ethidium and kn 62

ethidium has been researched along with kn 62 in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (16.67)18.2507
2000's10 (83.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cornish, JE; Gargett, CE; Wiley, JS1
Dubyak, GR; Humphreys, BD; Rice, J; Surprenant, A; Virginio, C1
Hibell, AD; Humphrey, PP; Michel, AD; Thompson, KM; Xing, M1
Baraldi, PG; del Carmen Nuñez, M; Di Virgilio, F; Falzoni, S; Morelli, A; Romagnoli, R1
Adinolfi, E; Baricordi, R; Di Virgilio, F; Falzoni, S; Ferrari, D; Forchap, S; Minelli, M; Pizzirani, C; Sitta, B; Turchet, L1
Christopherson, RI; Fuller, SJ; Georgiou, JG; Martin, CJ; Skarratt, KK; Sluyter, R; Wiley, JS1
Baraldi, PG; Borea, PA; Cara, CL; Carrion, MD; Cruz-Lopez, O; Fogli, E; Gessi, S; Moorman, AR; Preti, D; Romagnoli, R; Sacchetto, V; Tabrizi, MA1
Fuller, SJ; Georgiou, JG; Gu, BJ; Jursik, C; Sluyter, R; Wiley, JS1
Dehaye, JP; Garcia-Marcos, M; Marino, A; Otto, A; Pochet, S; Seil, M1
Chambers, LJ; Michel, AD; Walter, DS1
Di Virgilio, F; Gulinelli, S; Pellegatti, P; Pizzirani, C; Skerlavaj, B; Tomasinsig, L; Tossi, A; Zanetti, M1
Kim, JH; Kim, WK; Kim, YC; Lee, GE; Lee, HS; Lee, SD1

Other Studies

12 other study(ies) available for ethidium and kn 62

ArticleYear
ATP, a partial agonist for the P2Z receptor of human lymphocytes.
    British journal of pharmacology, 1997, Volume: 122, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Affinity Labels; Barium; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethidium; Flow Cytometry; Humans; In Vitro Techniques; Ion Channels; Leukemia, Lymphocytic, Chronic, B-Cell; Linear Models; Lymphocytes; Purinergic P2 Receptor Agonists; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Structure-Activity Relationship; Thionucleotides

1997
Isoquinolines as antagonists of the P2X7 nucleotide receptor: high selectivity for the human versus rat receptor homologues.
    Molecular pharmacology, 1998, Volume: 54, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Cells, Cultured; Chimera; Enzyme Inhibitors; Ethidium; Fluorescent Dyes; Humans; Ion Transport; Isoquinolines; Leukocytes; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7

1998
Complexities of measuring antagonist potency at P2X(7) receptor orthologs.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 296, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Amiloride; Animals; Benzoxazoles; Buffers; Cations, Divalent; Cell Adhesion; Cells, Cultured; Drug Interactions; Enzyme Inhibitors; Ethidium; Fluorescent Dyes; Humans; Kinetics; Mice; Platelet Aggregation Inhibitors; Purinergic P2 Receptor Antagonists; Pyridoxal Phosphate; Quinolinium Compounds; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Rosaniline Dyes; Serum Albumin, Bovine; Sodium Chloride; Species Specificity; Temperature

2001
Synthesis and biological activity of N-arylpiperazine-modified analogues of KN-62, a potent antagonist of the purinergic P2X7 receptor.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Arylsulfonates; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Ethidium; Humans; Interleukin-1; Macrophages; Monocytes; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2X7; Structure-Activity Relationship; Tyrosine

2003
The antibiotic polymyxin B modulates P2X7 receptor function.
    Journal of immunology (Baltimore, Md. : 1950), 2004, Oct-01, Volume: 173, Issue:7

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Amino Acid Sequence; Animals; Anti-Bacterial Agents; Calcium; Cell Line; Cell Line, Tumor; Cell Survival; Dose-Response Relationship, Drug; Drug Synergism; Ethidium; Humans; Intracellular Fluid; K562 Cells; Leukemia, Lymphocytic, Chronic, B-Cell; Macrophages; Mice; Molecular Sequence Data; Oxidation-Reduction; Polymyxin B; Purinergic P2 Receptor Antagonists; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Transfection

2004
Human epidermal and monocyte-derived langerhans cells express functional P2X receptors.
    The Journal of investigative dermatology, 2005, Volume: 125, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Biological Transport; Epidermal Cells; Ethidium; Humans; Keratinocytes; Langerhans Cells; Monocytes; Polymorphism, Genetic; Receptors, IgE; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Skin

2005
From tyrosine to glycine: synthesis and biological activity of potent antagonists of the purinergic P2X7 receptor.
    Journal of medicinal chemistry, 2007, Jul-26, Volume: 50, Issue:15

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; beta-Alanine; Calcium; Cell Line; Cell Membrane; Cell Membrane Permeability; Ethidium; Fluorescent Dyes; Glycine; Humans; Isoquinolines; Naphthalenes; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2X7; Recombinant Proteins; Structure-Activity Relationship; Sulfonamides; Sulfones; Tyrosine

2007
A quantitative method for routine measurement of cell surface P2X7 receptor function in leucocyte subsets by two-colour time-resolved flow cytometry.
    Journal of immunological methods, 2007, Aug-31, Volume: 325, Issue:1-2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; B-Lymphocytes; Barium; Biological Transport; Calcium; Chlorides; Enzyme Inhibitors; Ethidium; Flow Cytometry; Humans; Killer Cells, Natural; Leukocytes, Mononuclear; Monocytes; Potassium; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Reproducibility of Results; Sodium; T-Lymphocytes; Temperature

2007
Contribution of two ionotropic purinergic receptors to ATP responses in submandibular gland ductal cells.
    Cellular signalling, 2007, Volume: 19, Issue:10

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Biological Transport; Calcium; Carbachol; Ethidium; Interleukin-1beta; Mice; Mice, Knockout; Phospholipases A2; Receptors, Purinergic P2; Receptors, Purinergic P2X4; Receptors, Purinergic P2X7; Saliva; Submandibular Gland

2007
Negative and positive allosteric modulators of the P2X(7) receptor.
    British journal of pharmacology, 2008, Volume: 153, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Allosteric Regulation; Animals; Binding Sites; Cell Line; Dose-Response Relationship, Drug; Ethidium; Glycine; Humans; Molecular Structure; Piperazines; Protein Conformation; Pyridoxal Phosphate; Quinolines; Radioligand Assay; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Recombinant Proteins; Species Specificity; Time Factors; Transfection; Vanadates

2008
The human cathelicidin LL-37 modulates the activities of the P2X7 receptor in a structure-dependent manner.
    The Journal of biological chemistry, 2008, Nov-07, Volume: 283, Issue:45

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphate; Animals; Antimicrobial Cationic Peptides; Calcium; Calcium Signaling; Cathelicidins; Cell Proliferation; Enzyme Inhibitors; Ethidium; Fibroblasts; Gene Expression Regulation; Humans; Mice; NIH 3T3 Cells; Protein Structure, Secondary; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Structure-Activity Relationship

2008
Synthesis and structure-activity relationships of novel, substituted 5,6-dihydrodibenzo[a,g]quinolizinium P2X7 antagonists.
    Bioorganic & medicinal chemistry letters, 2009, Feb-01, Volume: 19, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Berberine Alkaloids; Cell Differentiation; Cell Line; Chemistry, Pharmaceutical; Drug Design; Ethidium; Humans; Interleukin-1beta; Lipopolysaccharides; Models, Chemical; Purinergic P2 Receptor Antagonists; Quinolizines; Receptors, Purinergic P2X7; Structure-Activity Relationship

2009