Compounds > estrone-3-o-sulfamate
Page last updated: 2024-09-03

estrone-3-o-sulfamate and sulfamic acid

estrone-3-o-sulfamate has been researched along with sulfamic acid in 7 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)		Trials
(estrone-3-o-sulfamate)		Recent Studies (post-2010)
(estrone-3-o-sulfamate)		Studies
(sulfamic acid)		Trials
(sulfamic acid)		Recent Studies (post-2010) (sulfamic acid)
890153770191

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (71.43)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Casini, A; Montero, JL; Scozzafava, A; Supuran, CT; Vullo, D; Winum, JY1
Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, M2
Fujii, T; Iwashita, S; Koizumi, N; Nakagawa, T; Okada, M; Takegawa, S1
Chander, SK; Potter, BV; Purohit, A; Reed, MJ; Woo, LW1
Edwards, DR; Wolfenden, R1
Potter, BV; Thomas, MP1

Other Studies

7 other study(ies) available for estrone-3-o-sulfamate and sulfamic acid

ArticleYear
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antigens, Neoplasm; Arylsulfatases; Biomarkers, Tumor; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cytosol; Enzyme Inhibitors; Estrone; Humans; Membrane Proteins; Neoplasm Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids

2003
Novel inhibitors of the enzyme estrone sulfatase (ES).
    Bioorganic & medicinal chemistry letters, 2001, Mar-26, Volume: 11, Issue:6

    Topics: Alkanes; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Ketones; Mesylates; Sulfatases; Sulfonamides; Sulfonic Acids

2001
Acid dissociation constant, a potential physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES).
    Bioorganic & medicinal chemistry letters, 2001, Apr-09, Volume: 11, Issue:7

    Topics: Estrogens; Estrone; Inhibitory Concentration 50; Kinetics; Phenols; Structure-Activity Relationship; Sulfatases; Sulfonic Acids

2001
Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
    The Journal of steroid biochemistry and molecular biology, 2003, Volume: 87, Issue:2-3

    Topics: Animals; Biphenyl Compounds; Breast Neoplasms; Cell Line, Tumor; Enzyme Inhibitors; Estradiol; Estrogen Receptor alpha; Estrone; Female; Humans; Liver; Organ Size; Rats; Rats, Sprague-Dawley; Receptors, Estrogen; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Uterus

2003
The role of steroid sulphatase in regulating the oestrogenicity of oestrogen sulphamates.
    Biochemical and biophysical research communications, 2004, Sep-10, Volume: 322, Issue:1

    Topics: Animals; Coumarins; Drug Combinations; Estrogens; Estrone; Female; Homeostasis; Organ Size; Ovariectomy; Rats; Rats, Wistar; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids; Uterus

2004
Proton-in-flight mechanism for the spontaneous hydrolysis of N-methyl O-phenyl sulfamate: implications for the design of steroid sulfatase inhibitors.
    The Journal of organic chemistry, 2012, May-04, Volume: 77, Issue:9

    Topics: Arylsulfatases; Catalysis; Coumarins; Esters; Estrone; Hydrogen-Ion Concentration; Hydrolysis; Kinetics; Molecular Structure; Steryl-Sulfatase; Sulfonamides; Sulfonic Acids

2012
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators

2015