ethylketocyclazocine has been researched along with dynorphins in 69 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 58 (84.06) | 18.7374 |
1990's | 11 (15.94) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Gannon, RL; Terrian, DM | 1 |
Jhamandas, K; Lapierre, C; Lemaire, S; Martinka, GP; Sabourin, L | 1 |
Kinouchi, K; Pasternak, GW | 1 |
Shea-Donohue, T; Touzeau, PL | 1 |
Hoss, W; Periyasamy, S | 1 |
Hirobe, M; Konno, F; Takayanagi, I; Toru, T | 1 |
Garzon, J; Landahl, HD; Lee, NM | 1 |
Su, TP | 1 |
Moises, HC; Walker, JM | 1 |
Way, EL; Yamasaki, Y | 1 |
Herz, A; Schiller, PW; Schulz, R; Shearman, GT | 1 |
Bicknell, RJ; Chapman, C; Leng, G | 1 |
Bryant, HU; Lowy, MT; Malven, PV; Steele, TD; Yim, GK | 1 |
Cooper, SJ; Jackson, A; Kirkham, TC | 1 |
Cho, N; Hirobe, M; Koike, K; Konno, F; Okumura, K; Takayanagi, I | 1 |
Illes, P; Ramme, D | 1 |
Geppert, M; Illes, P; Jackisch, R | 1 |
Buder, M; Fuder, H; Riers, HD; Rothacher, G | 1 |
Brenner, AS; Geppert, M; Illes, P; Jackisch, R | 1 |
Kirby, GC; McQueen, DS | 1 |
Baskin, DS; Hosobuchi, Y; Kuroda, H; Lee, NM; Loh, HH; Matsui, T | 1 |
Burks, TF; Deupree, D; Hruby, V; Hsiao, S; Mosberg, HI; Porreca, F; Spencer, RL | 1 |
Cho, N; Hirobe, M; Kobayashi, C; Konno, F; Morimoto, R; Takayanagi, I | 1 |
Inoki, R; Kudo, T; Ohkubo, T; Shibata, M; Takahashi, H | 1 |
Lipkowski, AW; Portoghese, PS; Takemori, AE | 1 |
Schmauss, C | 1 |
Dickenson, AH; Knox, RJ | 1 |
Bhargava, HN; Das, S | 1 |
Benyhe, S; Borsodi, A; Hepp, J; Khan, A; Medzihradszky, K; Simon, J; Szücs, M; Wollemann, M | 1 |
Inoki, R; Maeda, S; Nakamae, J | 2 |
Belisle, S; Bellabarba, D; Gallo-Payet, N; Lehoux, JG; Lemaire, S; Petit, A | 1 |
Bryant, HU; Malven, PV; Steele, TD; Yim, GK | 1 |
Alvinerie, M; Bueno, L; Gue, M; Honde, C; Junien, JL; Pascaud, X | 1 |
Borsodi, A; Lajtha, A; Zawilska, J | 1 |
Candeletti, S; Cavicchini, E; Ferri, S; Romualdi, P; Spampinato, S; Speroni, E | 1 |
Berzetei, IP; Duckles, SP; Fong, A; Yamamura, HI | 1 |
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Yoshimura, K | 3 |
Chavkin, C; Goldstein, A; James, IF | 1 |
Miller, RJ | 1 |
Herz, A; Pfeiffer, A | 1 |
Piercey, MF; Schroeder, LA; Varner, K | 1 |
Tung, AS; Yaksh, TL | 1 |
Huidobro-Toro, JP; Way, EL; Yoshimura, K | 1 |
Herz, A | 1 |
Lee, NM | 1 |
Kamerling, SG; Martin, WR; Wettstein, JG; Wu, KM | 1 |
Huidobro-Toro, JP; Lee, NM; Loh, HH; Way, EL; Zhu, YX | 1 |
Cros, J; Pontonnier, G; Porthe, G; Tafani, M; Valette, A | 1 |
Garzón, J; Gerhart, J; Lee, NM; Loh, HH; Sánchez-Blázquez, P | 1 |
Billington, CJ; Gerritsen, GC; Levine, AS; Morley, JE | 1 |
Pairet, M; Ruckebusch, Y | 1 |
Rezvani, A; Way, EL | 1 |
Gosnell, BA; Grace, M; Kneip, J; Levine, AS; Morley, JE | 1 |
Han, JS; Xie, GX | 2 |
Burkard, WP; Flück, N; Müller, PM | 1 |
Fujino, M; Negishi, K; Oka, T; Sawa, A; Suda, M; Wakimasu, M | 1 |
Laurent, S; Schmitt, H | 2 |
Goldstein, A; Han, JS; Xie, GX | 1 |
Barnard, EA; Benyhe, S; Borsodi, A; Simon, J; Wollemann, M | 1 |
Berzetei-Gurske, IP; Brandt, SR; Polgar, WE; Toll, L; Webster, JL | 1 |
Hogenboom, F; Mulder, AH; Schoffelmeer, AN | 1 |
Benyhe, S; Borsodi, A; Hepp, J; Ketevan, A; Medzihradszky, K; Simon, J | 1 |
Butelman, ER; Kreek, MJ; Vivian, JA; Woods, JH; Yu, J | 1 |
Akil, H; Goldstein, A; Mansour, A; Meng, F; Thompson, RC; Watson, SJ; Xie, GX | 1 |
3 review(s) available for ethylketocyclazocine and dynorphins
Article | Year |
---|---|
Endorphins and food intake: kappa opioid receptor agonists and hyperphagia.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Butorphanol; Choice Behavior; Cyclazocine; Diuresis; Drinking; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Humans; Morphine; Narcotic Antagonists; Phenazocine; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Satiety Response | 1985 |
Multiple opiate receptors for multiple opioid peptides.
Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dogs; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Male; Mice; Morphine; Naloxone; Neuromuscular Junction; Phenazocine; Rabbits; Radioligand Assay; Rats; Receptors, Opioid; Synaptic Transmission | 1982 |
Multiple opiate receptors and their functional significance.
Topics: Animals; beta-Endorphin; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Morphine; Receptors, Opioid; Tissue Distribution | 1983 |
66 other study(ies) available for ethylketocyclazocine and dynorphins
Article | Year |
---|---|
Kappa opioid agonists inhibit transmitter release from guinea pig hippocampal mossy fiber synaptosomes.
Topics: Animals; Azocines; Calcium; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Potassium; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptosomes | 1992 |
Dynorphin A-(1-13)-Tyr14-Leu15-Phe16-Asn17-Gly18-Pro19 : a potent and selective kappa opioid peptide.
Topics: Amino Acid Sequence; Animals; Dynorphins; Ethylketocyclazocine; Guinea Pigs; Kinetics; Male; Mice; Molecular Sequence Data; Muscle Contraction; Nociceptors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1991 |
Evidence for kappa 1 opioid receptor multiplicity in the guinea pig cerebellum.
Topics: Animals; Benzeneacetamides; Binding Sites; Binding, Competitive; Cerebellum; Dynorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Tritium | 1991 |
Kappa agonists inhibit gastric emptying but not acid secretion in rhesus monkeys.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Antihypertensive Agents; Cyclazocine; Dynorphins; Ethylketocyclazocine; Gastric Acid; Gastric Emptying; Macaca mulatta; Male; Narcotics; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Sodium | 1990 |
Kappa opioid receptors stimulate phosphoinositide turnover in rat brain.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Dynorphins; Enkephalins; Ethylketocyclazocine; Male; Phosphatidylinositols; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1990 |
Kappa-receptor mechanisms in synaptosomal Ca uptake.
Topics: Animals; Calcium; Calcium Radioisotopes; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Morphine; Nalorphine; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Synaptosomes | 1989 |
Computer analysis of the effect of beta-endorphin and dynorphin and related compounds on opioid binding to mouse brain membrane.
Topics: Animals; beta-Endorphin; Binding, Competitive; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Mice; Models, Neurological; Receptors, Opioid | 1989 |
Further demonstration of kappa opioid binding sites in the brain: evidence for heterogeneity.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzodiazepines; Binding Sites; Brain; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Levallorphan; Peptide Fragments; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism | 1985 |
Electrophysiological effects of dynorphin peptides on hippocampal pyramidal cells in rat.
Topics: Animals; Cyclazocine; Dynorphins; Electrophysiology; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; gamma-Aminobutyric Acid; Hippocampus; Male; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid | 1985 |
Inhibition of Ca++-ATPase of rat erythrocyte membranes by k-opioid agonists.
Topics: Animals; beta-Endorphin; Calcium-Transporting ATPases; Cyclazocine; Dynorphins; Endorphins; Erythrocyte Membrane; Ethylketocyclazocine; Levorphanol; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
Generalization tests with intraventricularly applied pro-enkephalin B-derived peptides in rats trained to discriminate the opioid kappa receptor agonist ethylketocyclazocine.
Topics: Animals; beta-Endorphin; Cyclazocine; Discrimination Learning; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Generalization, Stimulus; Injections, Intraventricular; Male; Protein Precursors; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
Effects of opioid agonists and antagonists on oxytocin and vasopressin release in vitro.
Topics: Animals; Arginine Vasopressin; Benzomorphans; beta-Endorphin; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Male; Naloxone; Oxytocin; Peptide Fragments; Pituitary Gland, Posterior; Rats; Rats, Inbred Strains | 1985 |
Effects of 2% sodium chloride imbibition on various opiate related hyperphagic conditions.
Topics: Animals; Cyclazocine; Deoxyglucose; Dynorphins; Ethylketocyclazocine; Feeding Behavior; Insulin; Male; Naloxone; Narcotics; Rats; Rats, Inbred Strains; Receptors, Opioid; Sodium Chloride; Time Factors | 1985 |
Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor.
Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Guanosine Triphosphate; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Nalorphine; Naloxone; Peptide Fragments; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sodium; Synaptosomes; Vas Deferens | 1985 |
Differential effect of stimulation strength in mouse vas deferens on inhibition of neuroeffector transmission by receptor type selective opioids.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Cyclazocine; Dynorphins; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Morphine Derivatives; Muscle, Smooth; Neuromuscular Junction; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Synaptic Transmission | 1986 |
Characterization of opioid receptors modulating noradrenaline release in the hippocampus of the rabbit.
Topics: Animals; Benzomorphans; Clonidine; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hippocampus; Morphine; Norepinephrine; Rabbits; Receptors, Opioid | 1986 |
On the opioid receptor subtype inhibiting the evoked release of 3H-noradrenaline from guinea-pig atria in vitro.
Topics: Animals; Atropine; Benzomorphans; Binding, Competitive; Corticosterone; Cyclazocine; Desipramine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Guinea Pigs; Heart Atria; In Vitro Techniques; Morphine; Myocardium; Naloxone; Norepinephrine; Peptide Fragments; Phentolamine; Receptors, Opioid; Receptors, Opioid, kappa; Synapses | 1986 |
Presynaptic opioid receptors modulating acetylcholine release in the hippocampus of the rabbit.
Topics: Acetylcholine; Animals; Benzomorphans; Choline; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Hippocampus; Naloxone; Peptide Fragments; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa; Synapses | 1986 |
Characterization of opioid receptors in the cat carotid body involved in chemosensory depression in vivo.
Topics: Animals; Carotid Body; Cats; Chemoreceptor Cells; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; Ethylketocyclazocine; Hypercapnia; Hypoxia; Peptide Fragments; Receptors, Opioid | 1986 |
Effects of dynorphin1-13 on opiate binding and dopamine and GABA uptake in stroked cat brain.
Topics: Animals; Brain; Brain Ischemia; Cats; Cyclazocine; Disease Models, Animal; Dopamine; Dynorphins; Ethylketocyclazocine; gamma-Aminobutyric Acid; Kinetics; Male; Peptide Fragments; Receptors, Opioid | 1986 |
Centrally-administered opioid selective agonists inhibit drinking in the rat.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain; Cyclazocine; Drinking Behavior; Dynorphins; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Male; Morphine; Naloxone; Peptide Fragments; Pyrrolidines; Rats; Receptors, Opioid | 1986 |
Pharmacological effects of nalorphine and nalorphine-7,8-oxide (nalorphine-epoxide): interaction of the intrinsic activity, affinity and pharmacological responses.
Topics: Analgesics; Animals; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Nalorphine; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid | 1986 |
[Peripheral analgesic actions of opioid peptides and morphine analogues].
Topics: Analgesics, Opioid; Animals; Cyclazocine; Dynorphins; Enkephalin, Methionine; Ethylketocyclazocine; Levallorphan; Lidocaine; Male; Mice; Morphine; Naloxone; Pain; Peptide Fragments | 1986 |
Binaltorphimine and nor-binaltorphimine, potent and selective kappa-opioid receptor antagonists.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Chemical Phenomena; Chemistry; Cyclazocine; Dynorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Male; Mice; Morphine; Naloxone; Naltrexone; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, kappa | 1987 |
Spinal kappa-opioid receptor-mediated antinociception is stimulus-specific.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzodiazepines; Benzomorphans; Cyclazocine; Drug Tolerance; Dynorphins; Ethylketocyclazocine; Injections, Spinal; Male; Morphine; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord | 1987 |
Effects of selective and non-selective kappa-opioid receptor agonists on cutaneous C-fibre-evoked responses of rat dorsal horn neurones.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Action Potentials; Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Electric Stimulation; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Nerve Fibers; Pain; Peptide Fragments; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Skin; Spinal Cord; Time Factors | 1987 |
Inhibition of [3H][3-MeHis2]thyrotropin releasing hormone recognition sites in the rat brain by tifluadom, a kappa opiate receptor agonist.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analysis of Variance; Animals; Benzodiazepines; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Kinetics; Male; Peptide Fragments; Pyrrolidines; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Thyrotropin-Releasing Hormone; Thyrotropin-Releasing Hormone | 1987 |
Purification of a kappa-opioid receptor subtype from frog brain.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Brain Chemistry; Chromatography, Gel; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Membranes; Molecular Weight; Naloxone; Peptide Fragments; Pyrrolidines; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Solubility | 1987 |
Positive inotropic action of kappa opiate agonists, ethylketocyclazocine and dynorphin-A(1-13), in isolated rat atrium.
Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Ethylketocyclazocine; Heart; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Peptide Fragments; Rats; Rats, Inbred Strains; Stimulation, Chemical | 1987 |
Functional opioid receptor sites in human placentas.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Cyclazocine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gonadotropin-Releasing Hormone; Humans; Kinetics; Placenta; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Thyrotropin-Releasing Hormone | 1988 |
Inhibition of cardiac Na+, K+-ATPase activity by dynorphin-A and ethylketocyclazocine.
Topics: Adenosine Triphosphate; Animals; Cyclazocine; Dynorphins; Enzyme Activation; Ethylketocyclazocine; Male; Myocardium; Naloxone; Peptide Fragments; Potassium; Rats; Rats, Inbred Strains; Sodium; Sodium-Potassium-Exchanging ATPase | 1988 |
Nocturnal depletion of hypothalamic dynorphin in anorexic Walker-256 tumor-bearing rats.
Topics: Animals; Anorexia; Carcinoma 256, Walker; Circadian Rhythm; Cyclazocine; Dynorphins; Eating; Ethylketocyclazocine; Feeding and Eating Disorders; Hypothalamus; Male; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1988 |
CNS blockade of acoustic stress-induced gastric motor inhibition by kappa-opiate agonists in dogs.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Acoustic Stimulation; Adrenocorticotropic Hormone; Analgesics; Animals; Cyclazocine; Dogs; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Ethylketocyclazocine; Gastrointestinal Motility; Hydrocortisone; Pyrrolidines; Stress, Physiological | 1988 |
Selective protection of benzomorphan binding sites against inactivation by N-ethylmaleimide. Evidence for kappa-opioid receptors in frog brain.
Topics: Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dynorphins; Ethylketocyclazocine; Ethylmaleimide; Morphinans; Peptide Fragments; Rana esculenta; Receptors, Opioid; Sodium Chloride | 1988 |
Investigations on dynorphin structurally-related opioid peptides. I. Impact on nociceptive transmission. II. Regulation of pituitary content.
Topics: Animals; Benzomorphans; Cyclazocine; Dynorphins; Estradiol; Ethylketocyclazocine; Female; Hypothalamo-Hypophyseal System; Male; Ovary; Pain; Pain Measurement; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1988 |
Characterization of kappa opioid receptors in the rabbit ear artery.
Topics: Animals; Benzeneacetamides; Benzomorphans; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle, Smooth, Vascular; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1988 |
Dynorphin interaction at the kappa-opiate site.
Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Receptors, Opioid; Receptors, Opioid, kappa | 1981 |
Dynorphin is a specific endogenous ligand of the kappa opioid receptor.
Topics: Analgesics, Opioid; Animals; Binding, Competitive; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Ligands; Morphine Derivatives; Myenteric Plexus; Naloxone; Peptide Fragments; Receptors, Opioid | 1982 |
Kappa opioid properties of dynorphin and its peptide fragments on the guinea-pig Ileum.
Topics: Animals; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Receptors, Opioid; Receptors, Opioid, kappa | 1982 |
Discrimination of three opiate receptor binding sites with the use of a computerized curve-fitting technique.
Topics: Animals; Binding, Competitive; Brain; Computers; Cyclazocine; Dihydromorphine; Diprenorphine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Phenazocine; Rats; Receptors, Opioid | 1982 |
Analgesic activity of intraspinally administered dynorphin and ethylketocyclazocine.
Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Injections; Male; Mice; Spinal Cord | 1982 |
Activation of K-opiate sites by dynorphin in the myenteric plexus.
Topics: Animals; Cyclazocine; Drug Tolerance; Dynorphins; Electric Stimulation; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa | 1982 |
In vivo evidence for multiple opiate receptors mediating analgesia in the rat spinal cord.
Topics: Animals; Cyclazocine; Dose-Response Relationship, Drug; Dynorphins; Endorphins; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Injections, Spinal; Male; Naloxone; Pain; Phenazocine; Rats; Rats, Inbred Strains; Receptors, Opioid; Spinal Cord | 1982 |
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum.
Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists | 1982 |
Is dynorphin a k ligand?
Topics: Animals; Brain; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Receptors, Opioid; Receptors, Opioid, kappa | 1983 |
Possible medullary kappa hyperalgesic mechanism. I. A new potential role for endogenous opioid peptides in pain perception.
Topics: Animals; Cyclazocine; Dogs; Dynorphins; Endorphins; Ethylketocyclazocine; Medulla Oblongata; Naloxone; Pain; Receptors, Opioid; Reflex | 1983 |
Dynorphin inhibition of the neurotensin contractile activity on the myenteric plexus.
Topics: Animals; Atropine; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Nerve Tissue Proteins; Neurotensin; Peptide Fragments; Receptors, Opioid; Tetrodotoxin | 1984 |
Placental kappa binding site : interaction with dynorphin and its possible implication in hCG secretion.
Topics: Analgesics, Opioid; Chorionic Gonadotropin; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; Female; Humans; Peptide Fragments; Placenta; Pregnancy; Receptors, Opioid; Receptors, Opioid, kappa | 1983 |
Dynorphin A: inhibitory effect on other opiate ligand bindings in the mouse brain.
Topics: Animals; Brain; Cyclazocine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Naloxone; Narcotics; Peptide Fragments; Receptors, Opioid; Sodium Chloride | 1984 |
Feeding systems in Chinese hamsters.
Topics: Animals; Brain; Calcitonin; Circadian Rhythm; Cricetinae; Cyclazocine; Diabetes Mellitus; Dynorphins; Eating; Endorphins; Ethylketocyclazocine; Feeding Behavior; Haloperidol; Mesocricetus; Naloxone; Peptide Fragments; Phenazocine; Sincalide; Starvation | 1984 |
Opioid receptor agonists in the rabbit colon: comparison of in vivo and in vitro studies.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Colon; Cyclazocine; Dynorphins; Electric Conductivity; Enkephalins; Ethylketocyclazocine; Fentanyl; Male; Morphine; Naloxone; Narcotics; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1984 |
Dynorphin-(1-13) restores the potency of morphine on the tolerant guinea pig ileum.
Topics: Animals; beta-Endorphin; Cyclazocine; Drug Interactions; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments | 1984 |
The effect of ovariectomy, estradiol and progesterone on opioid modulation of feeding.
Topics: Animals; Appetite Regulation; Brain; Castration; Cyclazocine; Dynorphins; Eating; Estradiol; Ethylketocyclazocine; Female; Naloxone; Progesterone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1984 |
[Dynorphin: analgesic effect via kappa receptors in the spinal cord of rats].
Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Ethylketocyclazocine; Female; Naloxone; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Spinal Cord | 1984 |
Characteristics of 3H-tifluadom binding in guinea-pig brain membranes.
Topics: Animals; Benzodiazepines; Benzomorphans; Binding Sites; Brain; Cyclazocine; Dihydromorphine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Male; Morphine; Receptors, Opioid | 1984 |
[Dynorphin: analgesic effect via kappa receptors in spinal cord of the spinal cords of rats].
Topics: Analgesics; Animals; Cyclazocine; Dynorphins; Ethylketocyclazocine; Female; Morphine; Naloxone; Pain; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Sensory Thresholds; Spinal Cord | 1984 |
Evidence that dynorphin-(1-13) acts as an agonist on opioid kappa-receptors.
Topics: Animals; Cyclazocine; Dynorphins; Electric Stimulation; Endorphins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Naloxone; Peptide Fragments; Rabbits; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vas Deferens | 1982 |
Central cardiovascular effects of kappa agonists dynorphin-(1-13) and ethylketocyclazocine in the anaesthetized rat.
Topics: Animals; beta-Endorphin; Blood Pressure; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Heart Rate; Male; Naloxone; Peptide Fragments; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Vagus Nerve | 1983 |
Opposite central cardiovascular effects of various morphine-like drugs and opiate peptides in the rat.
Topics: Animals; Blood Pressure; Brain; Cyclazocine; Dynorphins; Endorphins; Enkephalin, Methionine; Ethylketocyclazocine; Fentanyl; Heart Rate; Male; Peptide Fragments; Rats; Rats, Inbred Strains | 1983 |
Analgesia induced by intrathecal injection of dynorphin B in the rat.
Topics: Analgesics; Animals; Cyclazocine; Dose-Response Relationship, Drug; Drug Tolerance; Dynorphins; Endorphins; Enkephalin, Leucine; Ethylketocyclazocine; Female; Injections, Spinal; Morphine; Naloxone; Rats | 1984 |
[3H]dynorphin1-8 binding sites in frog (Rana esculenta) brain membranes.
Topics: Amino Acid Sequence; Animals; Brain; Cell Membrane; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Naloxone; Peptide Fragments; Rana esculenta; Receptors, Opioid; Sodium Chloride; Tritium | 1994 |
Comparison of kappa 2-opioid receptors in guinea pig brain and guinea pig ileum membranes.
Topics: Analgesics; Animals; Benzomorphans; Brain Chemistry; Dynorphins; Ethylketocyclazocine; Guanylyl Imidodiphosphate; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Ligands; Male; Membranes; Myenteric Plexus; Receptors, Opioid, kappa | 1993 |
Kappa1- and kappa2-opioid receptors mediating presynaptic inhibition of dopamine and acetylcholine release in rat neostriatum.
Topics: Acetylcholine; Animals; Benzeneacetamides; Dopamine; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Male; N-Methylaspartate; Naloxone; Neostriatum; Neural Inhibition; Peptide Fragments; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1997 |
Affinity labelling of frog brain opioid receptors by dynorphin(1-10) chloromethyl ketone.
Topics: Affinity Labels; Amino Acid Chloromethyl Ketones; Analgesics, Opioid; Animals; Binding, Competitive; Brain Chemistry; Dihydromorphine; Dynorphins; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Membrane Proteins; Peptide Fragments; Radioligand Assay; Rana esculenta; Receptors, Opioid; Receptors, Opioid, kappa; Tritium | 1997 |
Systemic effects of E-2078, a stabilized dynorphin A(1-8) analog, in rhesus monkeys.
Topics: Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Conditioning, Operant; Discrimination, Psychological; Diuresis; Dynorphins; Ethylketocyclazocine; Female; Food; Injections, Intramuscular; Injections, Subcutaneous; Macaca mulatta; Male; Pain Measurement; Peptide Fragments; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1999 |
Cloning and pharmacological characterization of a rat kappa opioid receptor.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Amino Acid Sequence; Analgesics; Animals; Benzeneacetamides; Cell Line; Cell Membrane; Cloning, Molecular; Corpus Striatum; Cyclic AMP; DNA Primers; DNA, Complementary; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Gene Library; In Situ Hybridization; Inositol 1,4,5-Trisphosphate; Kinetics; Ligands; Molecular Sequence Data; Pyrrolidines; Rats; Receptors, Opioid, kappa; Restriction Mapping; RNA, Messenger; Transfection | 1993 |