ethylketocyclazocine has been researched along with etorphine in 35 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 30 (85.71) | 18.7374 |
1990's | 4 (11.43) | 18.2507 |
2000's | 1 (2.86) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Coale, EH; Hein, DW; Herling, S; Valentino, RJ; Woods, JH | 1 |
Cruciani, RA; Munson, PJ; Pesce, GO; Rodbard, D | 1 |
Ahmed, MS; Cavinato, AG; Maulik, D; Zhou, DH | 1 |
Blake, JW; DeQuick, D; Kamerling, S; Tai, C; Tobin, T; Weckman, TJ; Wood, T | 1 |
Bowen, WD; Copeland, CF; Kooper, GN; Levinson, NR | 1 |
Su, TP | 1 |
Carino, MA; Horita, A; Yamawaki, S | 1 |
Buder, M; Fuder, H; Riers, HD; Rothacher, G | 1 |
Barchfeld-Rothschild, CC; Medzihradsky, F | 1 |
Cruciani, RA; Gainer, H; Lang, MA; Pesce, GO; Rodbard, D; Russell, JT | 1 |
Adler, MW; Geller, EB; Rowan, CH | 1 |
Holford, NH; Rosenbaum, JS; Sadée, W | 1 |
Bunn, SJ; Hanley, MR; Wilkin, GP | 1 |
Boudouresque, F; Bourhim, N; Cantau, P; Castanas, E; Giraud, P; Oliver, C | 1 |
Cros, J; Gouardères, C; Kopp, N; Quirion, R | 1 |
Fischel, SV; Medzihradsky, F | 1 |
Brown, SR; Cote, TE; Cox, BM; Puttfarcken, P; Werling, LL | 1 |
Brown, SR; Cox, BM; Puttfarcken, P; Werling, LL | 1 |
Hynes, MD; Leander, JD; Reel, JK; Zimmerman, DM | 1 |
Gardner, EL; Vaysse, PJ; Zukin, RS | 1 |
Catt, KJ; Dufau, ML; Stojilković, SS | 1 |
Delay-Goyet, P; Roques, BP; Zajac, JM | 1 |
Bradford, HF; White, EJ | 1 |
Cros, J; Porthé, G; Valette, A | 1 |
Dahlstrom, PJ; Fischel, SV; Medzihradsky, F; Mitsos, SE; Woods, JH | 1 |
Audigier, Y; Cros, J; Gouardéres, C | 1 |
Guidotti, A; Saiani, L | 1 |
Attali, B; Audigier, Y; Cros, J; Gouardères, C; Mazarguil, H | 1 |
Brown, DR; Holtzman, SG; Locke, KW | 1 |
Ahmed, MS | 1 |
Herling, S; Woods, JH | 1 |
Bakogeorgou, E; Castanas, E; Hatzoglou, A | 1 |
Calvo, F; Castanas, E; Hatzoglou, A; Martin, PM; Panagiotou, S | 1 |
Bakogeorgou, E; Castanas, E; Dussert, C; Hatzoglou, A; Martin, PM; Panagiotou, S; Papakonstanti, E; Stournaras, C; Wallet, F | 1 |
Benaderet, TS; Bishop-Mathis, K; Dersch, CM; Partilla, JS; Prisinzano, TE; Rothman, RB; Simpson, DS; Wang, X; Xu, H | 1 |
1 review(s) available for ethylketocyclazocine and etorphine
Article | Year |
---|---|
Narcotic analgesics, their detection and pain measurement in the horse: a review.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Butorphanol; Chromatography, Thin Layer; Cyclazocine; Ethylketocyclazocine; Etorphine; Fentanyl; Horses; Morphine; Pain Measurement; Pentazocine; Pyrrolidines; Radioimmunoassay; Receptors, Opioid | 1989 |
34 other study(ies) available for ethylketocyclazocine and etorphine
Article | Year |
---|---|
Narcotic drug discriminations by rhesus monkeys and pigeons.
Topics: Animals; Columbidae; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalins; Ethylketocyclazocine; Etorphine; Hormones; Macaca; Macaca mulatta; Naltrexone; Narcotics; Phenazocine | 1979 |
Computer modeling of subtypes of kappa opioid receptors in adrenal medulla.
Topics: Adrenal Medulla; Animals; Binding, Competitive; Cattle; Computer Simulation; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; In Vitro Techniques; Kinetics; Models, Biological; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa | 1990 |
Opioid binding properties of the purified kappa receptor from human placenta.
Topics: Benzomorphans; Binding, Competitive; Chromatography; Cyclazocine; Electrophoresis, Polyacrylamide Gel; Ethylketocyclazocine; Etorphine; Humans; Molecular Weight; Naloxone; Narcotics; Placenta; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, kappa | 1989 |
Photoaffinity labeling of opiate receptors using intrinsically photoactive 3H-opiates.
Topics: Affinity Labels; Animals; Benzomorphans; Binding Sites; Cholic Acids; Cyclazocine; Ethylketocyclazocine; Etorphine; In Vitro Techniques; Light; Male; Narcotics; Rats; Rats, Inbred Strains; Receptors, Opioid; Tritium | 1988 |
Further demonstration of kappa opioid binding sites in the brain: evidence for heterogeneity.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Binding Sites; Brain; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Levallorphan; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism | 1985 |
Analeptic effect of opiate receptor agonists in rabbits.
Topics: Animals; Arousal; Brain; Central Nervous System Stimulants; Codeine; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Methionine; Ethylketocyclazocine; Etorphine; Male; Meperidine; Methadone; Morphine; Naltrexone; Narcotics; Phenazocine; Rabbits; Receptors, Opioid; Reflex | 1985 |
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro.
Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses | 1986 |
Heterogeneity of opioid receptor binding in brain slices.
Topics: Analgesics, Opioid; Animals; Brain; Corpus Striatum; Cyclazocine; Dihydromorphine; Ethylketocyclazocine; Etorphine; In Vitro Techniques; Male; Morphinans; Morphine Derivatives; Rats; Rats, Inbred Strains; Receptors, Opioid | 1987 |
Opioid receptors of bovine posterior pituitary neurosecretosomes are exclusively kappa.
Topics: Analgesics, Opioid; Animals; Cattle; Cyclazocine; Cytoplasmic Granules; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Kinetics; Morphinans; Pituitary Gland, Posterior; Receptors, Opioid; Receptors, Opioid, kappa | 1986 |
Body temperature effects of opioids in rats: intracerebroventricular administration.
Topics: Animals; beta-Endorphin; Body Temperature; Cyclazocine; Dose-Response Relationship, Drug; Endorphins; Ethylketocyclazocine; Etorphine; Heroin; Injections, Intraventricular; Injections, Subcutaneous; Male; Morphine; Naloxone; Narcotics; Pentazocine; Phenazocine; Rats; Rats, Inbred Strains | 1986 |
In vivo receptor binding of opioid drugs at the mu site.
Topics: Animals; Brain; Cyclazocine; Ethylketocyclazocine; Etorphine; Female; Guanosine Triphosphate; In Vitro Techniques; Narcotic Antagonists; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, mu; Sodium; Tritium | 1985 |
Evidence for a kappa-opioid receptor on pituitary astrocytes: an autoradiographic study.
Topics: Animals; Astrocytes; Autoradiography; Binding Sites; Binding, Competitive; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Pituitary Gland; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
Interaction of opiates with opioid binding sites in the bovine adrenal medulla: II. Interaction with kappa sites.
Topics: Adrenal Medulla; Animals; Benzomorphans; Binding Sites; Calcium; Cattle; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Ethylketocyclazocine; Ethylmaleimide; Etorphine; Guinea Pigs; Kinetics; Lithium; Manganese; Narcotics; Oligopeptides; Phospholipases A; Potassium; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Stereoisomerism | 1985 |
Kappa opioid receptors in human lumbo-sacral spinal cord.
Topics: Adult; Aged; Binding Sites; Cyclazocine; Endorphins; Ethylketocyclazocine; Etorphine; Female; Humans; Lumbosacral Region; Male; Middle Aged; Narcotics; Osmolar Concentration; Receptors, Opioid; Spinal Cord | 1986 |
Interaction between [3H]ethylketocyclazocine and [3H]etorphine and opioid receptors in membranes from rat brain. A kinetic analysis.
Topics: Animals; Brain; Computers; Cyclazocine; Drug Interactions; Ethylketocyclazocine; Etorphine; Kinetics; Ligands; Membranes; Morphinans; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1986 |
Sodium regulation of agonist binding at opioid receptors. I. Effects of sodium replacement on binding at mu- and delta-type receptors in 7315c and NG108-15 cells and cell membranes.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Glioma; Guinea Pigs; Monensin; Naloxone; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Sodium | 1986 |
Sodium regulation of agonist binding at opioid receptors. II. Effects of sodium replacement on opioid binding in guinea pig cortical membranes.
Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Guinea Pigs; Male; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium | 1986 |
Use of beta-funaltrexamine to determine mu opioid receptor involvement in the analgesic activity of various opioid ligands.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Biological Assay; Buprenorphine; Butorphanol; Cyclazocine; Dose-Response Relationship, Drug; Ethylketocyclazocine; Etorphine; Fentanyl; Methadone; Mice; Morphine; Muscle Contraction; Nalbuphine; Nalorphine; Naltrexone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, mu | 1987 |
Modulation of rat brain opioid receptors by cannabinoids.
Topics: Animals; Cannabinoids; Cyclazocine; Dihydromorphine; Dose-Response Relationship, Drug; Dronabinol; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Etorphine; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Spiperone | 1987 |
Opiate receptor subtypes in the rat hypothalamus and neurointermediate lobe.
Topics: Animals; Binding, Competitive; Cyclazocine; Ethylketocyclazocine; Etorphine; Female; Hypothalamus; Kinetics; Naloxone; Phencyclidine; Pituitary Gland; Rats; Rats, Inbred Strains; Receptors, Opioid; Temperature | 1987 |
Differences of binding characteristics of non-selective opiates towards mu and delta receptor types.
Topics: Animals; Binding, Competitive; Brain; Cell Membrane; Cerebellum; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Etorphine; Male; Oligopeptides; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu | 1987 |
Uptake of opioid drugs by rat cerebrocortical brain slices.
Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Ethylketocyclazocine; Etorphine; Kinetics; Membrane Lipids; Morphinans; Morphine; Rats; Rats, Inbred Strains | 1986 |
Kappa opiate binding sites in human placenta.
Topics: Analgesics, Opioid; Binding, Competitive; Cell Membrane; Cyclazocine; Ethylketocyclazocine; Etorphine; Female; Humans; Kinetics; Placenta; Potassium; Pregnancy; Receptors, Opioid; Receptors, Opioid, kappa; Sodium | 1981 |
Resolution in the receptor binding of putative mu and kappa opiates.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Cell Membrane; Columbidae; Cyclazocine; Ethylketocyclazocine; Etorphine; Kinetics; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Species Specificity | 1984 |
Benzomorphan binding sites in rat lumbo-sacral spinal cord.
Topics: Animals; Benzomorphans; Binding Sites; Cyclazocine; Ethylketocyclazocine; Etorphine; In Vitro Techniques; Kinetics; Lumbosacral Region; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord | 1982 |
Opiate receptor-mediated inhibition of catecholamine release in primary cultures of bovine adrenal chromaffin cells.
Topics: Acetylcholine; Adrenal Medulla; Animals; beta-Endorphin; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Phenazocine; Receptors, Opioid | 1982 |
Evidence for multiple "Kappa" binding sites by use of opioid peptides in the guinea-pig lumbo-sacral spinal cord.
Topics: Animals; Binding Sites; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord | 1982 |
Effects of opiate antagonists and putative mu- and kappa-agonists on milk intake in rat and squirrel monkey.
Topics: Animals; Buprenorphine; Cyclazocine; Diazepam; Diprenorphine; Drinking; Ethylketocyclazocine; Etorphine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Taste | 1982 |
Characterization of solubilized opiate receptors from human placenta.
Topics: Binding, Competitive; Chemical Phenomena; Chemistry, Physical; Cyclazocine; Ethylketocyclazocine; Etorphine; Female; Humans; Naloxone; Placenta; Pregnancy; Receptors, Opioid; Solubility | 1983 |
Discriminative stimulus effects of etorphine in Rhesus monkeys.
Topics: Animals; Codeine; Cyclazocine; Discrimination Learning; Ethylketocyclazocine; Etorphine; Macaca mulatta; Male; Meperidine; Morphinans; Morphine; Pentazocine; Phenazocine; Sodium Chloride | 1981 |
The antiproliferative effect of opioid receptor agonists on the T47D human breast cancer cell line, is partially mediated through opioid receptors.
Topics: Adenocarcinoma; Amino Acid Sequence; Binding Sites; Breast Neoplasms; Cell Division; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Humans; Molecular Sequence Data; Morphine; Narcotic Antagonists; Opioid Peptides; Receptors, Opioid; Tumor Cells, Cultured | 1996 |
Modulation of the estrogen-regulated proteins cathepsin D and pS2 by opioid agonists in hormone-sensitive breast cancer cell lines (MCF7 and T47D): evidence for an interaction between the two systems.
Topics: Breast Neoplasms; Cathepsin D; Cell Division; Cycloheximide; Cytosol; Diprenorphine; Dose-Response Relationship, Drug; Estradiol; Ethylketocyclazocine; Etorphine; Female; Humans; Inhibitory Concentration 50; Narcotic Antagonists; Narcotics; Neoplasms, Hormone-Dependent; Protein Synthesis Inhibitors; Proteins; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins | 1998 |
Opioid agonists modify breast cancer cell proliferation by blocking cells to the G2/M phase of the cycle: involvement of cytoskeletal elements.
Topics: Actins; Analgesics, Opioid; Breast Neoplasms; Cytoskeleton; Ethylketocyclazocine; Etorphine; G2 Phase; Humans; Mitosis; Tumor Cells, Cultured | 1999 |
Differential effects of opioid agonists on G protein expression in CHO cells expressing cloned human opioid receptors.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzamides; Blotting, Western; CHO Cells; Cricetinae; Cricetulus; Diterpenes, Clerodane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Female; Furans; Gene Expression; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Morphine; Oligopeptides; Piperazines; Pyrones; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 2008 |