estrone-3-o-sulfamate has been researched along with tibolone in 3 studies
| Studies (estrone-3-o-sulfamate) | Trials (estrone-3-o-sulfamate) | Recent Studies (post-2010) (estrone-3-o-sulfamate) | Studies (tibolone) | Trials (tibolone) | Recent Studies (post-2010) (tibolone) |
|---|---|---|---|---|---|
| 89 | 0 | 15 | 927 | 336 | 162 |
| Protein | Taxonomy | estrone-3-o-sulfamate (IC50) | tibolone (IC50) |
|---|---|---|---|
| Estrogen receptor | Homo sapiens (human) | 0.4333 | |
| Androgen receptor | Rattus norvegicus (Norway rat) | 0.113 | |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | 0.0907 | |
| Cytochrome P450 2C19 | Homo sapiens (human) | 3 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 3 (100.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| de Gooyer, ME; Ederveen, AG; Kleyn, GT; Kloosterboer, HJ; Smits, KC; Verheul, HA | 1 |
| Day, JM; Potter, BV; Purohit, A; Raobaikady, B; Reed, MJ | 1 |
| Parsons, MF; Purohit, A; Raobaikady, B; Reed, MJ | 1 |
3 other study(ies) available for estrone-3-o-sulfamate and tibolone
| Article | Year |
|---|---|
Tibolone: a compound with tissue specific inhibitory effects on sulfatase.
Topics: Animals; Antineoplastic Agents, Hormonal; Breast; Cell Line; Endometrium; Enzyme Inhibitors; Estrone; Female; Humans; Norpregnenes; Organ Specificity; Osteoblasts; Sulfatases; Tumor Cells, Cultured | 2001 |
The nature of inhibition of steroid sulphatase activity by tibolone and its metabolites.
Topics: Enzyme Inhibitors; Estrogen Replacement Therapy; Estrone; Female; Humans; Kinetics; Microsomes; Norpregnenes; Placenta; Pregnancy; Steryl-Sulfatase | 2005 |
Tibolone and its delta-4, 7alpha-methyl norethisterone metabolite are reversible inhibitors of human aromatase.
Topics: Aromatase; Aromatase Inhibitors; Dose-Response Relationship, Drug; Estrone; Humans; Models, Biological; Norethindrone; Norpregnenes; Time Factors; Tumor Cells, Cultured | 2007 |