etazolate has been researched along with gamma-aminobutyric acid in 16 studies
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 16 (100.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Risley, EA; Williams, M | 1 |
Mehta, AK; Ticku, MK | 1 |
Maksay, G; Ticku, MK | 1 |
Olsen, RW; Snowman, AM | 1 |
Braunwalder, A; Cheney, DL; Loo, P; Wood, PL; Yokoyama, N | 1 |
Karobath, M; Placheta, P | 1 |
Drexler, G; Karobath, M; Supavilai, P | 1 |
Drexler, G; Karobath, M; Sieghart, W; Supavilai, P | 1 |
Goodwin, FK; Marangos, PJ; Paul, SM; Skolnick, P | 1 |
Barnes, DM; Dichter, MA; White, WF | 1 |
Williams, M | 1 |
Borea, PA; Karobath, M; Supavilai, P | 1 |
Agnati, LF; Andersson, K; Eneroth, P; Fuxe, K; Karobath, M; Köhler, C; Krogsgaard-Larsen, P; Ogren, SO; Pérez de la Mora, M | 1 |
Karobath, M; Supavilai, P | 2 |
Leeb-Lundberg, F; Olsen, RW; Snowman, A | 1 |
3 review(s) available for etazolate and gamma-aminobutyric acid
Article | Year |
---|---|
Anxioselective anxiolytics.
Topics: Adenosine; Animals; Anti-Anxiety Agents; Anxiety; Azabicyclo Compounds; Benzodiazepines; Brain Chemistry; Drug Interactions; Etazolate; gamma-Aminobutyric Acid; Humans; Molecular Weight; Piperazines; Pyrazoles; Pyridazines; Quinolines; Receptors, Cell Surface; Receptors, GABA-A; Structure-Activity Relationship | 1983 |
Distinction of benzodiazepine receptor agonists and inverse agonists by binding studies in vitro.
Topics: Affinity Labels; Animals; Anti-Anxiety Agents; Benzodiazepines; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Etazolate; gamma-Aminobutyric Acid; Humans; In Vitro Techniques; Muscimol; Rats; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
GABA and benzodiazepine receptors. Studies on their localization in the hippocampus and their interaction with central dopamine neurons in the rat brain.
Topics: Animals; Brain; Dopamine; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Muscimol; Neural Pathways; Neurons; Neurons, Afferent; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A | 1981 |
13 other study(ies) available for etazolate and gamma-aminobutyric acid
Article | Year |
---|---|
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical | 1979 |
Characteristics of flunitrazepam binding to intact primary cultured spinal cord neurons and its modulation by GABAergic drugs.
Topics: Animals; Benzodiazepines; Binding, Competitive; Carbolines; Cells, Cultured; Embryo, Mammalian; Etazolate; Etomidate; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Neurons; Pentobarbital; Receptors, GABA-A; Spinal Cord | 1987 |
Dissociation of [35S]t-butylbicyclophosphorothionate binding differentiates convulsant and depressant drugs that modulate GABAergic transmission.
Topics: Animals; Barbiturates; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cell Membrane; Central Nervous System Depressants; Cerebral Cortex; Convulsants; Etazolate; Etomidate; gamma-Aminobutyric Acid; Kinetics; Male; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Avermectin B1a modulation of gamma-aminobutyric acid/benzodiazepine receptor binding in mammalian brain.
Topics: Animals; Bicuculline; Brain; Cattle; Cell Membrane; Cerebral Cortex; Etazolate; gamma-Aminobutyric Acid; Isonicotinic Acids; Ivermectin; Lactones; Muscimol; Pentobarbital; Rats; Receptors, GABA-A | 1985 |
In vitro characterization of benzodiazepine receptor agonists, antagonists, inverse agonists and agonist/antagonists.
Topics: Animals; Brain; Chlorides; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Muscimol; Rats; Receptors, GABA-A | 1984 |
In vitro modulation by SQ 20009 and SQ 65396 of GABA receptor binding in rat CNS membranes.
Topics: Animals; Anti-Anxiety Agents; Brain; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nerve Tissue Proteins; Nicotinic Acids; Pyrazoles; Pyridines; Rats; Receptors, Cell Surface | 1980 |
Modulation by picrotoxin and IPTBO of 3H-flunitrazepam binding to the GABA/benzodiazepine receptor complex of rat cerebellum.
Topics: Animals; Anti-Anxiety Agents; Bicuculline; Binding Sites; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Male; Membranes; Organophosphorus Compounds; Picrotoxin; Rats; Receptors, Drug; Receptors, GABA-A; Temperature | 1981 |
Properties of benzodiazepine receptors in rat retina.
Topics: Animals; Anthelmintics; Anti-Anxiety Agents; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Ivermectin; Lactones; Molecular Weight; Pyridazines; Rats; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter; Retina | 1982 |
Biological substrates of anxiety: benzodiazepine receptors and endogenous ligands.
Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Benzodiazepines; Brain; Carbolines; Chlorides; Etazolate; Ethanol; gamma-Aminobutyric Acid; Humans; Molecular Weight; Niacinamide; Pentobarbital; Purines; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A | 1982 |
Etazolate (SQ20009): electrophysiology and effects on [3H]flunitrazepam binding in cultured cortical neurons.
Topics: Animals; Anti-Anxiety Agents; Binding Sites; Cells, Cultured; Cerebral Cortex; Electric Conductivity; Electrophysiology; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; Kinetics; Neurons; Nicotinic Acids; Rats; Synapses | 1983 |
In vitro modulation by avermectin B1a of the GABA/benzodiazepine receptor complex of rat cerebellum.
Topics: Animals; Cerebellum; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Ivermectin; Lactones; Octoxynol; Polyethylene Glycols; Pyrazoles; Rats; Receptors, Cell Surface; Receptors, Drug; Receptors, GABA-A | 1981 |
Interaction of SQ 20009 and GABA-like drugs as modulators of benzodiazepine receptor binding.
Topics: Animals; Benzodiazepines; Cerebellum; Drug Interactions; Etazolate; Flunitrazepam; gamma-Aminobutyric Acid; In Vitro Techniques; Membranes; Muscimol; Nicotinic Acids; Rats; Receptors, Drug | 1980 |
Perturbation of benzodiazepine receptor binding by pyrazolopyridines involves picrotoxinin/barbiturate receptor sites.
Topics: Animals; Benzodiazepines; Binding Sites; Brain; Etazolate; gamma-Aminobutyric Acid; Phenobarbital; Picrotoxin; Pyrazoles; Rats; Rats, Inbred Strains; Receptors, Drug; Sesterterpenes | 1981 |