Page last updated: 2024-08-23

ethylketocyclazocine and diprenorphine

ethylketocyclazocine has been researched along with diprenorphine in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-199014 (66.67)18.7374
1990's6 (28.57)18.2507
2000's1 (4.76)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, C; Li, JG; Liu-Chen, LY; Luo, LY; Zhu, J1
Bartness, TJ; Billington, CJ; Herman, BH; Levine, AS; Morley, JE1
Imai, T; Kamikubo, K; Miura, K; Miura, Y; Miyashita, T; Murase, H; Nakamura, S; Niwa, M; Satoh, T; Tomita, A1
Falke, NE; Fischer, EG; Martin, R1
Mack, KJ; Weyhenmeyer, JA1
Grace, M; Kneip, J; Levine, AS; Morley, JE; Shearman, GT; Zeugner, H1
DeRossett, SE; Holtzman, SG2
Bidlack, JM; Denton, RR1
Brown, SR; Cox, BM; Puttfarcken, P; Werling, LL1
Spoerlein, MT; Szewczak, MR1
Corbett, AD; Gillan, MG; Kosterlitz, HW; McKnight, AT; Paterson, SJ; Robson, LE1
Herz, A; Pfeiffer, A1
Chang, KJ; Cuatrecasas, P; Hazum, E1
Brown, DR; Holtzman, SG; Locke, KW1
Dykstra, LA1
Castanas, E; Hatzoglou, A; Kampa, M; Loukas, S; Martin, P; Martin, PM1
Bakogeorgou, E; Castanas, E; Hatzoglou, A1
Calvo, F; Castanas, E; Hatzoglou, A; Martin, PM; Panagiotou, S1
Castanas, E; Denizot, A; Dermitzaki, I; Gravanis, A; Hatzoglou, A; Henry, JF; Kampa, M; Margioris, AN; Oliver, C1
Castanas, E; Kampa, M; Kouroumalis, E; Nifli, AP; Notas, G; Papasava, D; Thermos, K; Xidakis, K1

Other Studies

21 other study(ies) available for ethylketocyclazocine and diprenorphine

ArticleYear
Activation of the cloned human kappa opioid receptor by agonists enhances [35S]GTPgammaS binding to membranes: determination of potencies and efficacies of ligands.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adenylate Cyclase Toxin; Animals; Binding Sites; Cell Membrane; CHO Cells; Cholera Toxin; Cloning, Molecular; Cricetinae; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Humans; Kinetics; Magnesium; Pertussis Toxin; Pyrrolidines; Receptors, Opioid, kappa; Recombinant Proteins; Sodium; Sulfur Radioisotopes; Virulence Factors, Bordetella

1997
Effects of the opiate antagonists diprenorphine and naloxone and of selected opiate agonists on feeding behavior in guinea pigs.
    Life sciences, 1990, Volume: 46, Issue:2

    Topics: Animals; Butorphanol; Circadian Rhythm; Cyclazocine; Diprenorphine; Ethylketocyclazocine; Feeding Behavior; Guinea Pigs; Morphinans; Morphine; Naloxone; Narcotic Antagonists; Narcotics; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Varying expression of opioid receptors and GTP-binding proteins in human pheochromocytomas.
    NIDA research monograph, 1986, Volume: 75

    Topics: Adrenal Gland Neoplasms; beta-Endorphin; Cell Membrane; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; GTP-Binding Proteins; Humans; Pheochromocytoma; Receptors, Opioid

1986
Stereospecific opiate binding in living human polymorphonuclear leucocytes.
    Cell biology international reports, 1985, Volume: 9, Issue:11

    Topics: Analgesics, Opioid; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Granulocytes; Humans; Kinetics; Naloxone; Neutrophils; Receptors, Opioid

1985
Binding characteristics of kappa opioids in rat brain. A comparison of in vitro binding paradigms.
    Neuropharmacology, 1985, Volume: 24, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cyclazocine; Diprenorphine; Ethylketocyclazocine; Kinetics; Male; Morphinans; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
The kappa opioid receptor and food intake.
    European journal of pharmacology, 1985, May-28, Volume: 112, Issue:1

    Topics: Animals; Benzodiazepines; Benzomorphans; Butorphanol; Cyclazocine; Diprenorphine; Eating; Ethylketocyclazocine; Haloperidol; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism; Time Factors

1985
Effects of opiate antagonists and putative kappa agonists on unpunished and punished operant behavior in the rat.
    Psychopharmacology, 1985, Volume: 86, Issue:4

    Topics: Animals; Conditioning, Operant; Cyclazocine; Diprenorphine; Ethylketocyclazocine; Male; Naloxone; Narcotic Antagonists; Punishment; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1985
A monoclonal antibody capable of modulating opioid binding to rat neural membranes.
    The Journal of biological chemistry, 1985, Dec-15, Volume: 260, Issue:29

    Topics: Animals; Antibodies, Monoclonal; Cell Line; Cyclazocine; Dihydromorphine; Diprenorphine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Flunitrazepam; Immunoglobulin M; Kinetics; Male; Mice; Mice, Inbred BALB C; Molecular Weight; Naloxone; Narcotics; Nerve Tissue; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Opioid

1985
Discriminative stimulus effects of the opioid antagonist diprenorphine in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Cyclazocine; Diprenorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ethylketocyclazocine; Generalization, Stimulus; Morphinans; Naloxone; Narcotic Antagonists; Phenazocine; Psychotropic Drugs; Receptors, Neurotransmitter; Receptors, Opioid; Receptors, Phencyclidine; Saimiri

1986
Sodium regulation of agonist binding at opioid receptors. II. Effects of sodium replacement on opioid binding in guinea pig cortical membranes.
    Molecular pharmacology, 1986, Volume: 30, Issue:2

    Topics: Animals; Cell Membrane; Cerebral Cortex; Cyclazocine; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Etorphine; Guinea Pigs; Male; Oligopeptides; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sodium

1986
Opiate-induced turning in rats after injection into the ventral tegmental area.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 25, Issue:5

    Topics: Animals; Cyclazocine; Diprenorphine; Endorphins; Ethylketocyclazocine; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Stereotyped Behavior; Tegmentum Mesencephali

1986
Radioligands for probing opioid receptors.
    Journal of receptor research, 1984, Volume: 4, Issue:1-6

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzomorphans; Binding Sites; Brain; Cyclazocine; Diprenorphine; Enkephalin, Leucine; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Naloxone; Pro-Opiomelanocortin; Protein Precursors; Pyrrolidines; Radioligand Assay; Rats; Receptors, Opioid; Vas Deferens

1984
Discrimination of three opiate receptor binding sites with the use of a computerized curve-fitting technique.
    Molecular pharmacology, 1982, Volume: 21, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Computers; Cyclazocine; Dihydromorphine; Diprenorphine; Dynorphins; Endorphins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Phenazocine; Rats; Receptors, Opioid

1982
Possible role of distinct morphine and enkephalin receptors in mediating actins of benzomorphan drugs (putative kappa and sigma agonists).
    Proceedings of the National Academy of Sciences of the United States of America, 1980, Volume: 77, Issue:8

    Topics: Animals; Benzomorphans; Brain; Cyclazocine; Diprenorphine; Endorphins; Enkephalins; Ethylketocyclazocine; Guanosine Triphosphate; Morphinans; Morphine; Naloxone; Neuroblastoma; Rats; Receptors, Opioid; Sodium; Synaptic Membranes

1980
Effects of opiate antagonists and putative mu- and kappa-agonists on milk intake in rat and squirrel monkey.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6

    Topics: Animals; Buprenorphine; Cyclazocine; Diazepam; Diprenorphine; Drinking; Ethylketocyclazocine; Etorphine; Male; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Saimiri; Taste

1982
Development of enhanced sensitivity to naloxone.
    Life sciences, 1983, Nov-21, Volume: 33, Issue:21

    Topics: Animals; Buprenorphine; Cyclazocine; Diprenorphine; Dose-Response Relationship, Drug; Drug Interactions; Ethylketocyclazocine; Male; Meperidine; Naloxone; Phencyclidine; Reaction Time; Saimiri

1983
Identification of a novel opioid peptide (Tyr-Val-Pro-Phe-Pro) derived from human alpha S1 casein (alpha S1-casomorphin, and alpha S1-casomorphin amide).
    The Biochemical journal, 1996, Nov-01, Volume: 319 ( Pt 3)

    Topics: Amino Acid Sequence; Binding, Competitive; Breast Neoplasms; Caseins; Cell Division; Cell Line; Diprenorphine; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Female; Humans; Kinetics; Peptide Fragments; Receptors, Opioid, kappa

1996
Taxol inhibits opioid binding on T47D human breast cancer cells.
    Biochemical and biophysical research communications, 1997, Jun-09, Volume: 235, Issue:1

    Topics: Amino Acid Sequence; Analgesics, Opioid; Antineoplastic Agents, Phytogenic; Binding Sites; Binding, Competitive; Breast Neoplasms; Diprenorphine; Ethylketocyclazocine; Humans; Molecular Sequence Data; Paclitaxel; Receptors, Opioid; Receptors, Opioid, kappa; Sequence Alignment; Tubulin; Tumor Cells, Cultured

1997
Modulation of the estrogen-regulated proteins cathepsin D and pS2 by opioid agonists in hormone-sensitive breast cancer cell lines (MCF7 and T47D): evidence for an interaction between the two systems.
    Journal of cellular biochemistry, 1998, Dec-01, Volume: 71, Issue:3

    Topics: Breast Neoplasms; Cathepsin D; Cell Division; Cycloheximide; Cytosol; Diprenorphine; Dose-Response Relationship, Drug; Estradiol; Ethylketocyclazocine; Etorphine; Female; Humans; Inhibitory Concentration 50; Narcotic Antagonists; Narcotics; Neoplasms, Hormone-Dependent; Protein Synthesis Inhibitors; Proteins; Trefoil Factor-1; Tumor Cells, Cultured; Tumor Suppressor Proteins

1998
Kappa1-opioid binding sites are the dominant opioid binding sites in surgical specimens of human pheochromocytomas and in a human pheochromocytoma (KAT45) cell line.
    European journal of pharmacology, 1999, Jan-08, Volume: 364, Issue:2-3

    Topics: Analgesics, Opioid; Binding Sites; Binding, Competitive; Catecholamines; Cell Membrane; Diprenorphine; Dopamine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Epinephrine; Ethylketocyclazocine; Humans; Narcotic Antagonists; Norepinephrine; Opioid Peptides; Pheochromocytoma; Radioligand Assay; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tritium; Tumor Cells, Cultured

1999
The inhibitory effect of opioids on HepG2 cells is mediated via interaction with somatostatin receptors.
    European journal of pharmacology, 2007, Jan-19, Volume: 555, Issue:1

    Topics: Analgesics, Opioid; Apoptosis; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Diprenorphine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Humans; Narcotic Antagonists; Octreotide; Receptors, Opioid; Receptors, Somatostatin; RNA, Messenger; Somatostatin

2007