Page last updated: 2024-08-17

estrone and piperidines

estrone has been researched along with piperidines in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (25.00)18.2507
2000's5 (62.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
de Launoit, Y; Dufour, M; Labrie, F; Simard, J; Veilleux, R1
Eckhardt, U; Hagenbuch, B; Höchli, M; Landmann, L; Meier, PJ; Schroeder, A; Stieger, B; Tynes, R1
Candas, B; Couillard, S; Gutman, M; Labrie, C; Labrie, F; Roy, J1
Albain, KS; Anderson, J; Arneson, DW; Bacus, JW; Beenken, SW; Browne, D; Budd, GT; Burak, WE; Fabian, CJ; Fruehauf, JP; Ganz, PA; Grizzle, WE; Hyams, DM; Johnson, KA; Kimler, BF; Lagios, MD; Mayo, MS; O'Shaughnessy, JA; Sauter, ER; Tawfik, OW1
Heal, DJ1
Alemany, M; Cabot, C; Fernández-López, JA; Ferrer-Lorente, R1
Brun, ME; Funk, C; Grimm, HP; Kansy, M; Lavé, T; Poirier, A; Portmann, R; Senner, F1
Asahi, S; Ebihara, T; Kondo, T; Moriwaki, T; Moriya, Y; Tagawa, Y; Takeuchi, T1

Trials

1 trial(s) available for estrone and piperidines

ArticleYear
Breast cancer chemoprevention phase I evaluation of biomarker modulation by arzoxifene, a third generation selective estrogen receptor modulator.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2004, Aug-15, Volume: 10, Issue:16

    Topics: Anticarcinogenic Agents; Biopsy; Breast Neoplasms; Dose-Response Relationship, Drug; Estradiol; Estrone; Female; Hormones; Humans; Middle Aged; Patient Selection; Piperidines; Postmenopause; Reoperation; Selective Estrogen Receptor Modulators; Thiophenes

2004

Other Studies

7 other study(ies) available for estrone and piperidines

ArticleYear
Characteristics of the biphasic action of androgens and of the potent antiproliferative effects of the new pure antiestrogen EM-139 on cell cycle kinetic parameters in LNCaP human prostatic cancer cells.
    Cancer research, 1991, Oct-01, Volume: 51, Issue:19

    Topics: Androgens; Androstane-3,17-diol; Binding, Competitive; Cell Cycle; Dihydrotestosterone; Dose-Response Relationship, Drug; Drug Antagonism; Estradiol; Estrogen Antagonists; Estrone; Flow Cytometry; Flutamide; Humans; In Vitro Techniques; Male; Metribolone; Piperidines; Prostatic Neoplasms; Raloxifene Hydrochloride; Tamoxifen; Testosterone; Time Factors; Tumor Cells, Cultured

1991
Polyspecific substrate uptake by the hepatic organic anion transporter Oatp1 in stably transfected CHO cells.
    The American journal of physiology, 1999, Volume: 276, Issue:4

    Topics: Animals; Anion Transport Proteins; Carrier Proteins; CHO Cells; Cholic Acid; Cricetinae; Dehydroepiandrosterone Sulfate; Dipeptides; Estradiol; Estrone; Glycocholic Acid; HeLa Cells; Humans; Kinetics; Liver; Ochratoxins; Ouabain; Piperidines; Rats; Recombinant Proteins; Substrate Specificity; Sulfobromophthalein; Taurochenodeoxycholic Acid; Taurocholic Acid; Transfection; Xenopus laevis

1999
Comparison of the effects of EM-652 (SCH57068), tamoxifen, toremifene, droloxifene, idoxifene, GW-5638 and raloxifene on the growth of human ZR-75-1 breast tumors in nude mice.
    International journal of cancer, 2002, May-10, Volume: 99, Issue:2

    Topics: Animals; Breast Neoplasms; Cell Division; Cell Size; Cinnamates; Endometrium; Epithelial Cells; Estrogen Antagonists; Estrone; Female; Humans; Kinetics; Mice; Mice, Nude; Neoplasm Transplantation; Ovariectomy; Piperidines; Raloxifene Hydrochloride; Stilbenes; Tamoxifen; Toremifene; Tumor Cells, Cultured

2002
Obesity drug development - CBI's 2nd Annual Summit.
    IDrugs : the investigational drugs journal, 2006, Volume: 9, Issue:10

    Topics: Adipocytes; Animals; Anti-Obesity Agents; Cannabinoid Receptor Modulators; Disease Models, Animal; Drug Design; Estrone; Fatty Acids; Humans; Obesity; Oleic Acids; Oxidation-Reduction; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant

2006
Effects of combined oleoyl-estrone and rimonabant on overweight rats.
    Journal of pharmacological sciences, 2007, Volume: 104, Issue:2

    Topics: Animals; Anti-Obesity Agents; Appetite; Blood Glucose; Cholecystokinin; Cholesterol; Drug Synergism; Drug Therapy, Combination; Eating; Energy Metabolism; Estrone; Fatty Acids, Nonesterified; Ghrelin; Glucagon-Like Peptide 1; Insulin; Leptin; Male; Obesity; Oleic Acids; Overweight; Peptide Hormones; Piperidines; Pyrazoles; Rats; Rats, Wistar; Rimonabant; Triglycerides

2007
Design, data analysis, and simulation of in vitro drug transport kinetic experiments using a mechanistic in vitro model.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:12

    Topics: Algorithms; Animals; Biological Transport, Active; CHO Cells; Computer Simulation; Cricetinae; Cricetulus; Diffusion; Estrone; Fatty Acids, Monounsaturated; Fluvastatin; Hepatocytes; Indoles; Kinetics; Male; Membranes, Artificial; Models, Biological; Naphthalenes; Oligopeptides; Organic Anion Transporters; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Piperidines; Quinolines; Rats; Rats, Wistar; Sincalide; Temperature; Terfenadine

2008
Characterization of Transporters in the Hepatic Uptake of TAK-475 M-I, a Squalene Synthase Inhibitor, in Rats and Humans.
    Drug research, 2016, Volume: 66, Issue:6

    Topics: Animals; Carbon Radioisotopes; Cells, Cultured; Cyclosporine; Estrone; Farnesyl-Diphosphate Farnesyltransferase; Hepatocytes; Humans; Liver; Oxazepines; Piperidines; Rats

2016