estrone-3-o-sulfamate has been researched along with letrozole in 2 studies
Studies (estrone-3-o-sulfamate) | Trials (estrone-3-o-sulfamate) | Recent Studies (post-2010) (estrone-3-o-sulfamate) | Studies (letrozole) | Trials (letrozole) | Recent Studies (post-2010) (letrozole) |
---|---|---|---|---|---|
89 | 0 | 15 | 2,612 | 612 | 1,602 |
Protein | Taxonomy | estrone-3-o-sulfamate (IC50) | letrozole (IC50) |
---|---|---|---|
Steryl-sulfatase | Homo sapiens (human) | 0.0009 | |
Aromatase | Homo sapiens (human) | 0.009 | |
Cytochrome P450 11B1, mitochondrial | Homo sapiens (human) | 2.62 | |
Cytochrome P450 11B2, mitochondrial | Homo sapiens (human) | 1.42 | |
Amine oxidase [flavin-containing] A | Rattus norvegicus (Norway rat) | 0.0009 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Acharya, KR; Chander, SK; Cozier, G; Jackson, T; Leonard, P; Potter, BV; Purohit, A; Putey, A; Reed, MJ; Woo, LW | 1 |
Potter, BV; Thomas, MP | 1 |
2 other study(ies) available for estrone-3-o-sulfamate and letrozole
Article | Year |
---|---|
Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template.
Topics: Animals; Aromatase Inhibitors; Biphenyl Compounds; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Female; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Rats; Rats, Wistar; Spectrometry, Mass, Electrospray Ionization; Steryl-Sulfatase; Structure-Activity Relationship; Triazoles | 2010 |
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators | 2015 |