Page last updated: 2024-09-03

estrone-3-o-sulfamate and 2-methoxyestrone

estrone-3-o-sulfamate has been researched along with 2-methoxyestrone in 3 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)
Trials
(estrone-3-o-sulfamate)
Recent Studies (post-2010)
(estrone-3-o-sulfamate)
Studies
(2-methoxyestrone)
Trials
(2-methoxyestrone)
Recent Studies (post-2010) (2-methoxyestrone)
890154926

Protein Interaction Comparison

ProteinTaxonomyestrone-3-o-sulfamate (IC50)2-methoxyestrone (IC50)
17-beta-hydroxysteroid dehydrogenase type 1Homo sapiens (human)0.207

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hejaz, HA; Leese, MP; Mahon, MF; Newman, SP; Potter, BV; Purohit, A; Reed, MJ1
Cortés-Benítez, F; Dutour, R; Poirier, D; Roy, J1
MacCarthy-Morrogh, L; Packham, G; Purohit, A; Reed, MJ; Townsend, PA1

Other Studies

3 other study(ies) available for estrone-3-o-sulfamate and 2-methoxyestrone

ArticleYear
A-ring-substituted estrogen-3-O-sulfamates: potent multitargeted anticancer agents.
    Journal of medicinal chemistry, 2005, Aug-11, Volume: 48, Issue:16

    Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Estradiol; Estrone; Female; Humans; Mice; Molecular Structure; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Transplantation, Heterologous

2005
Targeting cytochrome P450 (CYP) 1B1 with steroid derivatives.
    Bioorganic & medicinal chemistry letters, 2016, 11-01, Volume: 26, Issue:21

    Topics: Cytochrome P-450 CYP1B1; Cytochrome P-450 Enzyme Inhibitors; Estrogens; Humans; Inhibitory Concentration 50; Molecular Docking Simulation; Structure-Activity Relationship

2016
Differential effects of estrone and estrone-3-O-sulfamate derivatives on mitotic. Arrest, apoptosis, and microtubule assembly in human breast cancer cells.
    Cancer research, 2000, Oct-01, Volume: 60, Issue:19

    Topics: Antineoplastic Agents; Apoptosis; Breast Neoplasms; Cell Cycle; Cell Division; Estrone; Humans; Hydroxyestrones; Microtubules; Mitosis; Tubulin; Tumor Cells, Cultured

2000