Page last updated: 2024-08-23

ethylketocyclazocine and ketazocine

ethylketocyclazocine has been researched along with ketazocine in 104 studies

Research

Studies (104)

TimeframeStudies, this research(%)All Research%
pre-199084 (80.77)18.7374
1990's17 (16.35)18.2507
2000's2 (1.92)29.6817
2010's1 (0.96)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Eades, CG; Gilbert, PE; Huppler, RE; Martin, WR; Thompson, JA1
Gulati, K; Ray, A; Sharma, KK2
Barr, GA; Miya, DY; Paredes, W1
Gent, JP; Goodchild, CS; Serrao, JM1
Funder, JW; Jefferys, D1
Cone, EJ; Vaupel, DB1
Shea-Donohue, T; Touzeau, PL1
Hoss, W; Periyasamy, S1
Bartness, TJ; Billington, CJ; Herman, BH; Levine, AS; Morley, JE1
LoPresti, D; Porreca, F; Ward, SJ1
Edwards, M; Gent, JP; Goodchild, CS; Serrao, JM1
Clark, WC; Haertzen, CA; Janal, MN; Kumor, KM1
Chahl, LA1
Balster, RL1
DiBona, GF; Jones, SY; Kapusta, DR1
Cameron, DP; Ma, A; Ma, V1
Dykstra, LA; Massie, CA1
Caudill, A; Condon, RE; Szurszewski, JH; Telford, GL1
Bryant, HU; Lowy, MT; Malven, PV; Steele, TD; Yim, GK1
Cooper, SJ; Jackson, A; Kirkham, TC1
Bryant, HU; Malven, PV; Steele, TD; Yim, GK1
Hirst, M; Kavaliers, M2
Boublik, J; Funder, JW; Jefferys, D1
Hayes, A; Kelly, A1
Gosnell, BA; Levine, AS; Morley, JE; Waggoner, DW1
DeRossett, SE; Holtzman, SG1
Kitchen, I; McDowell, J1
Hirst, M; Kavaliers, M; Rangeley, RW; Teskey, GC1
Haertzen, CA; Jasinski, D; Johnson, RE; Kocher, T; Kumor, KM1
Goldberg, S; Haertzen, C; Johnson, RE; Kumor, K; Su, TP; Vaupel, B1
Barr, GA; Erickson, KL; Paredes, W; Zukin, RS1
Barr, GA; Giordano, J2
Bagley, RB; Compton, DR; Katzen, JS; Martin, BR1
Kadlec, O; Masek, K; Sebestová, L; Seferna, I1
Kadlec, O; Masek, K; Seferna, I1
Gosnell, BA; Levine, AS; Morley, JE; Romsos, DR2
Hart, JC; Leander, JD; Zerbe, RL1
Haertzen, CA; Jasinski, DR; Johnson, RE; Kumor, KM1
Maher, TJ; Moya-Huff, FA1
Dykstra, LA; Picker, M1
Baragatti, G; Caron, F; Gavend, MM; Gavend, MR; Pastrello, D; Serre-Debeauvais, F1
Brocklehurst, C; Devia, C; Moerschbaecher, JM1
Dykstra, LA; Heise, JW; Picker, M1
Beck, T; Krieglstein, J1
Buchwald, WD; Cone, EJ; Kumor, K; Yousefnejad, D1
Bergman, J; Hassoun, J; Schuster, CR1
Leander, JD5
Bryant, HU; Malven, PV; Yim, GK1
Gosnell, BA; Levine, AS; Morley, JE2
Khazan, N; Young, GA3
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Yoshimura, K3
Miller, RJ1
Sewell, RD; Spencer, PS; Upton, N1
Herz, A1
Ben-Sreti, MM; Gonzalez, JP; Sewell, RD1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Zhu, YX1
Gosnell, BA; Grace, M; Kneip, J; Levine, AS; Morley, JE2
Pasternak, GW1
Akkerman, AM; Bakel, HC; Büscher, H; Hill, RC; Maurer, R; Petcher, TJ; Römer, D; Welle, HB1
Harris, RA; Snell, D1
Grace, M; Kniep, J; Levine, AS; Morley, JE1
Hirst, M; Tepperman, FS1
Brown, DR; Holtzman, SG; Locke, KW1
Kandasamy, SB; Williams, BA1
Cicero, TJ; Meyer, ER; Owens, DP; Schmoeker, PF1
Grace, M; Kneip, J; Levine, AS; Morley, JE; Zeugner, H1
Boublik, JH; Clements, JA; Funder, JW; Herington, AC1
Altura, BM; Altura, BT; Quirion, R1
Bajorek, JG; Lee, RJ; Lomax, P1
Holtzman, SG; White, JM1
Cowan, A; Porreca, F; Raffa, RB; Tallarida, RJ1
Dykstra, LA2
Lowy, MT; Yim, GK1
Haertzen, CA; Henningfield, JE; Hickey, JE; Jasinski, DR; Johnson, RE; Kumor, K1
Kitchen, I1
Chaillet, P; Costentin, J; Marçais-Collado, H1
Colpaert, FC; Janssen, PA1
Isaacson, RL; Lanthorn, TH1
Iwamoto, ET1
Dykstra, LA; Milar, KS1
Moerschbaecher, JM; Thompson, DM1
Castañeda-Hernández, G; Flores-Murrieta, FJ; Granados-Soto, V; Hong, E; López-Muñoz, FJ1
Bandoli, G; Grassi, A; Pappalardo, GC1
Funder, JW; Jefferys, DE1
Gulati, K; Puri, S; Ray, A; Sen, P1
Gulati, K1
Bakthavachalam, V; Bidlack, JM; Cohen, DJ; Gao, P; Mello, NK; Negus, SS; Neumeyer, JL; Zong, R1
Brandt, W; Cambareri, A; Englberger, W; Friderichs, E; Haurand, M; Holzgrabe, U; Kögel, B; Kuhl, U; Siener, T; Strassburger, W1
Devaud, JM; Farina, WM; Fernández, VM; Giurfa, M1

Reviews

3 review(s) available for ethylketocyclazocine and ketazocine

ArticleYear
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response

1985
Multiple opiate receptors for multiple opioid peptides.
    Medical biology, 1982, Volume: 60, Issue:1

    Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission

1982
Multiple opiate receptors and their functional significance.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Morphine; Receptors, Opioid; Tissue Distribution

1983

Trials

3 trial(s) available for ethylketocyclazocine and ketazocine

ArticleYear
Multidimensional scaling of subjective judgements of drug similarities among ketocyclazocine, morphine, cyclazocine, naloxone and placebo.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:2

    Topics: Adult; Cyclazocine; Ethylketocyclazocine; Generalization, Stimulus; Humans; Male; Models, Psychological; Morphine; Naloxone

1990
Human psychopharmacology of ketocyclazocine as compared with cyclazocine, morphine and placebo.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:3

    Topics: Adult; Blood Pressure; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Euphoria; Hallucinations; Humans; Male; Morphine; Placebos; Pupil; Receptors, Opioid; Receptors, Opioid, kappa; Substance-Related Disorders; Time Factors

1986
The psychopharmacologic and prolactin response after large doses of naloxone in man.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:4

    Topics: Adult; Blood Pressure; Body Temperature; Cyclazocine; Discrimination, Psychological; Ethylketocyclazocine; Humans; Male; Models, Theoretical; Morphine; Naloxone; Prolactin; Pulse; Pupil; Respiration

1988

Other Studies

98 other study(ies) available for ethylketocyclazocine and ketazocine

ArticleYear
The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog.
    The Journal of pharmacology and experimental therapeutics, 1976, Volume: 197, Issue:3

    Topics: Animals; Apomorphine; Cyclazocine; Cyclopropanes; Dextropropoxyphene; Dogs; Ethylketocyclazocine; Humans; Morphinans; Morphine; Morphine Dependence; Nalorphine; Naltrexone; Phenazocine; Spinal Cord

1976
Effects of acute and chronic ketocyclazocine and its modulation by oxytocin or vasopressin on food intake in rats.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 41, Issue:1

    Topics: Animals; Arginine Vasopressin; Drug Tolerance; Eating; Ethylketocyclazocine; Light; Male; Oxytocin; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Time Factors; Vasopressins

1992
Effects of acute or chronic opioid agonists and their modulation by diurnal rhythmicity and satiety states on food intake in rats.
    Indian journal of experimental biology, 1992, Volume: 30, Issue:3

    Topics: Animals; Circadian Rhythm; Eating; Ethylketocyclazocine; Male; Morphine; Rats; Rats, Inbred Strains; Satiety Response; Time Factors

1992
Analgesic effects of intraventricular and intrathecal injection of morphine and ketocyclazocine in the infant rat.
    Brain research, 1992, Jul-03, Volume: 584, Issue:1-2

    Topics: Analgesics; Animals; Animals, Newborn; Behavior, Animal; Cold Temperature; Ethylketocyclazocine; Hot Temperature; Injections, Intraventricular; Injections, Spinal; Morphine; Postural Balance; Rats; Reaction Time; Reflex; Respiration; Spinal Cord

1992
Reversal by naloxone of spinal antinociceptive effects of fentanyl, ketocyclazocine and midazolam.
    European journal of anaesthesiology, 1991, Volume: 8, Issue:5

    Topics: Analgesia, Epidural; Animals; Catheters, Indwelling; Dose-Response Relationship, Drug; Drug Tolerance; Electric Stimulation; Ethylketocyclazocine; Fentanyl; Flumazenil; Injections, Spinal; Lumbar Vertebrae; Male; Midazolam; Naloxone; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Opioid; Sensory Thresholds

1991
The forced swimming test: effects of glucose administration on the response to food deprivation and adrenalectomy.
    European journal of pharmacology, 1991, Dec-03, Volume: 205, Issue:3

    Topics: Adrenal Glands; Adrenalectomy; Animals; Behavior, Animal; Dexamethasone; Ethylketocyclazocine; Food Deprivation; Glucose; Male; Movement; Physical Exertion; Rats; Rats, Inbred Strains; Swimming; Time Factors

1991
Pharmacodynamic and pharmacokinetic actions of ketocyclazocine enantiomers in the dog: absence of sigma- or phencyclidine-like activity.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Dogs; Dose-Response Relationship, Drug; Drug Administration Schedule; Ethylketocyclazocine; Female; Morphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, sigma; Stereoisomerism; Time Factors

1991
Kappa agonists inhibit gastric emptying but not acid secretion in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Antihypertensive Agents; Cyclazocine; Dynorphins; Ethylketocyclazocine; Gastric Acid; Gastric Emptying; Macaca mulatta; Male; Narcotics; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Sodium

1990
Kappa opioid receptors stimulate phosphoinositide turnover in rat brain.
    Life sciences, 1990, Volume: 47, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Dynorphins; Enkephalins; Ethylketocyclazocine; Male; Phosphatidylinositols; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1990
Effects of the opiate antagonists diprenorphine and naloxone and of selected opiate agonists on feeding behavior in guinea pigs.
    Life sciences, 1990, Volume: 46, Issue:2

    Topics: Animals; Butorphanol; Circadian Rhythm; Cyclazocine; Diprenorphine; Ethylketocyclazocine; Feeding Behavior; Guinea Pigs; Morphinans; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Opioid agonist affinity in the guinea-pig ileum and mouse vas deferens.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Methadone; Mice; Morphine; Morphine Derivatives; Naltrexone; Receptors, Opioid; Vas Deferens

1990
On the mechanism by which midazolam causes spinally mediated analgesia.
    Anesthesiology, 1990, Volume: 73, Issue:2

    Topics: Analgesia, Epidural; Animals; Bicuculline; Cyclazocine; Dose-Response Relationship, Drug; Electric Stimulation; Ethylketocyclazocine; Fentanyl; Flumazenil; Male; Midazolam; Pain; Rats; Rats, Inbred Strains; Receptors, GABA-A; Sensory Thresholds

1990
Withdrawal responses of guinea-pig isolated ileum following brief exposure to opiates and opioid peptides.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:4

    Topics: Animals; Benzomorphans; Buprenorphine; Cyclazocine; Endorphins; Ethylketocyclazocine; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle, Smooth; Naloxone; Narcotics; Substance P; Substance Withdrawal Syndrome

1986
Substitution and antagonism in rats trained to discriminate (+)-N-allylnormetazocine from saline.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 249, Issue:3

    Topics: Animals; Binding Sites; Butaclamol; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Haloperidol; Male; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Phencyclidine

1989
Role of renal nerves in excretory responses to administration of kappa agonists in conscious spontaneously hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Diuresis; Ethylketocyclazocine; Hemodynamics; Hypertension; Kidney; Male; Pyrrolidines; Rats; Rats, Inbred SHR; Receptors, Opioid; Receptors, Opioid, kappa; Sympathetic Nervous System

1989
Regulation of feeding behaviour in monosodium glutamate (MSG) treated mice.
    Life sciences, 1988, Volume: 42, Issue:15

    Topics: Animals; Animals, Newborn; Benzomorphans; Cyclazocine; Eating; Ethylketocyclazocine; Glutamates; Mice; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Glutamate

1988
Antagonism of the analgesic effects of mu and kappa opioid agonists in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Azocines; Benzomorphans; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Fentanyl; Male; Methadone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri

1988
Ketocyclazocine, a kappa-opioid receptor agonist, and control of intestinal myoelectric activity in dogs.
    The American journal of physiology, 1988, Volume: 255, Issue:5 Pt 1

    Topics: Animals; Cyclazocine; Dogs; Electromyography; Ethylketocyclazocine; Intestine, Small; Muscle, Smooth; Receptors, Opioid; Receptors, Opioid, kappa; Stomach

1988
Effects of 2% sodium chloride imbibition on various opiate related hyperphagic conditions.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:3

    Topics: Animals; Cyclazocine; Deoxyglucose; Dynorphins; Ethylketocyclazocine; Feeding Behavior; Insulin; Male; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride; Time Factors

1985
Nocturnal depletion of hypothalamic dynorphin in anorexic Walker-256 tumor-bearing rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:3

    Topics: Animals; Anorexia; Carcinoma 256, Walker; Circadian Rhythm; Cyclazocine; Dynorphins; Eating; Ethylketocyclazocine; Feeding and Eating Disorders; Hypothalamus; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1988
The influence of opiate agonists on day-night feeding rhythms in young and old mice.
    Brain research, 1985, Feb-04, Volume: 326, Issue:1

    Topics: Aging; Animals; Cyclazocine; Endorphins; Ethylketocyclazocine; Feeding Behavior; Male; Mice; Morphine; Naloxone; Periodicity; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1985
A kappa-selective opioidergic pathway is involved in the reversal of a behavioural effect of adrenalectomy.
    European journal of pharmacology, 1985, Jan-08, Volume: 107, Issue:3

    Topics: Adrenalectomy; Animals; Benzomorphans; Cyclazocine; Enkephalins; Ethylketocyclazocine; Immobilization; Male; Memory; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1985
Profile of activity of kappa receptor agonists in the rabbit vas deferens.
    European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Ethylketocyclazocine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
The pineal gland and opiate-induced feeding.
    Physiology & behavior, 1985, Volume: 34, Issue:1

    Topics: Animals; Butorphanol; Cyclazocine; Endorphins; Ethylketocyclazocine; Feeding Behavior; Male; Melatonin; Morphine; Naloxone; Pineal Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
Effects of opiate antagonists and putative kappa agonists on unpunished and punished operant behavior in the rat.
    Psychopharmacology, 1985, Volume: 86, Issue:4

    Topics: Animals; Conditioning, Operant; Cyclazocine; Diprenorphine; Ethylketocyclazocine; Male; Naloxone; Narcotic Antagonists; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
Impairment of ketocyclazocine antinociception in rats by perinatal lead exposure.
    Toxicology letters, 1985, Volume: 26, Issue:2-3

    Topics: Animals; Animals, Newborn; Animals, Suckling; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Lead; Lead Poisoning; Pain; Pregnancy; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sensory Thresholds

1985
Mu- and kappa-opiate agonists modulate ingestive behaviors in the slug, Limax maximus.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Ethylketocyclazocine; Feeding Behavior; Mollusca; Morphine; Narcotic Antagonists; Narcotics; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Time Factors

1986
Studies of kappa agonist.
    NIDA research monograph, 1986, Volume: 67

    Topics: Animals; Brain; Cyclazocine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Humans; Morphine; Naloxone; Receptors, Opioid; Receptors, Opioid, kappa

1986
Kappa opioid receptor-mediated analgesia in the developing rat.
    Brain research, 1986, Volume: 394, Issue:2

    Topics: Age Factors; Animals; Brain; Cyclazocine; Drug Tolerance; Ethylketocyclazocine; Hot Temperature; Morphine; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986
Food hoarding and ingestion in the deer mouse, Peromyscus maniculatus: selective responses to mu and kappa opiate agonists.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Endorphins; Ethylketocyclazocine; Feeding Behavior; Food Deprivation; Male; Morphine; Peromyscus; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1986
Morphine- and ketocyclazocine-induced analgesia in the developing rat: differences due to type of noxious stimulus and body topography.
    Brain research, 1987, Volume: 429, Issue:2

    Topics: Age Factors; Analgesics; Animals; Animals, Suckling; Central Nervous System; Cyclazocine; Ethylketocyclazocine; Morphine; Naloxone; Pain; Pain Measurement; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1987
(+)- and (-)-N-allylnormetazocine binding sites in mouse brain: in vitro and in vivo characterization and regional distribution.
    Life sciences, 1987, Jun-01, Volume: 40, Issue:22

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Ethylketocyclazocine; Haloperidol; In Vitro Techniques; Mice; Naloxone; Phenazocine; Phencyclidine; Receptors, Opioid; Receptors, sigma; Stereoisomerism

1987
The topography and dynamics of cholinergic transmission in the myenteric plexus-smooth muscle preparation of the guinea-pig ileum; the effect of ketocyclazocine, a kappa opiate ligand.
    Physiologia Bohemoslovaca, 1987, Volume: 36, Issue:1

    Topics: Acetylcholine; Animals; Cyclazocine; Electric Stimulation; Electromyography; Ethylketocyclazocine; Guinea Pigs; Ileum; Ligands; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Parasympathetic Nervous System; Synaptic Transmission

1987
The topography of cholinergic transmission in the mechanism of drug action at muscarinic synapses of the guinea-pig ileum.
    European journal of pharmacology, 1987, Apr-14, Volume: 136, Issue:2

    Topics: Action Potentials; Animals; Axons; Cholinergic Fibers; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Synaptic Transmission

1987
Opiates and medial hypothalamic knife cuts cause hyperphagia through different mechanisms.
    Behavioral neuroscience, 1985, Volume: 99, Issue:6

    Topics: Animals; Brain Mapping; Butorphanol; Cyclazocine; Dietary Carbohydrates; Dietary Fats; Eating; Ethylketocyclazocine; Hypothalamus, Middle; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid

1985
Kappa agonist-induced diuresis: evidence for stereoselectivity, strain differences, independence of hydration variables and a result of decreased plasma vasopressin levels.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 242, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Butorphanol; Cyclazocine; Diuresis; Drinking; Ethylketocyclazocine; Female; Male; Nalorphine; Pyrrolidines; Rats; Rats, Inbred Strains; Rats, Zucker; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Vasopressins; Water Deprivation

1987
Phenylpropanolamine decreases food intake in rats made hyperphagic by various stimuli.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:1

    Topics: Animals; Appetite Depressants; Cyclazocine; Deoxyglucose; Dextroamphetamine; Eating; Ethylketocyclazocine; Feeding and Eating Disorders; Food Deprivation; Hyperphagia; Insulin; Male; Motor Activity; Phenylpropanolamine; Rats; Rats, Inbred Strains

1987
Comparison of the discriminative stimulus properties of U50,488 and morphine in pigeons.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Columbidae; Cyclazocine; Dextroamphetamine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Female; Fentanyl; Methadone; Morphine; Naloxone; Phenazocine; Phencyclidine; Pyrrolidines; Time Factors

1987
Neurochemical actions of ethylketocyclazocine and ketocyclazocine in different regions of rat brain.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 1987, Volume: 41, Issue:7

    Topics: Animals; Brain; Cyclazocine; Dopamine; Ethylketocyclazocine; Male; Norepinephrine; Rats; Rats, Inbred Strains; Serotonin

1987
Differential antagonism by naltrexone of the effects of opioids on a fixed-ratio discrimination in rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1

    Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naltrexone; Narcotic Antagonists; Narcotics; Pentazocine; Rats

1988
Effects of neonatal spinal cord serotonin depletion on opiate-induced analgesia in tests of thermal and mechanical pain.
    Brain research, 1988, Jun-01, Volume: 469, Issue:1-2

    Topics: 5,7-Dihydroxytryptamine; Analgesia; Animals; Animals, Newborn; Cyclazocine; Desipramine; Dihydroxytryptamines; Ethylketocyclazocine; Hot Temperature; Morphine; Pain; Physical Stimulation; Rats; Serotonin; Spinal Cord

1988
Effects of kappa opiate agonists, cholecystokinin and bombesin on intake of diets varying in carbohydrate-to-fat ratio in rats.
    The Journal of nutrition, 1987, Volume: 117, Issue:5

    Topics: Animals; Body Weight; Bombesin; Butorphanol; Cyclazocine; Dietary Carbohydrates; Dietary Fats; Eating; Energy Intake; Ethylketocyclazocine; Food Preferences; Male; Naloxone; Rats; Rats, Inbred Strains; Sincalide

1987
Evaluation of the effects of opioid agonists and antagonists under a fixed-consecutive-number schedule in rats.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Male; Methadone; Morphine; Naloxone; Narcotics; Phenazocine; Pyrrolidines; Rats; Reinforcement Schedule

1987
The effects of tifluadom and ketazocine on behaviour, dopamine turnover in the basal ganglia and local cerebral glucose utilization of rats.
    Brain research, 1986, Sep-03, Volume: 381, Issue:2

    Topics: Animals; Benzodiazepines; Brain; Corpus Striatum; Cyclazocine; Dopamine; Ethylketocyclazocine; Glucose; Male; Motor Activity; Nucleus Accumbens; Rats; Rats, Inbred Strains

1986
Determination of ketocyclazocine in human plasma by gas chromatography-negative-ion chemical-ionization mass spectrometry.
    Journal of chromatography, 1986, Nov-28, Volume: 383, Issue:1

    Topics: Cyclazocine; Ethylketocyclazocine; Gas Chromatography-Mass Spectrometry; Humans; Indicators and Reagents; Injections, Intramuscular

1986
Behavioral effects of selected opiates and phencyclidine in the nondependent and cyclazocine-dependent rhesus monkey.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Ethylketocyclazocine; Food; Macaca mulatta; Male; Naloxone; Phenazocine; Phencyclidine; Stereoisomerism; Substance-Related Disorders

1985
Kappa opioid agonists and antagonists: effects on drinking and urinary output.
    Appetite, 1984, Volume: 5, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Clonidine; Cyclazocine; Drinking; Ethylketocyclazocine; Naloxone; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Urination; Vasopressins

1984
Differential inhibition by propranolol of feeding induced in rats by various stimuli.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:4

    Topics: Animals; Cyclazocine; Deoxyglucose; Dose-Response Relationship, Drug; Eating; Ethylketocyclazocine; Insulin; Male; Naloxone; Propranolol; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1984
Lesions of the globus pallidus and striatum attenuate ketocyclazocine-induced feeding.
    Physiology & behavior, 1984, Volume: 33, Issue:3

    Topics: Animals; Brain Mapping; Corpus Striatum; Cyclazocine; Endorphins; Ethylketocyclazocine; Feeding Behavior; Globus Pallidus; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1984
Differential neuropharmacological effects of mu, kappa and sigma opioid agonists on cortical EEG power spectra in the rat. Stereospecificity and naloxone antagonism.
    Neuropharmacology, 1984, Volume: 23, Issue:10

    Topics: Animals; Cerebral Cortex; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Methadone; Molecular Conformation; Morphine; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma

1984
Effects of full and partial kappa agonists and mu agonists on urine output of normally hydrated rats.
    Neuropeptides, 1984, Volume: 5, Issue:1-3

    Topics: Animals; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Naltrexone; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1984
Dynorphin interaction at the kappa-opiate site.
    European journal of pharmacology, 1981, Jun-19, Volume: 72, Issue:2-3

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Receptors, Opioid; Receptors, Opioid, kappa

1981
Kappa opioid properties of dynorphin and its peptide fragments on the guinea-pig Ileum.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:1

    Topics: Animals; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Receptors, Opioid; Receptors, Opioid, kappa

1982
Activation of K-opiate sites by dynorphin in the myenteric plexus.
    Advances in biochemical psychopharmacology, 1982, Volume: 33

    Topics: Animals; Cyclazocine; Drug Tolerance; Dynorphins; Electric Stimulation; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa

1982
Effects of ketazocine, ethylketazocine and phenazocine on schedule-controlled behavior: antagonism by naloxone.
    Neuropharmacology, 1982, Volume: 21, Issue:9

    Topics: Analgesics, Opioid; Animals; Columbidae; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Naloxone; Phenazocine

1982
Analgesic actions of mu- and kappa-opiate agonists in rats.
    Archives internationales de pharmacodynamie et de therapie, 1983, Volume: 262, Issue:2

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Hot Temperature; Male; Nociceptors; Pain; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1983
Effects of elevated calcium and calcium antagonists on 6,7-benzomorphan-induced analgesia.
    European journal of pharmacology, 1983, Jun-17, Volume: 90, Issue:4

    Topics: Analgesia; Analgesics; Analgesics, Opioid; Animals; Benzomorphans; Calcium; Calcium Channel Blockers; Cyclazocine; Egtazic Acid; Ethylketocyclazocine; Gallopamil; Male; Mice; Morphinans; Pentazocine; Phenazocine

1983
Further study of kappa opioids on increased urination.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cyclazocine; Diuresis; Ethylketocyclazocine; Male; Morphinans; Naloxone; Narcotic Antagonists; Narcotics; Piperidines; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Urination

1983
Dynorphin inhibition of the neurotensin contractile activity on the myenteric plexus.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:2

    Topics: Animals; Atropine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Nerve Tissue Proteins; Neurotensin; Peptide Fragments; Receptors, Opioid; Tetrodotoxin

1984
The effect of ovariectomy, estradiol and progesterone on opioid modulation of feeding.
    Physiology & behavior, 1984, Volume: 33, Issue:2

    Topics: Animals; Appetite Regulation; Brain; Castration; Cyclazocine; Dynorphins; Eating; Estradiol; Ethylketocyclazocine; Female; Naloxone; Progesterone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1984
Multiple opiate receptors: [3H]ethylketocyclazocine receptor binding and ketocyclazocine analgesia.
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:6

    Topics: Analgesics; Animals; Brain; Cyclazocine; Dihydromorphine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Mice; Morphine; Motor Activity; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa

1980
Bremazocine: a potent, long-acting opiate kappa-agonist.
    Life sciences, 1980, Sep-15, Volume: 27, Issue:11

    Topics: Analgesia; Animals; Benzomorphans; Brain; Cyclazocine; Electric Stimulation; Ethylketocyclazocine; Guinea Pigs; Ileum; Macaca mulatta; Male; Mice; Morphinans; Morphine; Naloxone; Pentazocine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1980
Interactions between narcotic agonists, partial agonists andd antagonists evaluated by punished an unpunished behavior in the rat.
    Psychopharmacology, 1982, Volume: 76, Issue:2

    Topics: Animals; Conditioning, Psychological; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Narcotics; Phenazocine; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid

1982
A kappa opioid effect: increased urination in the rat.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Diuretics; Ethylketocyclazocine; Male; Narcotic Antagonists; Narcotics; Phencyclidine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1983
An investigation of the role of kappa opiate receptor agonists in the initiation of feeding.
    Life sciences, 1982, Dec-06, Volume: 31, Issue:23

    Topics: Animals; Circadian Rhythm; Cyclazocine; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Starvation; Time Factors

1982
Concerning the specificity of the hypothalamic opiate receptor responsible for food intake in the rat.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6

    Topics: Animals; Body Temperature Regulation; Codeine; Cyclazocine; Dextrorphan; Eating; Ethylketocyclazocine; Levorphanol; Male; Morphine; Naloxone; Phencyclidine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Ventromedial Hypothalamic Nucleus

1982
Effects of opiate antagonists and putative mu- and kappa-agonists on milk intake in rat and squirrel monkey.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6

    Topics: Animals; Buprenorphine; Cyclazocine; Diazepam; Diprenorphine; Drinking; Ethylketocyclazocine; Etorphine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Taste

1982
Peptide and non-peptide opioid-induced hyperthermia in rabbits.
    Brain research, 1983, Apr-11, Volume: 265, Issue:1

    Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptides; Phenazocine; Rats

1983
Differential stereospecific effects of mu, kappa, and sigma opioid agonists on cortical EEG power spectra in the rat.
    NIDA research monograph, 1983, Volume: 43

    Topics: Animals; Cerebral Cortex; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Methadone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma; Stereoisomerism

1983
Opiate-induced enhancement of the effects of naloxone on serum luteinizing hormone levels in the male rat: specificity for Mu agonists.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Binding, Competitive; Cyclazocine; Ethanol; Ethylketocyclazocine; Kinetics; Luteinizing Hormone; Male; Morphine; Naloxone; Pentobarbital; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
The effect of the opioid-benzodiazepine, tifluadom, on ingestive behaviors.
    European journal of pharmacology, 1983, Sep-30, Volume: 93, Issue:3-4

    Topics: Animals; Benzodiazepines; Butorphanol; Cyclazocine; Drinking Behavior; Ethylketocyclazocine; Feeding Behavior; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1983
Opiate binding sites in bovine adrenal medulla.
    Journal of receptor research, 1983, Volume: 3, Issue:4

    Topics: Adrenal Medulla; Animals; Binding Sites; Brain; Brain Chemistry; Cattle; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
N-allylnormetazocine (SKF-10,047): the induction of feeding by a putative sigma agonist.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:5

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Eating; Ethylketocyclazocine; Male; Morphine; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid

1983
The kappa opioid receptor, ingestive behaviors and the obese mouse (ob/ob).
    Physiology & behavior, 1983, Volume: 31, Issue:5

    Topics: Animals; Appetite; Benzodiazepines; Body Weight; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Drinking; Eating; Ethylketocyclazocine; Male; Mice; Mice, Obese; Receptors, Opioid; Receptors, Opioid, kappa

1983
Identification of benzomorphan-kappa opiate receptors in cerebral arteries which subserve relaxation.
    British journal of pharmacology, 1984, Volume: 82, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Cerebral Arteries; Cyclazocine; Dinoprost; Dogs; Drug Interactions; Ethylketocyclazocine; Female; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phencyclidine; Prostaglandins F; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1984
Similar anticonvulsant, but unique, behavioural effects of opioid agonists in the seizure-sensitive Mongolian gerbil.
    Neuropharmacology, 1984, Volume: 23, Issue:5

    Topics: Animals; Anticonvulsants; Behavior, Animal; Cyclazocine; Electroencephalography; Ethylketocyclazocine; Female; Gerbillinae; Male; Morphine; Narcotics; Phenazocine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures

1984
Further characterization of the three-choice morphine, cyclazocine and saline discrimination paradigm: opioids with agonist and antagonist properties.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Animals; Cyclazocine; Discrimination Learning; Discrimination, Psychological; Ethylketocyclazocine; Male; Morphine; Narcotic Antagonists; Narcotics; Phenazocine; Phencyclidine; Rats; Sodium Chloride; Stereoisomerism

1983
Ketazocines and morphine: effects on gastrointestinal transit after central and peripheral administration.
    Life sciences, 1983, Apr-11, Volume: 32, Issue:15

    Topics: Animals; Cyclazocine; Ethylketocyclazocine; Gastrointestinal Motility; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Phenazocine; Rats; Rats, Inbred Strains

1983
Self-administration of ketocyclazocine and ethylketocyclazocine by the rat.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:4

    Topics: Animals; Cyclazocine; Drug Tolerance; Electroencephalography; Ethylketocyclazocine; Female; Humans; Injections, Intravenous; Opioid-Related Disorders; Rats; Rats, Inbred Strains; Self Administration

1983
Effects of ketocyclazocine and ethylketocyclazocine on electric shock titration.
    European journal of pharmacology, 1983, Oct-14, Volume: 94, Issue:1-2

    Topics: Animals; Behavior, Animal; Cyclazocine; Dose-Response Relationship, Drug; Drug Interactions; Drug Tolerance; Electroshock; Ethylketocyclazocine; Morphine; Naloxone; Saimiri

1983
Stimulation of food intake following opiate agonists in rats but not hamsters.
    Psychopharmacology, 1983, Volume: 81, Issue:1

    Topics: Animals; Cricetinae; Cyclazocine; Dose-Response Relationship, Drug; Drinking Behavior; Ethylketocyclazocine; Feeding Behavior; Male; Meperidine; Mesocricetus; Morphine; Narcotics; Rats; Rats, Inbred Strains; Species Specificity

1983
Progress report from the NIDA Addiction Research Center Baltimore, Maryland (1984).
    NIDA research monograph, 1984, Volume: 55

    Topics: Blood Pressure; Body Temperature; Compulsive Behavior; Cyclazocine; Discrimination Learning; Endorphins; Ethylketocyclazocine; Euphoria; Gambling; Glucose; Heart Rate; Humans; Morphine; Naloxone; Nicotine; Perception; Respiration; Substance-Related Disorders; Time Factors

1984
Modification of an analgesy meter for paw-pressure antinociceptive testing in neonatal rats.
    Journal of pharmacological methods, 1984, Volume: 12, Issue:4

    Topics: Aging; Analgesics; Animals; Animals, Newborn; Cyclazocine; Drug Evaluation, Preclinical; Ethylketocyclazocine; Foot; Pressure; Rats; Tail

1984
Development of enhanced sensitivity to naloxone.
    Life sciences, 1983, Nov-21, Volume: 33, Issue:21

    Topics: Animals; Buprenorphine; Cyclazocine; Diprenorphine; Dose-Response Relationship, Drug; Drug Interactions; Ethylketocyclazocine; Male; Meperidine; Naloxone; Phencyclidine; Reaction Time; Saimiri

1983
Catatonic or hypotonic immobility induced in mice by intracerebroventricular injection of mu or kappa opioid receptor agonists as well as enkephalins or inhibitors of their degradation.
    Life sciences, 1983, Nov-21, Volume: 33, Issue:21

    Topics: Animals; Benzomorphans; Catatonia; Cyclazocine; Enkephalins; Ethylketocyclazocine; Fentanyl; Humans; Immobilization; Injections, Intraventricular; Male; Mice; Morphine; Naloxone; Narcotic Antagonists; Narcotics

1983
Agonist and antagonist effects of prototype opiate drugs in rats discriminating fentanyl from saline: characteristics of partial generalization.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Animals; Conditioning, Operant; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Fentanyl; Male; Morphine; Nalorphine; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Sodium Chloride

1984
Hippocampal involvement in the pharmacologic induction of withdrawal-like behaviors.
    Federation proceedings, 1981, Volume: 40, Issue:5

    Topics: Animals; Cyclazocine; Endorphins; Enkephalin, Methionine; Enkephalins; Escape Reaction; Ethylketocyclazocine; Hippocampus; Humans; Injections, Intraventricular; Kainic Acid; Morphine Dependence; Pyrrolidines; Rats; Serotonin; Shivering; Substance Withdrawal Syndrome; Valproic Acid

1981
Pharmacologic effects of N-allylnormetazocine (SKF-10047).
    NIDA research monograph, 1981, Volume: 34

    Topics: Analgesics; Animals; Behavior, Animal; Clonidine; Cyclazocine; Ethylketocyclazocine; Male; Morphine; Motor Activity; Phenazocine; Rats; Receptors, Dopamine; Spiperone

1981
Effects of ketocyclazocine alone and in combination with naloxone on schedule-controlled responding in squirrel monkeys.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 18, Issue:3

    Topics: Animals; Conditioning, Operant; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Male; Naloxone; Reinforcement Schedule; Saimiri

1983
Differential effects of prototype opioid agonists on the acquisition of conditional discriminations in monkeys.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Animals; Behavior, Animal; Conditioning, Psychological; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Erythrocebus patas; Ethylketocyclazocine; Male; Morphine; Pentazocine; Phenazocine; Psychomotor Performance

1983
Evidence against the participation of mu- and kappa-opioid receptors in the analgesic activity of ketorolac in rats.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:6

    Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Ethylketocyclazocine; Female; Ketorolac; Morphine; Movement Disorders; Naloxone; Pain Measurement; Rats; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu; Time Factors; Tolmetin

1995
X-ray molecular structures and theoretical conformational studies of narcotic analgesics alpha-(-)-N-cis-3-chloroallyl-normetazocine, ethylketazocine, and ketazocine.
    Journal of pharmaceutical sciences, 1993, Volume: 82, Issue:8

    Topics: Analgesics, Opioid; Benzomorphans; Crystallography; Ethylketocyclazocine; Molecular Conformation; Stereoisomerism

1993
The thyroadrenal axis, food deprivation and retention of a behavioural response.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: Adrenal Glands; Adrenalectomy; Animals; Behavior, Animal; Dexamethasone; Ethylketocyclazocine; Food Deprivation; Male; Rats; Rats, Sprague-Dawley; Thyroid Gland; Thyroxine

1993
Role of kappa opioid receptors during stress responsiveness in rats.
    Indian journal of experimental biology, 1993, Volume: 31, Issue:2

    Topics: Animals; Benzomorphans; Corticosterone; Ethylketocyclazocine; Male; Naltrexone; Narcotic Antagonists; Rats; Rats, Wistar; Receptors, Opioid, kappa; Stomach Ulcer; Stress, Physiological

1993
Differential effects of intrahypothalamic administration of opioids on food intake in naive and tolerant rats.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:4

    Topics: Animals; Eating; Ethylketocyclazocine; Hypothalamus; Male; Morphine; Naltrexone; Narcotics; Rats; Rats, Wistar; Time Factors

1995
Synthesis and opioid receptor affinity of morphinan and benzomorphan derivatives: mixed kappa agonists and mu agonists/antagonists as potential pharmacotherapeutics for cocaine dependence.
    Journal of medicinal chemistry, 2000, Jan-13, Volume: 43, Issue:1

    Topics: Acetic Acid; Animals; Benzomorphans; Brain; Dose-Response Relationship, Drug; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Injections, Intraventricular; Male; Mice; Mice, Inbred ICR; Morphinans; Morphine; Narcotic Antagonists; Pain; Pain Measurement; Reaction Time; Receptors, Opioid, kappa; Receptors, Opioid, mu

2000
Diazabicyclononanones, a potent class of kappa opioid analgesics.
    Farmaco (Societa chimica italiana : 1989), 2002, Volume: 57, Issue:7

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Brain; Carboxylic Acids; Ethylketocyclazocine; Models, Molecular; Molecular Structure; Pyridines; Quantitative Structure-Activity Relationship; Rats; Receptors, Opioid, kappa

2002
Latent inhibition in an insect: the role of aminergic signaling.
    Learning & memory (Cold Spring Harbor, N.Y.), 2012, Nov-16, Volume: 19, Issue:12

    Topics: Analysis of Variance; Animals; Bees; Conditioning, Classical; Dibenzazepines; Dopamine; Dopamine Antagonists; Ethylketocyclazocine; Extinction, Psychological; Fluphenazine; Habituation, Psychophysiologic; Histamine H1 Antagonists; Imidazoles; Inhibition, Psychological; Ketanserin; Methysergide; Odorants; Serotonin; Serotonin Antagonists; Smell

2012