinase Inhibitors; Demecolcine; Doxorubicin; Drug Resistance, Neoplasm; Etoposide; Fluorouracil; Gene Expression Regulation, Neoplastic; Genes, p53; Humans; Intracellular Membranes; Membrane Potentials; Mitochondria; Neoplasm Proteins; Recombination, Genetic; Resveratrol; Stilbenes; Thiazoles; Toluene; Tumor Cells, Cultured; Tumor Suppressor Protein p53

2001
PTEN protects p53 from Mdm2 and sensitizes cancer cells to chemotherapy.
    The Journal of biological chemistry, 2002, Feb-15, Volume: 277, Issue:7

    Topics: Blotting, Western; Cell Cycle; Cell Line; Cell Nucleus; Cloning, Molecular; Coloring Agents; Cytoplasm; DNA Damage; Dose-Response Relationship, Drug; Down-Regulation; Etoposide; Genes, Reporter; Glioblastoma; Humans; Microscopy, Confocal; Mutation; Neoplasms; Nuclear Proteins; Phosphoric Monoester Hydrolases; Precipitin Tests; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-mdm2; PTEN Phosphohydrolase; Retroviridae; Signal Transduction; Tetrazolium Salts; Thiazoles; Transcription, Genetic; Transduction, Genetic; Tumor Cells, Cultured; Tumor Suppressor Protein p53; Tumor Suppressor Proteins

2002
Pifithrin-alpha, an inhibitor of p53, enhances the genetic instability induced by etoposide (VP16) in human lymphoblastoid cells treated in vitro.
    Mutation research, 2002, Feb-20, Volume: 499, Issue:2

    Topics: Antineoplastic Agents, Phytogenic; Benzothiazoles; Cell Cycle; Cell Survival; Chromosome Aberrations; DNA Fragmentation; Dose-Response Relationship, Drug; Drug Synergism; Etoposide; Flow Cytometry; Humans; In Vitro Techniques; Karyotyping; Lymphocytes; Thiazoles; Time Factors; Toluene; Tumor Cells, Cultured; Tumor Suppressor Protein p53

2002
Sensitivity to anticancer agents and resistance mechanisms in clear cell carcinoma of the ovary.
    Japanese journal of cancer research : Gann, 2002, Volume: 93, Issue:6

    Topics: Adenocarcinoma, Clear Cell; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Camptothecin; Cisplatin; Coloring Agents; DNA Topoisomerases, Type I; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Etoposide; Female; Glutathione; Humans; Inhibitory Concentration 50; Irinotecan; Mitochondrial Proteins; Mitomycin; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Ovarian Neoplasms; Paclitaxel; Reverse Transcriptase Polymerase Chain Reaction; Ribosomal Proteins; RNA, Messenger; Saccharomyces cerevisiae Proteins; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
SN-38 induces cell cycle arrest and apoptosis in human testicular cancer.
    European urology, 2002, Volume: 42, Issue:4

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Blotting, Western; Camptothecin; Cell Cycle; Cell Line; Cisplatin; DNA; Etoposide; G1 Phase; Humans; In Situ Nick-End Labeling; Irinotecan; Male; Testicular Neoplasms; Tetrazolium Salts; Thiazoles

2002
Cellular drug resistance in childhood acute myeloid leukemia is related to chromosomal abnormalities.
    Blood, 2002, Nov-01, Volume: 100, Issue:9

    Topics: Acute Disease; Adolescent; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Child; Child, Preschool; Chromosome Aberrations; Chromosome Inversion; Chromosomes, Human; Cladribine; Cytarabine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Female; Humans; Infant; Leukemia, Myeloid; Male; Neoplastic Stem Cells; Recurrence; Remission Induction; Tetrazolium Salts; Thiazoles; Translocation, Genetic; Trisomy

2002
DR1-like element in human topoisomerase IIalpha gene involved in enhancement of etoposide-induced apoptosis by PPARgamma ligand.
    Experimental hematology, 2003, Volume: 31, Issue:4

    Topics: Antigens, Neoplasm; Apoptosis; Chromans; DNA Topoisomerases, Type II; DNA-Binding Proteins; Electrophoretic Mobility Shift Assay; Etoposide; Flow Cytometry; Gene Expression; Humans; Jurkat Cells; Leukemia; Ligands; Mutagenesis; Phosphoproteins; Promoter Regions, Genetic; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Thiazoles; Thiazolidinediones; Topoisomerase II Inhibitors; Transcription Factors; Transfection; Troglitazone; Tumor Cells, Cultured

2003
p53 is present in synapses where it mediates mitochondrial dysfunction and synaptic degeneration in response to DNA damage, and oxidative and excitotoxic insults.
    Neuromolecular medicine, 2003, Volume: 3, Issue:3

    Topics: Animals; Benzothiazoles; Brain; Cells, Cultured; DNA Damage; Etoposide; Membrane Potentials; Mice; Mitochondria; Neurodegenerative Diseases; Neuroprotective Agents; Neurotoxins; Nucleic Acid Synthesis Inhibitors; Oxidative Stress; Phosphorylation; Presynaptic Terminals; Reactive Oxygen Species; Synapsins; Synaptosomes; Thiazoles; Toluene; Tumor Suppressor Protein p53

2003
Enhancement of chemotherapeutic response of tumor cells by a heme oxygenase inhibitor, pegylated zinc protoporphyrin.
    International journal of cancer, 2004, Volume: 109, Issue:1

    Topics: Animals; Annexin A5; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Apoptosis; Body Weight; Camptothecin; Cell Line, Tumor; Cisplatin; Coloring Agents; Dose-Response Relationship, Drug; Doxorubicin; Drug Synergism; Etoposide; Heme Oxygenase (Decyclizing); Humans; Hydrogen Peroxide; Male; Metalloporphyrins; Mice; Mitomycin; Neoplasms; Oxidants; Oxidation-Reduction; Oxidative Stress; Oxygen; Polyethylene Glycols; Proline; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles

2004
Chemotherapeutic potential of plant alkaloids and multidrug resistance mechanisms in malignant fibrous histiocytoma of the heart.
    Oncology reports, 2004, Volume: 11, Issue:3

    Topics: Alkaloids; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Separation; Cell Survival; Cells, Cultured; Coloring Agents; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Flow Cytometry; Heart Neoplasms; Histiocytoma, Benign Fibrous; Humans; Inhibitory Concentration 50; Paclitaxel; Phenotype; Plant Extracts; Soft Tissue Neoplasms; Tetrazolium Salts; Thiazoles; Vault Ribonucleoprotein Particles; Vincristine

2004
Down-regulation of sphingosine kinase-1 by DNA damage: dependence on proteases and p53.
    The Journal of biological chemistry, 2004, May-07, Volume: 279, Issue:19

    Topics: Apoptosis; Blotting, Western; Cell Division; Cell Line, Tumor; Cell Survival; Coloring Agents; Dactinomycin; DNA Damage; Dose-Response Relationship, Drug; Down-Regulation; Doxorubicin; Endopeptidases; Enzyme Inhibitors; Etoposide; Gamma Rays; Humans; Mass Spectrometry; Models, Biological; Phosphotransferases (Alcohol Group Acceptor); Proto-Oncogene Proteins c-bcl-2; Reverse Transcriptase Polymerase Chain Reaction; RNA Processing, Post-Transcriptional; RNA, Messenger; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Transcription, Genetic; Tumor Suppressor Protein p53; Up-Regulation

2004
Interference by anti-cancer chemotherapeutic agents in the MTT-tumor chemosensitivity assay.
    Chemotherapy, 2004, Volume: 50, Issue:1

    Topics: Antineoplastic Agents; Cisplatin; Colorimetry; Drug Interactions; Drug Screening Assays, Antitumor; Etoposide; Tetrazolium Salts; Thiazoles

2004
Caspase-2 can function upstream of bid cleavage in the TRAIL apoptosis pathway.
    The Journal of biological chemistry, 2004, Aug-13, Volume: 279, Issue:33

    Topics: Animals; Apoptosis; Apoptosis Regulatory Proteins; bcl-2-Associated X Protein; BH3 Interacting Domain Death Agonist Protein; Blotting, Western; Carrier Proteins; Caspase 2; Caspase 3; Caspase 7; Caspase 8; Caspases; Cell Death; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Etoposide; Gene Silencing; Humans; Membrane Glycoproteins; Mitochondria; Models, Biological; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; RNA Interference; RNA, Small Interfering; Staurosporine; Tetrazolium Salts; Thiazoles; Time Factors; TNF-Related Apoptosis-Inducing Ligand; Transfection; Tumor Necrosis Factor-alpha

2004
The DNA double-stranded break repair protein endo-exonuclease as a therapeutic target for cancer.
    Molecular cancer therapeutics, 2004, Volume: 3, Issue:8

    Topics: Animals; Antimetabolites, Antineoplastic; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Carcinoma, Lewis Lung; Cell Line, Tumor; Cell Survival; Cisplatin; Coloring Agents; DNA; DNA Damage; DNA Repair; Down-Regulation; Drug Evaluation, Preclinical; Endonucleases; Etoposide; Exonucleases; Fluorouracil; HeLa Cells; Humans; Kinetics; Mice; Mitomycin; Neoplasms; Pentamidine; Plasmids; Recombination, Genetic; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Time Factors

2004
Identification of a novel cardenolide (2''-oxovoruscharin) from Calotropis procera and the hemisynthesis of novel derivatives displaying potent in vitro antitumor activities and high in vivo tolerance: structure-activity relationship analyses.
    Journal of medicinal chemistry, 2005, Feb-10, Volume: 48, Issue:3

    Topics: Animals; Antineoplastic Agents; Calotropis; Camptothecin; Cardenolides; Cell Line, Tumor; Cell Proliferation; Cerebral Cortex; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Etoposide; Humans; Irinotecan; Magnetic Resonance Spectroscopy; Maximum Tolerated Dose; Mice; Organoplatinum Compounds; Oxaliplatin; Paclitaxel; Sodium-Potassium-Exchanging ATPase; Structure-Activity Relationship; Swine; Thiazoles

2005
Novel cyclized Pifithrin-alpha p53 inactivators: synthesis and biological studies.
    Bioorganic & medicinal chemistry letters, 2005, Mar-15, Volume: 15, Issue:6

    Topics: Animals; Benzothiazoles; Cerebral Cortex; Drug Stability; Etoposide; Mice; Models, Chemical; Molecular Structure; Neurons; Structure-Activity Relationship; Thiazoles; Toluene; Tumor Suppressor Protein p53

2005
Neuroprotective activity of the mGluR5 antagonists MPEP and MTEP against acute excitotoxicity differs and does not reflect actions at mGluR5 receptors.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Apoptosis; Cell Survival; Cells, Cultured; Cerebral Cortex; Dizocilpine Maleate; Dose-Response Relationship, Drug; Etoposide; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glutamic Acid; Glycine; Hydrolysis; Male; Membrane Potentials; Mice; Mice, Knockout; N-Methylaspartate; Neurons; Neuroprotective Agents; Phenylacetates; Phosphatidylinositols; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Thiazoles

2005
Insulin-like growth factor-I decreased etoposide-induced apoptosis in glioma cells by increasing bcl-2 expression and decreasing CPP32 activity.
    Neurological research, 2005, Volume: 27, Issue:1

    Topics: Apoptosis; Benzimidazoles; Blotting, Southern; Blotting, Western; Caspase 3; Caspases; Cell Count; Cell Line, Tumor; Cell Proliferation; Colorimetry; Cyclin D1; DNA Fragmentation; Dose-Response Relationship, Drug; Drug Interactions; Endopeptidases; Etoposide; Gene Expression Regulation, Neoplastic; Glioma; Humans; Insulin-Like Growth Factor I; Nerve Tissue Proteins; Nucleic Acid Synthesis Inhibitors; Oligodeoxyribonucleotides, Antisense; Receptor, IGF Type 1; Tetrazolium Salts; Thiazoles; Time Factors; Transfection

2005
Role of IL-6 in neuroendocrine differentiation and chemosensitivity of non-small cell lung cancer.
    American journal of physiology. Lung cellular and molecular physiology, 2005, Volume: 289, Issue:3

    Topics: Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Carcinoma, Non-Small-Cell Lung; Cell Count; Cell Differentiation; Cell Division; Cell Line, Tumor; Cisplatin; Coloring Agents; Down-Regulation; ErbB Receptors; Etoposide; Humans; Interleukin-6; Lung Neoplasms; Neurosecretory Systems; Phosphopyruvate Hydratase; Receptors, Interleukin-6; Recombinant Proteins; Signal Transduction; Tetrazolium Salts; Thiazoles

2005
Sesquiterpenes with various carbon skeletons from Ligularia virgaurea spp. oligocephala.
    Die Pharmazie, 2006, Volume: 61, Issue:3

    Topics: Antineoplastic Agents, Phytogenic; Asteraceae; Cell Line, Tumor; Etoposide; HL-60 Cells; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Plant Extracts; Sesquiterpenes; Spectrometry, Mass, Electrospray Ionization; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Tetrazolium Salts; Thiazoles

2006
Imino-tetrahydro-benzothiazole derivatives as p53 inhibitors: discovery of a highly potent in vivo inhibitor and its action mechanism.
    Journal of medicinal chemistry, 2006, Jun-15, Volume: 49, Issue:12

    Topics: Administration, Topical; Animals; Antineoplastic Agents; Apoptosis; Axotomy; Benzothiazoles; Cells, Cultured; Cyclin-Dependent Kinase Inhibitor p21; Drug Design; Drug Stability; Etoposide; Imines; Male; Mice; Neocortex; Neuroprotective Agents; Optic Nerve; Phosphorylation; Prodrugs; Rats; Rats, Wistar; Retinal Ganglion Cells; Thiazoles; Toluene; Tumor Suppressor Protein p53; Vitreous Body

2006
A novel mechanism of methylglyoxal cytotoxicity in neuroglial cells.
    Journal of neurochemistry, 2009, Volume: 108, Issue:1

    Topics: Animals; Antineoplastic Agents, Phytogenic; Cell Survival; Cells, Cultured; Cytokine Receptor gp130; Dose-Response Relationship, Drug; Etoposide; Flow Cytometry; Hydrogen Peroxide; Interleukin-6; Neuroglia; Protein Binding; Protein Processing, Post-Translational; Protein Transport; Pyruvaldehyde; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Signal Transduction; STAT3 Transcription Factor; Tetrazolium Salts; Thiazoles; Time Factors; Transfection

2009
Acyl-CoA synthetase as a cancer survival factor: its inhibition enhances the efficacy of etoposide.
    Cancer science, 2009, Volume: 100, Issue:8

    Topics: Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Benzimidazoles; Caspases; Catalysis; Cell Line, Tumor; Cell Survival; Coenzyme A Ligases; Cytochrome c Group; Dose-Response Relationship, Drug; Etoposide; Fluorescent Antibody Technique; Fluorescent Dyes; Glioma; Humans; Indoles; Injections, Subcutaneous; Isoenzymes; Mice; Mice, Nude; Neoplasm Transplantation; Subcellular Fractions; Tetrazolium Salts; Thiazoles; Triazenes; Tumor Burden; Xenograft Model Antitumor Assays

2009
Voreloxin is an anticancer quinolone derivative that intercalates DNA and poisons topoisomerase II.
    PloS one, 2010, Apr-15, Volume: 5, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Cell Line, Tumor; DNA; DNA Damage; DNA Fragmentation; DNA Topoisomerases, Type II; Drug Delivery Systems; Etoposide; G2 Phase; Humans; Intercalating Agents; Naphthyridines; Quinolones; Thiazoles

2010
Preferential antitumor effect of the Src inhibitor dasatinib associated with a decreased proportion of aldehyde dehydrogenase 1-positive cells in breast cancer cells of the basal B subtype.
    BMC cancer, 2010, Oct-20, Volume: 10

    Topics: Aldehyde Dehydrogenase; Antineoplastic Agents; Apoptosis; Breast Neoplasms; Cell Line, Tumor; Dasatinib; DNA Damage; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Enzyme Inhibitors; Etoposide; Humans; Inhibitory Concentration 50; Neoplastic Stem Cells; Pyrimidines; src-Family Kinases; Thiazoles

2010
Pro-apoptotic role of integrin β3 in glioma cells.
    Journal of neurochemistry, 2011, Volume: 117, Issue:3

    Topics: Animals; Antineoplastic Agents, Alkylating; Apoptosis; Carmustine; Cell Line, Tumor; Drug Interactions; Enzyme Inhibitors; Etoposide; Flow Cytometry; Free Radical Scavengers; Gene Expression Regulation, Neoplastic; Glioma; Humans; Integrin beta3; Nitric Oxide; Rats; RNA, Messenger; Signal Transduction; Statistics as Topic; Tetrazolium Salts; Thiazoles; Vitronectin

2011
Bcl-2 is a better therapeutic target than c-Myc, but attacking both could be a more effective treatment strategy for B-cell lymphoma with concurrent Bcl-2 and c-Myc overexpression.
    Experimental hematology, 2011, Volume: 39, Issue:8

    Topics: Aniline Compounds; Antineoplastic Agents; Blotting, Western; Cell Line, Tumor; Cell Survival; Chromosomes, Human, Pair 14; Chromosomes, Human, Pair 18; Cytarabine; Dose-Response Relationship, Drug; Doxorubicin; Drug Synergism; Etoposide; Gene Expression Regulation, Neoplastic; Humans; Lymphoma, Large B-Cell, Diffuse; MicroRNAs; Proto-Oncogene Proteins c-bcl-2; Proto-Oncogene Proteins c-myc; Reverse Transcriptase Polymerase Chain Reaction; Spectral Karyotyping; Sulfonamides; Thiazoles; Translocation, Genetic

2011
Depletion of HDAC6 enhances cisplatin-induced DNA damage and apoptosis in non-small cell lung cancer cells.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: Animals; Apoptosis; Carcinoma, Non-Small-Cell Lung; Cell Cycle; Cell Line, Tumor; Cisplatin; Comet Assay; DNA Damage; Doxorubicin; Etoposide; Female; Histone Deacetylase 6; Histone Deacetylases; Humans; Immunoblotting; Immunohistochemistry; Inhibitory Concentration 50; Lung Neoplasms; Mice; Mice, Nude; Neoplasm Transplantation; Tetrazolium Salts; Thiazoles

2012
Colloidal formulations of etoposide based on poly(butyl cyanoacrylate) nanoparticles: preparation, physicochemical properties and cytotoxicity.
    Colloids and surfaces. B, Biointerfaces, 2013, Jan-01, Volume: 101

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Benzimidazoles; Cell Line, Tumor; Chemistry, Pharmaceutical; Colloids; Coloring Agents; Enbucrilate; Etoposide; Fluorescent Dyes; Humans; Indicators and Reagents; Light; Microscopy, Electron, Scanning; Nanoparticles; Particle Size; Scattering, Radiation; Tetrazolium Salts; Thiazoles

2013
HIF1 regulates WSB-1 expression to promote hypoxia-induced chemoresistance in hepatocellular carcinoma cells.
    FEBS letters, 2013, Aug-19, Volume: 587, Issue:16

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Carcinoma, Hepatocellular; Carrier Proteins; Cell Hypoxia; DNA Damage; Drug Resistance, Neoplasm; Etoposide; Gene Expression Regulation, Neoplastic; Hep G2 Cells; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Intracellular Signaling Peptides and Proteins; Liver Neoplasms; Promoter Regions, Genetic; Protein Serine-Threonine Kinases; Proteins; RNA Interference; RNA, Small Interfering; Tetrazolium Salts; Thiazoles

2013
Fifteenth biannual report of the Cochrane Haematological Malignancies Group--focus on non-Hodgkin's lymphoma.
    Journal of the National Cancer Institute, 2013, Aug-07, Volume: 105, Issue:15

    Topics: Adult; Aged; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Bleomycin; Cyclophosphamide; Dasatinib; Doxorubicin; Etoposide; Hodgkin Disease; Humans; Imatinib Mesylate; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Lymphoma, Non-Hodgkin; Middle Aged; Multicenter Studies as Topic; Multiple Myeloma; Neoplasm Staging; Piperazines; Platelet Transfusion; Prednisone; Primary Prevention; Procarbazine; Pyrimidines; Randomized Controlled Trials as Topic; Rituximab; Stem Cell Transplantation; Survival Analysis; Thiazoles; Thrombocytopenia; Transplantation, Autologous; Treatment Outcome; Vincristine; Vindesine

2013
In vitro chemosensitivity assay of ascites in epithelial ovarian cancer.
    European journal of gynaecological oncology, 2013, Volume: 34, Issue:6

    Topics: Antineoplastic Agents; Ascites; Carboplatin; Carcinoma, Ovarian Epithelial; Coloring Agents; Deoxycytidine; Disease Progression; Drug Screening Assays, Antitumor; Epirubicin; Etoposide; Female; Fluorouracil; Gemcitabine; Humans; Kaplan-Meier Estimate; Ki-67 Antigen; Middle Aged; Neoplasms, Glandular and Epithelial; Ovarian Neoplasms; Paclitaxel; Predictive Value of Tests; Retrospective Studies; Survival Rate; Tetrazolium Salts; Thiazoles; Time Factors; Tumor Cells, Cultured; Tumor Suppressor Protein p53

2013
Genotoxic potential of selected cytostatic drugs in human and zebrafish cells.
    Environmental science and pollution research international, 2016, Volume: 23, Issue:15

    Topics: Acridine Orange; Animals; Cell Line; Cell Survival; Cisplatin; Cytostatic Agents; Ethidium; Etoposide; Fluorouracil; Hep G2 Cells; Humans; Lymphocytes; Tetrazolium Salts; Thiazoles; Zebrafish

2016
Residual Cdk1/2 activity after DNA damage promotes senescence.
    Aging cell, 2017, Volume: 16, Issue:3

    Topics: Antigens, CD; Cadherins; CDC2 Protein Kinase; Cell Line; Cell Line, Tumor; Cell Size; Cell Survival; Cellular Senescence; Cyclin B1; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinase Inhibitor p21; DNA Damage; Epithelial Cells; Etoposide; G2 Phase Cell Cycle Checkpoints; Gene Expression Regulation; Humans; Osteoblasts; Pteridines; Purines; Quinolines; Retinal Pigment Epithelium; Signal Transduction; Single-Cell Analysis; Thiazoles

2017
Identification of Smac mimetics as novel substrates for p-glycoprotein.
    Cancer letters, 2019, Volume: 440-441

    Topics: Apoptosis Regulatory Proteins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biomimetic Materials; Cell Line, Tumor; Dipeptides; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Humans; Indoles; Inhibitor of Apoptosis Proteins; Intracellular Signaling Peptides and Proteins; Mitochondrial Proteins; Neuroblastoma; Oligopeptides; Rhabdomyosarcoma; Thiazoles; Up-Regulation; Vincristine

2019
Benzisothiazolone Derivatives Exhibit Cytotoxicity in Hodgkin's Lymphoma Cells through NF-κB Inhibition and are Synergistic with Doxorubicin and Etoposide.
    Anti-cancer agents in medicinal chemistry, 2020, Volume: 20, Issue:6

    Topics: A549 Cells; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Movement; Doxorubicin; Drug Synergism; Etoposide; Hodgkin Disease; Humans; NF-kappa B; Thiazoles

2020
Facile One-Pot Multicomponent Synthesis of Pyrazolo-Thiazole Substituted Pyridines with Potential Anti-Proliferative Activity: Synthesis, In Vitro and In Silico Studies.
    Molecules (Basel, Switzerland), 2021, May-22, Volume: 26, Issue:11

    Topics: Antineoplastic Agents; Cell Line, Tumor; Chemistry Techniques, Synthetic; Computer Simulation; DNA Topoisomerases, Type II; Drug Screening Assays, Antitumor; Etoposide; HeLa Cells; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mass Spectrometry; Molecular Docking Simulation; PC-3 Cells; Pyrazoles; Pyridines; Spectrophotometry, Infrared; Thiazoles

2021