Page last updated: 2024-08-23

ethylketocyclazocine and mr 2266

ethylketocyclazocine has been researched along with mr 2266 in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-199026 (92.86)18.7374
1990's2 (7.14)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bueno, L; Gué, M; Junien, JL1
Dykstra, LA; Picker, MJ1
Cameron, DP; Ma, A; Ma, V1
Bicknell, RJ; Chapman, C; Leng, G1
Buder, M; Fuder, H; Riers, HD; Rothacher, G1
Buéno, L; Gué, M; Hondé, C; Junien, JL; Pascaud, X1
Berzetei, IP; Duckles, SP; Fong, A; Yamamura, HI1
Portoghese, PS; Takemori, AE1
Boublik, J; Funder, JW; Jefferys, D1
Bettermann, R; Illes, P1
Aoki, K; Ishii, K; Kajiwara, M; Matsumiya, T; Numata, H; Oka, T1
Hiramatsu, M; Kameyama, T; Nabeshima, T2
Ahmed, MS; Horst, MA1
Calcagnetti, DJ; Cramer, CP; Fanselow, MS; Helmstetter, FJ1
Cooper, SJ; Turkish, S1
Fitzjarrell, AT; Heath, RG; Walker, CF1
Huidobro-Toro, JP; Parada, S1
Corbett, AD; Gillan, MG; Kosterlitz, HW; McKnight, AT; Paterson, SJ; Robson, LE1
Huidobro-Toro, JP; Way, EL; Yoshimura, K1
Leander, JD1
Gautret, B; Schmitt, H1
Akkerman, AM; Bakel, HC; Büscher, H; Hill, RC; Maurer, R; Petcher, TJ; Römer, D; Welle, HB1
Kosterlitz, HW; Paterson, SJ; Robson, LE1
Herz, A; Shearman, GT1
Ishizuka, Y; Kajiwara, M; Matsumiya, T; Negishi, K; Oka, T; Watanabe, Y1
Gulati, K; Puri, S; Ray, A; Sen, P1
Rabkin, SW1

Other Studies

28 other study(ies) available for ethylketocyclazocine and mr 2266

ArticleYear
Central and peripheral opioid modulation of gastric relaxation induced by feeding in dogs.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cyclazocine; Dogs; Dose-Response Relationship, Drug; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Morphine; Muscle Relaxation; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Stomach; Vagotomy; Vagus Nerve

1989
Discriminative stimulus effects of mu and kappa opioids in the pigeon: analysis of the effects of full and partial mu and kappa agonists.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Columbidae; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Morphinans; Naloxone; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1989
Regulation of feeding behaviour in monosodium glutamate (MSG) treated mice.
    Life sciences, 1988, Volume: 42, Issue:15

    Topics: Animals; Animals, Newborn; Benzomorphans; Cyclazocine; Eating; Ethylketocyclazocine; Glutamates; Mice; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Glutamate

1988
Effects of opioid agonists and antagonists on oxytocin and vasopressin release in vitro.
    Neuroendocrinology, 1985, Volume: 41, Issue:2

    Topics: Animals; Arginine Vasopressin; Benzomorphans; beta-Endorphin; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Naloxone; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains

1985
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1986
Peripheral antagonistic action of trimebutine and kappa opioid substances on acoustic stress-induced gastric motor inhibition in dogs.
    European journal of pharmacology, 1988, Jan-27, Volume: 146, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acoustic Stimulation; Analgesics; Analgesics, Opioid; Animals; Benzoates; Benzomorphans; Cyclazocine; Dogs; Ethylketocyclazocine; Gastrointestinal Motility; Injections, Intravenous; Injections, Intraventricular; Naloxone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stress, Psychological; Trimebutine

1988
Characterization of kappa opioid receptors in the rabbit ear artery.
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: Animals; Benzeneacetamides; Benzomorphans; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle, Smooth, Vascular; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1988
TENA, a selective kappa opioid receptor antagonist.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Azocines; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
A kappa-selective opioidergic pathway is involved in the reversal of a behavioural effect of adrenalectomy.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Adrenalectomy; Animals; Benzomorphans; Cyclazocine; Enkephalins; Ethylketocyclazocine; Immobilization; Male; Memory; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
Classification of presynaptic opioid receptors in the rabbit ear artery by competitive antagonists.
    European journal of pharmacology, 1986, Mar-11, Volume: 122, Issue:1

    Topics: Animals; Arteries; Benzomorphans; Binding, Competitive; Biological Assay; Cyclazocine; Ear; Enkephalin, Leucine; Ethylketocyclazocine; In Vitro Techniques; Naloxone; Rabbits; Receptors, Opioid; Synaptic Membranes

1986
Agonist and antagonist actions of buprenorphine on three types of opioid receptor in isolated preparations.
    Japanese journal of pharmacology, 1986, Volume: 40, Issue:1

    Topics: Animals; Benzomorphans; Buprenorphine; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Morphinans; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Species Specificity; Time Factors; Vas Deferens

1986
Phencyclidine-induced stereotyped behaviors after injection of ethylketocyclazocine, Mr 2266 and naltrexone in rats.
    Brain research, 1986, Jul-23, Volume: 378, Issue:2

    Topics: Animals; Benzomorphans; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Male; Motor Skills; Naltrexone; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Stereotyped Behavior

1986
Opioid receptors of human placental villi modulate acetylcholine release.
    Life sciences, 1986, Aug-11, Volume: 39, Issue:6

    Topics: Acetylcholine; Animals; Benzomorphans; Cyclazocine; Endorphins; Ethylketocyclazocine; Humans; Organ Culture Techniques; Placenta; Rats; Receptors, Opioid

1986
Involvement of opioid receptors in hypo- and hyperthermic effects induced by phencyclidine in mice.
    Journal of pharmacobio-dynamics, 1986, Volume: 9, Issue:5

    Topics: Animals; Benzomorphans; Body Temperature; Cyclazocine; Ethylketocyclazocine; Hyperthermia, Induced; Hypothermia, Induced; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Phenazocine; Phencyclidine; Receptors, Opioid

1986
Ethylketocyclazocine and bremazocine analgesia in neonatal rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Analgesia; Analgesics; Animals; Animals, Newborn; Benzomorphans; Cyclazocine; Ethylketocyclazocine; Female; Male; Morphinans; Naltrexone; Narcotic Antagonists; Rats

1988
Effects of a kappa receptor agonist, ethylketocyclazocine, on water consumption in water-deprived and nondeprived rats in diurnal and nocturnal tests.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:1

    Topics: Animals; Benzomorphans; Circadian Rhythm; Cyclazocine; Drinking Behavior; Ethylketocyclazocine; Male; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Water Deprivation

1984
Kappa opiate receptor agonists: effects on behavior and on brain function and structure in rhesus monkeys.
    Biological psychiatry, 1984, Volume: 19, Issue:7

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Behavior, Animal; Benzomorphans; Brain; Computers; Cyclazocine; Dose-Response Relationship, Drug; Electroencephalography; Ethylketocyclazocine; Evoked Potentials; Macaca mulatta; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1984
Kappa-opiates and urination: pharmacological evidence for an endogenous role of the kappa-opiate receptor in fluid and electrolyte balance.
    European journal of pharmacology, 1984, Dec-15, Volume: 107, Issue:1

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Female; Injections, Intraperitoneal; Morphinans; Morphine; Naloxone; Potassium; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium; Water-Electrolyte Balance

1984
Radioligands for probing opioid receptors.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Pro-Opiomelanocortin; Protein Precursors; Pyrrolidines; Radioligand Assay; Rats; Receptors, Opioid; Vas Deferens

1984
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists

1982
Further study of kappa opioids on increased urination.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Male; Morphinans; Naloxone; Narcotic Antagonists; Narcotics; Piperidines; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Urination

1983
Cardiac slowing induced by peripheral kappa-opiate receptor stimulation in rats.
    European journal of pharmacology, 1984, Jun-15, Volume: 102, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Benzomorphans; Cyclazocine; Electrocardiography; Ethylketocyclazocine; Heart Rate; Hemodynamics; Injections, Intravenous; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Time Factors; Vagotomy

1984
Bremazocine: a potent, long-acting opiate kappa-agonist.
    Life sciences, 1980, Sep-15, Volume: 27, Issue:11

    Topics: Analgesia; Animals; Benzomorphans; Brain; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; Macaca mulatta; Male; Mice; Morphinans; Morphine; Naloxone; Pentazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1980
Characterization of the kappa-subtype of the opiate receptor in the guinea-pig brain.
    British journal of pharmacology, 1981, Volume: 73, Issue:4

    Topics: Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Naloxone; Naltrexone; Narcotics; Phenoxybenzamine; Receptors, Opioid

1981
Evidence that the discriminative stimulus properties of fentanyl and ethylketocyclazocine are mediated by an interaction with different opiate receptors.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 221, Issue:3

    Topics: Animals; Benzomorphans; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Fentanyl; Male; Rats; Rats, Inbred Strains; Receptors, Opioid

1982
The choice of opiate receptor subtype by neo-endorphins.
    European journal of pharmacology, 1982, Apr-23, Volume: 79, Issue:3-4

    Topics: Animals; Benzomorphans; beta-Endorphin; Cyclazocine; Drug Interactions; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Naloxone; Protein Precursors; Rabbits; Receptors, Opioid

1982
Role of kappa opioid receptors during stress responsiveness in rats.
    Indian journal of experimental biology, 1993, Volume: 31, Issue:2

    Topics: Animals; Benzomorphans; Corticosterone; Ethylketocyclazocine; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Wistar; Receptors, Opioid, kappa; Stomach Ulcer; Stress, Physiological

1993
The opioid agonist ethylketocyclazocine accentuates epinephrine-induced cardiac arrhythmias in the rat through an action in the brain.
    Brain research bulletin, 1993, Volume: 31, Issue:3-4

    Topics: Animals; Arrhythmias, Cardiac; Benzomorphans; Blood Pressure; Brain; Dose-Response Relationship, Drug; Electrocardiography; Epinephrine; Ethylketocyclazocine; Injections; Male; Narcotic Antagonists; Rats; Rats, Wistar

1993