Page last updated: 2024-09-03

etomoxir and cerulenin

etomoxir has been researched along with cerulenin in 4 studies

Compound Research Comparison

Studies
(etomoxir)
Trials
(etomoxir)
Recent Studies (post-2010)
(etomoxir)
Studies
(cerulenin)
Trials
(cerulenin)
Recent Studies (post-2010) (cerulenin)
2608935240105

Protein Interaction Comparison

ProteinTaxonomyetomoxir (IC50)cerulenin (IC50)
Fatty acid synthaseHomo sapiens (human)5.8
Protease Human immunodeficiency virus 12.5

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kuhajda, FP; Pinn, ML; Thupari, JN1
Cheng, H; Sharp, GW; Straub, SG1
Downs, SM; Klinger, J; Mosey, JL1
Cózar-Castellano, I; Joumady, I; Perdomo, G; Sáez-Benito, A; Tirado-Vélez, JM1

Other Studies

4 other study(ies) available for etomoxir and cerulenin

ArticleYear
Fatty acid synthase inhibition in human breast cancer cells leads to malonyl-CoA-induced inhibition of fatty acid oxidation and cytotoxicity.
    Biochemical and biophysical research communications, 2001, Jul-13, Volume: 285, Issue:2

    Topics: Acetyl-CoA Carboxylase; Apoptosis; Breast Neoplasms; Carnitine O-Palmitoyltransferase; Cell Survival; Cerulenin; Enzyme Inhibitors; Epoxy Compounds; Fatty Acid Synthases; Fatty Acids; Female; Furans; Humans; Hypolipidemic Agents; Kinetics; Malonyl Coenzyme A; Models, Biological; Oxidation-Reduction; Tumor Cells, Cultured

2001
Protein acylation in the inhibition of insulin secretion by norepinephrine, somatostatin, galanin, and PGE2.
    American journal of physiology. Endocrinology and metabolism, 2003, Volume: 285, Issue:2

    Topics: Acylation; Acyltransferases; Animals; Cerulenin; Cyclic AMP; Dinoprostone; Enzyme Activation; Enzyme Inhibitors; Epoxy Compounds; Fatty Acids, Unsaturated; Galanin; GTP-Binding Proteins; Hypoglycemic Agents; Insulin; Insulin Secretion; Lipid Metabolism; Male; Norepinephrine; Oxidation-Reduction; Palmitates; Palmitic Acid; Proteins; Rats; Rats, Sprague-Dawley; Somatostatin

2003
Fatty acid oxidation and meiotic resumption in mouse oocytes.
    Molecular reproduction and development, 2009, Volume: 76, Issue:9

    Topics: 4-Butyrolactone; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Carnitine; Carnitine O-Palmitoyltransferase; Cerulenin; Cumulus Cells; Epoxy Compounds; Fatty Acids; Female; Malonyl Coenzyme A; Meiosis; Mice; Mice, Inbred C57BL; Oocytes; Oxidation-Reduction; Palmitic Acid; Ribonucleotides

2009
Inhibition of fatty acid metabolism reduces human myeloma cells proliferation.
    PloS one, 2012, Volume: 7, Issue:9

    Topics: Antimetabolites, Antineoplastic; Apoptosis; Boronic Acids; Bortezomib; Carbohydrate Metabolism; Cell Cycle Proteins; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cerulenin; Cyclin-Dependent Kinase Inhibitor p21; Drug Synergism; Epoxy Compounds; Fatty Acids; G1 Phase Cell Cycle Checkpoints; Glucose; Humans; Lactones; Lipid Metabolism; Multiple Myeloma; Orlistat; Oxidation-Reduction; Pyrazines; Retinoblastoma Protein

2012