Compounds > estrone-3-o-sulfamate

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estrone-3-o-sulfamate and 4-methylcoumarin 7-o-sulfamate

estrone-3-o-sulfamate has been researched along with 4-methylcoumarin 7-o-sulfamate in 16 studies

Compound Research Comparison

Studies (estrone-3-o-sulfamate)	Trials (estrone-3-o-sulfamate)	Recent Studies (post-2010) (estrone-3-o-sulfamate)	Studies (4-methylcoumarin 7-o-sulfamate)	Trials (4-methylcoumarin 7-o-sulfamate)	Recent Studies (post-2010) (4-methylcoumarin 7-o-sulfamate)
89	0	15	17	0	4

Protein Interaction Comparison

Protein	Taxonomy	estrone-3-o-sulfamate (IC50)	4-methylcoumarin 7-o-sulfamate (IC50)
Steryl-sulfatase	Homo sapiens (human)		0.5489

Research

Studies (16)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	2 (12.50)	18.2507
2000's	10 (62.50)	29.6817
2010's	3 (18.75)	24.3611
2020's	1 (6.25)	2.80

Authors

Authors	Studies
Potter, BV; Purohit, A; Reed, MJ; Woo, LW	1
Ahmed, S; James, K	1
Auer, M; Bilban, M; Billich, A; Nussbaumer, P	1
Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, M	2
Ahmed, S; James, K; Owen, CP; Patel, CK; Patel, MB	1
Ahmed, S; James, K; Owen, CP; Patel, CK; Sampson, L	1
Gräfe, U; Härtl, A; Heinisch, L; Jütten, P; Schumann, W; Ulbricht, H; Werner, W	1
Ahmed, S; James, K; Owen, CP; Patel, CK	1
Ahmed, S; James, K; Owen, CP	1
Ahmed, S; Owen, CP; Patel, CK	1
Cecchi, A; Hill, B; Liu, Y; Scozzafava, A; Supuran, CT; Taylor, SD; Vullo, D	1
Potter, BV; Thomas, MP	1
Daśko, M; Demkowicz, S; Kubiński, K; Masłyk, M; Misiak, M; Przybyłowska, M; Rachon, J; Składanowski, A	1
Abduelkarem, AR; Anbar, HS; El-Gamal, MI; Kobeissi, S; Mohammad, M; Ossama, A; Zaraei, SO	1
Biernacki, K; Ciupak, O; Daśko, M; Demkowicz, S; Kozak, W; Kubiński, K; Martyna, A; Masłyk, M; Nocentini, A; Rachon, J; Rak, J; Śliwka-Kaszyńska, M; Supuran, CT; Świtalska, M; Wietrzyk, J	1

Reviews

1 review(s) available for estrone-3-o-sulfamate and 4-methylcoumarin 7-o-sulfamate

Article	Year
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations. European journal of medicinal chemistry, 2019, Oct-01, Volume: 179 Topics: Anti-Bacterial Agents; Drug Discovery; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Sulfonic Acids	2019

Other Studies

15 other study(ies) available for estrone-3-o-sulfamate and 4-methylcoumarin 7-o-sulfamate

Article	Year
Active site directed inhibition of estrone sulfatase by nonsteroidal coumarin sulfamates. Journal of medicinal chemistry, 1996, Mar-29, Volume: 39, Issue:7 Topics: Binding Sites; Breast Neoplasms; Coumarins; Enzyme Inhibitors; Humans; Microsomes; Placenta; Sulfatases; Sulfonamides; Tumor Cells, Cultured	1996
Derivation of a possible transition-state for the reaction catalysed by the enzyme estrone Sulfatase (ES). Bioorganic & medicinal chemistry letters, 1999, Jun-21, Volume: 9, Issue:12 Topics: Binding Sites; Catalysis; Enzyme Inhibitors; Models, Molecular; Structure-Activity Relationship; Substrate Specificity; Sulfatases	1999
New fluorogenic substrate for the first continuous steroid sulfatase assay. Bioorganic & medicinal chemistry letters, 2000, May-01, Volume: 10, Issue:9 Topics: Arylsulfatases; Chemical Phenomena; Chemistry, Physical; Coumarins; Enzyme Inhibitors; Fluorescent Dyes; Fluorometry; Humans; Kinetics; Recombinant Proteins; Steryl-Sulfatase; Structure-Activity Relationship; Sulfatases	2000
Novel inhibitors of the enzyme estrone sulfatase (ES). Bioorganic & medicinal chemistry letters, 2001, Mar-26, Volume: 11, Issue:6 Topics: Alkanes; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Ketones; Mesylates; Sulfatases; Sulfonamides; Sulfonic Acids	2001
Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES). Bioorganic & medicinal chemistry letters, 2001, Sep-17, Volume: 11, Issue:18 Topics: Chemistry, Physical; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Models, Biological; Models, Chemical; Structure-Activity Relationship; Sulfatases; Sulfonamides	2001
Determination and use of a transition state for the enzyme estrone sulfatase (ES) from a proposed reaction mechanism. Bioorganic & medicinal chemistry letters, 2001, Dec-03, Volume: 11, Issue:23 Topics: Catalytic Domain; Coumarins; Enzyme Inhibitors; Estrone; Inhibitory Concentration 50; Models, Molecular; Protein Conformation; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids	2001
The mechanism of the irreversible inhibition of estrone sulfatase (ES) through the consideration of a range of methane- and amino-sulfonate-based compounds. Bioorganic & medicinal chemistry letters, 2002, May-06, Volume: 12, Issue:9 Topics: Enzyme Inhibitors; Methane; Sulfatases; Sulfonic Acids	2002
A novel type of nonsteroidal estrone sulfatase inhibitors. Bioorganic & medicinal chemistry letters, 2002, May-20, Volume: 12, Issue:10 Topics: Cytosine; Drug Design; Enzyme Inhibitors; Kinetics; Lactones; Naphthacenes; Purines; Quinones; Structure-Activity Relationship; Sulfatases	2002
Design, synthesis and biochemical evaluation of AC ring mimics as novel inhibitors of the enzyme estrone sulfatase (ES). Bioorganic & medicinal chemistry letters, 2002, May-20, Volume: 12, Issue:10 Topics: Coumarins; Drug Design; Enzyme Inhibitors; Kinetics; Models, Molecular; Molecular Conformation; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids	2002
Inhibition of estrone sulfatase (ES) by derivatives of 4-[(aminosulfonyl)oxy] benzoic acid. Bioorganic & medicinal chemistry letters, 2002, Sep-02, Volume: 12, Issue:17 Topics: Antineoplastic Agents; Benzoates; Humans; Hydrophobic and Hydrophilic Interactions; Inhibitory Concentration 50; Structure-Activity Relationship; Sulfatases	2002
Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acid. Bioorganic & medicinal chemistry letters, 2004, Feb-09, Volume: 14, Issue:3 Topics: Antineoplastic Agents; Benzoic Acid; Coumarins; Enzyme Inhibitors; Esters; Inhibitory Concentration 50; Structure-Activity Relationship; Sulfatases; Sulfonamides; Sulfonic Acids	2004
Carbonic anhydrase inhibitors: inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamides. Bioorganic & medicinal chemistry letters, 2005, Dec-01, Volume: 15, Issue:23 Topics: Antigens, Neoplasm; Carbonic Anhydrase I; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Carbonic Anhydrase IX; Carbonic Anhydrase V; Carbonic Anhydrases; Humans; Hydrocarbons, Fluorinated; Isoenzymes; Sulfonamides	2005
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health. Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19 Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators	2015
Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors. European journal of medicinal chemistry, 2017, Mar-10, Volume: 128 Topics: Breast Neoplasms; Coumarins; Enzyme Inhibitors; Female; Halogenation; Humans; Placenta; Pregnancy; Receptors, Estrogen; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonamides; Tumor Cells, Cultured	2017
Development of Sulfamoylated 4-(1-Phenyl-1 Journal of medicinal chemistry, 2022, 03-24, Volume: 65, Issue:6 Topics: Animals; Breast Neoplasms; Enzyme Inhibitors; Female; Humans; MCF-7 Cells; Mice; Phenol; Steryl-Sulfatase; Structure-Activity Relationship	2022