Page last updated: 2024-09-03

estrone-3-o-sulfamate and methazolamide

estrone-3-o-sulfamate has been researched along with methazolamide in 2 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)
Trials
(estrone-3-o-sulfamate)
Recent Studies (post-2010)
(estrone-3-o-sulfamate)
Studies
(methazolamide)
Trials
(methazolamide)
Recent Studies (post-2010) (methazolamide)
8901545623114

Protein Interaction Comparison

ProteinTaxonomyestrone-3-o-sulfamate (IC50)methazolamide (IC50)
Carbonic anhydrase 12Homo sapiens (human)0.02
Tyrosine-protein kinase ABL1Homo sapiens (human)0.014
Carbonic anhydrase 1Homo sapiens (human)0.0469
Carbonic anhydrase 2Homo sapiens (human)0.0347
Carbonic anhydrase 3Homo sapiens (human)0.02
Cathepsin BBos taurus (cattle)0.02
Dihydrofolate reductaseEscherichia coli K-120.014
Carbonic anhydrase 4Homo sapiens (human)0.0792
Carbonic anhydrase 6Homo sapiens (human)0.02
Cyclin-dependent kinase 2Homo sapiens (human)0.014
Carbonic anhydrase 5A, mitochondrialHomo sapiens (human)0.02
Carbonic anhydrase 7Homo sapiens (human)0.02
Carbonic anhydrase 9Homo sapiens (human)0.0158
Carbonic anhydrase 13Homo sapiens (human)0.02
Carbonic anhydrase 4Bos taurus (cattle)0.036
Carbonic anhydrase 14Homo sapiens (human)0.02
Carbonic anhydrase 5B, mitochondrialHomo sapiens (human)0.02

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Casini, A; Montero, JL; Scozzafava, A; Supuran, CT; Vullo, D; Winum, JY1
Abbate, F; Casini, A; Ciattini, S; Coetzee, A; Scozzafava, A; Supuran, CT1

Other Studies

2 other study(ies) available for estrone-3-o-sulfamate and methazolamide

ArticleYear
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antigens, Neoplasm; Arylsulfatases; Biomarkers, Tumor; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cytosol; Enzyme Inhibitors; Estrone; Humans; Membrane Proteins; Neoplasm Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids

2003
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with the antipsychotic drug sulpiride.
    Bioorganic & medicinal chemistry letters, 2004, Jan-19, Volume: 14, Issue:2

    Topics: Antipsychotic Agents; Binding Sites; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Crystallography, X-Ray; Humans; Isoenzymes; Sulpiride

2004