estrone has been researched along with warfarin in 33 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 4 (12.12) | 18.7374 |
| 1990's | 2 (6.06) | 18.2507 |
| 2000's | 17 (51.52) | 29.6817 |
| 2010's | 10 (30.30) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Caron, G; Ermondi, G | 1 |
| Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
| Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ | 1 |
| Ekins, S; Williams, AJ; Xu, JJ | 1 |
| Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
| Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
| Elias, E; Iqbal, S; Vickers, C | 1 |
| Copas, DK; Cummings, AJ; Kaelin, AC; Landon, MJ; Rosankiewicz, JR | 1 |
| Eto, Y; Herschkowitz, NN; Rampini, S; Wiesmann, U | 1 |
| Cittanova, N; Desfosses, B; Dessen, P; Herve, F; Moenner, M; Urios, P | 1 |
| Kostian, ML; Lehtimäki, J; Mäkelä, S; Poutanen, M; Santti, R; Vihko, R | 1 |
| Potter, BV; Purohit, A; Reed, MJ; Woo, LW | 1 |
| Malini, B; Potter, BV; Purohit, A; Reed, MJ; Woo, LL | 1 |
| Barrow, D; Hejaz, HA; Nicholson, RI; Potter, BV; Purohit, A; Reed, MJ; Woo, LW | 1 |
| Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, M | 2 |
| Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, MB | 1 |
| Ahmed, S; James, K; Owen, CP; Patel, CK | 1 |
| Ahmed, S; James, K; Owen, CP | 2 |
| Ho, Y; Potter, BV; Purohit, A; Reed, MJ; Robinson, J; Vicker, N; Woo, LL | 1 |
| DOWBEN, RM; HSIA, DY; RIABOV, S | 1 |
| Chander, SK; Potter, BV; Purohit, A; Reed, MJ; Woo, LW | 1 |
| Newman, SP; Potter, BV; Purohit, A; Reed, MJ; Woo, LW | 1 |
| Coombes, RC; Dobbs, N; Elliott, M; Kulinskaya, E; Potter, BV; Purohit, A; Reed, MJ; Stanczyk, FZ; Stanway, SJ; Sufi, S; Vigushin, D; Ward, R; Wilson, RH; Woo, LW | 1 |
| Ahmed, V; Liu, Y; Silvestro, C; Taylor, SD | 1 |
| Akinaga, S; Anazawa, H; Ishida, H; Kuwabara, T; Li, PK; Murakata, C; Nakata, T; Sato, N; Shiotsu, Y; Suzuki, M; Takebayashi, M; Tanaka, H; Terasaki, Y | 1 |
| Häusler, S; Schneiter, R; Stieger, B; Treiber, A | 1 |
| Ishida, H; Nakata, T; Shiotsu, Y | 1 |
| Edwards, DR; Wolfenden, R | 1 |
| Dawson, PA; Lan, T; Oberlies, NH; Paine, MF; Scarlett, YV; Vandermolen, KM; Widmer, WW; Won, CS | 1 |
| Potter, BV; Thomas, MP | 1 |
| Finel, M; Ge, GB; Järvinen, E; Troberg, J; Yang, L | 1 |
4 review(s) available for estrone and warfarin
| Article | Year |
|---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Steroid sulfatase: molecular biology, regulation, and inhibition.
Topics: Animals; Breast Neoplasms; Clinical Trials, Phase I as Topic; Coumarins; Enzyme Inhibitors; Estrone; Female; Humans; Models, Molecular; Neoplasms, Hormone-Dependent; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids | 2005 |
[Steroid sulfatase inhibitor].
Topics: Animals; Breast Neoplasms; Clinical Trials as Topic; Coumarins; Drug Design; Enzyme Inhibitors; Estradiol; Estrogens; Estrone; Female; Humans; Steryl-Sulfatase; Sulfonamides | 2010 |
Estrogen O-sulfamates and their analogues: Clinical steroid sulfatase inhibitors with broad potential.
Topics: Animals; Coumarins; Enzyme Inhibitors; Estradiol; Estrogens; Estrone; Humans; Models, Molecular; Steryl-Sulfatase; Sulfonamides | 2015 |
2 trial(s) available for estrone and warfarin
| Article | Year |
|---|---|
Phase I study of STX 64 (667 Coumate) in breast cancer patients: the first study of a steroid sulfatase inhibitor.
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Androstenediol; Breast Neoplasms; Coumarins; Dose-Response Relationship, Drug; Estradiol; Estrone; Female; Humans; Maximum Tolerated Dose; Middle Aged; Neoplasm Metastasis; Neoplasms, Hormone-Dependent; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Testosterone | 2006 |
A modified grapefruit juice eliminates two compound classes as major mediators of the grapefruit juice-fexofenadine interaction: an in vitro-in vivo "connect".
Topics: Adult; Animals; Anti-Allergic Agents; Beverages; Chlorocebus aethiops; Citrus paradisi; COS Cells; Coumarins; Cross-Over Studies; Estrone; Female; Flavonoids; Food-Drug Interactions; Fruit; HEK293 Cells; Humans; Male; Middle Aged; Organic Anion Transporters; Terfenadine; Young Adult | 2013 |
27 other study(ies) available for estrone and warfarin
| Article | Year |
|---|---|
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water | 2005 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Developing structure-activity relationships for the prediction of hepatotoxicity.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes | 2010 |
A predictive ligand-based Bayesian model for human drug-induced liver injury.
Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Drug metabolism in end-stage liver disease. In vitro activities of some phase I and phase II enzymes.
Topics: Adolescent; Adult; Aminopyrine; Child; Coumarins; Cytochrome P-450 Enzyme System; Estrone; Female; Humans; Lithocholic Acid; Liver Diseases; Liver Function Tests; Male; Middle Aged; Oxazines; Pharmaceutical Preparations; Sulfotransferases | 1990 |
The transfer and metabolism of 7-ethoxycoumarin and androstenedione during the in vitro perfusion of the human placental lobule.
Topics: Androstenedione; Coumarins; Estrone; Female; Humans; In Vitro Techniques; Kinetics; Perfusion; Placenta; Pregnancy; Testosterone; Umbelliferones | 1988 |
Enzymic studies of sulphatases in tissues of the normal human and in metachromatic leukodystrophy with multiple sulphatase deficiencies: arylsulphatases A, B and C, cerebroside sulphatase, psychosine sulphatase and steroid sulphatases.
Topics: Adult; Brain; Cerebrosides; Child; Child, Preschool; Cholesterol; Chromatography, Thin Layer; Coumarins; Dehydroepiandrosterone; Estrone; Galactose; Galactosidases; Genetic Variation; Glycosides; Hexosaminidases; Humans; Hydrogen-Ion Concentration; Infant; Isoelectric Focusing; Kidney; Kinetics; Leukodystrophy, Metachromatic; Liver; Lysophosphatidylcholines; Lysosomes; Organ Specificity; Polyethylene Glycols; Solubility; Sphingosine; Sulfatases; Tritium | 1974 |
Interaction between rat alpha 1 fetoprotein and fluorescent derivatives of estrone in relation to the position and type of the fluorescent label.
Topics: alpha-Fetoproteins; Animals; Binding Sites; Binding, Competitive; Coumarins; Dansyl Compounds; Estrone; Fetal Blood; Fluorescent Dyes; Rats; Spectrometry, Fluorescence; Structure-Activity Relationship | 1983 |
Estrogen-specific 17 beta-hydroxysteroid oxidoreductase type 1 (E.C. 1.1.1.62) as a possible target for the action of phytoestrogens.
Topics: 17-Hydroxysteroid Dehydrogenases; Breast Neoplasms; Cell Division; Coumarins; Estradiol; Estrogens, Non-Steroidal; Estrone; Flavonoids; Glycyrrhetinic Acid; Humans; Isoflavones; Phytoestrogens; Plant Preparations; Sitosterols; Tumor Cells, Cultured | 1995 |
In vivo inhibition of estrone sulfatase activity and growth of nitrosomethylurea-induced mammary tumors by 667 COUMATE.
Topics: Animals; Antineoplastic Agents; Cell Division; Coumarins; Estrone; Female; Humans; Liver; Mammary Neoplasms, Experimental; Methylnitrosourea; Ovariectomy; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids; Time Factors; Uterus | 2000 |
Potent active site-directed inhibition of steroid sulphatase by tricyclic coumarin-based sulphamates.
Topics: Alanine; Antineoplastic Agents; Arylsulfatases; Binding Sites; Breast Neoplasms; Coumarins; Dehydroepiandrosterone Sulfate; Dose-Response Relationship, Drug; Estrone; Female; Glycine; Heterocyclic Compounds, 3-Ring; Humans; Hydrogen Bonding; Kinetics; Microsomes; Models, Molecular; Placenta; Postmenopause; Steryl-Sulfatase; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids | 2000 |
Non-steroidal and steroidal sulfamates: new drugs for cancer therapy.
Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Coumarins; Enzyme Inhibitors; Estrogens; Estrone; Female; Humans; Kinetics; Oxepins; Rats; Rats, Wistar; Sulfatases; Sulfonamides; Sulfonic Acids; Tumor Cells, Cultured | 2001 |
Novel inhibitors of the enzyme estrone sulfatase (ES).
Topics: Alkanes; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Ketones; Mesylates; Sulfatases; Sulfonamides; Sulfonic Acids | 2001 |
Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
Topics: Chemistry, Physical; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Models, Biological; Models, Chemical; Structure-Activity Relationship; Sulfatases; Sulfonamides | 2001 |
Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism.
Topics: Catalytic Domain; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids | 2001 |
Synthesis and biochemical evaluation of novel and potent inhibitors of the enzyme oestrone sulphatase (ES).
Topics: Coumarins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrone; Humans; Hydrolysis; Inhibitory Concentration 50; Kinetics; Microsomes; Models, Chemical; Placenta; Spectrophotometry, Infrared; Sulfatases; Sulfonamides; Time Factors | 2002 |
The design, synthesis, and biochemical evaluation of derivatives of biphenyl sulfamate-based compounds as novel inhibitors of estrone sulfatase.
Topics: Catalysis; Coumarins; Enzyme Inhibitors; Estrone; Models, Chemical; Models, Molecular; Sulfatases; Sulfonamides | 2002 |
Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES).
Topics: Coumarins; Drug Design; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Kinetics; Models, Chemical; Models, Molecular; Molecular Conformation; Molecular Mimicry; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids | 2002 |
Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II.
Topics: Binding Sites; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Coumarins; Estrone; Humans; Inhibitory Concentration 50; Models, Molecular; Steroids; Structure-Activity Relationship; Substrate Specificity; Sulfatases; Sulfonamides; Sulfonic Acids | 2003 |
INHIBITION OF GLUCURONOSYL TRANSFERASE BY STEROID HORMONES.
Topics: Amino Alcohols; Androgens; Cholesterol; Cortisone; Coumarins; Enzyme Inhibitors; Estradiol; Estriol; Estrone; Glucosyltransferases; Glucuronates; Glucuronosyltransferase; Guinea Pigs; Hormones; Hydroxyprogesterones; Methyltestosterone; Nandrolone; Nitrophenols; Pregnanediol; Pregnenolone; Progesterone; Research; Steroids; Testosterone | 1963 |
The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
Topics: Animals; Coumarins; Drug Combinations; Estrogens; Estrone; Female; Homeostasis; Organ Size; Ovariectomy; Rats; Rats, Wistar; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Uterus | 2004 |
Boronic acids as inhibitors of steroid sulfatase.
Topics: Boronic Acids; Chromones; Coumarins; Enzyme Inhibitors; Estrone; Humans; Molecular Structure; Steryl-Sulfatase; Structure-Activity Relationship | 2006 |
A novel steroidal selective steroid sulfatase inhibitor KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells in vitro and in animal models.
Topics: Administration, Oral; Animals; Breast Neoplasms; Cell Proliferation; Coumarins; Cricetinae; Disease Models, Animal; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Estrone; Female; Gene Expression Regulation, Enzymologic; Humans; Leukocytes; Methylnitrosourea; Molecular Structure; Rats; Rats, Sprague-Dawley; Receptors, Progesterone; Signal Transduction; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Tamoxifen; Tumor Cells, Cultured | 2007 |
Bosentan is a substrate of human OATP1B1 and OATP1B3: inhibition of hepatic uptake as the common mechanism of its interactions with cyclosporin A, rifampicin, and sildenafil.
Topics: Animals; Aryl Hydrocarbon Hydroxylases; Biological Transport; Bosentan; CHO Cells; Cricetinae; Cricetulus; Cyclosporine; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dehydroepiandrosterone Sulfate; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrone; Humans; Liver-Specific Organic Anion Transporter 1; Molecular Structure; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Piperazines; Purines; Pyrimidines; Rifampin; Sildenafil Citrate; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfonamides; Sulfones; Warfarin | 2007 |
Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
Topics: Arylsulfatases; Catalysis; Coumarins; Esters; Estrone; Hydrogen-Ion Concentration; Hydrolysis; Kinetics; Molecular Structure; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids | 2012 |
UGT1A10 Is a High Activity and Important Extrahepatic Enzyme: Why Has Its Role in Intestinal Glucuronidation Been Frequently Underestimated?
Topics: Animals; Blotting, Western; Camptothecin; Chromatography, High Pressure Liquid; Coumarins; Diclofenac; Estradiol; Estrone; Flavonoids; Glucuronosyltransferase; Humans; Hymecromone; Intestinal Mucosa; Irinotecan; Kinetics; Microsomes, Liver | 2017 |