etazolate and gamma-aminobutyric acid

etazolate has been researched along with gamma-aminobutyric acid in 16 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-199016 (100.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Risley, EA; Williams, M1
Mehta, AK; Ticku, MK1
Maksay, G; Ticku, MK1
Olsen, RW; Snowman, AM1
Braunwalder, A; Cheney, DL; Loo, P; Wood, PL; Yokoyama, N1
Karobath, M; Placheta, P1
Drexler, G; Karobath, M; Supavilai, P1
Drexler, G; Karobath, M; Sieghart, W; Supavilai, P1
Goodwin, FK; Marangos, PJ; Paul, SM; Skolnick, P1
Barnes, DM; Dichter, MA; White, WF1
Williams, M1
Borea, PA; Karobath, M; Supavilai, P1
Agnati, LF; Andersson, K; Eneroth, P; Fuxe, K; Karobath, M; Köhler, C; Krogsgaard-Larsen, P; Ogren, SO; Pérez de la Mora, M1
Karobath, M; Supavilai, P2
Leeb-Lundberg, F; Olsen, RW; Snowman, A1

Reviews

3 review(s) available for etazolate and gamma-aminobutyric acid

ArticleYear
Anxioselective anxiolytics.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:5

    Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety; Azabicyclo Compounds; Benzodiazepines; Brain Chemistry; Drug Interactions; Etazolate; gamma-Aminobutyric Acid; Humans; Molecular Weight; Piperazines; Pyrazoles; Pyridazines; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship

1983
Distinction of benzodiazepine receptor agonists and inverse agonists by binding studies in vitro.
    Advances in biochemical psychopharmacology, 1983, Volume: 38

    Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Etazolate; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Muscimol; Rats; Receptors, Cell Surface; Receptors, GABA-A

1983
GABA and benzodiazepine receptors. Studies on their localization in the hippocampus and their interaction with central dopamine neurons in the rat brain.
    Advances in biochemical psychopharmacology, 1981, Volume: 26

    Topics: Animals; Brain; Dopamine; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Muscimol; Neural Pathways; Neurons; Neurons, Afferent; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1981

Other Studies

13 other study(ies) available for etazolate and gamma-aminobutyric acid

ArticleYear
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
    Life sciences, 1979, Feb-26, Volume: 24, Issue:9

    Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical

1979
Characteristics of flunitrazepam binding to intact primary cultured spinal cord neurons and its modulation by GABAergic drugs.
    Journal of neurochemistry, 1987, Volume: 49, Issue:5

    Topics: Animals; Benzodiazepines; Binding, Competitive; Carbolines; Cells, Cultured; Embryo, Mammalian; Etazolate; Etomidate; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Neurons; Pentobarbital; Receptors, GABA-A; Spinal Cord

1987
Dissociation of [35S]t-butylbicyclophosphorothionate binding differentiates convulsant and depressant drugs that modulate GABAergic transmission.
    Journal of neurochemistry, 1985, Volume: 44, Issue:2

    Topics: Animals; Barbiturates; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Central Nervous System Depressants; Cerebral Cortex; Convulsants; Etazolate; Etomidate; gamma-Aminobutyric Acid; Kinetics; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Avermectin B1a modulation of gamma-aminobutyric acid/benzodiazepine receptor binding in mammalian brain.
    Journal of neurochemistry, 1985, Volume: 44, Issue:4

    Topics: Animals; Bicuculline; Brain; Cattle; Cell Membrane; Cerebral Cortex; Etazolate; gamma-Aminobutyric Acid; Isonicotinic Acids; Ivermectin; Lactones; Muscimol; Pentobarbital; Rats; Receptors, GABA-A

1985
In vitro characterization of benzodiazepine receptor agonists, antagonists, inverse agonists and agonist/antagonists.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 231, Issue:3

    Topics: Animals; Brain; Chlorides; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Muscimol; Rats; Receptors, GABA-A

1984
In vitro modulation by SQ 20009 and SQ 65396 of GABA receptor binding in rat CNS membranes.
    European journal of pharmacology, 1980, Mar-21, Volume: 62, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Brain; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nerve Tissue Proteins; Nicotinic Acids; Pyrazoles; Pyridines; Rats; Receptors, Cell Surface

1980
Modulation by picrotoxin and IPTBO of 3H-flunitrazepam binding to the GABA/benzodiazepine receptor complex of rat cerebellum.
    Life sciences, 1981, Jan-19, Volume: 28, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membranes; Organophosphorus Compounds; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Temperature

1981
Properties of benzodiazepine receptors in rat retina.
    Experimental eye research, 1982, Volume: 34, Issue:6

    Topics: Animals; Anthelmintics; Anti-Anxiety Agents; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Ivermectin; Lactones; Molecular Weight; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Retina

1982
Biological substrates of anxiety: benzodiazepine receptors and endogenous ligands.
    L'Encephale, 1982, Volume: 8, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Brain; Carbolines; Chlorides; Etazolate; Ethanol; gamma-Aminobutyric Acid; Humans; Molecular Weight; Niacinamide; Pentobarbital; Purines; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1982
Etazolate (SQ20009): electrophysiology and effects on [3H]flunitrazepam binding in cultured cortical neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1983, Volume: 3, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Binding Sites; Cells, Cultured; Cerebral Cortex; Electric Conductivity; Electrophysiology; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Neurons; Nicotinic Acids; Rats; Synapses

1983
In vitro modulation by avermectin B1a of the GABA/benzodiazepine receptor complex of rat cerebellum.
    Journal of neurochemistry, 1981, Volume: 36, Issue:3

    Topics: Animals; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ivermectin; Lactones; Octoxynol; Polyethylene Glycols; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A

1981
Interaction of SQ 20009 and GABA-like drugs as modulators of benzodiazepine receptor binding.
    European journal of pharmacology, 1980, Mar-21, Volume: 62, Issue:2-3

    Topics: Animals; Benzodiazepines; Cerebellum; Drug Interactions; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Membranes; Muscimol; Nicotinic Acids; Rats; Receptors, Drug

1980
Perturbation of benzodiazepine receptor binding by pyrazolopyridines involves picrotoxinin/barbiturate receptor sites.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1981, Volume: 1, Issue:5

    Topics: Animals; Benzodiazepines; Binding Sites; Brain; Etazolate; gamma-Aminobutyric Acid; Phenobarbital; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Drug; Sesterterpenes

1981