Page last updated: 2024-09-03

estrone-3-o-sulfamate and ethoxzolamide

estrone-3-o-sulfamate has been researched along with ethoxzolamide in 3 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)
Trials
(estrone-3-o-sulfamate)
Recent Studies (post-2010)
(estrone-3-o-sulfamate)
Studies
(ethoxzolamide)
Trials
(ethoxzolamide)
Recent Studies (post-2010) (ethoxzolamide)
89015357394

Protein Interaction Comparison

ProteinTaxonomyestrone-3-o-sulfamate (IC50)ethoxzolamide (IC50)
Carbonic anhydrase 1Homo sapiens (human)0.0417
Carbonic anhydrase 2Homo sapiens (human)0.0023
Carbonic anhydrase 9Homo sapiens (human)0.0006

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Casini, A; Montero, JL; Scozzafava, A; Supuran, CT; Vullo, D; Winum, JY1
Abbate, F; Casini, A; Montero, JL; Potter, BV; Scozzafava, A; Supuran, CT; Winum, JY1
Cavdar, H; Durdagi, S; Ekinci, D; Sentürk, M; Supuran, CT; Talaz, O1

Other Studies

3 other study(ies) available for estrone-3-o-sulfamate and ethoxzolamide

ArticleYear
Carbonic anhydrase inhibitors. Inhibition of cytosolic isozymes I and II and transmembrane, tumor-associated isozyme IX with sulfamates including EMATE also acting as steroid sulfatase inhibitors.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antigens, Neoplasm; Arylsulfatases; Biomarkers, Tumor; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase IX; Carbonic Anhydrases; Cytosol; Enzyme Inhibitors; Estrone; Humans; Membrane Proteins; Neoplasm Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids

2003
Carbonic anhydrase inhibitors: X-ray crystallographic structure of the adduct of human isozyme II with EMATE, a dual inhibitor of carbonic anhydrases and steroid sulfatase.
    Bioorganic & medicinal chemistry letters, 2004, Jan-05, Volume: 14, Issue:1

    Topics: Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Crystallography, X-Ray; Estrone; Humans; Isoenzymes; Steryl-Sulfatase

2004
Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI.
    European journal of medicinal chemistry, 2012, Volume: 49

    Topics: Animals; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Cattle; Humans; Indoles; Models, Molecular; Protein Isoforms; Structure-Activity Relationship

2012