Compounds > estrone
Page last updated: 2024-08-17

estrone and rifampin

estrone has been researched along with rifampin in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.76)18.7374
1990's0 (0.00)18.2507
2000's5 (29.41)29.6817
2010's10 (58.82)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Strassburg, CP; Tukey, RH1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Oliveri, V1
Bakke, P; Gulsvik, A; Lønning, PE; Olsen, B; Thorsen, T1
Breuer, H; Nocke-Finck, L; Reimers, D1
Ayrton, A; Friedberg, TH; Goh, LB; Morgan, P; Ross, J; Spears, KJ; Stenhouse, A; Ward, CJ; Wolf, CR1
Häusler, S; Schneiter, R; Stieger, B; Treiber, A1
Gui, C; Hagenbuch, B; Miao, Y; Mock, M; Stieger, B; Thompson, L; Wahlgren, B1
Ho, RH; Kim, RB; Meyer zu Schwabedissen, HE; Tirona, RG; Yip, CS1
Annaert, PP; Augustijns, PF; Baes, M; De Bruyn, T; Peeters, A; Sahi, J; Ye, ZW1
Blode, H; Kunz, M; Mellinger, U; Parke, S; Rohde, B; Zeun, S; Zimmermann, T1
Hong, M; Huang, J; Liu, X; Sun, Y; Zhan, K; Zhang, Z1
Hu, Y; Juréus, A; Juric, S; Lundquist, P; Sohlenius-Sternbeck, AK1

Reviews

4 review(s) available for estrone and rifampin

ArticleYear
Human UDP-glucuronosyltransferases: metabolism, expression, and disease.
    Annual review of pharmacology and toxicology, 2000, Volume: 40

    Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic

2000
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Toward the discovery and development of effective modulators of α-synuclein amyloid aggregation.
    European journal of medicinal chemistry, 2019, Apr-01, Volume: 167

    Topics: alpha-Synuclein; Amyloidogenic Proteins; Drug Discovery; Humans; Protein Aggregation, Pathological; Structure-Activity Relationship

2019

Trials

2 trial(s) available for estrone and rifampin

ArticleYear
[Effects of rifampicin on the menstrual cycle and on oestrogen excretion in patients taking oral contraceptives].
    Deutsche medizinische Wochenschrift (1946), 1973, Aug-11, Volume: 98, Issue:33

    Topics: Adolescent; Adult; Clinical Trials as Topic; Contraceptives, Oral; Estriol; Estrogens; Estrone; Ethambutol; Ethinyl Estradiol; Female; Humans; Isoniazid; Menstruation Disturbances; Pregnancy; Rifampin; Streptomycin; Tuberculosis, Pulmonary

1973
Evaluation of the effects of rifampicin, ketoconazole and erythromycin on the steady-state pharmacokinetics of the components of a novel oral contraceptive containing estradiol valerate and dienogest in healthy postmenopausal women.
    Contraception, 2012, Volume: 86, Issue:4

    Topics: Aged; Anti-Infective Agents; Biotransformation; Contraceptives, Oral, Combined; Contraceptives, Oral, Hormonal; Cross-Over Studies; Cytochrome P-450 CYP3A; Drug Combinations; Drug Interactions; Enzyme Induction; Erythromycin; Estradiol; Estrogen Replacement Therapy; Estrone; Female; Humans; Ketoconazole; Middle Aged; Nandrolone; Postmenopause; Rifampin

2012

Other Studies

11 other study(ies) available for estrone and rifampin

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Plasma levels of estradiol, estrone, estrone sulfate and sex hormone binding globulin in patients receiving rifampicin.
    Journal of steroid biochemistry, 1989, Volume: 33, Issue:4A

    Topics: Adult; Aged; Aged, 80 and over; Estradiol; Estrogens; Estrone; Female; Humans; Male; Middle Aged; Rifampin; Sex Hormone-Binding Globulin

1989
Directional trans-epithelial transport of organic anions in porcine LLC-PK1 cells that co-express human OATP1B1 (OATP-C) and MRP2.
    Biochemical pharmacology, 2005, Feb-01, Volume: 69, Issue:3

    Topics: Animals; Biological Transport; Epithelium; Estradiol; Estrone; Liver-Specific Organic Anion Transporter 1; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Rifampin; Swine; Transfection

2005
Bosentan is a substrate of human OATP1B1 and OATP1B3: inhibition of hepatic uptake as the common mechanism of its interactions with cyclosporin A, rifampicin, and sildenafil.
    Drug metabolism and disposition: the biological fate of chemicals, 2007, Volume: 35, Issue:8

    Topics: Animals; Aryl Hydrocarbon Hydroxylases; Biological Transport; Bosentan; CHO Cells; Cricetinae; Cricetulus; Cyclosporine; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dehydroepiandrosterone Sulfate; Drug Interactions; Enzyme Inhibitors; Estradiol; Estrone; Humans; Liver-Specific Organic Anion Transporter 1; Molecular Structure; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Piperazines; Purines; Pyrimidines; Rifampin; Sildenafil Citrate; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfonamides; Sulfones; Warfarin

2007
Effect of pregnane X receptor ligands on transport mediated by human OATP1B1 and OATP1B3.
    European journal of pharmacology, 2008, Apr-14, Volume: 584, Issue:1

    Topics: Animals; CHO Cells; Chromans; Clotrimazole; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Drug Interactions; Estradiol; Estrone; Humans; Kinetics; Ligands; Liver-Specific Organic Anion Transporter 1; Mifepristone; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Paclitaxel; Pregnane X Receptor; Receptors, Steroid; Rifampin; Solute Carrier Organic Anion Transporter Family Member 1B3; Thiazolidinediones; Transfection; Troglitazone; Xenobiotics

2008
Interplay between the nuclear receptor pregnane X receptor and the uptake transporter organic anion transporter polypeptide 1A2 selectively enhances estrogen effects in breast cancer.
    Cancer research, 2008, Nov-15, Volume: 68, Issue:22

    Topics: Breast; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Chromatin Immunoprecipitation; Constitutive Androstane Receptor; Dipeptides; Estrogens; Estrone; Female; Humans; Neoplasm Staging; Organic Anion Transporters; Pregnane X Receptor; Promoter Regions, Genetic; Pyridines; Receptors, Cytoplasmic and Nuclear; Receptors, Estrogen; Receptors, Steroid; Rifampin; RNA, Messenger; Transcription Factors

2008
Determination of OATP-, NTCP- and OCT-mediated substrate uptake activities in individual and pooled batches of cryopreserved human hepatocytes.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2011, Jul-17, Volume: 43, Issue:4

    Topics: 1-Methyl-4-phenylpyridinium; Adolescent; Adult; Biological Transport; Corticosterone; Cryopreservation; Digoxin; Estradiol; Estrone; Hepatocytes; Humans; Male; Membrane Transport Proteins; Middle Aged; Organic Anion Transporters; Organic Anion Transporters, Sodium-Dependent; Organic Anion Transporters, Sodium-Independent; Organic Cation Transport Proteins; Organic Cation Transporter 1; Prazosin; Rifampin; RNA, Messenger; Solute Carrier Organic Anion Transporter Family Member 1B3; Symporters; Taurocholic Acid

2011
Identification of multiple binding sites for substrate transport in bovine organic anion transporting polypeptide 1a2.
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:3

    Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Cattle; Estrone; HEK293 Cells; Humans; Hydrogen-Ion Concentration; Kinetics; Methotrexate; Organic Anion Transporters; Protein Structure, Secondary; Recombinant Proteins; Rifampin; Sulfobromophthalein; Taurocholic Acid; Transfection

2013
The utility of cold-preserved human hepatocytes in studies on cytochrome P450 induction and hepatic drug transport.
    Xenobiotica; the fate of foreign compounds in biological systems, 2013, Volume: 43, Issue:9

    Topics: Cell Culture Techniques; Cell Survival; Cells, Cultured; Cytochrome P-450 CYP3A; Estrone; Fluorobenzenes; Hepatocytes; Humans; Ipratropium; Liver; Organic Anion Transporters; Phenobarbital; Pyrimidines; Rifampin; RNA, Messenger; Rosuvastatin Calcium; Sulfonamides; Taurocholic Acid

2013