Page last updated: 2024-08-17

estrone and pitavastatin

estrone has been researched along with pitavastatin in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (55.56)29.6817
2010's4 (44.44)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Hirano, M; Maeda, K; Shitara, Y; Sugiyama, Y2
Hirano, M; Kusuhara, H; Maeda, K; Matsushima, S; Nozaki, Y; Sugiyama, Y1
Grime, K; Riley, RJ; Webborn, PJ1
Brun, ME; Funk, C; Grimm, HP; Kansy, M; Lavé, T; Poirier, A; Portmann, R; Senner, F1
Choi, MK; Choi, YL; Deng, JW; Shin, HJ; Shin, JG; Song, IS1
Owen, A; Riley, RJ; Soars, AC; Soars, MG; White, P; Williamson, B1

Reviews

1 review(s) available for estrone and pitavastatin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

8 other study(ies) available for estrone and pitavastatin

ArticleYear
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Contribution of OATP2 (OATP1B1) and OATP8 (OATP1B3) to the hepatic uptake of pitavastatin in humans.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 311, Issue:1

    Topics: Biological Transport; Blotting, Western; Cells, Cultured; Drug Interactions; Estrone; Hepatocytes; Humans; Liver; Liver-Specific Organic Anion Transporter 1; Organic Anion Transporters, Sodium-Independent; Quinolines; Sincalide; Sodium; Solute Carrier Organic Anion Transporter Family Member 1B3

2004
Involvement of BCRP (ABCG2) in the biliary excretion of pitavastatin.
    Molecular pharmacology, 2005, Volume: 68, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Bile; Cell Line; Dogs; Estrone; Humans; Male; Mice; Multidrug Resistance-Associated Protein 2; Neoplasm Proteins; Quinolines; Rats; Rats, Sprague-Dawley

2005
Drug-drug interaction between pitavastatin and various drugs via OATP1B1.
    Drug metabolism and disposition: the biological fate of chemicals, 2006, Volume: 34, Issue:7

    Topics: Cell Line; Cyclosporine; Drug Interactions; Estradiol; Estrone; Hepatocytes; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Kinetics; Liver-Specific Organic Anion Transporter 1; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Quinolines; Solute Carrier Organic Anion Transporter Family Member 1B3; Transfection

2006
Functional consequences of active hepatic uptake on cytochrome P450 inhibition in rat and human hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:8

    Topics: Animals; Atorvastatin; Cells, Cultured; Culture Media; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Diclofenac; Enzyme Inhibitors; Estrone; Hepatocytes; Heptanoic Acids; Humans; Hydroxylation; Liver; Midazolam; Pyrroles; Quinolines; Rats; Recombinant Proteins; Tritium

2008
Design, data analysis, and simulation of in vitro drug transport kinetic experiments using a mechanistic in vitro model.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:12

    Topics: Algorithms; Animals; Biological Transport, Active; CHO Cells; Computer Simulation; Cricetinae; Cricetulus; Diffusion; Estrone; Fatty Acids, Monounsaturated; Fluvastatin; Hepatocytes; Indoles; Kinetics; Male; Membranes, Artificial; Models, Biological; Naphthalenes; Oligopeptides; Organic Anion Transporters; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Piperidines; Quinolines; Rats; Rats, Wistar; Sincalide; Temperature; Terfenadine

2008
Differential effect of genetic variants of Na(+)-taurocholate co-transporting polypeptide (NTCP) and organic anion-transporting polypeptide 1B1 (OATP1B1) on the uptake of HMG-CoA reductase inhibitors.
    Xenobiotica; the fate of foreign compounds in biological systems, 2011, Volume: 41, Issue:1

    Topics: Animals; Atorvastatin; Estrone; Fluorobenzenes; Genetic Variation; Heptanoic Acids; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Liver-Specific Organic Anion Transporter 1; Oocytes; Organic Anion Transporters; Organic Anion Transporters, Sodium-Dependent; Pyrimidines; Pyrroles; Quinolines; Rosuvastatin Calcium; Sulfonamides; Symporters; Taurocholic Acid; Xenopus laevis

2011
Dissecting the relative contribution of OATP1B1-mediated uptake of xenobiotics into human hepatocytes using siRNA.
    Xenobiotica; the fate of foreign compounds in biological systems, 2013, Volume: 43, Issue:10

    Topics: Base Sequence; Cells, Cultured; Cytochrome P-450 CYP3A; Drug Interactions; Estrone; Female; Fluorobenzenes; Hepatocytes; Humans; Imidazoles; Liver-Specific Organic Anion Transporter 1; Male; Molecular Sequence Data; Organic Anion Transporters; Pyrimidines; Quinolines; RNA, Small Interfering; Rosuvastatin Calcium; Sulfonamides; Tetrazoles; Valine; Valsartan; Xenobiotics

2013