Page last updated: 2024-09-03

estrone-3-o-sulfamate and 2-ethylestradiol sulfamate

estrone-3-o-sulfamate has been researched along with 2-ethylestradiol sulfamate in 4 studies

Compound Research Comparison

Studies
(estrone-3-o-sulfamate)
Trials
(estrone-3-o-sulfamate)
Recent Studies (post-2010)
(estrone-3-o-sulfamate)
Studies
(2-ethylestradiol sulfamate)
Trials
(2-ethylestradiol sulfamate)
Recent Studies (post-2010) (2-ethylestradiol sulfamate)
890151305

Protein Interaction Comparison

ProteinTaxonomyestrone-3-o-sulfamate (IC50)2-ethylestradiol sulfamate (IC50)
Carbonic anhydrase 2Homo sapiens (human)0.29
Steryl-sulfataseHomo sapiens (human)1

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (50.00)29.6817
2010's2 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ho, Y; Potter, BV; Purohit, A; Reed, MJ; Robinson, J; Vicker, N; Woo, LL1
De Simone, G; Di Fiore, A; Leblond, B; Leese, MP; Newman, SP; Potter, BV; Purohit, A; Reed, MJ; Smith, A; Supuran, CT1
Potter, BV; Thomas, MP1
Abduelkarem, AR; Anbar, HS; El-Gamal, MI; Kobeissi, S; Mohammad, M; Ossama, A; Zaraei, SO1

Reviews

1 review(s) available for estrone-3-o-sulfamate and 2-ethylestradiol sulfamate

ArticleYear
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations.
    European journal of medicinal chemistry, 2019, Oct-01, Volume: 179

    Topics: Anti-Bacterial Agents; Drug Discovery; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Sulfonic Acids

2019

Other Studies

3 other study(ies) available for estrone-3-o-sulfamate and 2-ethylestradiol sulfamate

ArticleYear
Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II.
    Bioorganic & medicinal chemistry letters, 2003, Mar-10, Volume: 13, Issue:5

    Topics: Binding Sites; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Coumarins; Estrone; Humans; Inhibitory Concentration 50; Models, Molecular; Steroids; Structure-Activity Relationship; Substrate Specificity; Sulfatases; Sulfonamides; Sulfonic Acids

2003
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
    Journal of medicinal chemistry, 2006, Dec-28, Volume: 49, Issue:26

    Topics: Animals; Antineoplastic Agents; Binding Sites; Breast Neoplasms; Carbonic Anhydrase II; Carcinoma, Lewis Lung; Cell Proliferation; Crystallography, X-Ray; Estradiol; Female; Humans; Mice; Mice, Nude; Models, Molecular; Neovascularization, Pathologic; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Survival Rate; Tumor Cells, Cultured; Xenograft Model Antitumor Assays; Zinc

2006
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
    Journal of medicinal chemistry, 2015, Oct-08, Volume: 58, Issue:19

    Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators

2015