Compounds > estrone-3-o-sulfamate
Page last updated: 2024-09-03

estrone-3-o-sulfamate and estrone sulfate

estrone-3-o-sulfamate has been researched along with estrone sulfate in 5 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)		Trials
(estrone-3-o-sulfamate)		Recent Studies (post-2010)
(estrone-3-o-sulfamate)		Studies
(estrone sulfate)		Trials
(estrone sulfate)		Recent Studies (post-2010) (estrone sulfate)
8901592670201

Protein Interaction Comparison

ProteinTaxonomyestrone-3-o-sulfamate (IC50)estrone sulfate (IC50)
Steryl-sulfataseHomo sapiens (human)7.6

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Boivin, RP; Labrie, F; Lachance, R; Luu-The, V; Poirier, D1
Dauvois, S; Parker, MG; Potter, BV; Purohit, A; Reed, MJ; Williams, GJ1
Hejaz, HA; Hummelinck, AE; Potter, BV; Purohit, A; Reed, MJ; Vernon, KA; Woo, LW1
Kabler, H; Li, PK; Sarap, J; Selcer, KW; Xiao, Z1
Fujii, T; Iwashita, S; Koizumi, N; Nakagawa, T; Okada, M; Takegawa, S1

Other Studies

5 other study(ies) available for estrone-3-o-sulfamate and estrone sulfate

ArticleYear
Structure-activity relationships of 17alpha-derivatives of estradiol as inhibitors of steroid sulfatase.
    Journal of medicinal chemistry, 2000, Nov-16, Volume: 43, Issue:23

    Topics: Arylsulfatases; Cell Line; Enzyme Inhibitors; Estradiol; Humans; Steryl-Sulfatase; Structure-Activity Relationship; Transfection

2000
The hydrolysis of oestrone sulphate and dehydroepiandrosterone sulphate by human steroid sulphatase expressed in transfected COS-1 cells.
    The Journal of steroid biochemistry and molecular biology, 1994, Volume: 50, Issue:1-2

    Topics: Animals; Arylsulfatases; Catalysis; Cell Line; Chlorocebus aethiops; Dehydroepiandrosterone; Dehydroepiandrosterone Sulfate; Estrogens, Conjugated (USP); Estrone; Female; Humans; Hydrolysis; Placenta; Steryl-Sulfatase; Transfection

1994
The development of A-ring modified analogues of oestrone-3-O-sulphamate as potent steroid sulphatase inhibitors with reduced oestrogenicity.
    The Journal of steroid biochemistry and molecular biology, 1998, Volume: 64, Issue:5-6

    Topics: Animals; Arylsulfatases; Breast Neoplasms; Enzyme Inhibitors; Estrone; Female; Microsomes; Molecular Structure; Organ Size; Ovariectomy; Placenta; Rats; Rats, Inbred Strains; Steryl-Sulfatase; Uterus

1998
Inhibition of steryl sulfatase activity in LNCaP human prostate cancer cells.
    Steroids, 2002, Volume: 67, Issue:10

    Topics: Arylsulfatases; Breast Neoplasms; Danazol; Dehydroepiandrosterone Sulfate; Enzyme Inhibitors; Estrone; Female; Humans; Kinetics; Male; Microsomes; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonamides; Tumor Cells, Cultured; Tyramine

2002
Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
    The Journal of steroid biochemistry and molecular biology, 2003, Volume: 87, Issue:2-3

    Topics: Animals; Biphenyl Compounds; Breast Neoplasms; Cell Line, Tumor; Enzyme Inhibitors; Estradiol; Estrogen Receptor alpha; Estrone; Female; Humans; Liver; Organ Size; Rats; Rats, Sprague-Dawley; Receptors, Estrogen; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Uterus

2003