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ethylketocyclazocine and enkephalin, leucine-2-alanine

ethylketocyclazocine has been researched along with enkephalin, leucine-2-alanine in 91 studies

Research

Studies (91)

Timeframe	Studies, this research(%)	All Research%
pre-1990	76 (83.52)	18.7374
1990's	13 (14.29)	18.2507
2000's	2 (2.20)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Kuhar, MJ; Wamsley, JK; Zarbin, MA	1
Benyhe, S; Borsodi, A; Varga, E; Wollemann, M	1
LoPresti, D; Porreca, F; Ward, SJ	1
Cruciani, RA; Munson, PJ; Pesce, GO; Rodbard, D	1
deGroat, WC; Hisamitsu, T; Nagel, J; Roppolo, JR; Thor, KB; Tuttle, P	1
Brantl, V; Liebmann, C; Schrader, U	1
Bhargava, HN; Ramarao, P	1
Garzon, J; Landahl, HD; Lee, NM	1
Rauch, RJ; Stephenson, JD; Stolerman, IP	1
De Souza, EB; Kuhar, MJ; Schmidt, WK	1
Imai, T; Kamikubo, K; Miura, K; Miura, Y; Miyashita, T; Murase, H; Nakamura, S; Niwa, M; Satoh, T; Tomita, A	1
Larson, DL; Lipkowski, AW; Nagase, H; Portoghese, PS; Takemori, AE	1
Ishizuka, Y; Oka, T	1
Bertelli, GM; Borea, PA; Gilli, G	1
Cicero, TJ; Nock, B; O'Connor, LH; Rajpara, A	1
Nagase, H; Portoghese, PS; Takemori, AE	1
Ho, BY; Naeseth, JS; Portoghese, PS; Takemori, AE	1
Su, TP	1
Bicknell, RJ; Chapman, C; Leng, G	1
Falke, NE; Fischer, EG; Martin, R	1
Illes, P; Ramme, D	1
Geppert, M; Illes, P; Jackisch, R	1
Buder, M; Fuder, H; Riers, HD; Rothacher, G	1
Brenner, AS; Geppert, M; Illes, P; Jackisch, R	1
Kirby, GC; McQueen, DS	1
Lipkowski, AW; Portoghese, PS; Takemori, AE	1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K	1
Benyhe, S; Borsodi, A; Hepp, J; Khan, A; Medzihradszky, K; Simon, J; Szücs, M; Wollemann, M	1
Cruciani, RA; Gainer, H; Lang, MA; Pesce, GO; Rodbard, D; Russell, JT	1
Goodman, SR; McLaughlin, PJ; Zagon, IS	1
Coscia, CJ; Roth, BL; Spain, JW	1
Portoghese, PS; Takemori, AE	2
Hammonds, RG; Ho, CL; Li, CH	1
Ensinger, HA	1
Neil, A	1
Brown, SR; Cox, BM; Werling, LL; Zarr, GD	2
Dewar, D; Jenner, P; Marsden, CD	2
Bunn, SJ; Hanley, MR; Wilkin, GP	1
Krall, S; Lynch, WC; Paden, CM; Watt, J	1
Boudouresque, F; Bourhim, N; Cantau, P; Castanas, E; Giraud, P; Oliver, C	1
Hirobe, M; Konno, F; Sato, Y; Takayanagi, I; Togashi, K	1
Bidlack, JM; Denton, RR	1
Bell, RD; Cicero, TJ	1
Itzhak, Y; Pasternak, GW	1
Glasel, JA; Myers, WE	1
Su, TP; Weissman, AD; Yeh, SY	1
Simon, EJ	1
Faden, AI; Krumins, SA	1
Brown, SR; Cote, TE; Cox, BM; Puttfarcken, P; Werling, LL	1
Brown, SR; Cox, BM; Puttfarcken, P; Werling, LL	1
Liu-Chen, LY; Tam, SW	1
Bakalkin, GIa; Iarygin, KN; Kobylianskiĭ, AG; Nesterenko, PN; Pivovarov, AS	1
Portoghese, PS; Schoenecker, JW; Takemori, AE	1
Krumins, SA	1
Lovett, JA; Portoghese, PS	1
Bardon, T; Ruckebusch, Y	1
Bardon, T; Pairet, M; Ruckebusch, Y	1
Garzón, J; Lee, NM; Sánchez-Blázquez, P	1
Loh, HH; Stokes, KB	1
Dawson, G; McLawhon, RW; Miller, RJ; West, RE	2
Ben-Sreti, MM; Sewell, RD	1
Tung, AS; Yaksh, TL	1
Goodman, RR; Snyder, SH	1
Fujibayashi, K; Iwama, T; Kubota, A; Satoh, M; Takagi, H; Wada, T; Yasui, M	1
Burkard, WP; Flück, N; Müller, PM	1
Gähwiler, BH; Maurer, R	1
Kosterlitz, HW; Paterson, SJ; Robson, LE	1
Lajtha, A; Reith, ME; Sershen, H; Vadasz, C	1
Herz, A; Shearman, GT	1
Nishimura, S; Pasternak, GW	1
Guidotti, A; Saiani, L	1
Takemori, AE; Ward, SJ	1
Attali, B; Audigier, Y; Cros, J; Gouardères, C; Mazarguil, H	1
Johnson, N; Pasternak, GW	1
Boublik, JH; Clements, JA; Funder, JW; Herington, AC	1
Killian, A; Mack, KJ; Weyhenmeyer, JA	1
Fan, XT; Kitamura, K; Liu, XF; Oka, T; Taniguchi, T	1
Castanas, E; Gravanis, A; Hatzoglou, A; Margioris, AN; Zoumakis, E	1
Barg, J; Nah, SY; Saya, D; Vogel, Z	1
Bakogeorgou, E; Castanas, E; Hatzoglou, A	1
Castanas, E; Hatzoglou, A; Kampa, M; Loukas, S; Martin, P; Martin, PM	1
Farouz-Grant, F; Portoghese, PS	1
Benyhe, S; Borsodi, A; Hepp, J; Ketevan, A; Medzihradszky, K; Simon, J	1
Elde, R; Kshirsagar, T; Law, PY; Nakano, AH; Portoghese, PS	1
Castanas, E; Denizot, A; Dermitzaki, I; Gravanis, A; Hatzoglou, A; Henry, JF; Kampa, M; Margioris, AN; Oliver, C	1
Castanas, E; Kampa, M; Kouroumalis, E; Nifli, AP; Notas, G; Papasava, D; Thermos, K; Xidakis, K	1
Benaderet, TS; Bishop-Mathis, K; Dersch, CM; Partilla, JS; Prisinzano, TE; Rothman, RB; Simpson, DS; Wang, X; Xu, H	1

Reviews

2 review(s) available for ethylketocyclazocine and enkephalin, leucine-2-alanine

Article	Year
Classification of opioid and 5-hydroxytryptamine receptors by means of discriminative drug effects. Neuropharmacology, 1987, Volume: 26, Issue:7B Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Conditioning, Classical; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Lysergic Acid Diethylamide; Narcotics; Nicotine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, Serotonin; Research Design; Tetrahydronaphthalenes	1987
Recent studies on opioid receptors: heterogeneity and purification. Annals of the New York Academy of Sciences, 1986, Volume: 463 Topics: Alcohols; Animals; Brain Chemistry; Centrifugation, Density Gradient; Chromatography, Affinity; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Ethylmaleimide; Humans; Lectins; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Solubility; Tritium; Wheat Germ Agglutinins	1986

Article

Year

Classification of opioid and 5-hydroxytryptamine receptors by means of discriminative drug effects.

Neuropharmacology, 1987, Volume: 26, Issue:7B

Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Conditioning, Classical; Cyclazocine; Discrimination Learning; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Lysergic Acid Diethylamide; Narcotics; Nicotine; Piperazines; Pyrimidines; Receptors, Opioid; Receptors, Serotonin; Research Design; Tetrahydronaphthalenes

1987

Recent studies on opioid receptors: heterogeneity and purification.

Annals of the New York Academy of Sciences, 1986, Volume: 463

Topics: Alcohols; Animals; Brain Chemistry; Centrifugation, Density Gradient; Chromatography, Affinity; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Ethylmaleimide; Humans; Lectins; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Solubility; Tritium; Wheat Germ Agglutinins

1986

Other Studies

89 other study(ies) available for ethylketocyclazocine and enkephalin, leucine-2-alanine

Article	Year
Anterograde transport of opioid receptors in rat vagus nerves and dorsal roots of spinal nerves: pharmacology and sensitivity to sodium and guanine nucleotides. Experimental brain research, 1990, Volume: 81, Issue:2 Topics: Animals; Axonal Transport; Colchicine; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guanosine Triphosphate; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride; Spinal Nerve Roots; Vagus Nerve	1990
The occurrence of different kappa opioid receptors (K1 and K2) in frog (Rana esculenta) brain membranes. Acta physiologica Hungarica, 1990, Volume: 76, Issue:4 Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Ligands; Morphinans; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa	1990
Opioid agonist affinity in the guinea-pig ileum and mouse vas deferens. European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Methadone; Mice; Morphine; Morphine Derivatives; Naltrexone; Receptors, Opioid; Vas Deferens	1990
Computer modeling of subtypes of kappa opioid receptors in adrenal medulla. European journal of pharmacology, 1990, Jul-17, Volume: 182, Issue:3 Topics: Adrenal Medulla; Animals; Binding, Competitive; Cattle; Computer Simulation; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; In Vitro Techniques; Kinetics; Models, Biological; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa	1990
Selective inhibitory effects of ethylketocyclazocine on reflex pathways to the external urethral sphincter of the cat. The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:3 Topics: Animals; Cats; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Morphine; Naloxone; Oligopeptides; Receptors, Opioid; Receptors, Opioid, kappa; Reflex; Urethra; Urinary Bladder; Urinary Incontinence	1989
Opioid receptor affinities of the blood-derived tetrapeptides hemorphin and cytochrophin. European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3 Topics: Animals; Brain Chemistry; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; Guinea Pigs; Hemoglobins; In Vitro Techniques; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1989
Antagonism of kappa opioid mediated effects in the rat by cyclo(Leu-Gly). Life sciences, 1989, Volume: 45, Issue:26 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cerebral Cortex; Cyclazocine; Diuresis; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Neuropeptides; Peptides, Cyclic; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord	1989
Computer analysis of the effect of beta-endorphin and dynorphin and related compounds on opioid binding to mouse brain membrane. Computers in biology and medicine, 1989, Volume: 19, Issue:3 Topics: Animals; beta-Endorphin; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Mice; Models, Neurological; Receptors, Opioid	1989
Nalbuphine: an autoradiographic opioid receptor binding profile in the central nervous system of an agonist/antagonist analgesic. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:1 Topics: Analgesia; Animals; Autoradiography; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Haplorhini; Male; Morphinans; Nalbuphine; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1988
Varying expression of opioid receptors and GTP-binding proteins in human pheochromocytomas. NIDA research monograph, 1986, Volume: 75 Topics: Adrenal Gland Neoplasms; beta-Endorphin; Cell Membrane; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; GTP-Binding Proteins; Humans; Pheochromocytoma; Receptors, Opioid	1986
Binaltorphimine-related bivalent ligands and their kappa opioid receptor antagonist selectivity. Journal of medicinal chemistry, 1988, Volume: 31, Issue:4 Topics: Animals; Chemical Phenomena; Chemistry; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Models, Molecular; Morphine; Muscle, Smooth; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa; Structure-Activity Relationship	1988
Relation of diltiazem binding sites to opioid receptor subtypes in the guinea-pig brain. The Tokai journal of experimental and clinical medicine, 1987, Volume: 12, Issue:1 Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Diltiazem; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Naloxone; Radioligand Assay; Receptors, Opioid	1987
Temperature dependence of the binding of mu, delta and kappa agonists to the opiate receptors in guinea-pig brain. European journal of pharmacology, 1988, Feb-09, Volume: 146, Issue:2-3 Topics: Animals; Brain; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Temperature	1988
[3H]U-69593 labels a subtype of kappa opiate receptor with characteristics different from that labeled by [3H]ethylketocyclazocine. Life sciences, 1988, Volume: 42, Issue:23 Topics: Animals; Benzeneacetamides; Binding, Competitive; Brain; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride; Temperature; Tritium	1988
Only one pharmacophore is required for the kappa opioid antagonist selectivity of norbinaltorphimine. Journal of medicinal chemistry, 1988, Volume: 31, Issue:7 Topics: Animals; Chemical Phenomena; Chemistry; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Morphine; Naltrexone; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Structure-Activity Relationship; Vas Deferens	1988
Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays. The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesia; Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naltrexone; Oligopeptides; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa	1988
Further demonstration of kappa opioid binding sites in the brain: evidence for heterogeneity. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Binding Sites; Brain; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Levallorphan; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism	1985
Effects of opioid agonists and antagonists on oxytocin and vasopressin release in vitro. Neuroendocrinology, 1985, Volume: 41, Issue:2 Topics: Animals; Arginine Vasopressin; Benzomorphans; beta-Endorphin; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Naloxone; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains	1985
Stereospecific opiate binding in living human polymorphonuclear leucocytes. Cell biology international reports, 1985, Volume: 9, Issue:11 Topics: Analgesics, Opioid; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Granulocytes; Humans; Kinetics; Naloxone; Neutrophils; Receptors, Opioid	1985
Differential effect of stimulation strength in mouse vas deferens on inhibition of neuroeffector transmission by receptor type selective opioids. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cyclazocine; Dynorphins; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Morphine Derivatives; Muscle, Smooth; Neuromuscular Junction; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Synaptic Transmission	1986
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit. Journal of neurochemistry, 1986, Volume: 46, Issue:6 Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid	1986
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2 Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1986
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit. Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2 Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses	1986
Characterization of opioid receptors in the cat carotid body involved in chemosensory depression in vivo. British journal of pharmacology, 1986, Volume: 88, Issue:4 Topics: Animals; Carotid Body; Cats; Chemoreceptor Cells; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hypercapnia; Hypoxia; Peptide Fragments; Receptors, Opioid	1986
Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists. Life sciences, 1987, Mar-30, Volume: 40, Issue:13 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Chemical Phenomena; Chemistry; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa	1987
Involvement of opioid receptors in phencyclidine-induced enhancement of brain histamine turnover in mice. Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:3 Topics: Analgesics, Opioid; Animals; Brain; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Haloperidol; Histamine; Histidine Decarboxylase; Ketamine; Male; Methylhistidines; Mice; Naloxone; Pargyline; Phenazocine; Phencyclidine; Receptors, Opioid	1987
Purification of a kappa-opioid receptor subtype from frog brain. Neuropeptides, 1987, Volume: 10, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain Chemistry; Chromatography, Gel; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Membranes; Molecular Weight; Naloxone; Peptide Fragments; Pyrrolidines; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Solubility	1987
Opioid receptors of bovine posterior pituitary neurosecretosomes are exclusively kappa. NIDA research monograph, 1986, Volume: 75 Topics: Analgesics, Opioid; Animals; Cattle; Cyclazocine; Cytoplasmic Granules; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Kinetics; Morphinans; Pituitary Gland, Posterior; Receptors, Opioid; Receptors, Opioid, kappa	1986
Characterization of opioid binding sites in murine neuroblastoma. Brain research, 1988, May-24, Volume: 449, Issue:1-2 Topics: Analgesics, Opioid; Animals; Binding, Competitive; Cell Line; Clone Cells; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Kinetics; Ligands; Mice; Neuroblastoma; Receptors, Opioid	1988
Differential ontogeny of multiple opioid receptors (mu, delta, and kappa). The Journal of neuroscience : the official journal of the Society for Neuroscience, 1985, Volume: 5, Issue:3 Topics: Animals; Animals, Newborn; Brain; Computers; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tritium	1985
TENA, a selective kappa opioid receptor antagonist. Life sciences, 1985, Feb-25, Volume: 36, Issue:8 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Azocines; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens	1985
Opiate receptor binding profile in the rabbit cerebellum and brain membranes. Biochemical pharmacology, 1985, Apr-01, Volume: 34, Issue:7 Topics: Animals; beta-Endorphin; Binding Sites; Binding, Competitive; Brain; Cerebellum; Cold Temperature; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Rabbits; Receptors, Opioid; Sodium; Tritium	1985
Differentiating aspects of opioid receptor binding by [3H](-) (1R,5R,9R,2''S)-5,9-dimethyl-2-tetrahydrofurfuryl-2'-hydroxy-6,7- benzomorphan hydrochloride ([3H]Mr 2034), a drug preferentially acting on kappa-receptors. Arzneimittel-Forschung, 1985, Volume: 35, Issue:1A Topics: Animals; Benzomorphans; Binding, Competitive; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Morphinans; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1985
Detection and characterization of four binding sites for opioids in the mouse brain. Acta pharmacologica et toxicologica, 1985, Volume: 56, Issue:2 Topics: Animals; Binding Sites; Brain Chemistry; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Models, Biological; Naloxone; Receptors, Opioid; Software; Tritium	1985
Opioid binding to rat and guinea-pig neural membranes in the presence of physiological cations at 37 degrees C. The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:3 Topics: Animals; Brain; Cations; Cyclazocine; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guanosine Triphosphate; Guinea Pigs; In Vitro Techniques; Male; Narcotics; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Temperature; Tritium	1985
Behavioural effects in rats of unilateral and bilateral injections of opiate receptor agonists into the globus pallidus. Neuroscience, 1985, Volume: 15, Issue:1 Topics: Animals; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Globus Pallidus; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1985
Evidence for a kappa-opioid receptor on pituitary astrocytes: an autoradiographic study. Neuroscience letters, 1985, Apr-19, Volume: 55, Issue:3 Topics: Animals; Astrocytes; Autoradiography; Binding Sites; Binding, Competitive; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Pituitary Gland; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1985
Autoradiographic localization of kappa opiate receptors in CNS taste and feeding areas. Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5 Topics: Animals; Autoradiography; Binding, Competitive; Brain; Corpus Striatum; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Feeding Behavior; Limbic System; Male; Morphine; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Taste	1985
Interaction of opiates with opioid binding sites in the bovine adrenal medulla: II. Interaction with kappa sites. Journal of neurochemistry, 1985, Volume: 45, Issue:3 Topics: Adrenal Medulla; Animals; Benzomorphans; Binding Sites; Calcium; Cattle; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Ethylketocyclazocine; Ethylmaleimide; Etorphine; Guinea Pigs; Kinetics; Lithium; Manganese; Narcotics; Oligopeptides; Phospholipases A; Potassium; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Stereoisomerism	1985
Interactions of codeine-7,8-oxide (codeine-epoxide), as a new metabolite of codeine, with multiple opiate receptors. General pharmacology, 1985, Volume: 16, Issue:4 Topics: Animals; Brain; Cell Membrane; Codeine; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guanosine Triphosphate; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride	1985
A monoclonal antibody capable of modulating opioid binding to rat neural membranes. The Journal of biological chemistry, 1985, Dec-15, Volume: 260, Issue:29 Topics: Animals; Antibodies, Monoclonal; Cell Line; Cyclazocine; Dihydromorphine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Flunitrazepam; Immunoglobulin M; Kinetics; Male; Mice; Mice, Inbred BALB C; Molecular Weight; Naloxone; Narcotics; Nerve Tissue; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Opioid	1985
A radiolabeled-ligand-binding technique for the characterization of opioid receptors in the intact mouse vas deferens. Analytical biochemistry, 1985, Volume: 150, Issue:1 Topics: Animals; Binding, Competitive; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Male; Mice; Morphine; Naltrexone; Radioligand Assay; Receptors, Opioid; Vas Deferens	1985
Kappa-opiate binding to rat brain and guinea pig cerebellum: sensitivity towards ions and nucleotides. Neuroscience letters, 1986, Feb-14, Volume: 64, Issue:1 Topics: Animals; Brain; Cerebellum; Cyclazocine; Electrolytes; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guanine Nucleotides; Guinea Pigs; Rats; Receptors, Opioid; Receptors, Opioid, kappa	1986
Subclass specificity of anti-idiotypic anti-opiate receptor antibodies in rat brain, guinea pig cerebellum, & neuroblastoma x glioma (NG 108-15). Life sciences, 1986, May-12, Volume: 38, Issue:19 Topics: Animals; Antibodies, Anti-Idiotypic; Binding, Competitive; Cell Line; Cerebellum; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Morphine; Neurilemma; Neurons; Rats; Receptors, Opioid	1986
Endogenous ligands for sigma opioid receptors in the brain ("sigmaphin"): evidence from binding assays. Life sciences, 1986, Jun-16, Volume: 38, Issue:24 Topics: Animals; Binding, Competitive; Brain; Chromatography, Gel; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Naloxone; Phenazocine; Phencyclidine; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Phencyclidine; Receptors, sigma	1986
Traumatic injury alters opiate receptor binding in rat spinal cord. Annals of neurology, 1986, Volume: 19, Issue:5 Topics: Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord; Spinal Cord Injuries	1986
Sodium regulation of agonist binding at opioid receptors. I. Effects of sodium replacement on binding at mu- and delta-type receptors in 7315c and NG108-15 cells and cell membranes. Molecular pharmacology, 1986, Volume: 30, Issue:2 Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Glioma; Guinea Pigs; Monensin; Naloxone; Neuroblastoma; Pituitary Neoplasms; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Sodium	1986
Sodium regulation of agonist binding at opioid receptors. II. Effects of sodium replacement on opioid binding in guinea pig cortical membranes. Molecular pharmacology, 1986, Volume: 30, Issue:2 Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Guinea Pigs; Male; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium	1986
Opioid ligand binding sites in the spinal cord of the guinea-pig. Neuropharmacology, 1986, Volume: 25, Issue:5 Topics: Animals; Binding, Competitive; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1986
Reversible and irreversible binding of beta-funaltrexamine to mu, delta and kappa opioid receptors in guinea pig brain membranes. The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2 Topics: Animals; Brain; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Ethylmaleimide; Guinea Pigs; Kinetics; Male; Membranes; Naloxone; Naltrexone; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium Chloride	1986
[Differences in opioid binding in the left and right visual cortex of the turtle]. Doklady Akademii nauk SSSR, 1986, Volume: 291, Issue:2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Functional Laterality; Receptors, Opioid; Turtles; Visual Cortex	1986
Nonequilibrium opioid antagonist activity of 6,14-dideoxynaltrexone derivatives. Journal of medicinal chemistry, 1987, Volume: 30, Issue:6 Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Mice; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Structure-Activity Relationship	1987
Opioid receptor binding in rat spinal cord. Neurochemical research, 1987, Volume: 12, Issue:3 Topics: Animals; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Ligands; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord	1987
Synthesis and evaluation of melphalan-containing N,N-dialkylenkephalin analogues as irreversible antagonists of the delta opioid receptor. Journal of medicinal chemistry, 1987, Volume: 30, Issue:9 Topics: Alkylation; Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Melphalan; Mice; Morphine; Muscle, Smooth; Receptors, Opioid; Receptors, Opioid, delta; Structure-Activity Relationship	1987
Effects of opioid agonist drugs on the in vitro release of 3H-GABA, 3H-dopamine and 3H-5HT from slices of rat globus pallidus. Biochemical pharmacology, 1987, May-15, Volume: 36, Issue:10 Topics: Animals; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dopamine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; gamma-Aminobutyric Acid; Globus Pallidus; Potassium Chloride; Rats; Rats, Inbred Strains; Serotonin	1987
Comparative effects of opiate agonists on proximal and distal colonic motility in dogs. European journal of pharmacology, 1985, Apr-16, Volume: 110, Issue:3 Topics: Animals; Colon; Cyclazocine; Dogs; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Fentanyl; Gastrointestinal Motility; Injections, Intravenous; Injections, Spinal; Narcotics; Time Factors	1985
Opioid control of the ruminant stomach motility: functional importance of mu, kappa and delta receptors. Life sciences, 1984, Oct-22, Volume: 35, Issue:17 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Gastrointestinal Motility; Morphine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sheep; Stomach	1984
[3H]Ethylketocyclazocine binding to mouse brain membranes: evidence for a kappa opioid receptor type. The Journal of pharmacology and experimental therapeutics, 1984, Volume: 231, Issue:1 Topics: Animals; Brain; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1984
Altered opiate receptor binding in synaptosomes: implication of phosphorylation. Proceedings of the Western Pharmacology Society, 1984, Volume: 27 Topics: Animals; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Phosphorylation; Receptors, Opioid; Synaptosomes	1984
Comparative antagonism by naltrexone and naloxone of mu, kappa, and delta agonists. European journal of pharmacology, 1984, Sep-03, Volume: 104, Issue:1-2 Topics: Animals; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle, Smooth; Naloxone; Naltrexone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens	1984
Distinct high-affinity binding sites for benzomorphan drugs and enkephalin in a neuroblastoma--brain hybrid cell line. Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:7 Topics: Analgesics, Opioid; Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cell Line; Cyclazocine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hybrid Cells; Kinetics; Morphinans; Neuroblastoma; Phenazocine; Rats; Receptors, Opioid	1981
Stereospecific inhibition of oxotremorine-induced antinociception by (+)-isomers of opioid antagonists: comparison with opioid receptor agonists. The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:8 Topics: Animals; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Mice; Morphine; Narcotic Antagonists; Nociceptors; Oxotremorine; Receptors, Opioid; Stereoisomerism	1982
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord. Brain research, 1982, Sep-09, Volume: 247, Issue:1 Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord	1982
Kappa opiate receptors localized by autoradiography to deep layers of cerebral cortex: relation to sedative effects. Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:18 Topics: Analgesics; Analgesics, Opioid; Animals; Autoradiography; Benzomorphans; Brain Stem; Cerebral Cortex; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Morphine; Organ Specificity; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1982
Comparison of analgesic potencies of mu, delta and kappa agonists locally applied to various CNS regions relevant to analgesia in rats. Life sciences, 1983, Volume: 33 Suppl 1 Topics: Analgesics, Opioid; Animals; Brain Stem; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	1983
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes. Journal of receptor research, 1984, Volume: 4, Issue:1-6 Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid	1984
Involvement of mu-receptors in the opioid-induced generation of bursting discharges in hippocampal pyramidal cells. Regulatory peptides, 1981, Volume: 2, Issue:2 Topics: Animals; Benzomorphans; Culture Techniques; Cyclazocine; D-Ala(2),MePhe(4),Met(0)-ol-enkephalin; Dose-Response Relationship, Drug; Electrophysiology; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Membrane Potentials; Morphinans; Rats; Receptors, Opioid; Receptors, Opioid, mu	1981
Characterization of the kappa-subtype of the opiate receptor in the guinea-pig brain. British journal of pharmacology, 1981, Volume: 73, Issue:4 Topics: Animals; Benzomorphans; Binding Sites; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Naloxone; Naltrexone; Narcotics; Phenoxybenzamine; Receptors, Opioid	1981
Strain differences in opiate receptors in mouse brain. European journal of pharmacology, 1981, Sep-24, Volume: 74, Issue:4 Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Naloxone; Receptors, Opioid; Species Specificity	1981
D-Ala2,D-Leu5-enkephalin generalizes to a discriminative stimulus produced by fentanyl but not ethylketocyclazocine. Pharmacology, biochemistry, and behavior, 1982, Volume: 16, Issue:2 Topics: Animals; Cyclazocine; Discrimination, Psychological; Endorphins; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Fentanyl; Generalization, Stimulus; Male; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid	1982
Opiate and opioid peptide binding in rat goldfish: further evidence for opiate receptor heterogeneity. Brain research, 1982, Sep-23, Volume: 248, Issue:1 Topics: Animals; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Goldfish; Male; Naloxone; Narcotics; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma	1982
Opiate receptor-mediated inhibition of catecholamine release in primary cultures of bovine adrenal chromaffin cells. Journal of neurochemistry, 1982, Volume: 39, Issue:6 Topics: Acetylcholine; Adrenal Medulla; Animals; beta-Endorphin; Catecholamines; Cattle; Cells, Cultured; Chromaffin Granules; Chromaffin System; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Phenazocine; Receptors, Opioid	1982
Relative involvement of receptor subtypes in opioid-induced inhibition of gastrointestinal transit in mice. The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2 Topics: Animals; Charcoal; Cyclazocine; Drug Interactions; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Gastrointestinal Motility; Male; Mice; Morphine; Nalorphine; Naltrexone; Receptors, Opioid	1983
Evidence for multiple "Kappa" binding sites by use of opioid peptides in the guinea-pig lumbo-sacral spinal cord. Neuropeptides, 1982, Volume: 3, Issue:1 Topics: Animals; Binding Sites; Cyclazocine; Dihydromorphine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Radioligand Assay; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord	1982
The binding to rat brain homogenates of Mr2034, a universal opiate. Life sciences, 1983, Sep-05, Volume: 33, Issue:10 Topics: Animals; Benzomorphans; Brain; Cyclazocine; Dihydromorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Morphinans; Naloxone; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid	1983
Opiate binding sites in bovine adrenal medulla. Journal of receptor research, 1983, Volume: 3, Issue:4 Topics: Adrenal Medulla; Animals; Binding Sites; Brain; Brain Chemistry; Cattle; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid	1983
Comparison of mu, delta, and kappa opiate binding sites in rat brain and spinal cord. Life sciences, 1984, Jan-16, Volume: 34, Issue:3 Topics: Animals; Binding Sites; Brain; Cell Membrane; Cyclazocine; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord	1984
[3H]ethylketocyclazocine binding to NCB-20 hybrid neurotumor cells. Molecular pharmacology, 1983, Volume: 23, Issue:2 Topics: Animals; Binding, Competitive; Brain; Cricetinae; Cricetulus; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Hybrid Cells; Kinetics; Neuroblastoma; Trypsin	1983
A method to estimate the potency of the mu-component of an opioid having mixed mu-, and kappa- and/or delta-agonist activities. Psychopharmacology, 1995, Volume: 117, Issue:2 Topics: Animals; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Female; Male; Mice; Mice, Inbred ICR; Morphine; Naloxone; Postural Balance; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reflex	1995
Identification and characterization of opioid-binding sites present in the Ishikawa human endometrial adenocarcinoma cell line. The Journal of clinical endocrinology and metabolism, 1995, Volume: 80, Issue:2 Topics: Acids; Adenocarcinoma; Binding Sites; Endometrial Neoplasms; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; Humans; Narcotics; Tumor Cells, Cultured	1995
Opiate receptor agonists regulate phosphorylation of synapsin I in cocultures of rat spinal cord and dorsal root ganglion. Proceedings of the National Academy of Sciences of the United States of America, 1993, May-01, Volume: 90, Issue:9 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Cell Communication; Cells, Cultured; Colforsin; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Ganglia, Spinal; Isoproterenol; Kinetics; Male; Morphine; Naloxone; Neurons; Phosphates; Phosphoproteins; Phosphorylation; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid; Serotonin; Spinal Cord; Synapsins; Synaptosomes	1993
The antiproliferative effect of opioid receptor agonists on the T47D human breast cancer cell line, is partially mediated through opioid receptors. European journal of pharmacology, 1996, Jan-25, Volume: 296, Issue:2 Topics: Adenocarcinoma; Amino Acid Sequence; Binding Sites; Breast Neoplasms; Cell Division; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Humans; Molecular Sequence Data; Morphine; Narcotic Antagonists; Opioid Peptides; Receptors, Opioid; Tumor Cells, Cultured	1996
Identification of a novel opioid peptide (Tyr-Val-Pro-Phe-Pro) derived from human alpha S1 casein (alpha S1-casomorphin, and alpha S1-casomorphin amide). The Biochemical journal, 1996, Nov-01, Volume: 319 ( Pt 3) Topics: Amino Acid Sequence; Binding, Competitive; Breast Neoplasms; Caseins; Cell Division; Cell Line; Diprenorphine; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; Humans; Kinetics; Peptide Fragments; Receptors, Opioid, kappa	1996
Pyrrolomorphinans as delta opioid receptor antagonists. The role of steric hindrance in conferring selectivity. Journal of medicinal chemistry, 1997, Jun-20, Volume: 40, Issue:13 Topics: Animals; Electric Stimulation; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Models, Chemical; Morphinans; Morphine; Muscle, Smooth; Pyrroles; Receptors, Opioid, delta; Stereoisomerism	1997
Affinity labelling of frog brain opioid receptors by dynorphin(1-10) chloromethyl ketone. Neuropeptides, 1997, Volume: 31, Issue:1 Topics: Affinity Labels; Amino Acid Chloromethyl Ketones; Analgesics, Opioid; Animals; Binding, Competitive; Brain Chemistry; Dihydromorphine; Dynorphins; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Membrane Proteins; Peptide Fragments; Radioligand Assay; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Tritium	1997
NTI4F: a non-peptide fluorescent probe selective for functional delta opioid receptors. Neuroscience letters, 1998, Jun-19, Volume: 249, Issue:2-3 Topics: Animals; Bridged-Ring Compounds; Cell Line; Dogs; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Fluorescent Dyes; Imides; Microscopy, Confocal; Microscopy, Fluorescence; Morphine; Naltrexone; Receptors, Opioid, delta; Transfection	1998
Kappa1-opioid binding sites are the dominant opioid binding sites in surgical specimens of human pheochromocytomas and in a human pheochromocytoma (KAT45) cell line. European journal of pharmacology, 1999, Jan-08, Volume: 364, Issue:2-3 Topics: Analgesics, Opioid; Binding Sites; Binding, Competitive; Catecholamines; Cell Membrane; Diprenorphine; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Epinephrine; Ethylketocyclazocine; Humans; Narcotic Antagonists; Norepinephrine; Opioid Peptides; Pheochromocytoma; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tritium; Tumor Cells, Cultured	1999
The inhibitory effect of opioids on HepG2 cells is mediated via interaction with somatostatin receptors. European journal of pharmacology, 2007, Jan-19, Volume: 555, Issue:1 Topics: Analgesics, Opioid; Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Humans; Narcotic Antagonists; Octreotide; Receptors, Opioid; Receptors, Somatostatin; RNA, Messenger; Somatostatin	2007
Differential effects of opioid agonists on G protein expression in CHO cells expressing cloned human opioid receptors. Brain research bulletin, 2008, Sep-05, Volume: 77, Issue:1 Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzamides; Blotting, Western; CHO Cells; Cricetinae; Cricetulus; Diterpenes, Clerodane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Female; Furans; Gene Expression; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Morphine; Oligopeptides; Piperazines; Pyrones; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu	2008