ethylmaleimide has been researched along with guanylyl imidodiphosphate in 75 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 49 (65.33) | 18.7374 |
1990's | 23 (30.67) | 18.2507 |
2000's | 3 (4.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Ferguson, KM; Gilman, AG; Howlett, AC; Ross, EM | 1 |
Gilman, AG; Howlett, AC; Ross, EM | 1 |
Bourne, HR; Johnson, GL; Kaslow, HR | 1 |
LaPorte, DC; Storm, DR; Toscano, WA; Westcott, KR | 1 |
Nakata, H | 1 |
Albrecht, FE; Eisner, GM; Felder, RA; Horiuchi, A; Jose, PA | 1 |
Emerit, MB; Gozlan, H; Hamon, M; Miquel, MC | 1 |
Dattatreyamurty, B; Reichert, LE; Zhang, SB | 1 |
Allende, G; Canela, EI; Franco, R; Lluis, C; Mallol, J | 1 |
Jagadeesh, G; Phan, NT; Sulakhe, PV | 1 |
Carroll, AG; Rhoads, AR; Wagner, PD | 1 |
Dawson, RM; Poretski, M | 1 |
Jagadeesh, G; Phan, NT; Rao, TS; Sulakhe, PV; Veeranjaneyulu, A | 1 |
Gharib, A; Lagarde, M; Reynaud, D; Sarda, N | 1 |
Ashby, B | 1 |
Kukovetz, WR; Schmidt, K | 1 |
Green, RD; Leung, E | 1 |
Ariani, K; Ciaranello, RD; Hamblin, MW; Stratford, CA; Tan, GL | 1 |
Itzhak, Y | 1 |
Berlan, M; Galitzky, J; Lafontan, M; Paris, H | 1 |
Ferrendelli, CA; Hanchett, HE; Hollifield, MA; Lorenzi, MV; Potter, LT | 1 |
Gharib, A; Ou, L; Pacheco, H; Reynaud, D; Sarda, N | 1 |
Codina, J; Herberg, JT; Iyengar, R; Premont, RT; Rich, KA | 1 |
Ito, Y; Makimura, M; Murakoshi, Y | 1 |
Bick, RJ; Chu, A; Entman, ML; Tate, CA; Van Winkle, WB | 1 |
Asano, T; Ogasawara, N | 1 |
Coscia, CJ; Spain, JW | 1 |
Musacchio, JM; Sharma, PM | 1 |
Cooper, DM; Perez-Reyes, E | 1 |
Flynn, DD; Potter, LT | 1 |
Aiyar, N; Crooke, ST; Nambi, P; Stassen, FL | 1 |
Dwyer, TM; Farley, JM; Mohan, PM; Yang, CM | 1 |
Braun, AP; Sperelakis, N | 1 |
Ammon, HP; Kühn, M; Trier, JK | 1 |
Tolkovsky, AM | 1 |
Roeske, WR; Watson, M; Yamamura, HI | 1 |
Franck, H; Keck, E; Krüskemper, HL; van Valen, F | 1 |
Daly, JW; Seamon, KB; Vaillancourt, R | 1 |
Childers, SR | 1 |
Roeske, WR; Vickroy, TW; Watson, M; Yamamura, HI | 1 |
Lad, PM; Nielsen, TB; Preston, MS; Rodbell, M | 1 |
Braun, S; Levitzki, A; Tolkovsky, AM | 1 |
Arnaud, CD; Nissenson, RA; Teitelbaum, AP | 1 |
Green, RD; Yeung, SM | 1 |
Braun, S; Feder, D; Gal, A; Levitzki, A | 1 |
Coscia, CJ; Roth, BL | 1 |
Seamon, KB; Wetzel, B | 1 |
Harden, TK; Martin, MW; Smith, MM | 1 |
Bitensky, MW; Kosack, CM; Malina, RL; Rasenick, MM; Stein, PJ; Wheeler, GL | 1 |
Krall, JF | 1 |
Fung, BK; Ho, YK | 1 |
Haga, T; Ichiyama, A; Nukada, T | 1 |
Roeske, WR; Vickroy, TW; Yamamura, HI | 1 |
Hosey, MM; McMahon, KK | 1 |
Drummond, GI; Nambi, P | 1 |
Ehlert, FJ; Roeske, WR; Yamamura, HI | 1 |
Drummond, GI | 1 |
Drummond, GI; Nambi, P; Sano, M | 1 |
Neufeld, G; Schramm, M; Weinberg, N | 1 |
Kimura, K; Sidhu, A; Vachvanichsanong, P | 1 |
Ishige, K; Ito, Y; Makimura, M; Murakoshi, Y | 1 |
Jakobs, KH; Mura, R; Niroomand, F; Piacentini, L | 1 |
Allegrucci, C; Mezzasoma, I; Minelli, A | 1 |
Spindler, KD; Spindler-Barth, M; Wegener, S | 1 |
Giusti, L; Lucacchini, A; Mazzoni, MR; Rossi, E; Taddei, S | 1 |
Cowburn, RF; Einblad, B; Fastbom, J; García-Jiménez, A | 1 |
Grüb, S; Hartig, R; Janetzko, A; Shoeman, RL; Traub, P | 1 |
Dhalla, NS; Elimban, V; Persad, S; Siddiqui, F | 1 |
Constantino, MD; Cunha, RA; Ribeiro, JA | 1 |
Cowburn, RF; Fastbom, J; Garcia-Jiménez, A; Winblad, B | 1 |
Chiu, ML; Waeber, C | 1 |
Childers, SR; Sim-Selley, LJ; Xiao, R | 1 |
Giusto, NM; Pasquaré, SJ; Roque, ME; Salvador, GA | 1 |
Bigini, G; Ceccarelli, F; Chericoni, S; Giusti, L; Lucacchini, A; Mazzoni, MR; Taddei, S | 1 |
Di Scala-Guenot, D; Evrard, ME; Strosser, MT | 1 |
1 review(s) available for ethylmaleimide and guanylyl imidodiphosphate
Article | Year |
---|---|
Differential regulation of putative M1/M2 muscarinic receptors: implications for different receptor-effector coupling mechanisms.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adenylyl Cyclases; Animals; Benzodiazepinones; Cerebral Cortex; Chemical Phenomena; Chemistry; Ethylmaleimide; Guanine Nucleotides; Guanylyl Imidodiphosphate; In Vitro Techniques; Molecular Conformation; Myocardium; Pilocarpine; Pirenzepine; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic | 1984 |
74 other study(ies) available for ethylmaleimide and guanylyl imidodiphosphate
Article | Year |
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Reconstitution of hormone-sensitive adenylate cyclase activity with resolved components of the enzyme.
Topics: Adenylyl Cyclases; Cell Line; Cell Membrane; Drug Stability; Ethylmaleimide; Fluorides; Guanylyl Imidodiphosphate; Hot Temperature; Isoproterenol; Magnesium; Manganese; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cell Surface | 1978 |
Identification and partial characterization of some components of hormone-stimulated adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cells, Cultured; Ethylmaleimide; Guanylyl Imidodiphosphate; Hot Temperature; Liver Neoplasms, Experimental; Lymphoma; Neoplasms, Experimental; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cyclic AMP | 1979 |
Reconstitution of cholera toxin-activated adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Binding Sites; Cell Line; Cholera Toxin; Enzyme Activation; Ethylmaleimide; Fluorides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Macromolecular Substances; Mutation | 1978 |
Evidence for a dissociable protein subunit required for calmodulin stimulation of brain adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Calcium-Binding Proteins; Calmodulin; Cattle; Cerebral Cortex; Enzyme Activation; Ethylmaleimide; Fluorides; Guanylyl Imidodiphosphate; Macromolecular Substances; Structure-Activity Relationship; Temperature; Trypsin | 1979 |
Biochemical and immunological characterization of A1 adenosine receptors purified from human brain membranes.
Topics: Adenosine; Animals; Antibodies; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Chromatography; Chromatography, Affinity; Durapatite; Ethylmaleimide; Guanylyl Imidodiphosphate; Humans; Hydroxyapatites; Kinetics; Rats; Receptors, Purinergic | 1992 |
Renal dopamine receptors and pre- and post-cAMP-mediated Na+ transport defect in spontaneously hypertensive rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Biological Transport; Carrier Proteins; Cyclic AMP; Dopamine Agents; Ethylmaleimide; Fenoldopam; Guanylyl Imidodiphosphate; Kidney; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Dopamine; Sodium; Sodium-Hydrogen Exchangers; Thionucleotides | 1992 |
The GTP-insensitive component of high-affinity [3H]8-hydroxy-2-(di-n-propylamino)tetralin binding in the rat hippocampus corresponds to an oxidized state of the 5-hydroxytryptamine1A receptor.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Dithiothreitol; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hippocampus; Male; Oxidation-Reduction; Rats; Receptors, Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes; Tetrathionic Acid; Tritium | 1991 |
Differential roles of high and low affinity guanosine 5'-triphosphate binding sites in the regulation of follicle-stimulating hormone binding to receptor and signal transduction in bovine calf testis membranes.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Cattle; Cell Membrane; Cholera Toxin; Colforsin; Enzyme Activation; Ethylmaleimide; Follicle Stimulating Hormone; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Receptors, FSH; Signal Transduction; Testis | 1991 |
N-ethylmaleimide affects agonist binding to A1 adenosine receptors differently in the presence than in the absence of ligand.
Topics: Adenine; Animals; Brain; Dithionitrobenzoic Acid; Ethylmaleimide; Guanylyl Imidodiphosphate; Hydroxymercuribenzoates; Kinetics; Ligands; Phenylisopropyladenosine; Receptors, Purinergic; Swine; Xanthines | 1991 |
Two distinct, divalent cation-sensitive, antagonist binding states of heart muscarinic receptors: differential modulation by guanine nucleotide.
Topics: Animals; Calcium; Cations, Divalent; Edetic Acid; Egtazic Acid; Ethylmaleimide; Guanine Nucleotides; Guanylyl Imidodiphosphate; Heart; In Vitro Techniques; Kinetics; Magnesium; Male; Myocardium; Parasympatholytics; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic; Subcellular Fractions | 1990 |
Hydrolysis-resistant GTP analogs stimulate catecholamine release from digitonin-permeabilized PC12 cells.
Topics: Adenosine Triphosphate; Adrenal Gland Neoplasms; Animals; Calcium; Cell Membrane Permeability; Digitonin; Ethylmaleimide; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hydrolysis; Kinetics; Norepinephrine; Pheochromocytoma; Rats; Signal Transduction; Tetradecanoylphorbol Acetate; Thionucleotides; Tumor Cells, Cultured | 1990 |
Opposing effects of N-ethylmaleimide on the affinity of carbachol for muscarinic cholinoceptors of guinea-pig atrium.
Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; Guinea Pigs; Heart Atria; Premedication; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Temperature | 1990 |
MgCl2-sensitive and Gpp(NH)p-sensitive antagonist binding states of rat heart muscarinic receptors: preferential detection at ambient temperature assay and location in two subcellular fractions.
Topics: Animals; Dithiothreitol; Ethylmaleimide; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Magnesium Chloride; Male; Microsomes; Myocardium; N-Methylscopolamine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine Derivatives; Temperature | 1990 |
Characterization of A-2 receptors in postmortem human pineal gland.
Topics: Adenosine; Autopsy; Cell Membrane; Ethylmaleimide; Guanylyl Imidodiphosphate; Humans; Kinetics; Pineal Gland; Radioligand Assay; Receptors, Purinergic | 1990 |
Kinetic evidence indicating separate stimulatory and inhibitory prostaglandin receptors on platelet membranes.
Topics: Adenylyl Cyclases; Alprostadil; Blood Platelets; Cell Membrane; Cell-Free System; Cyclic AMP; Epoprostenol; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; Iloprost; Kinetics; Prostaglandin D2; Prostaglandins D; Receptors, Prostaglandin | 1986 |
Mediation of the cardiac effects of forskolin by specific binding sites.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Colforsin; Ethylmaleimide; Female; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Rate; Hot Temperature; In Vitro Techniques; Magnesium; Magnesium Chloride; Male; Myocardial Contraction; Trypsin | 1989 |
Density gradient profiles of A1 adenosine receptors labeled by agonist and antagonist radioligands before and after detergent solubilization.
Topics: Adenosine; Adenosine Deaminase; Animals; Cattle; Cell Membrane; Centrifugation, Density Gradient; Cerebral Cortex; Ethylmaleimide; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Iodobenzenes; Ligands; Macromolecular Substances; Receptors, Purinergic; Solubility; Xanthines | 1989 |
G protein dependent alterations in [125I]iodocyanopindolol and +/- cyanopindolol binding at 5-HT1B binding sites in rat brain membranes.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Dihydroergotamine; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Iodocyanopindolol; Magnesium Sulfate; Pindolol; Rats; Receptors, Serotonin | 1989 |
Multiple affinity binding states of the sigma receptor: effect of GTP-binding protein-modifying agents.
Topics: Animals; Binding, Competitive; Chlorpromazine; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Pentazocine; Pertussis Toxin; Piperidines; Rats; Receptors, Opioid; Receptors, sigma; Virulence Factors, Bordetella | 1989 |
Human fat cell alpha-2 adrenoceptors. II. Comparative study of partial and full agonist binding parameters using [3H]clonidine and [3H]UK-14,304.
Topics: Adipose Tissue; Adrenergic alpha-Agonists; Allosteric Regulation; Binding, Competitive; Brimonidine Tartrate; Clonidine; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Kinetics; Magnesium; Quinoxalines; Receptors, Adrenergic, alpha; Yohimbine | 1989 |
Tetrahydroaminoacridine and other allosteric antagonists of hippocampal M1 muscarine receptors.
Topics: Allosteric Regulation; Aminoacridines; Animals; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; In Vitro Techniques; N-Methylscopolamine; Parasympatholytics; Pirenzepine; Protein Conformation; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Solubility; Tacrine | 1989 |
Identification of adenosine receptor in rat pineal gland: evidence for A-2 selectivity.
Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cell Membrane; Ethylmaleimide; Guanylyl Imidodiphosphate; Male; Phenylisopropyladenosine; Pineal Gland; Rats; Rats, Inbred Strains; Receptors, Purinergic; S-Adenosylhomocysteine | 1989 |
Glucagon receptor-mediated activation of Gs is accompanied by subunit dissociation.
Topics: Adenylyl Cyclases; Centrifugation, Density Gradient; Ethylmaleimide; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Liver; Macromolecular Substances; Magnesium; Receptors, Gastrointestinal Hormone; Receptors, Glucagon; Thionucleotides | 1988 |
[Characterization of opioid receptor from bullfrog brain].
Topics: Animals; Binding, Competitive; Brain; Carps; Chickens; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Levorphanol; Mice; Naloxone; Rana catesbeiana; Rats; Receptors, Opioid; Solubility; Surface-Active Agents | 1988 |
Nucleotide specificity of cardiac sarcoplasmic reticulum. GTP-induced calcium accumulation and GTPase activity.
Topics: Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; Calcium; Dogs; Ethylmaleimide; GTP Phosphohydrolases; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hydrogen-Ion Concentration; Hydrolysis; Kinetics; Mersalyl; Mitochondria, Heart; Myocardium; Phosphoric Monoester Hydrolases; Sarcolemma; Sarcoplasmic Reticulum | 1985 |
Uncoupling of gamma-aminobutyric acid B receptors from GTP-binding proteins by N-ethylmaleimide: effect of N-ethylmaleimide on purified GTP-binding proteins.
Topics: Adenosine Diphosphate Ribose; Animals; Cattle; Ethylmaleimide; gamma-Aminobutyric Acid; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Magnesium; Pertussis Toxin; Receptors, GABA-A; Thionucleotides; Tritium; Virulence Factors, Bordetella | 1986 |
Multiple interconvertible affinity states for the delta opioid agonist-receptor complex.
Topics: Animals; Cattle; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; Kinetics; Morphine; Naltrexone; Receptors, Opioid; Receptors, Opioid, delta; Synaptic Membranes | 1987 |
N-ethylmaleimide blocks the modulatory effects of divalent cations and guanine nucleotides on the brain substance P receptor.
Topics: Animals; Brain Chemistry; Cations, Divalent; Ethylmaleimide; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Membranes; Nerve Tissue Proteins; Physalaemin; Rats; Receptors, Neurokinin-1; Receptors, Neurotransmitter | 1987 |
Interaction of the inhibitory GTP regulatory component with soluble cerebral cortical adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Animals; Arabinonucleotides; Cell Membrane; Centrifugation, Density Gradient; Cerebral Cortex; Chromatography, Gel; Egtazic Acid; Ethylmaleimide; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Rats; Rats, Inbred Strains; Temperature; Thionucleotides | 1986 |
Effect of solubilization on the distinct binding properties of muscarine receptors from rabbit hippocampus and brainstem.
Topics: Animals; Brain Stem; Carbachol; Edetic Acid; Ethylmaleimide; Guanylyl Imidodiphosphate; Hippocampus; In Vitro Techniques; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Solubility | 1986 |
Effects of N-ethylmaleimide on arginine vasopressin-induced responses in an established smooth muscle cell line.
Topics: Animals; Aorta, Thoracic; Arginine Vasopressin; Calcium; Cell Membrane; Ethylmaleimide; GTP Phosphohydrolases; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Male; Muscle, Smooth, Vascular; Phosphatidylinositols; Rats | 1987 |
Changes in affinity states during down-regulation of muscarinic receptors in tracheal smooth muscle of organophosphate-treated swine.
Topics: Animals; Carbachol; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Isoflurophate; Magnesium; Male; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine; Trachea | 1988 |
Attenuation by N-ethylmaleimide treatment of the cholinergically induced shortening of action potential duration in guinea pig right atrium.
Topics: Action Potentials; Animals; Electrophysiology; Ethylmaleimide; Guanylyl Imidodiphosphate; Guinea Pigs; Heart; Heart Atria; Heart Conduction System; Male; Oxotremorine; Rabbits | 1988 |
Adenylate cyclase in membrane fractions of RIN-A2-cells: studies with forskolin, NaF, GppNHp and NEM.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Cells, Cultured; Colforsin; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Rats; Sodium Fluoride | 1988 |
Modulation of guanine nucleotide affinity does not affect the first order rate constant of activation of adenylate cyclase in native membranes.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Enzyme Activation; Ethylmaleimide; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Intracellular Membranes; Kinetics; Male; Mathematics; Models, Biological; Rats; Synaptosomes; Thionucleotides | 1986 |
[3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. II. Characterization and regulation of antagonist binding to putative muscarinic subtypes.
Topics: Animals; Benzodiazepinones; Buffers; Cerebral Cortex; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Myocardium; Parasympatholytics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1986 |
Selective effects of gold (III) on parathyroid hormone-, prostaglandin E2- and guanine nucleotide-sensitive adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Chick Embryo; Dinoprostone; Dose-Response Relationship, Drug; Ethylmaleimide; Gold; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Magnesium; Osteoblasts; Parathyroid Hormone; Prostaglandins E | 1985 |
Modulation of forskolin binding to rat brain membranes.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Brain; Cations, Divalent; Cations, Monovalent; Cell Membrane; Chymotrypsin; Colforsin; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Rats; Sodium Fluoride; Trypsin | 1985 |
Interaction of opiate receptor binding sites and guanine nucleotide regulatory sites: selective protection from N-ethylmaleimide.
Topics: Adenylyl Imidodiphosphate; Animals; Binding Sites; Brain; Diprenorphine; Enkephalin, Methionine; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Opioid | 1984 |
Characteristics of the guanine nucleotide regulatory component of adenylate cyclase in human erythrocyte membranes.
Topics: Adenylyl Cyclases; Animals; Chemical Phenomena; Chemistry; Cholera Toxin; Erythrocyte Membrane; Erythrocytes; Ethylmaleimide; Fluorides; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Humans; Mice; Molecular Weight; NAD; Protein Binding; Rats; Receptors, Adrenergic, beta; Turkeys | 1980 |
Kinetics of interaction between beta-receptors, GTP protein, and the catalytic unit of turkey erythrocyte adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Enzyme Activation; Epinephrine; Erythrocyte Membrane; Erythrocytes; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanylyl Imidodiphosphate; Kinetics; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Cell Surface; Turkeys | 1982 |
Coupling of the canine renal parathyroid hormone receptor to adenylate cyclase: modulation by guanyl nucleotides and N-ethylmaleimide.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Dogs; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kidney; Kinetics; Parathyroid Hormone; Peptide Fragments; Receptors, Cell Surface; Receptors, Parathyroid Hormone; Teriparatide | 1982 |
Agonist and antagonist affinities for inhibitory adenosine receptors are reciprocally affected by 5'-guanylylimidodiphosphate or N-ethylmaleimide.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Ethylmaleimide; Female; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Hippocampus; Male; Phenylisopropyladenosine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Purinergic | 1983 |
Reconstitution of a functional beta-adrenergic receptor using cholate and a novel method for its functional assay.
Topics: Adenylyl Cyclases; Animals; Cholic Acids; Erythrocyte Membrane; Ethylmaleimide; Guanylyl Imidodiphosphate; Receptors, Adrenergic; Receptors, Adrenergic, beta; Solubility; Turkeys | 1983 |
Microsomal opiate receptors: characterization of smooth microsomal and synaptic membrane opiate receptors.
Topics: Animals; Brain; Dihydromorphine; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Intracellular Membranes; Manganese; Microsomes; Morphine; Naloxone; Rats; Receptors, Opioid; Synaptic Membranes | 1984 |
Interaction of forskolin with dually regulated adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Blood Platelets; Cell Line; Colforsin; Diterpenes; Drug Interactions; Enzyme Activation; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hormones; Humans; Lymphoma; Manganese; Mice; Receptors, Cell Surface | 1984 |
Modulation of muscarinic cholinergic receptor affinity for antagonists in rat heart.
Topics: Animals; Binding, Competitive; Cold Temperature; Computers; Ethylmaleimide; Female; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Magnesium; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thionucleotides | 1984 |
Photoaffinity identification of colchicine-solubilized regulatory subunit from rat brain adenylate cyclase.
Topics: Adenylyl Cyclases; Affinity Labels; Animals; Azides; Brain; Colchicine; Enzyme Activation; Ethylmaleimide; GTP-Binding Proteins; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Rats; Rats, Inbred Strains; Synaptic Membranes; Vinblastine | 1984 |
A kinetic analysis of activation of smooth muscle adenylate cyclase by forskolin.
Topics: Adenylyl Cyclases; Animals; Antihypertensive Agents; Colforsin; Diterpenes; Enzyme Activation; Ethylmaleimide; Female; Guanylyl Imidodiphosphate; Kinetics; Magnesium; Muscle, Smooth; Rats; Uterus | 1984 |
Characterization of transducin from bovine retinal rod outer segments. The role of sulfhydryl groups.
Topics: Amino Acids; Animals; Cattle; Dithionitrobenzoic Acid; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Membrane Proteins; Nitrobenzoates; Photoreceptor Cells; Rod Cell Outer Segment; Sulfhydryl Compounds; Transducin; Tritium | 1984 |
Muscarinic receptors in porcine caudate nucleus. II. Different effects of N-ethylmaleimide on [3H]cis-methyldioxolane binding to heat-labile (guanyl nucleotide-sensitive) sites and heat-stable (guanyl nucleotide-insensitive) sites.
Topics: Animals; Caudate Nucleus; Dioxolanes; Ethylmaleimide; Guanine Nucleotides; Guanylyl Imidodiphosphate; Hot Temperature; In Vitro Techniques; Nickel; Receptors, Muscarinic; Swine; Trypsin | 1983 |
Differential regulation of high-affinity agonist binding to muscarinic sites in the rat heart, cerebellum, and cerebral cortex.
Topics: Animals; Cerebellum; Cerebral Cortex; Ethylmaleimide; Guanylyl Imidodiphosphate; Magnesium; Male; Myocardium; Rats; Receptors, Muscarinic; Sodium | 1983 |
Potentiation of monovalent cation effects on ligand binding to cardiac muscarinic receptors in N-ethylmaleimide treated membranes.
Topics: Ammonia; Animals; Cations, Monovalent; Chick Embryo; Drug Synergism; Ethylmaleimide; Guanylyl Imidodiphosphate; Myocardium; Oxotremorine; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic | 1983 |
Proteolysis of skeletal muscle adenylate cyclase. Destruction and reconstitution of fluoride and guanylnucleotide sensitivity.
Topics: Adenylyl Cyclases; Animals; Cell Membrane; Ethylmaleimide; Fluorides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Muscles; Rabbits; Sodium Fluoride; Subtilisins | 1980 |
Regulation of muscarinic receptor binding by guanine nucleotides and N-ethylmaleimide.
Topics: Animals; Binding, Competitive; Brain; Dioxolanes; Ethylmaleimide; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Kinetics; Male; Parasympathomimetics; Quinuclidinyl Benzilate; Rats; Receptors, Cholinergic; Receptors, Muscarinic | 1980 |
Inactivation of cardiac adenylate cyclase by oxidation, trivalent arsenicals, and N-ethylmaleimide.
Topics: Adenylyl Cyclase Inhibitors; Animals; Arsenicals; Cell Membrane; Dithiothreitol; Ethylmaleimide; Fluorides; Guanylyl Imidodiphosphate; Hydrogen Peroxide; Kinetics; Myocardium; Oxidation-Reduction; Rabbits | 1981 |
Skeletal muscle adenylate cyclase: reconstitution of fluoride and guanylnucleotide sensitivity.
Topics: Adenylyl Cyclases; Animals; Detergents; Ethylmaleimide; Fluorides; Guanine Nucleotides; Guanylyl Imidodiphosphate; Hot Temperature; Muscles; Myocardium; Rabbits; Solubility | 1980 |
Hybridization of adenylate cyclase components by membrane fusion and the effect of selective digestion by trypsin.
Topics: Adenylyl Cyclases; Animals; Cell Fusion; Cell Membrane; Erythrocyte Membrane; Erythrocytes; Ethylmaleimide; Guanylyl Imidodiphosphate; Isoproterenol; Leukemia, Experimental; Mice; Trypsin; Turkeys | 1980 |
Induction of G protein-independent agonist high-affinity binding sites of D-1 dopamine receptors by beta-mercaptoethanol.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Binding Sites; Cell Membrane; Corpus Striatum; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Kinetics; Macromolecular Substances; Male; Mercaptoethanol; Molecular Weight; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1 | 1994 |
Inhibitory effects of NaCl and guanyl-5'yl-imidodiphosphate (GppNHp) on [3H]naloxone binding to kappa-opioid receptors in guinea pig cerebellum.
Topics: Animals; Benzeneacetamides; Binding Sites; Cerebellum; Cerebral Cortex; Corpus Striatum; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylmaleimide; Guanylyl Imidodiphosphate; Guinea Pigs; Male; Naloxone; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa; Sodium Chloride | 1993 |
Stable GDP analog-induced inactivation of G(i) proteins promotes cardiac adenylyl cyclase inhibition by guanosine 5'-(beta gamma-imino)triphosphate and muscarinic acetylcholine receptor.
Topics: Adenylyl Cyclase Inhibitors; Animals; Carbachol; Dogs; Ethylmaleimide; GTP-Binding Proteins; Guanosine Diphosphate; Guanylyl Imidodiphosphate; Magnesium; Manganese; Myocardium; Receptors, Muscarinic; Sarcolemma; Thionucleotides | 1996 |
[3H]-(R)-N6-Phenylisopropyladenosine agonist binding to the solubilized A1 adenosine receptor from bovine epididymal spermatozoa.
Topics: Animals; Cattle; Cell Membrane; Epididymis; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Ligands; Male; Phenylisopropyladenosine; Receptors, Purinergic P1; Signal Transduction; Spermatozoa | 1997 |
A muscarinic acetylcholine receptor, present in the epithelial cell line from Chironomus tentans.
Topics: Animals; Atropine; Binding Sites; Binding, Competitive; Blotting, Western; Carbachol; Cell Line; Chironomidae; Ecdysterone; Epithelium; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Oxotremorine; Pirenzepine; Quinuclidinyl Benzilate; Receptors, Cholinergic | 1996 |
Role of cysteine residues of rat A2a adenosine receptors in agonist binding.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cell Membrane; Corpus Striatum; Cysteine; Dithiothreitol; Ethylmaleimide; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Sulfhydryl Reagents | 1997 |
Inhibition of [3H]forskolin binding by Gpp[NH]p may reflect adenylyl cyclase coupling to Gi.
Topics: Adenylyl Cyclases; Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Cerebellum; Colforsin; Corpus Striatum; Enzyme Inhibitors; Ethylmaleimide; GTP-Binding Protein alpha Subunits, Gi-Go; Guanylyl Imidodiphosphate; Male; Rats; Rats, Sprague-Dawley; Tritium | 1998 |
Active nuclear import of single-stranded oligonucleotides and their complexes with non-karyophilic macromolecules.
Topics: Animals; Biological Transport, Active; Cell Membrane Permeability; Cell Nucleus; Cells, Cultured; Digitonin; DNA, Single-Stranded; Ethylmaleimide; Fibroblasts; Fluorescein-5-isothiocyanate; Guanylyl Imidodiphosphate; Humans; Macropodidae; Mice; Microinjections; Microscopy, Confocal; Nuclear Envelope; Oligodeoxyribonucleotides; Proteins; Serum Albumin, Bovine; Streptavidin; Wheat Germ Agglutinins | 1998 |
Alterations in cardiac membrane beta-adrenoceptors and adenylyl cyclase due to hypochlorous acid.
Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Ascorbic Acid; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hypochlorous Acid; Immunoblotting; Isoproterenol; Lipid Peroxidation; Methionine; Myocardium; Pertussis Toxin; Pindolol; Propane; Rats; Receptors, Adrenergic; Sodium Fluoride; Virulence Factors, Bordetella | 1999 |
G protein coupling of CGS 21680 binding sites in the rat hippocampus and cortex is different from that of adenosine A1 and striatal A2A receptors.
Topics: Adenosine; Animals; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Cholera Toxin; Corpus Striatum; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Pertussis Toxin; Phenethylamines; Purinergic P1 Receptor Agonists; Pyrimidines; Rats; Rats, Wistar; Receptors, Purinergic P1; Triazines; Triazoles; Tritium; Virulence Factors, Bordetella | 1999 |
Inhibition of [3H]forskolin binding by Gpp[NH]p may reflect adenylate cyclase coupling to Gi.
Topics: Adenylyl Cyclases; Animals; Autoradiography; Brain; Cerebellum; Colforsin; Corpus Striatum; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Rats; Rats, Sprague-Dawley; Tritium | 1999 |
In vitro autoradiographic visualization of guanosine-5'-O-(3-[35S]thio)triphosphate binding stimulated by sphingosine 1-phosphate and lysophosphatidic acid.
Topics: Animals; Autoradiography; Binding Sites; Brain; Enzyme Inhibitors; Ethylmaleimide; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Guinea Pigs; Image Processing, Computer-Assisted; In Vitro Techniques; Lysophospholipids; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Sphingosine; Sulfur Radioisotopes | 1999 |
Anatomical distribution of sodium-dependent [(3)H]naloxone binding sites in rat brain.
Topics: Animals; Autoradiography; Binding Sites; Brain; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethylmaleimide; Guanylyl Imidodiphosphate; Kinetics; Male; Naloxone; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Sodium; Tissue Distribution; Tritium | 2000 |
Effect of light on phosphatidate phosphohydrolase activity of retina rod outer segments: the role of transducin.
Topics: Adenosine Diphosphate Ribose; Animals; Cattle; Cell Membrane; Cholera Toxin; Darkness; Ethylmaleimide; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanylyl Imidodiphosphate; Hydrolysis; Isoenzymes; Light; Lipoprotein Lipase; Pertussis Toxin; Phosphatidate Phosphatase; Rod Cell Outer Segment; Thionucleotides; Transducin; Virulence Factors, Bordetella | 2000 |
Alkylation of sulfhydryl groups on Galpha(s/olf) subunits by N-ethylmaleimide: regulation by guanine nucleotides.
Topics: Alkylation; Animals; Brain; Cell Membrane; Ethylmaleimide; GTP-Binding Protein alpha Subunits; Guanine Nucleotides; Guanylyl Imidodiphosphate; Heterotrimeric GTP-Binding Proteins; Kinetics; Protein Subunits; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sulfhydryl Compounds | 2003 |
Pharmacological characterization of oxytocin-binding sites in rat spinal cord membranes: comparison with embryonic cultured spinal cord neurones and astrocytes.
Topics: Aging; Animals; Astrocytes; Binding Sites; Ethylmaleimide; Guanylyl Imidodiphosphate; Magnesium; Neurons; Oxytocin; Rats; Rats, Wistar; Spinal Cord | 1997 |