estrone-3-o-sulfamate has been researched along with 2-ethylestradiol sulfamate in 4 studies
| Studies (estrone-3-o-sulfamate) | Trials (estrone-3-o-sulfamate) | Recent Studies (post-2010) (estrone-3-o-sulfamate) | Studies (2-ethylestradiol sulfamate) | Trials (2-ethylestradiol sulfamate) | Recent Studies (post-2010) (2-ethylestradiol sulfamate) |
|---|---|---|---|---|---|
| 89 | 0 | 15 | 13 | 0 | 5 |
| Protein | Taxonomy | estrone-3-o-sulfamate (IC50) | 2-ethylestradiol sulfamate (IC50) |
|---|---|---|---|
| Carbonic anhydrase 2 | Homo sapiens (human) | 0.29 | |
| Steryl-sulfatase | Homo sapiens (human) | 1 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (50.00) | 29.6817 |
| 2010's | 2 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Ho, Y; Potter, BV; Purohit, A; Reed, MJ; Robinson, J; Vicker, N; Woo, LL | 1 |
| De Simone, G; Di Fiore, A; Leblond, B; Leese, MP; Newman, SP; Potter, BV; Purohit, A; Reed, MJ; Smith, A; Supuran, CT | 1 |
| Potter, BV; Thomas, MP | 1 |
| Abduelkarem, AR; Anbar, HS; El-Gamal, MI; Kobeissi, S; Mohammad, M; Ossama, A; Zaraei, SO | 1 |
1 review(s) available for estrone-3-o-sulfamate and 2-ethylestradiol sulfamate
| Article | Year |
|---|---|
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations.
Topics: Anti-Bacterial Agents; Drug Discovery; Gram-Positive Bacteria; Microbial Sensitivity Tests; Molecular Structure; Sulfonic Acids | 2019 |
3 other study(ies) available for estrone-3-o-sulfamate and 2-ethylestradiol sulfamate
| Article | Year |
|---|---|
Docking studies of sulphamate inhibitors of estrone sulphatase in human carbonic anhydrase II.
Topics: Binding Sites; Carbonic Anhydrase II; Carbonic Anhydrase Inhibitors; Coumarins; Estrone; Humans; Inhibitory Concentration 50; Models, Molecular; Steroids; Structure-Activity Relationship; Substrate Specificity; Sulfatases; Sulfonamides; Sulfonic Acids | 2003 |
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
Topics: Animals; Antineoplastic Agents; Binding Sites; Breast Neoplasms; Carbonic Anhydrase II; Carcinoma, Lewis Lung; Cell Proliferation; Crystallography, X-Ray; Estradiol; Female; Humans; Mice; Mice, Nude; Models, Molecular; Neovascularization, Pathologic; Steryl-Sulfatase; Structure-Activity Relationship; Sulfonic Acids; Survival Rate; Tumor Cells, Cultured; Xenograft Model Antitumor Assays; Zinc | 2006 |
Discovery and Development of the Aryl O-Sulfamate Pharmacophore for Oncology and Women's Health.
Topics: Animals; Antineoplastic Agents; Aromatase Inhibitors; Breast Neoplasms; Drug Discovery; Endometriosis; Estrone; Female; Humans; Male; Molecular Targeted Therapy; Prostatic Neoplasms; Steryl-Sulfatase; Sulfonic Acids; Tubulin Modulators | 2015 |