Page last updated: 2024-08-17

estrone and ouabain

estrone has been researched along with ouabain in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19905 (31.25)18.7374
1990's3 (18.75)18.2507
2000's4 (25.00)29.6817
2010's4 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Baert, B; Beetens, J; Bodé, S; De Spiegeleer, B; Deconinck, E; Lambert, J; Slegers, G; Slodicka, M; Stoppie, P; Van Gele, M; Vander Heyden, Y1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Takagi, I1
Robinson, JD1
Atger, M; Baulieu, EE; Milgrom, E1
Hauser, G1
Alivisatos, SG; Deliconstantinos, G; Theodosiadis, GP1
Chiba, M; Geng, W; Hassen, AM; Lam, D; Pang, KS; Tan, E1
Ramirez, VD; Zheng, J1
Eckhardt, U; Hagenbuch, B; Höchli, M; Landmann, L; Meier, PJ; Schroeder, A; Stieger, B; Tynes, R1
Braun, EJ; Dudas, PL; Pelis, RM; Renfro, JL1
Abe, T; Goto, J; Hishinuma, T; Mano, N; Mikkaichi, T; Okada, M; Shimada, M; Sugie, M; Toyohara, T; Yamaguchi, H1

Reviews

1 review(s) available for estrone and ouabain

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Other Studies

15 other study(ies) available for estrone and ouabain

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Transdermal penetration behaviour of drugs: CART-clustering, QSPR and selection of model compounds.
    Bioorganic & medicinal chemistry, 2007, Nov-15, Volume: 15, Issue:22

    Topics: Anti-Inflammatory Agents; Cell Membrane Permeability; Cluster Analysis; Drug Evaluation, Preclinical; Humans; Models, Biological; Predictive Value of Tests; Quantitative Structure-Activity Relationship; Regression Analysis; Skin; Skin Absorption

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Effect of thyroid-stimulating hormone, estrogens and other thyroid-tropic substances in vitro on Na+, K+-activated ATP-ase of pig thyroid gland.
    The Japanese journal of physiology, 1968, Dec-15, Volume: 18, Issue:6

    Topics: Adenosine Triphosphatases; Animals; Cortisone; Depression, Chemical; Dexamethasone; Estradiol; Estriol; Estrogens; Estrone; Hexestrol; In Vitro Techniques; Iodides; Monoiodotyrosine; Ouabain; Potassium; Progesterone; Sodium; Swine; Testosterone; Thiocyanates; Thiouracil; Thiourea; Thyroid Gland; Thyrotropin

1968
Diethyl stilbestrol--mode of inhibition of the (Na + +K + )-dependent adenosine triphosphatase.
    Biochemical pharmacology, 1970, Volume: 19, Issue:5

    Topics: Adenosine Triphosphatases; Animals; Brain; Diethylstilbestrol; Estradiol; Estriol; Estrone; Hexestrol; Kinetics; Microsomes; Ouabain; Phenolphthaleins; Phloretin; Phosphoric Monoester Hydrolases; Potassium Chloride; Rats; Sodium Chloride

1970
Studies on estrogen entry into uterine cells and on estradiol-receptor complex attachment to the nucleus--is the entry of estrogen into uterine cells a protein-mediated process?
    Biochimica et biophysica acta, 1973, Sep-14, Volume: 320, Issue:2

    Topics: Animals; Binding Sites; Biological Transport; Cell Nucleus; Chromatography, Thin Layer; Cyanides; Cytosol; Dinitrophenols; Estradiol; Estriol; Estrone; Female; In Vitro Techniques; Iodoacetates; Kinetics; Oligomycins; Ouabain; Protein Binding; Rats; Receptors, Cell Surface; Sulfhydryl Reagents; Tritium; Uterus

1973
Myo-inositol transport in slices of rat kidney cortex. 3. Hormonal, metabolic, and efflux studies.
    Annals of the New York Academy of Sciences, 1969, Oct-17, Volume: 165, Issue:2

    Topics: Adenosine Triphosphate; Animals; Biological Transport, Active; Calcium; Carbon Dioxide; Carbon Isotopes; Castration; Cyanides; Dinitrophenols; Dogs; Estradiol; Estrone; Female; Glucose; Gonads; In Vitro Techniques; Inositol; Kidney; Kinetics; Magnesium; Male; Nitrogen; Ouabain; Oxaloacetates; Phlorhizin; Potassium; Rats; Sodium; Temperature; Tritium

1969
Specificity of binding of cholesterol, steroid hormones and other compounds in synaptosomal plasma membranes, and their effect on ouabain-sensitive ATPase.
    Biochimica et biophysica acta, 1981, May-20, Volume: 643, Issue:3

    Topics: 1-Octanol; Adenosine Triphosphatases; Animals; Binding Sites; Cholesterol; Dodecanol; Dogs; Estrone; Glycosides; Octanols; Ouabain; Progesterone; Synaptic Membranes; Testosterone

1981
Uptake of sulfate conjugates by isolated rat hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 1996, Volume: 24, Issue:7

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Biological Transport; Carrier Proteins; Choline; Estrogens, Conjugated (USP); Estrone; Harmine; Hymecromone; In Vitro Techniques; Liver; Male; Ouabain; Rats; Rats, Sprague-Dawley

1996
Rapid inhibition of rat brain mitochondrial proton F0F1-ATPase activity by estrogens: comparison with Na+, K+ -ATPase of porcine cortex.
    European journal of pharmacology, 1999, Feb-26, Volume: 368, Issue:1

    Topics: Animals; Brain; Cholesterol; Corticosterone; Dehydroepiandrosterone; Detergents; Diethylstilbestrol; Enzyme Inhibitors; Estrogens; Female; Hydroxyestrones; Microsomes; Mitochondria; Ouabain; Progesterone; Proton-Translocating ATPases; Rats; Rats, Sprague-Dawley; Sodium-Potassium-Exchanging ATPase; Solubility; Swine; Testosterone; Zeranol

1999
Polyspecific substrate uptake by the hepatic organic anion transporter Oatp1 in stably transfected CHO cells.
    The American journal of physiology, 1999, Volume: 276, Issue:4

    Topics: Animals; Anion Transport Proteins; Carrier Proteins; CHO Cells; Cholic Acid; Cricetinae; Dehydroepiandrosterone Sulfate; Dipeptides; Estradiol; Estrone; Glycocholic Acid; HeLa Cells; Humans; Kinetics; Liver; Ochratoxins; Ouabain; Piperidines; Rats; Recombinant Proteins; Substrate Specificity; Sulfobromophthalein; Taurochenodeoxycholic Acid; Taurocholic Acid; Transfection; Xenopus laevis

1999
Transepithelial urate transport by avian renal proximal tubule epithelium in primary culture.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 22

    Topics: Animals; Biological Transport, Active; Bromcresol Green; Carbon Radioisotopes; Chickens; Cimetidine; Cytochalasins; DNA Primers; Electric Impedance; Epithelium; Estrone; Glutarates; Hydrogen-Ion Concentration; Kidney Tubules, Proximal; Lithium; Membrane Potentials; Nocodazole; Organic Anion Transporters; Ouabain; p-Aminohippuric Acid; Probenecid; Reverse Transcriptase Polymerase Chain Reaction; Time Factors; Uric Acid

2005
Transport of estrone 3-sulfate mediated by organic anion transporter OATP4C1: estrone 3-sulfate binds to the different recognition site for digoxin in OATP4C1.
    Drug metabolism and pharmacokinetics, 2010, Volume: 25, Issue:3

    Topics: Animals; Binding, Competitive; Biological Transport; Cell Line; Chenodeoxycholic Acid; Cyclosporine; Digoxin; Dogs; Epithelial Cells; Estrone; Humans; Kidney; Organic Anion Transporters; Ouabain; Pharmacokinetics; Sulfobromophthalein; Triiodothyronine

2010