estrone-3-o-sulfamate has been researched along with topiramate in 3 studies
Studies (estrone-3-o-sulfamate) | Trials (estrone-3-o-sulfamate) | Recent Studies (post-2010) (estrone-3-o-sulfamate) | Studies (topiramate) | Trials (topiramate) | Recent Studies (post-2010) (topiramate) |
---|---|---|---|---|---|
89 | 0 | 15 | 3,197 | 557 | 1,329 |
Protein | Taxonomy | estrone-3-o-sulfamate (IC50) | topiramate (IC50) |
---|---|---|---|
Carbonic anhydrase 1 | Homo sapiens (human) | 0.25 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.8683 | |
Carbonic anhydrase 2 | Rattus norvegicus (Norway rat) | 1.4 | |
Carbonic anhydrase 4 | Bos taurus (cattle) | 0.054 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Casini, A; Montero, JL; Scozzafava, A; Supuran, CT; Vullo, D; Winum, JY | 1 |
Abbate, F; Casini, A; Ciattini, S; Coetzee, A; Scozzafava, A; Supuran, CT | 1 |
Alterio, V; De Simone, G; Di Fiore, A; Menchise, V; Pedone, C; Scozzafava, A; Supuran, CT | 1 |
3 other study(ies) available for estrone-3-o-sulfamate and topiramate
Article | Year |
---|---|
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
Topics: Antigens, Neoplasm; Arylsulfatases; Biomarkers, Tumor; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cytosol; Enzyme Inhibitors; Estrone; Humans; Membrane Proteins; Neoplasm Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids | 2003 |
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride.
Topics: Antipsychotic Agents; Binding Sites; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Crystallography, X-Ray; Humans; Isoenzymes; Sulpiride | 2004 |
Carbonic anhydrase inhibitors: stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II.
Topics: Antigens, Neoplasm; Antineoplastic Agents; Binding Sites; Biomarkers, Tumor; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cell Membrane Permeability; Crystallography, X-Ray; Humans; Isoenzymes; Models, Molecular; Molecular Structure; Protein Binding; Pyridinium Compounds; Quantitative Structure-Activity Relationship; Recombinant Proteins; Sulfonamides | 2005 |