estrone has been researched along with tamoxifen in 107 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 41 (38.32) | 18.7374 |
| 1990's | 31 (28.97) | 18.2507 |
| 2000's | 19 (17.76) | 29.6817 |
| 2010's | 14 (13.08) | 24.3611 |
| 2020's | 2 (1.87) | 2.80 |
| Authors | Studies |
|---|---|
| Ambros, R; Brandl, G; Mannschreck, A; Polossek, T; von Angerer, E; von Angerer, S | 1 |
| Knebel, NG; von Angerer, E | 1 |
| Prekajac, J; von Angerer, E | 1 |
| Bogden, A; Buchborn, H; Hartmann, RW; Kranzfelder, G; Schönenberger, H | 1 |
| Carlsson, B; Enmark, E; Grandien, K; Gustafsson, JA; Häggblad, J; Kuiper, GG; Nilsson, S | 1 |
| Bellavance, E; Luu-The, V; Poirier, D | 1 |
| Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
| Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ | 1 |
| Ekins, S; Williams, AJ; Xu, JJ | 1 |
| Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
| Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K | 1 |
| Geras, E; Gershengorn, MC; Marcus-Samuels, BE | 1 |
| Bolan, G; Lippman, M; Monaco, ME | 1 |
| Kennedy, BJ; Kiang, DT | 1 |
| Hisamatsu, K; Nomura, Y; Tashiro, H | 1 |
| Adessi, G; Jouvenot, M; Marechal, G; Ordener, C; Pellerin, I; Royez, M; Vuillermoz, C | 1 |
| Burton, R; Castleden, CM; Ekelund, P; Miodrag, A | 1 |
| de Launoit, Y; Dufour, M; Labrie, F; Simard, J; Veilleux, R | 1 |
| Sasson, S | 1 |
| Akami, T; Honjyo, H; Mitsuo, M; Naitoh, K; Oka, T; Okada, H; Yamamoto, T; Yasumura, T | 1 |
| Hayashi, K; Kosaki, G; Shimozuma, K; Tominaga, T; Yoshida, Y | 1 |
| Corna, D; Garattini, S; Pusineri, F; Remuzzi, G; Rossini, M; Viganò, G; Zoja, C | 1 |
| Gelly, C; Nguyen, BL; Pasqualini, JR | 1 |
| Courion, C; Dumas, MY; Fanidi, A; Laugier, C; Nemoz, G; Pacheco, H; Pageaux, JF; Prigent, AF | 1 |
| Bygdeman, M; Matlin, SA; Swahn, ML; Wu, ZY | 1 |
| Cantwell, BM; Carmichael, J; Dowsett, M; Harris, AL | 1 |
| Adessi, GL; Alkhalaf, M; Propper, A | 1 |
| Howe, RS; Lee, YH; Lyttle, CR; Sha, SJ; Sheehan, DM; Teuscher, C | 1 |
| Baird, DT; Lumsden, MA; West, CP | 1 |
| Lamberts, SW; Verleun, T | 1 |
| Gelly, C; Pasqualini, JR | 3 |
| Carlström, K; Pousette, A; Rannevik, G; Sköldefors, H; Theve, NO; Wilking, N | 1 |
| Fletcher, WS; Keenan, EJ; Pommier, RF; Woltering, EA | 1 |
| Jordan, VC; Robinson, SP | 1 |
| Honjyo, H; Oka, T; Okada, H; Yasumura, T | 1 |
| Kauppila, A; Kivinen, S; Stenbäck, F; Vihko, R; Vuopala, S | 1 |
| Gelly, C; Lecerf, F; Pasqualini, JR | 1 |
| Karácsony, G; Karcsú, S; Kocsis, J; László, FA | 1 |
| Benz, C; DeGregorio, M; Drakes, T; Gandara, D; Miller, B; Monroe, S; Wilbur, B | 1 |
| Adessi, GL; Alkhalaf, M; Chaminadas, G; Propper, AY | 1 |
| Reddel, RR; Sutherland, RL | 1 |
| Gorski, J; Hansen, JC | 1 |
| Dowsett, M; Harris, AL; Smith, IE; Stuart-Harris, R | 1 |
| Bozek, T; Carr, L; Dowsett, M; Gazet, JC; Jeffcoate, SL; Kurkure, A; McKinna, JA; Smith, IE; Stuart-Harris, R | 1 |
| Carlström, K; Sköldefors, H; Theve, NO; Wallgren, A; Wilking, N | 1 |
| Carlström, K; Döberl, A; Pousette, A; Rannevik, G; Wilking, N | 1 |
| Smith, IE; Stuart-Harris, RC | 1 |
| Davis, TE; Rose, DP | 1 |
| Guichard, A; Mignot, TM; Scheib, D | 1 |
| Fisher, B; Gunduz, N; Saffer, EA | 1 |
| Gross, M; Kuhl, H; Mehlis, W; Schneider, M; Stegmüller, M; Taubert, HD; Weber, W | 1 |
| Carlström, K; Sköldefors, H; Theve, NO; Wilking, N | 1 |
| Billiet, G; Bonte, J; Ide, P; Wynants, P | 1 |
| Bayard, F; Jozan, S; Kreitmann, B | 1 |
| Capony, F; Williams, DL | 1 |
| Samsel, J; Weniger, JP; Zeis, A | 1 |
| Gulino, A; Pasqualini, JR | 1 |
| Ekse, D; Geisler, J; Hösch, S; Lønning, PE | 1 |
| Diamandis, EP; Grass, L; Yu, H; Zarghami, N | 1 |
| Potter, BV; Purohit, A; Reed, MJ; Roberts, CJ; Williams, GJ | 1 |
| Geisler, J; Gundersen, S; Haarstad, H; Kvinnsland, S; Lønning, PE; Raabe, N | 1 |
| Adlercreutz, H; Ekse, D; Fotsis, T; Johannessen, DC; Lien, EA; Lønning, PE | 1 |
| Giannoulis, G; Hadziyannis, SJ; Manesis, EK; Vafiadou, I; Zoumboulis, P | 1 |
| Bhargava, S; Farooq, A; Murugesan, K; Vij, U | 1 |
| Borrás, M; el Khissiin, AH; Gol-Winkler, R; Hardy, L; Leclercq, G; Legros, N; Lempereur, F | 1 |
| Chetrite, G; Pasqualini, JR; Urabe, M | 1 |
| Biberger, C; von Angerer, E | 1 |
| Bender, W; Yu, FL | 2 |
| Ahmari, SE; Bryan-Poole, N; Evans, GF; Glasebrook, AL; Short, L; Zuckerman, SH | 1 |
| Fletcher, WS; Lum, SS; Pommier, RF; Woltering, EA | 1 |
| Eng, FC; Ferrara, J; Lee, HS; White, JH; Willson, TM | 1 |
| Belanger, A; Gauthier, S; Labrie, C; Labrie, F; Luo, S; Martel, C; Mérand, Y; Sourla, A | 1 |
| Bélanger, A; Candas, B; Couillard, S; Gutman, M; Labrie, C; Labrie, F | 1 |
| Gorodeski, GI | 1 |
| Adams, MR; Schwenke, DC; Wagner, JD | 1 |
| Guo, ZG; Niu, XL; Zhang, XW | 1 |
| Gaston, K; Taylor, A; Webster, K | 1 |
| Keller-Wood, M; Saoud, CJ; Stoner, TA; Wood, CE | 1 |
| Budziszewska, B; Jaworska-Feil, L; Kajta, M; Kubera, M; Lasoń, W; Leśkiewicz, M | 1 |
| Browne-Martin, K; Longcope, C | 1 |
| Candas, B; Couillard, S; Gutman, M; Labrie, C; Labrie, F; Roy, J | 1 |
| Imai, Y; Sugimoto, Y; Tsukahara, S; Tsuruo, T; Ueda, K | 1 |
| Deavers, MT; Gershenson, DM; Malpica, A; Parlow, AF; Silva, EG | 1 |
| Barry, WH; Li, F; Su, Z; Sugishita, K | 1 |
| Cosman, F; Lindsay, R; Mikhail, M; Nieves, J; Richart, RM; Scotti, RJ; Vardy, MD; Zion, M | 1 |
| Eugster, EA; Jou, HC; Pescovitz, OH; Plourde, P; Reiter, EO; Rubin, SD | 1 |
| Asnis, AG; Duncan, B; Francis, D; Hortobagyi, GN; Rivera, E; Schaaf, LJ; Valero, V | 1 |
| Alemany, M; Fernández-López, JA; Ferrer-Lorente, R; García-Peláez, B; Remesar, X | 1 |
| Cleary, JF; Havighurst, TC; Hutson, PR; Love, RR | 1 |
| Cleary, JF; Havighurst, TC; Hutson, PR; Love, RR; Rogers, E | 1 |
| Bågeman, E; Ingvar, C; Jernström, H; Klug, TL; Rose, C | 1 |
| Akinaga, S; Anazawa, H; Ishida, H; Kuwabara, T; Li, PK; Murakata, C; Nakata, T; Sato, N; Shiotsu, Y; Suzuki, M; Takebayashi, M; Tanaka, H; Terasaki, Y | 1 |
| A'Hern, RP; Cameron, DA; Dixon, JM; Dowsett, M; Folkerd, E; Macaskill, EJ; McHugh, M; Murray, J; Renshaw, L; Young, O | 1 |
| Ballard-Barbash, R; Baumgartner, KB; Baumgartner, RN; Bernstein, L; Gilliland, F; McTiernan, A; Neuhouser, ML; Nojomi, M; Stanczyk, F | 1 |
| Coombes, RC; Januszewski, A; Palmieri, C; Stanway, S | 1 |
| Bryk, M; Chatterton, RT; Habe-Evans, M; Khan, SA; Parker, NP; Scholtens, DM | 1 |
| Baker, AE; Corkery, DP; Dellaire, G; Hawco, CL; Marchal, E; Thompson, A; Uddin, MI | 1 |
| Cardozo, T; Fadiel, A; Hamza, A; Naftolin, F; Song, J; Tivon, D | 1 |
| Bhatta, P; Curpan, RF; Fernandes, DJ; Jordan, VC; Korostyshevskiy, VR; Maximov, PY; McDaniel, RE | 1 |
| Kong, D; Li, J; Li, N; Teng, Y; Wang, J; Wang, Y | 1 |
| Avella, A; Azaro, A; Bellet, M; Bohn, U; Catalán, G; Catalán, R; Ciruelos, E; Climent, MA; Ferrer, R; Fleming, GF; Francis, PA; González-Martin, A; Gray, KP; Láng, I; Lluch, A; Morales, J; Price, KN; Rajasekaran, A; Regan, MM; Vázquez, J | 1 |
| Altbach, M; Chalasani, P; Chow, HHS; Galons, JP; Huang, C; Maskarinec, G; Roe, DJ; Stopeck, A; Strom, MB; Thompson, PA; Thomson, CA; Wertheim, BC | 1 |
| Billen, J; Han, SN; Neven, P; Pauwels, S; Van Houdt, M | 1 |
| Bazgier, V; Berka, K; Holcakova, J; Hrstka, R; Kolarova, T; Kudova, E; Kvasnica, M; Oklestkova, J; Rarova, L; Strnad, M; Tichy, V; Vonka, P | 1 |
4 review(s) available for estrone and tamoxifen
| Article | Year |
|---|---|
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk | 2016 |
Equilibrium binding analysis of estrogen agonists and antagonists: relation to the activation of the estrogen receptor.
Topics: Clomiphene; Drug Interactions; Estradiol; Estriol; Estrogen Antagonists; Estrone; Humans; Receptors, Estrogen; Tamoxifen | 1991 |
Aminoglutethimide in the treatment of advanced breast cancer.
Topics: Adrenalectomy; Aged; Aminoglutethimide; Androstenedione; Breast Neoplasms; Clinical Trials as Topic; Dehydroepiandrosterone; Drug Therapy, Combination; Estradiol; Estrone; Female; Glucocorticoids; Humans; Hydrocortisone; Hypophysectomy; Menopause; Middle Aged; Neoplasm Metastasis; Tamoxifen | 1984 |
Irosustat: a first-generation steroid sulfatase inhibitor in breast cancer.
Topics: Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Clinical Trials, Phase II as Topic; Dehydroepiandrosterone Sulfate; Estradiol; Estrone; Female; Fulvestrant; Humans; Neoplasms, Hormone-Dependent; Steryl-Sulfatase; Sulfonic Acids; Tamoxifen | 2011 |
13 trial(s) available for estrone and tamoxifen
| Article | Year |
|---|---|
Tamoxifen and natural progesterone as supplements to low-dose postmenopausal estrogen therapy.
Topics: Alanine Transaminase; Aspartate Aminotransferases; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Estrone; Female; Hormones; Humans; Lipids; Menopause; Middle Aged; Progesterone; Tamoxifen | 1988 |
Aminoglutethimide in the treatment of advanced breast cancer.
Topics: Adrenalectomy; Aged; Aminoglutethimide; Androstenedione; Breast Neoplasms; Clinical Trials as Topic; Dehydroepiandrosterone; Drug Therapy, Combination; Estradiol; Estrone; Female; Glucocorticoids; Humans; Hydrocortisone; Hypophysectomy; Menopause; Middle Aged; Neoplasm Metastasis; Tamoxifen | 1984 |
Influence of droloxifene (3-hydroxytamoxifen), 40 mg daily, on plasma gonadotrophins, sex hormone binding globulin and estrogen levels in postmenopausal breast cancer patients.
Topics: Antineoplastic Agents, Hormonal; Breast Neoplasms; Estradiol; Estrogens; Estrone; Female; Follicle Stimulating Hormone; Follow-Up Studies; Humans; Luteinizing Hormone; Postmenopause; Sex Hormone-Binding Globulin; Tamoxifen; Time Factors | 1995 |
Influence of treatment with the anti-oestrogen 3-hydroxytamoxifen (droloxifene) on plasma sex hormone levels in postmenopausal patients with breast cancer.
Topics: Aged; Breast Neoplasms; Estradiol; Estrogen Antagonists; Estrogens, Conjugated (USP); Estrone; Female; Follicle Stimulating Hormone; Gonadal Steroid Hormones; Humans; Luteinizing Hormone; Middle Aged; Postmenopause; Sex Hormone-Binding Globulin; Tamoxifen; Time Factors | 1995 |
Treatment of hepatocellular carcinoma with combined suppression and inhibition of sex hormones: a randomized, controlled trial.
Topics: Analysis of Variance; Androgens; Carcinoma, Hepatocellular; Double-Blind Method; Drug Therapy, Combination; Estradiol; Estrone; Female; Flutamide; Follicle Stimulating Hormone; Follow-Up Studies; Humans; Liver Neoplasms; Luteinizing Hormone; Male; Middle Aged; Neoplasm Staging; Placebos; Probability; Survival Rate; Tamoxifen; Time Factors; Triptorelin Pamoate | 1995 |
Short-term urogenital effects of raloxifene, tamoxifen, and estrogen.
Topics: Aged; Atrophy; Double-Blind Method; Estradiol; Estrogens; Estrogens, Conjugated (USP); Estrone; Female; Humans; Menopause; Middle Aged; Placebos; Raloxifene Hydrochloride; Tamoxifen; Urethra; Uterine Prolapse; Vagina | 2003 |
Tamoxifen treatment for precocious puberty in McCune-Albright syndrome: a multicenter trial.
Topics: Cafe-au-Lait Spots; Estradiol; Estrogen Antagonists; Estrone; Female; Fibrous Dysplasia of Bone; Fibrous Dysplasia, Polyostotic; Follicle Stimulating Hormone; Humans; Hyperthyroidism; Insulin-Like Growth Factor I; Luteinizing Hormone; Prospective Studies; Puberty, Precocious; Tamoxifen; Time Factors | 2003 |
Pilot study evaluating the pharmacokinetics, pharmacodynamics, and safety of the combination of exemestane and tamoxifen.
Topics: Administration, Oral; Aged; Aged, 80 and over; Androstadienes; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Estradiol; Estrone; Female; History, 18th Century; Humans; Middle Aged; Neoplasm Metastasis; Neoplasm Staging; Pilot Projects; Tamoxifen | 2004 |
Endocrine effects of tamoxifen plus exemestane in postmenopausal women with breast cancer.
Topics: Adult; Aged; Alkaline Phosphatase; Androstadienes; Antineoplastic Combined Chemotherapy Protocols; Aromatase Inhibitors; Breast Neoplasms; Cholesterol, HDL; Estradiol; Estrogen Antagonists; Estrone; Exanthema; Female; Hot Flashes; Humans; Middle Aged; Postmenopause; Tamoxifen; Treatment Outcome | 2005 |
Effect of exemestane on tamoxifen pharmacokinetics in postmenopausal women treated for breast cancer.
Topics: Adult; Aged; Androstadienes; Antineoplastic Agents, Hormonal; Aromatase Inhibitors; Breast Neoplasms; Drug Interactions; Estradiol; Estrone; Female; Humans; Middle Aged; Postmenopause; Tamoxifen | 2005 |
Letrozole suppresses plasma estradiol and estrone sulphate more completely than anastrozole in postmenopausal women with breast cancer.
Topics: Adult; Aged; Aged, 80 and over; Anastrozole; Antineoplastic Agents; Breast Neoplasms; Chemotherapy, Adjuvant; Cross-Over Studies; Estradiol; Estrone; Female; Humans; Letrozole; Middle Aged; Nitriles; Postmenopause; Radioimmunoassay; Selective Estrogen Receptor Modulators; Tamoxifen; Treatment Outcome; Triazoles | 2008 |
Twelve-Month Estrogen Levels in Premenopausal Women With Hormone Receptor-Positive Breast Cancer Receiving Adjuvant Triptorelin Plus Exemestane or Tamoxifen in the Suppression of Ovarian Function Trial (SOFT): The SOFT-EST Substudy.
Topics: Adult; Androstadienes; Antineoplastic Agents, Hormonal; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Chemotherapy, Adjuvant; Estradiol; Estrogens; Estrone; Female; Follicle Stimulating Hormone; Humans; Luteinizing Hormone; Ovary; Tamoxifen; Triptorelin Pamoate | 2016 |
A randomized, placebo-controlled trial of diindolylmethane for breast cancer biomarker modulation in patients taking tamoxifen.
Topics: Adult; Antineoplastic Combined Chemotherapy Protocols; Biomarkers, Tumor; Breast Neoplasms; Double-Blind Method; Female; Humans; Hydroxyestrones; Indoles; Mammography; Middle Aged; Sex Hormone-Binding Globulin; Tamoxifen; Time Factors; Treatment Outcome | 2017 |
91 other study(ies) available for estrone and tamoxifen
| Article | Year |
|---|---|
6-Alkyl-12-formylindolo[2,1-a]isoquinolines. Syntheses, estrogen receptor binding affinities, and stereospecific cytostatic activity.
Topics: Animals; Antineoplastic Agents; Binding Sites; Cattle; Computer Simulation; Estrogen Antagonists; Female; Isoquinolines; Mammary Neoplasms, Experimental; Mice; Models, Molecular; Receptors, Estrogen; Stereoisomerism; Uterus | 1992 |
2-Phenylindole-linked [2-(aminoalkyl)pyridine]dichloroplatinum(II): complexes with a selective action on estrogen receptor positive mammary tumors.
Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Cattle; Cell Line; Female; Humans; Mammary Neoplasms, Experimental; Mice; Organoplatinum Compounds; Receptors, Estrogen; Structure-Activity Relationship | 1991 |
Benzo[a]carbazole derivatives. Synthesis, estrogen receptor binding affinities, and mammary tumor inhibiting activity.
Topics: Animals; Antineoplastic Agents; Carbazoles; Cattle; Cell Line; Estrogen Antagonists; Estrogens, Non-Steroidal; Female; Humans; In Vitro Techniques; Mammary Neoplasms, Experimental; Neoplasms, Hormone-Dependent; Organ Size; Rats; Rats, Inbred Strains; Receptors, Estrogen; Structure-Activity Relationship; Uterus | 1986 |
Potential antiestrogens. Synthesis and evaluation of mammary tumor inhibiting activity of 1,2-dialkyl-1,2-bis(3'-hydroxyphenyl)ethanes.
Topics: Animals; Antineoplastic Agents; Cell Line; Dose-Response Relationship, Drug; Estrogen Antagonists; Female; Hexestrol; Humans; Mammary Neoplasms, Experimental; Mice; Mice, Inbred Strains; Rats; Rats, Inbred Strains; Uterus | 1981 |
Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta.
Topics: Amino Acid Sequence; Animals; Female; Humans; Isomerism; Ligands; Male; Molecular Sequence Data; Rats; Receptors, Estrogen; RNA, Messenger; Tissue Distribution | 1997 |
Potent and selective steroidal inhibitors of 17beta-hydroxysteroid dehydrogenase type 7, an enzyme that catalyzes the reduction of the key hormones estrone and dihydrotestosterone.
Topics: 17-Hydroxysteroid Dehydrogenases; Androstane-3,17-diol; Androstanes; Biocatalysis; Cell Line; Dihydrotestosterone; Enzyme Inhibitors; Estradiol; Estrone; Humans; Inhibitory Concentration 50; Oxidation-Reduction; Substrate Specificity | 2009 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Developing structure-activity relationships for the prediction of hepatotoxicity.
Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes | 2010 |
A predictive ligand-based Bayesian model for human drug-induced liver injury.
Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Estrogens increase the number of thyrotropin-releasing hormone receptors on mammotropic cells in culture.
Topics: Cell Line; Diethylstilbestrol; Estradiol; Estrogens; Estrone; Prolactin; Receptors, Cell Surface; Receptors, Estrogen; Tamoxifen; Thyrotropin-Releasing Hormone | 1979 |
Effects of estrone, estradiol, and estriol on hormone-responsive human breast cancer in long-term tissue culture.
Topics: Binding, Competitive; Breast Neoplasms; Cell Nucleus; Culture Techniques; Cytoplasm; Drug Interactions; Estradiol; Estriol; Estrone; Humans; Receptors, Estrogen; Serine; Tamoxifen; Thymidine | 1977 |
Tamoxifen (antiestrogen) therapy in advanced breast cancer.
Topics: Adult; Aged; Breast Neoplasms; Estradiol; Estrone; Female; Humans; Menopause; Middle Aged; Neoplasm Metastasis; Prolactin; Receptors, Estrogen; Tamoxifen | 1977 |
[Aminoglutethimide and aminoglutethimide+tamoxifen treatment for advanced breast cancer].
Topics: Administration, Oral; Adult; Aged; Aged, 80 and over; Aminoglutethimide; Androstenedione; Breast Neoplasms; Drug Evaluation; Drug Therapy, Combination; Estrone; Female; Humans; Middle Aged; Survival Rate; Tamoxifen | 1992 |
Superinduction of c-fos gene expression by estrogen in cultured guinea-pig endometrial cells requires priming by a cycloheximide-dependent mechanism.
Topics: Androstenedione; Animals; Cells, Cultured; Cycloheximide; Diethylstilbestrol; Endometrium; Estradiol; Estriol; Estrone; Female; Gene Expression; Genes, fos; Guinea Pigs; Hydrocortisone; Kinetics; RNA, Messenger; Tamoxifen; Testosterone; Transcription, Genetic | 1992 |
Tamoxifen and partial oestrogen agonism in postmenopausal women.
Topics: Aged; Breast Neoplasms; Estradiol; Estrogens; Estrone; Female; Follicle Stimulating Hormone; Humans; Hydrogen-Ion Concentration; Luteinizing Hormone; Menopause; Tamoxifen; Vagina | 1991 |
Characteristics of the biphasic action of androgens and of the potent antiproliferative effects of the new pure antiestrogen EM-139 on cell cycle kinetic parameters in LNCaP human prostatic cancer cells.
Topics: Androgens; Androstane-3,17-diol; Binding, Competitive; Cell Cycle; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Antagonism; Estradiol; Estrogen Antagonists; Estrone; Flow Cytometry; Flutamide; Humans; In Vitro Techniques; Male; Metribolone; Piperidines; Prostatic Neoplasms; Raloxifene Hydrochloride; Tamoxifen; Testosterone; Time Factors; Tumor Cells, Cultured | 1991 |
The effect of adjuvant therapy with or without tamoxifen on the endocrine function of patients with breast cancer.
Topics: Aged; Antibiotics, Antineoplastic; Breast Neoplasms; Cyclophosphamide; Drug Evaluation; Drug Therapy, Combination; Estradiol; Estrone; Female; Follicle Stimulating Hormone; Gonadotropins; Humans; Luteinizing Hormone; Middle Aged; Progesterone; Tamoxifen | 1990 |
Effect of CGS 16949A plus tamoxifen on induced mammary tumours in rats.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Animals; Antineoplastic Combined Chemotherapy Protocols; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Estrone; Fadrozole; Female; Follicle Stimulating Hormone; Imidazoles; Luteinizing Hormone; Mammary Neoplasms, Experimental; Nitriles; Prolactin; Rats; Rats, Inbred Strains; Tamoxifen | 1990 |
17 beta-estradiol is the most active component of the conjugated estrogen mixture active on uremic bleeding by a receptor mechanism.
Topics: Animals; Clomiphene; Dose-Response Relationship, Drug; Estradiol; Estrogens, Conjugated (USP); Estrone; Hemorrhage; Male; Rats; Rats, Inbred Strains; Receptors, Estrogen; Tamoxifen; Uremia | 1990 |
Metabolism and biologic response of estrogen sulfates in hormone-dependent and hormone-independent mammary cancer cell lines. Effect of antiestrogens.
Topics: Breast Neoplasms; Estradiol; Estriol; Estrone; Female; Humans; Menstruation; Polyunsaturated Alkamides; Progesterone; Receptors, Progesterone; Tamoxifen; Tumor Cells, Cultured | 1990 |
Cyclic nucleotide phosphodiesterase activity in the quail oviduct: hormonal regulation and involvement in estrogen-induced growth.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Aging; Animals; Coturnix; Estradiol; Estriol; Estrogens; Estrone; Female; Kinetics; Oviducts; Tamoxifen | 1988 |
The effect of tamoxifen on the function and lifespan of the corpus luteum and on subsequent ovarian function.
Topics: 17-alpha-Hydroxyprogesterone; 20-alpha-Dihydroprogesterone; Adult; Corpus Luteum; Estradiol; Estrone; Female; Follicle Stimulating Hormone; Follow-Up Studies; Humans; Hydroxyprogesterones; Luteinizing Hormone; Menstruation; Progesterone; Prolactin; Tamoxifen | 1989 |
Zoladex: endocrine and therapeutic effects in post-menopausal breast cancer.
Topics: Adult; Aged; Aged, 80 and over; Breast Neoplasms; Buserelin; Estradiol; Estrone; Female; Goserelin; Humans; Menopause; Middle Aged; Tamoxifen | 1989 |
[Action of estradiol-17 beta, estrone sulfate and progesterone on the growth and differentiation of endometrial epithelial cells of the guinea pig in primary culture].
Topics: Animals; Cell Differentiation; Cell Division; Cells, Cultured; DNA; Endometrium; Epithelial Cells; Estradiol; Estrone; Female; Guinea Pigs; Progesterone; Sulfotransferases; Sulfurtransferases; Tamoxifen | 1989 |
Estrogen regulation of an eosinophil chemotactic factor in the immature rat uterus.
Topics: Animals; Biological Assay; Chemotactic Factors; Chemotaxis, Leukocyte; Eosinophils; Estradiol; Estriol; Estrogens; Estrone; Female; Peroxidase; Rats; Rats, Inbred Strains; Tamoxifen; Uterus | 1989 |
Tamoxifen prolongs luteal phase in premenopausal women but has no effect on the size of uterine fibroids.
Topics: Estrone; Female; Humans; Leiomyoma; Luteal Phase; Menopause; Pregnanediol; Progesterone; Sex Hormone-Binding Globulin; Tamoxifen; Uterine Neoplasms | 1989 |
Differences in the mechanism of the inhibitory actions of catecholestrogens, tamoxifen and high concentrations of estrogens on prolactin release by cultured rat pituitary tumor cells.
Topics: Animals; Dose-Response Relationship, Drug; Estradiol; Estrogen Antagonists; Estrogens, Catechol; Female; Hydroxyestrones; Pituitary Neoplasms; Prolactin; Rats; Rats, Inbred BUF; Secretory Rate; Tamoxifen; Tumor Cells, Cultured | 1987 |
Effect of tamoxifen and tamoxifen derivatives on the conversion of estrone-sulfate to estradiol in the R-27 cells, a tamoxifen-resistant line derived from MCF-7 human breast cancer cells.
Topics: Breast Neoplasms; Cell Line; Drug Resistance; Estradiol; Estrogens, Conjugated (USP); Estrone; Female; Humans; Kinetics; Tamoxifen; Tritium | 1988 |
Endocrine treatment of breast cancer: effects upon intratumoral estrone sulfate metabolism and peripheral steroid levels.
Topics: Aminoglutethimide; Breast Neoplasms; Danazol; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Drug Administration Schedule; Estrogens; Estrone; Female; Humans; Pregnadienes; Sex Hormone-Binding Globulin; Tamoxifen | 1986 |
The mechanism of hormone-sensitive breast cancer progression on antiestrogen therapy. Implications for treatment and protocol planning.
Topics: Adrenal Glands; Adrenalectomy; Adult; Aged; Breast Neoplasms; Castration; Dehydroepiandrosterone; Estradiol; Estrone; Female; Humans; Hypophysectomy; Middle Aged; Neoplasms, Hormone-Dependent; Receptors, Estrogen; Stimulation, Chemical; Tamoxifen | 1987 |
[Cancer of the breast, mechanism of action of anti-estrogens].
Topics: Breast Neoplasms; Cell Line, Transformed; Estradiol; Estrone; Neoplasms, Hormone-Dependent; Polyunsaturated Alkamides; Tamoxifen | 1988 |
Reversal of the antitumor effects of tamoxifen by progesterone in the 7,12-dimethylbenzanthracene-induced rat mammary carcinoma model.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Animals; Drug Interactions; Estradiol; Estrenes; Estrogens; Estrone; Mammary Neoplasms, Experimental; Mifepristone; Organ Size; Progesterone; Rats; Tamoxifen | 1987 |
[Serum estrone sulfate levels in patients with breast cancer].
Topics: Adult; Aged; Breast Neoplasms; Combined Modality Therapy; Estrone; Female; Humans; Kinetics; Menopause; Middle Aged; Postoperative Period; Radioimmunoassay; Reference Values; Tamoxifen | 1988 |
[Biological responses, ultrastructural changes and metabolism of estrone sulfate in line cells of human breast cancer: MCF-7].
Topics: Breast Neoplasms; Cell Line; Estrone; Female; Humans; Hydrolysis; Receptors, Progesterone; Tamoxifen | 1987 |
Effect of the anti-oestrogen tamoxifen on the development of renal cortical necrosis induced by oestrone + vasopressin administration in rats.
Topics: Animals; Cell Membrane; Epithelium; Estrone; Kidney Cortex; Kidney Cortex Necrosis; Lypressin; Male; Microscopy, Electron; Rats; Succinate Dehydrogenase; Tamoxifen | 1988 |
Effect of tamoxifen and tamoxifen derivatives on the conversion of estrone sulfate to estradiol in the MCF-7 mammary cancer cell line.
Topics: Breast Neoplasms; Cell Line; Estradiol; Estrone; Female; Humans; Tamoxifen; Tumor Cells, Cultured | 1988 |
Chemoendocrine therapy with prolonged estrogen priming in advanced breast cancer: endocrine pharmacokinetics and toxicity.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Estradiol; Estrone; Female; Fluorouracil; Humans; Kinetics; Leucovorin; Methotrexate; Middle Aged; Tamoxifen | 1987 |
Compared effects of oestrogens and oestrone sulphate on the epithelial cell surface of guinea-pig endometrium (in vivo and in vitro studies).
Topics: Animals; Endometrium; Epithelium; Estradiol; Estrogen Antagonists; Estrogens; Estrone; Female; Guinea Pigs; In Vitro Techniques; Microscopy, Electron, Scanning; Microvilli; Progesterone; Tamoxifen | 1987 |
Effects of pharmacological concentrations of estrogens on proliferation and cell cycle kinetics of human breast cancer cell lines in vitro.
Topics: Breast Neoplasms; Cell Cycle; Cell Division; Cell Line; Diethylstilbestrol; Estradiol; Estrogens; Estrone; Female; Humans; Receptors, Estrogen; Stereoisomerism; Tamoxifen | 1987 |
Conformational transitions of the estrogen receptor monomer. Effects of estrogens, antiestrogen, and temperature.
Topics: Animals; Diethylstilbestrol; Estradiol; Estrogen Antagonists; Estrogens; Estrone; Female; Kinetics; Mathematics; Protein Conformation; Rats; Receptors, Estrogen; Tamoxifen; Temperature | 1986 |
Role of aminoglutethimide in male breast cancer.
Topics: Aminoglutethimide; Breast Neoplasms; Drug Therapy, Combination; Estradiol; Estrone; Humans; Hydrocortisone; Lung Neoplasms; Male; Orchiectomy; Tamoxifen | 1986 |
Low-dose aminoglutethimide in treatment of advanced breast cancer.
Topics: Adrenal Glands; Aged; Aminoglutethimide; Breast Neoplasms; Castration; Dehydroepiandrosterone; Drug Evaluation; Estradiol; Estrone; Female; Humans; Middle Aged; Tamoxifen | 1984 |
Effects of tamoxifen on the serum levels of oestrogens and adrenocortical steroids in postmenopausal breast cancer patients.
Topics: Adrenal Cortex Hormones; Breast Neoplasms; Dehydroepiandrosterone; Estradiol; Estrogens; Estrone; Female; Humans; Hydrocortisone; Menopause; Tamoxifen | 1982 |
Inhibition of steroid sulfatase activity by danazol.
Topics: Aminoglutethimide; Breast Neoplasms; Carcinoma; Culture Techniques; Danazol; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Dihydrotestosterone; Estrogen Antagonists; Estrone; Female; Humans; Medroxyprogesterone; Medroxyprogesterone Acetate; Pregnadienes; Tamoxifen | 1984 |
Effects of adjuvant chemohormonal therapy on the ovarian and adrenal function of breast cancer patients.
Topics: Adrenal Cortex; Androstenedione; Antineoplastic Agents; Breast Neoplasms; Dehydroepiandrosterone; Drug Therapy, Combination; Estradiol; Estrone; Female; Follicle Stimulating Hormone; Humans; Luteinizing Hormone; Menstruation; Ovary; Prednisone; Sex Hormone-Binding Globulin; Tamoxifen | 1980 |
Effects of early tamoxifen treatment on hormonal content of 15-day quail embryo gonads.
Topics: Animals; Coturnix; Estradiol; Estrone; Female; Gonadal Steroid Hormones; Male; Ovary; Proteins; Quail; Tamoxifen; Testis; Testosterone | 1984 |
Interrelation between tumor cell proliferation and 17-fluoresceinated estrone binding following primary tumor removal, radiation, cyclophosphamide, or tamoxifen.
Topics: Animals; Cyclophosphamide; Estrone; Female; Fluorescent Dyes; Immunotherapy; Mammary Neoplasms, Experimental; Mice; Mice, Inbred Strains; Neoplasm Metastasis; Tamoxifen | 1983 |
The effect of sex steroids and hormonal contraceptives upon thymus and spleen on intact female rats.
Topics: Androgens; Animals; Clomiphene; Contraceptives, Oral; Contraceptives, Oral, Combined; Contraceptives, Oral, Hormonal; Diethylstilbestrol; Estradiol; Estriol; Estrogens; Estrone; Ethinyl Estradiol; Female; Gonadal Steroid Hormones; Progestins; Rats; Receptors, Estrogen; Spleen; Tamoxifen; Thymus Gland | 1983 |
Estradiol formation and estrogen receptors in breast tumor tissue: effects of tamoxifen on estrogen interconversions in breast tumor homogenate in vitro.
Topics: Breast Neoplasms; Estrone; Female; Humans; In Vitro Techniques; Receptors, Estrogen; Tamoxifen | 1984 |
Tamoxifen as a possible chemotherapeutic agent in endometrial adenocarcinoma.
Topics: Adenocarcinoma; Cells, Cultured; Estrone; Female; Follicle Stimulating Hormone; Humans; Luteinizing Hormone; Neoplasm Recurrence, Local; Receptors, Progesterone; Tamoxifen; Uterine Neoplasms | 1981 |
Different effects of oestradiol, oestriol, oestetrol and of oestrone on human breast cancer cells (MCF-7) in long term tissue culture.
Topics: Breast Neoplasms; Cell Division; Cell Line; Estetrol; Estradiol; Estriol; Estrone; Female; Humans; Levonorgestrel; Norgestrel; Progesterone; Receptors, Progesterone; Tamoxifen | 1981 |
Antiestrogen action in avian liver: the interaction of estrogens and antiestrogens in the regulation of apolipoprotein B synthesis.
Topics: Animals; Apolipoproteins; Apolipoproteins B; Chickens; Estradiol; Estradiol Congeners; Estriol; Estrogens; Estrone; Kinetics; Liver; Male; Nitromifene; Stilbenes; Tamoxifen | 1981 |
[Feminization of embryonic chicken testicle by diethylstilbestrol and antagonistic action of tamoxifen].
Topics: Androgen-Insensitivity Syndrome; Animals; Chick Embryo; Diethylstilbestrol; Estradiol; Estrogens; Estrone; Male; Tamoxifen; Testis | 1982 |
Specific binding and biological response of antiestrogens in the fetal uterus of the guinea pig.
Topics: Animals; Binding Sites; Binding, Competitive; Cytosol; Estradiol; Estrone; Female; Fetal Blood; Guinea Pigs; Nafoxidine; Organ Size; Pregnancy; Pyrrolidines; Receptors, Estrogen; Tamoxifen; Uterus | 1980 |
Induction of prostate specific antigen production by steroids and tamoxifen in breast cancer cell lines.
Topics: Blotting, Western; Breast Neoplasms; Chromatography, High Pressure Liquid; Estradiol; Estrone; Humans; Prostate-Specific Antigen; Steroids; Tamoxifen; Testosterone; Tumor Cells, Cultured | 1994 |
In vivo inhibition of oestrone sulphatase and dehydroepiandrosterone sulphatase by oestrone-3-O-sulphamate.
Topics: Animals; Arylsulfatases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estradiol; Estrone; Female; Fulvestrant; Liver; Mammary Neoplasms, Experimental; Rats; Rats, Wistar; Steryl-Sulfatase; Sulfatases; Tamoxifen; Time Factors | 1995 |
Influence of tamoxifen on sex hormones, gonadotrophins and sex hormone binding globulin in postmenopausal breast cancer patients.
Topics: Aged; Androgens; Breast Neoplasms; Estradiol; Estrogens; Estrone; Female; Follicle Stimulating Hormone; Gonadal Steroid Hormones; Gonadotropins, Pituitary; Humans; Luteinizing Hormone; Middle Aged; Postmenopause; Sex Hormone-Binding Globulin; Tamoxifen; Testosterone | 1995 |
Effect of tamoxifen, estradiol 17 beta on coenzymes NAD, NADPH and the metabolism of estradiol and estrone in rabbit uterus in vivo.
Topics: Animals; Estradiol; Estradiol Dehydrogenases; Estrone; Female; NAD; NADP; Rabbits; Tamoxifen; Uterus | 1993 |
Estradiol-induced down-regulation of estrogen receptor. Effect of various modulators of protein synthesis and expression.
Topics: Cycloheximide; Dactinomycin; Down-Regulation; Estradiol; Estrone; Half-Life; Humans; Intercalating Agents; Kinetics; Molecular Weight; Phosphoric Monoester Hydrolases; Protein Kinase Inhibitors; Protein Synthesis Inhibitors; Receptors, Estrogen; RNA, Messenger; Tamoxifen; Tritium; Tumor Cells, Cultured | 1994 |
Transformation of estrone, estradiol, and estrone sulfate in uterine and vaginal isolated cells of fetal guinea pig. Effect of various antiestrogens in the conversion of estrone sulfate to estradiol.
Topics: Animals; Cells, Cultured; Culture Media; DNA; Estradiol; Estrogen Antagonists; Estrone; Female; Guinea Pigs; Polyunsaturated Alkamides; Pregnancy; Tamoxifen; Uterus; Vagina | 1993 |
2-Phenylindoles with sulfur containing side chains. Estrogen receptor affinity, antiestrogenic potency, and antitumor activity.
Topics: Animals; Antineoplastic Agents, Hormonal; Breast Neoplasms; Cattle; Cell Division; Estradiol; Estrogen Antagonists; Estrone; Female; Fulvestrant; HeLa Cells; Humans; Indoles; Mammary Neoplasms, Experimental; Mice; Organ Size; Receptors, Estrogen; Sulfur; Tamoxifen; Transcriptional Activation; Tumor Cells, Cultured; Uterus; Vitellogenins | 1996 |
Activation of 17beta-estradiol and estrone by dimethyldioxirane and inhibition of rat liver nuclear and nucleolar RNA synthesis in vitro.
Topics: Animals; Cell Nucleolus; Cell Nucleus; Diethylstilbestrol; Epoxy Compounds; Estradiol; Estrone; Guanosine Monophosphate; Kinetics; Liver; Oxidation-Reduction; Rats; RNA; Tamoxifen | 1996 |
Estriol: a potent regulator of TNF and IL-6 expression in a murine model of endotoxemia.
Topics: Animals; Autoimmune Diseases; Cells, Cultured; Endotoxemia; Estradiol; Estriol; Estrogen Antagonists; Estrogens; Estrone; Female; Gene Expression Regulation; Humans; Incidence; Interleukin-6; Lipopolysaccharides; Macrophages, Peritoneal; Mice; Mice, Inbred BALB C; Mice, Inbred Strains; Mice, Mutant Strains; Polymerase Chain Reaction; RNA, Messenger; Tamoxifen; Tumor Necrosis Factor-alpha | 1996 |
Changes in serum estrogen levels in women during tamoxifen therapy.
Topics: Adult; Aged; Aged, 80 and over; Breast Neoplasms; Dehydroepiandrosterone; Estradiol; Estrogens; Estrone; Female; Humans; Menopause; Middle Aged; Prospective Studies; Tamoxifen | 1997 |
Probing the structure and function of the estrogen receptor ligand binding domain by analysis of mutants with altered transactivation characteristics.
Topics: Amino Acid Sequence; Animals; Cloning, Molecular; COS Cells; Estradiol; Estrogen Antagonists; Estrone; HSP90 Heat-Shock Proteins; Hydroxyestrones; Ligands; Molecular Sequence Data; Mutation; Nuclear Proteins; Polyunsaturated Alkamides; Receptors, Estrogen; Saccharomyces cerevisiae; Sequence Alignment; Tamoxifen; Transcriptional Activation | 1997 |
Comparative effects of 28-day treatment with the new anti-estrogen EM-800 and tamoxifen on estrogen-sensitive parameters in intact mice.
Topics: 17-Hydroxysteroid Dehydrogenases; Androstenedione; Animals; Atrophy; Benzopyrans; Drug Administration Schedule; Endometrium; Estradiol; Estrogen Antagonists; Estrone; Female; Mice; Mice, Inbred BALB C; Organ Size; Ovariectomy; Propionates; Receptors, Estrogen; Tamoxifen; Testosterone; Uterus; Vagina | 1997 |
Comparison of the effects of the antiestrogens EM-800 and tamoxifen on the growth of human breast ZR-75-1 cancer xenografts in nude mice.
Topics: Analysis of Variance; Animals; Antineoplastic Agents, Hormonal; Benzopyrans; Breast Neoplasms; Cell Division; Estrogen Antagonists; Estrone; Female; Humans; Mice; Mice, Nude; Ovariectomy; Propionates; Tamoxifen; Transplantation, Heterologous | 1998 |
Estrogen increases the permeability of the cultured human cervical epithelium by modulating cell deformability.
Topics: Actins; Cell Line; Cell Membrane Permeability; Cells, Cultured; Cervix Uteri; Chlorides; Diethylstilbestrol; Egtazic Acid; Epithelial Cells; Estradiol; Estriol; Estrogen Antagonists; Estrogens; Estrone; Female; Fulvestrant; Humans; Kinetics; Progesterone; Sodium; Tamoxifen | 1998 |
In vitro lipid peroxidation of LDL from postmenopausal cynomolgus macaques treated with female hormones.
Topics: Alkenes; alpha-Tocopherol; Amidines; Animals; Cholesterol, HDL; Copper; Estradiol; Estrogens, Conjugated (USP); Estrone; Female; gamma-Tocopherol; Lipid Peroxidation; Lipoproteins, LDL; Macaca fascicularis; Medroxyprogesterone Acetate; Molecular Weight; Multivariate Analysis; Tamoxifen | 1999 |
Estrogens induce apoptosis in mouse peritoneal macrophages.
Topics: Animals; Apoptosis; Cycloheximide; DNA Fragmentation; Estradiol; Estrogen Antagonists; Estrone; Female; Macrophages, Peritoneal; Mice; Protein Kinase C; Protein Synthesis Inhibitors; Staurosporine; Tamoxifen | 1997 |
Oestrogen and progesterone increase the levels of apoptosis induced by the human papillomavirus type 16 E2 and E7 proteins.
Topics: Apoptosis; DNA-Binding Proteins; Dose-Response Relationship, Drug; Estrogens; HeLa Cells; Humans; Hydroxyestrones; Indoles; Mifepristone; Oncogene Proteins, Viral; Papillomaviridae; Papillomavirus E7 Proteins; Progesterone; Receptors, Estrogen; Tamoxifen; Tumor Cells, Cultured | 2001 |
Estrogen and androgen influence hypothalamic AVP and CRF concentrations in fetal and adult sheep.
Topics: Androgens; Androstenedione; Animals; Arginine Vasopressin; Case-Control Studies; Corticotropin-Releasing Hormone; Estradiol; Estrogen Antagonists; Estrogens; Estrone; Female; Hypothalamus; Pregnancy; Sheep; Tamoxifen | 2001 |
Estrone, but not 17 beta-estradiol, attenuates kainate-induced seizures and toxicity in male mice.
Topics: Animals; Estradiol; Estrogen Antagonists; Estrone; Hippocampus; Immunity; Kainic Acid; Male; Mice; Neurons; Seizures; Tamoxifen | 2001 |
Regulation of sex hormone-binding globulin secretion in human hepatoma G2 cells.
Topics: Antineoplastic Agents, Hormonal; Carcinoma, Hepatocellular; Dose-Response Relationship, Drug; Estradiol; Estradiol Congeners; Estrone; Ethinyl Estradiol; Humans; Liver Neoplasms; Sex Hormone-Binding Globulin; Tamoxifen; Time Factors; Tumor Cells, Cultured | 2001 |
Comparison of the effects of EM-652 (SCH57068), tamoxifen, toremifene, droloxifene, idoxifene, GW-5638 and raloxifene on the growth of human ZR-75-1 breast tumors in nude mice.
Topics: Animals; Breast Neoplasms; Cell Division; Cell Size; Cinnamates; Endometrium; Epithelial Cells; Estrogen Antagonists; Estrone; Female; Humans; Kinetics; Mice; Mice, Nude; Neoplasm Transplantation; Ovariectomy; Piperidines; Raloxifene Hydrochloride; Stilbenes; Tamoxifen; Toremifene; Tumor Cells, Cultured | 2002 |
A proposed mechanism of tamoxifen in breast cancer prevention.
Topics: Animals; Anticarcinogenic Agents; Breast Neoplasms; DNA Adducts; Epoxy Compounds; Estradiol; Estrone; Female; Humans; Liver; Rats; RNA; Tamoxifen | 2002 |
Reversal of breast cancer resistance protein-mediated drug resistance by estrogen antagonists and agonists.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Breast Neoplasms; Cell Survival; Diethylstilbestrol; Drug Resistance, Neoplasm; Estrogen Antagonists; Estrogens; Estrone; Female; Humans; K562 Cells; Kinetics; Mitoxantrone; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Tamoxifen; Topotecan; Tumor Cells, Cultured | 2003 |
Calcifications in ovary and endometrium and their neoplasms.
Topics: Animals; Calcinosis; Chorionic Gonadotropin; Clomiphene; Dihydrotestosterone; Endometrial Neoplasms; Endometrium; Estradiol; Estrone; Female; Growth Hormone; Guinea Pigs; Hormones; Megestrol Acetate; Ovarian Neoplasms; Ovary; Prolactin; Tamoxifen; Testosterone | 2003 |
Anti-oxidant effects of estrogen reduce [Ca2+]i during metabolic inhibition.
Topics: 1,2-Dihydroxybenzene-3,5-Disulfonic Acid Disodium Salt; Animals; Antioxidants; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium-Transporting ATPases; Estriol; Estrogen Antagonists; Estrogens; Estrone; Male; Mice; Myocytes, Cardiac; Nifedipine; Sodium-Potassium-Exchanging ATPase; Tamoxifen; Testosterone | 2003 |
Tamoxifen does not prevent the mobilization of body lipids elicited by oleoyl-estrone.
Topics: Animals; Anti-Obesity Agents; Blood Glucose; Body Composition; Body Weight; Energy Intake; Energy Metabolism; Estradiol; Estrogen Antagonists; Estrone; Lipid Mobilization; Male; Oleic Acids; Rats; Rats, Wistar; Receptors, Estrogen; Tamoxifen; Triglycerides | 2004 |
Moderate coffee and alcohol consumption improves the estrogen metabolite profile in adjuvant treated breast cancer patients: a pilot study comparing pre- and post-operative levels.
Topics: Adjuvants, Pharmaceutic; Aged; Aged, 80 and over; Alcohol Drinking; Breast Neoplasms; Coffee; Cytochrome P-450 CYP1A2; Estrogen Antagonists; Estrogens; Female; Humans; Hydroxyestrones; Hydroxytestosterones; Middle Aged; Pilot Projects; Postoperative Period; Receptors, Estrogen; Tamoxifen | 2006 |
A novel steroidal selective steroid sulfatase inhibitor KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells in vitro and in animal models.
Topics: Administration, Oral; Animals; Breast Neoplasms; Cell Proliferation; Coumarins; Cricetinae; Disease Models, Animal; Enzyme Inhibitors; Estradiol; Estrogen Antagonists; Estrone; Female; Gene Expression Regulation, Enzymologic; Humans; Leukocytes; Methylnitrosourea; Molecular Structure; Rats; Rats, Sprague-Dawley; Receptors, Progesterone; Signal Transduction; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Tamoxifen; Tumor Cells, Cultured | 2007 |
Dietary fat, tamoxifen use and circulating sex hormones in postmenopausal breast cancer survivors.
Topics: Adult; Breast Neoplasms; Diet; Dietary Fats; Dietary Fats, Unsaturated; Estradiol; Estrogen Antagonists; Estrone; Female; Gonadal Steroid Hormones; Humans; Middle Aged; Neoplasm Staging; Postmenopause; Survivors; Tamoxifen; Testosterone | 2010 |
Breast ductal lavage for assessment of breast cancer biomarkers.
Topics: Adult; Aged; Analysis of Variance; Androstenedione; Antineoplastic Agents, Hormonal; Biomarkers, Tumor; Breast; Breast Neoplasms; Cathepsin D; Dehydroepiandrosterone; Epidermal Growth Factor; Estradiol; Estrone; Female; Humans; Immunoassay; Middle Aged; Postmenopause; Premenopause; Progesterone; Tamoxifen; Therapeutic Irrigation | 2010 |
Synthesis and biological evaluation of prodigiosene conjugates of porphyrin, estrone and 4-hydroxytamoxifen.
Topics: Cell Line, Tumor; Cell Proliferation; Cell Survival; Estrone; Humans; MCF-7 Cells; Molecular Structure; Neoplasms; Porphyrins; Prodigiosin; Tamoxifen | 2013 |
Phenytoin is an estrogen receptor α-selective modulator that interacts with helix 12.
Topics: Amino Acid Sequence; Anticonvulsants; Binding Sites; Binding, Competitive; Crystallography; Dose-Response Relationship, Drug; Estradiol; Estrogen Receptor alpha; Estrogen Receptor beta; Estrone; Gene Expression Regulation; Genes, Reporter; Humans; MCF-7 Cells; Molecular Docking Simulation; Molecular Sequence Data; Phenytoin; Protein Binding; Protein Structure, Secondary; Selective Estrogen Receptor Modulators; Tamoxifen; Transcription, Genetic; Transfection | 2015 |
Pharmacological relevance of endoxifen in a laboratory simulation of breast cancer in postmenopausal patients.
Topics: Aged; Antineoplastic Agents, Hormonal; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Cytochrome P-450 CYP2D6; Estradiol; Estrogen Receptor Modulators; Estrone; Female; Gene Expression Regulation, Neoplastic; Humans; MCF-7 Cells; Middle Aged; Postmenopause; Real-Time Polymerase Chain Reaction; Research Design; Tamoxifen | 2014 |
Evaluation and characterization of anti-estrogenic and anti-androgenic activities in soil samples along the Second Songhua River, China.
Topics: Androgen Antagonists; Biological Assay; China; Environmental Monitoring; Estrogens; Estrone; Receptors, Androgen; Rivers; Soil; Soil Pollutants; Tamoxifen; Water Pollutants, Chemical | 2015 |
Measurable Serum Estradiol and Estrone in Women 36-56 Years During Adjuvant Treatment With Aromatase Inhibitors for a Hormone Receptor-Positive Breast Cancer. Case Studies and Cross-sectional Study Using an Ultra-sensitive LC-MS/MS-Method.
Topics: Adult; Aromatase Inhibitors; Breast Neoplasms; Chromatography, Liquid; Cross-Sectional Studies; Estradiol; Estrogens; Estrone; Female; Gonadotropin-Releasing Hormone; Humans; Middle Aged; Retrospective Studies; Tamoxifen; Tandem Mass Spectrometry | 2023 |
Small change - big consequence: The impact of C15-C16 double bond in a D‑ring of estrone on estrogen receptor activity.
Topics: Breast Neoplasms; Cell Line, Tumor; Estradiol; Estrogen Receptor alpha; Estrone; Female; Fulvestrant; Humans; Molecular Docking Simulation; Receptors, Estrogen; Tamoxifen | 2023 |