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ethylketocyclazocine and dynorphins

ethylketocyclazocine has been researched along with dynorphins in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-199058 (84.06)18.7374
1990's11 (15.94)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gannon, RL; Terrian, DM1
Jhamandas, K; Lapierre, C; Lemaire, S; Martinka, GP; Sabourin, L1
Kinouchi, K; Pasternak, GW1
Shea-Donohue, T; Touzeau, PL1
Hoss, W; Periyasamy, S1
Hirobe, M; Konno, F; Takayanagi, I; Toru, T1
Garzon, J; Landahl, HD; Lee, NM1
Su, TP1
Moises, HC; Walker, JM1
Way, EL; Yamasaki, Y1
Herz, A; Schiller, PW; Schulz, R; Shearman, GT1
Bicknell, RJ; Chapman, C; Leng, G1
Bryant, HU; Lowy, MT; Malven, PV; Steele, TD; Yim, GK1
Cooper, SJ; Jackson, A; Kirkham, TC1
Cho, N; Hirobe, M; Koike, K; Konno, F; Okumura, K; Takayanagi, I1
Illes, P; Ramme, D1
Geppert, M; Illes, P; Jackisch, R1
Buder, M; Fuder, H; Riers, HD; Rothacher, G1
Brenner, AS; Geppert, M; Illes, P; Jackisch, R1
Kirby, GC; McQueen, DS1
Baskin, DS; Hosobuchi, Y; Kuroda, H; Lee, NM; Loh, HH; Matsui, T1
Burks, TF; Deupree, D; Hruby, V; Hsiao, S; Mosberg, HI; Porreca, F; Spencer, RL1
Cho, N; Hirobe, M; Kobayashi, C; Konno, F; Morimoto, R; Takayanagi, I1
Inoki, R; Kudo, T; Ohkubo, T; Shibata, M; Takahashi, H1
Lipkowski, AW; Portoghese, PS; Takemori, AE1
Schmauss, C1
Dickenson, AH; Knox, RJ1
Bhargava, HN; Das, S1
Benyhe, S; Borsodi, A; Hepp, J; Khan, A; Medzihradszky, K; Simon, J; Szücs, M; Wollemann, M1
Inoki, R; Maeda, S; Nakamae, J2
Belisle, S; Bellabarba, D; Gallo-Payet, N; Lehoux, JG; Lemaire, S; Petit, A1
Bryant, HU; Malven, PV; Steele, TD; Yim, GK1
Alvinerie, M; Bueno, L; Gue, M; Honde, C; Junien, JL; Pascaud, X1
Borsodi, A; Lajtha, A; Zawilska, J1
Candeletti, S; Cavicchini, E; Ferri, S; Romualdi, P; Spampinato, S; Speroni, E1
Berzetei, IP; Duckles, SP; Fong, A; Yamamura, HI1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Yoshimura, K3
Chavkin, C; Goldstein, A; James, IF1
Miller, RJ1
Herz, A; Pfeiffer, A1
Piercey, MF; Schroeder, LA; Varner, K1
Tung, AS; Yaksh, TL1
Huidobro-Toro, JP; Way, EL; Yoshimura, K1
Herz, A1
Lee, NM1
Kamerling, SG; Martin, WR; Wettstein, JG; Wu, KM1
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Zhu, YX1
Cros, J; Pontonnier, G; Porthe, G; Tafani, M; Valette, A1
Garzón, J; Gerhart, J; Lee, NM; Loh, HH; Sánchez-Blázquez, P1
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE1
Pairet, M; Ruckebusch, Y1
Rezvani, A; Way, EL1
Gosnell, BA; Grace, M; Kneip, J; Levine, AS; Morley, JE1
Han, JS; Xie, GX2
Burkard, WP; Flück, N; Müller, PM1
Fujino, M; Negishi, K; Oka, T; Sawa, A; Suda, M; Wakimasu, M1
Laurent, S; Schmitt, H2
Goldstein, A; Han, JS; Xie, GX1
Barnard, EA; Benyhe, S; Borsodi, A; Simon, J; Wollemann, M1
Berzetei-Gurske, IP; Brandt, SR; Polgar, WE; Toll, L; Webster, JL1
Hogenboom, F; Mulder, AH; Schoffelmeer, AN1
Benyhe, S; Borsodi, A; Hepp, J; Ketevan, A; Medzihradszky, K; Simon, J1
Butelman, ER; Kreek, MJ; Vivian, JA; Woods, JH; Yu, J1
Akil, H; Goldstein, A; Mansour, A; Meng, F; Thompson, RC; Watson, SJ; Xie, GX1

Reviews

3 review(s) available for ethylketocyclazocine and dynorphins

ArticleYear
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:5

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response

1985
Multiple opiate receptors for multiple opioid peptides.
    Medical biology, 1982, Volume: 60, Issue:1

    Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission

1982
Multiple opiate receptors and their functional significance.
    Journal of neural transmission. Supplementum, 1983, Volume: 18

    Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Morphine; Receptors, Opioid; Tissue Distribution

1983

Other Studies

66 other study(ies) available for ethylketocyclazocine and dynorphins

ArticleYear
Kappa opioid agonists inhibit transmitter release from guinea pig hippocampal mossy fiber synaptosomes.
    Neurochemical research, 1992, Volume: 17, Issue:8

    Topics: Animals; Azocines; Calcium; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Potassium; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptosomes

1992
Dynorphin A-(1-13)-Tyr14-Leu15-Phe16-Asn17-Gly18-Pro19 : a potent and selective kappa opioid peptide.
    European journal of pharmacology, 1991, Apr-17, Volume: 196, Issue:2

    Topics: Amino Acid Sequence; Animals; Dynorphins; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Mice; Molecular Sequence Data; Muscle Contraction; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1991
Evidence for kappa 1 opioid receptor multiplicity in the guinea pig cerebellum.
    European journal of pharmacology, 1991, Jun-19, Volume: 207, Issue:2

    Topics: Animals; Benzeneacetamides; Binding Sites; Binding, Competitive; Cerebellum; Dynorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Tritium

1991
Kappa agonists inhibit gastric emptying but not acid secretion in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Antihypertensive Agents; Cyclazocine; Dynorphins; Ethylketocyclazocine; Gastric Acid; Gastric Emptying; Macaca mulatta; Male; Narcotics; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Sodium

1990
Kappa opioid receptors stimulate phosphoinositide turnover in rat brain.
    Life sciences, 1990, Volume: 47, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Dynorphins; Enkephalins; Ethylketocyclazocine; Male; Phosphatidylinositols; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1990
Kappa-receptor mechanisms in synaptosomal Ca uptake.
    General pharmacology, 1989, Volume: 20, Issue:2

    Topics: Animals; Calcium; Calcium Radioisotopes; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Morphine; Nalorphine; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Synaptosomes

1989
Computer analysis of the effect of beta-endorphin and dynorphin and related compounds on opioid binding to mouse brain membrane.
    Computers in biology and medicine, 1989, Volume: 19, Issue:3

    Topics: Animals; beta-Endorphin; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Mice; Models, Neurological; Receptors, Opioid

1989
Further demonstration of kappa opioid binding sites in the brain: evidence for heterogeneity.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Binding Sites; Brain; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Levallorphan; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism

1985
Electrophysiological effects of dynorphin peptides on hippocampal pyramidal cells in rat.
    European journal of pharmacology, 1985, Jan-15, Volume: 108, Issue:1

    Topics: Animals; Cyclazocine; Dynorphins; Electrophysiology; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; gamma-Aminobutyric Acid; Hippocampus; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid

1985
Inhibition of Ca++-ATPase of rat erythrocyte membranes by k-opioid agonists.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Animals; beta-Endorphin; Calcium-Transporting ATPases; Cyclazocine; Dynorphins; Endorphins; Erythrocyte Membrane; Ethylketocyclazocine; Levorphanol; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
Generalization tests with intraventricularly applied pro-enkephalin B-derived peptides in rats trained to discriminate the opioid kappa receptor agonist ethylketocyclazocine.
    Psychopharmacology, 1985, Volume: 85, Issue:4

    Topics: Animals; beta-Endorphin; Cyclazocine; Discrimination Learning; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Generalization, Stimulus; Injections, Intraventricular; Male; Protein Precursors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
Effects of opioid agonists and antagonists on oxytocin and vasopressin release in vitro.
    Neuroendocrinology, 1985, Volume: 41, Issue:2

    Topics: Animals; Arginine Vasopressin; Benzomorphans; beta-Endorphin; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Naloxone; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains

1985
Effects of 2% sodium chloride imbibition on various opiate related hyperphagic conditions.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 23, Issue:3

    Topics: Animals; Cyclazocine; Deoxyglucose; Dynorphins; Ethylketocyclazocine; Feeding Behavior; Insulin; Male; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride; Time Factors

1985
Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor.
    General pharmacology, 1985, Volume: 16, Issue:6

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Peptide Fragments; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Synaptosomes; Vas Deferens

1985
Differential effect of stimulation strength in mouse vas deferens on inhibition of neuroeffector transmission by receptor type selective opioids.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cyclazocine; Dynorphins; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Morphine Derivatives; Muscle, Smooth; Neuromuscular Junction; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Synaptic Transmission

1986
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid

1986
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1986
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 332, Issue:2

    Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses

1986
Characterization of opioid receptors in the cat carotid body involved in chemosensory depression in vivo.
    British journal of pharmacology, 1986, Volume: 88, Issue:4

    Topics: Animals; Carotid Body; Cats; Chemoreceptor Cells; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hypercapnia; Hypoxia; Peptide Fragments; Receptors, Opioid

1986
Effects of dynorphin1-13 on opiate binding and dopamine and GABA uptake in stroked cat brain.
    Brain research, 1986, Jul-30, Volume: 379, Issue:1

    Topics: Animals; Brain; Brain Ischemia; Cats; Cyclazocine; Disease Models, Animal; Dopamine; Dynorphins; Ethylketocyclazocine; gamma-Aminobutyric Acid; Kinetics; Male; Peptide Fragments; Receptors, Opioid

1986
Centrally-administered opioid selective agonists inhibit drinking in the rat.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Drinking Behavior; Dynorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptide Fragments; Pyrrolidines; Rats; Receptors, Opioid

1986
Pharmacological effects of nalorphine and nalorphine-7,8-oxide (nalorphine-epoxide): interaction of the intrinsic activity, affinity and pharmacological responses.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 282, Issue:2

    Topics: Analgesics; Animals; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Nalorphine; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid

1986
[Peripheral analgesic actions of opioid peptides and morphine analogues].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1986, Volume: 88, Issue:2

    Topics: Analgesics, Opioid; Animals; Cyclazocine; Dynorphins; Enkephalin, Methionine; Ethylketocyclazocine; Levallorphan; Lidocaine; Male; Mice; Morphine; Naloxone; Pain; Peptide Fragments

1986
Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists.
    Life sciences, 1987, Mar-30, Volume: 40, Issue:13

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Chemical Phenomena; Chemistry; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa

1987
Spinal kappa-opioid receptor-mediated antinociception is stimulus-specific.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Dynorphins; Ethylketocyclazocine; Injections, Spinal; Male; Morphine; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord

1987
Effects of selective and non-selective kappa-opioid receptor agonists on cutaneous C-fibre-evoked responses of rat dorsal horn neurones.
    Brain research, 1987, Jul-07, Volume: 415, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Action Potentials; Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Nerve Fibers; Pain; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Skin; Spinal Cord; Time Factors

1987
Inhibition of [3H][3-MeHis2]thyrotropin releasing hormone recognition sites in the rat brain by tifluadom, a kappa opiate receptor agonist.
    Neuropharmacology, 1987, Volume: 26, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analysis of Variance; Animals; Benzodiazepines; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Kinetics; Male; Peptide Fragments; Pyrrolidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Thyrotropin-Releasing Hormone; Thyrotropin-Releasing Hormone

1987
Purification of a kappa-opioid receptor subtype from frog brain.
    Neuropeptides, 1987, Volume: 10, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain Chemistry; Chromatography, Gel; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Membranes; Molecular Weight; Naloxone; Peptide Fragments; Pyrrolidines; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Solubility

1987
Positive inotropic action of kappa opiate agonists, ethylketocyclazocine and dynorphin-A(1-13), in isolated rat atrium.
    Japanese journal of pharmacology, 1987, Volume: 45, Issue:1

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Ethylketocyclazocine; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Peptide Fragments; Rats; Rats, Inbred Strains; Stimulation, Chemical

1987
Functional opioid receptor sites in human placentas.
    The Journal of clinical endocrinology and metabolism, 1988, Volume: 66, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gonadotropin-Releasing Hormone; Humans; Kinetics; Placenta; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thyrotropin-Releasing Hormone

1988
Inhibition of cardiac Na+, K+-ATPase activity by dynorphin-A and ethylketocyclazocine.
    Life sciences, 1988, Volume: 42, Issue:4

    Topics: Adenosine Triphosphate; Animals; Cyclazocine; Dynorphins; Enzyme Activation; Ethylketocyclazocine; Male; Myocardium; Naloxone; Peptide Fragments; Potassium; Rats; Rats, Inbred Strains; Sodium; Sodium-Potassium-Exchanging ATPase

1988
Nocturnal depletion of hypothalamic dynorphin in anorexic Walker-256 tumor-bearing rats.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 29, Issue:3

    Topics: Animals; Anorexia; Carcinoma 256, Walker; Circadian Rhythm; Cyclazocine; Dynorphins; Eating; Ethylketocyclazocine; Feeding and Eating Disorders; Hypothalamus; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1988
CNS blockade of acoustic stress-induced gastric motor inhibition by kappa-opiate agonists in dogs.
    The American journal of physiology, 1988, Volume: 254, Issue:6 Pt 1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acoustic Stimulation; Adrenocorticotropic Hormone; Analgesics; Animals; Cyclazocine; Dogs; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gastrointestinal Motility; Hydrocortisone; Pyrrolidines; Stress, Physiological

1988
Selective protection of benzomorphan binding sites against inactivation by N-ethylmaleimide. Evidence for kappa-opioid receptors in frog brain.
    Journal of neurochemistry, 1988, Volume: 51, Issue:3

    Topics: Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Ethylmaleimide; Morphinans; Peptide Fragments; Rana esculenta; Receptors, Opioid; Sodium Chloride

1988
Investigations on dynorphin structurally-related opioid peptides. I. Impact on nociceptive transmission. II. Regulation of pituitary content.
    Annali dell'Istituto superiore di sanita, 1988, Volume: 24, Issue:3

    Topics: Animals; Benzomorphans; Cyclazocine; Dynorphins; Estradiol; Ethylketocyclazocine; Female; Hypothalamo-Hypophyseal System; Male; Ovary; Pain; Pain Measurement; Rats; Rats, Inbred Strains; Structure-Activity Relationship

1988
Characterization of kappa opioid receptors in the rabbit ear artery.
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: Animals; Benzeneacetamides; Benzomorphans; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle, Smooth, Vascular; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1988
Dynorphin interaction at the kappa-opiate site.
    European journal of pharmacology, 1981, Jun-19, Volume: 72, Issue:2-3

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Receptors, Opioid; Receptors, Opioid, kappa

1981
Dynorphin is a specific endogenous ligand of the kappa opioid receptor.
    Science (New York, N.Y.), 1982, Jan-22, Volume: 215, Issue:4531

    Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Ligands; Morphine Derivatives; Myenteric Plexus; Naloxone; Peptide Fragments; Receptors, Opioid

1982
Kappa opioid properties of dynorphin and its peptide fragments on the guinea-pig Ileum.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 222, Issue:1

    Topics: Animals; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Receptors, Opioid; Receptors, Opioid, kappa

1982
Discrimination of three opiate receptor binding sites with the use of a computerized curve-fitting technique.
    Molecular pharmacology, 1982, Volume: 21, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Computers; Cyclazocine; Dihydromorphine; Diprenorphine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Phenazocine; Rats; Receptors, Opioid

1982
Analgesic activity of intraspinally administered dynorphin and ethylketocyclazocine.
    European journal of pharmacology, 1982, May-21, Volume: 80, Issue:2-3

    Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Injections; Male; Mice; Spinal Cord

1982
Activation of K-opiate sites by dynorphin in the myenteric plexus.
    Advances in biochemical psychopharmacology, 1982, Volume: 33

    Topics: Animals; Cyclazocine; Drug Tolerance; Dynorphins; Electric Stimulation; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa

1982
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
    Brain research, 1982, Sep-09, Volume: 247, Issue:1

    Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord

1982
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists

1982
Is dynorphin a k ligand?
    Proceedings of the Western Pharmacology Society, 1983, Volume: 26

    Topics: Animals; Brain; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Receptors, Opioid; Receptors, Opioid, kappa

1983
Possible medullary kappa hyperalgesic mechanism. I. A new potential role for endogenous opioid peptides in pain perception.
    Life sciences, 1983, Oct-31, Volume: 33, Issue:18

    Topics: Animals; Cyclazocine; Dogs; Dynorphins; Endorphins; Ethylketocyclazocine; Medulla Oblongata; Naloxone; Pain; Receptors, Opioid; Reflex

1983
Dynorphin inhibition of the neurotensin contractile activity on the myenteric plexus.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 228, Issue:2

    Topics: Animals; Atropine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Nerve Tissue Proteins; Neurotensin; Peptide Fragments; Receptors, Opioid; Tetrodotoxin

1984
Placental kappa binding site : interaction with dynorphin and its possible implication in hCG secretion.
    Life sciences, 1983, Volume: 33 Suppl 1

    Topics: Analgesics, Opioid; Chorionic Gonadotropin; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Female; Humans; Peptide Fragments; Placenta; Pregnancy; Receptors, Opioid; Receptors, Opioid, kappa

1983
Dynorphin A: inhibitory effect on other opiate ligand bindings in the mouse brain.
    Biochemical pharmacology, 1984, Aug-15, Volume: 33, Issue:16

    Topics: Animals; Brain; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Naloxone; Narcotics; Peptide Fragments; Receptors, Opioid; Sodium Chloride

1984
Feeding systems in Chinese hamsters.
    The American journal of physiology, 1984, Volume: 247, Issue:3 Pt 2

    Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation

1984
Opioid receptor agonists in the rabbit colon: comparison of in vivo and in vitro studies.
    Life sciences, 1984, Oct-15, Volume: 35, Issue:16

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Colon; Cyclazocine; Dynorphins; Electric Conductivity; Enkephalins; Ethylketocyclazocine; Fentanyl; Male; Morphine; Naloxone; Narcotics; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1984
Dynorphin-(1-13) restores the potency of morphine on the tolerant guinea pig ileum.
    European journal of pharmacology, 1984, Jul-20, Volume: 102, Issue:3-4

    Topics: Animals; beta-Endorphin; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments

1984
The effect of ovariectomy, estradiol and progesterone on opioid modulation of feeding.
    Physiology & behavior, 1984, Volume: 33, Issue:2

    Topics: Animals; Appetite Regulation; Brain; Castration; Cyclazocine; Dynorphins; Eating; Estradiol; Ethylketocyclazocine; Female; Naloxone; Progesterone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1984
[Dynorphin: analgesic effect via kappa receptors in the spinal cord of rats].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1984, Volume: 5, Issue:4

    Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Ethylketocyclazocine; Female; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord

1984
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid

1984
[Dynorphin: analgesic effect via kappa receptors in spinal cord of the spinal cords of rats].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1984, Volume: 5, Issue:4

    Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Ethylketocyclazocine; Female; Morphine; Naloxone; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sensory Thresholds; Spinal Cord

1984
Evidence that dynorphin-(1-13) acts as an agonist on opioid kappa-receptors.
    European journal of pharmacology, 1982, Jan-22, Volume: 77, Issue:2-3

    Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens

1982
Central cardiovascular effects of kappa agonists dynorphin-(1-13) and ethylketocyclazocine in the anaesthetized rat.
    European journal of pharmacology, 1983, Dec-09, Volume: 96, Issue:1-2

    Topics: Animals; beta-Endorphin; Blood Pressure; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Heart Rate; Male; Naloxone; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vagus Nerve

1983
Opposite central cardiovascular effects of various morphine-like drugs and opiate peptides in the rat.
    European heart journal, 1983, Volume: 4 Suppl G

    Topics: Animals; Blood Pressure; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Heart Rate; Male; Peptide Fragments; Rats; Rats, Inbred Strains

1983
Analgesia induced by intrathecal injection of dynorphin B in the rat.
    Life sciences, 1984, Apr-16, Volume: 34, Issue:16

    Topics: Analgesics; Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Female; Injections, Spinal; Morphine; Naloxone; Rats

1984
[3H]dynorphin1-8 binding sites in frog (Rana esculenta) brain membranes.
    Neuropeptides, 1994, Volume: 26, Issue:5

    Topics: Amino Acid Sequence; Animals; Brain; Cell Membrane; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Naloxone; Peptide Fragments; Rana esculenta; Receptors, Opioid; Sodium Chloride; Tritium

1994
Comparison of kappa 2-opioid receptors in guinea pig brain and guinea pig ileum membranes.
    European journal of pharmacology, 1993, Feb-09, Volume: 231, Issue:2

    Topics: Analgesics; Animals; Benzomorphans; Brain Chemistry; Dynorphins; Ethylketocyclazocine; Guanylyl Imidodiphosphate; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Ligands; Male; Membranes; Myenteric Plexus; Receptors, Opioid, kappa

1993
Kappa1- and kappa2-opioid receptors mediating presynaptic inhibition of dopamine and acetylcholine release in rat neostriatum.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: Acetylcholine; Animals; Benzeneacetamides; Dopamine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; N-Methylaspartate; Naloxone; Neostriatum; Neural Inhibition; Peptide Fragments; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1997
Affinity labelling of frog brain opioid receptors by dynorphin(1-10) chloromethyl ketone.
    Neuropeptides, 1997, Volume: 31, Issue:1

    Topics: Affinity Labels; Amino Acid Chloromethyl Ketones; Analgesics, Opioid; Animals; Binding, Competitive; Brain Chemistry; Dihydromorphine; Dynorphins; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Membrane Proteins; Peptide Fragments; Radioligand Assay; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Tritium

1997
Systemic effects of E-2078, a stabilized dynorphin A(1-8) analog, in rhesus monkeys.
    Psychopharmacology, 1999, Volume: 143, Issue:2

    Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Conditioning, Operant; Discrimination, Psychological; Diuresis; Dynorphins; Ethylketocyclazocine; Female; Food; Injections, Intramuscular; Injections, Subcutaneous; Macaca mulatta; Male; Pain Measurement; Peptide Fragments; Receptors, Opioid, kappa; Receptors, Opioid, mu

1999
Cloning and pharmacological characterization of a rat kappa opioid receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Nov-01, Volume: 90, Issue:21

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Analgesics; Animals; Benzeneacetamides; Cell Line; Cell Membrane; Cloning, Molecular; Corpus Striatum; Cyclic AMP; DNA Primers; DNA, Complementary; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Gene Library; In Situ Hybridization; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Molecular Sequence Data; Pyrrolidines; Rats; Receptors, Opioid, kappa; Restriction Mapping; RNA, Messenger; Transfection

1993