eseroline has been researched along with naloxone in 8 studies
Studies (eseroline) | Trials (eseroline) | Recent Studies (post-2010) (eseroline) | Studies (naloxone) | Trials (naloxone) | Recent Studies (post-2010) (naloxone) |
---|---|---|---|---|---|
29 | 0 | 1 | 20,134 | 1,257 | 3,321 |
Protein | Taxonomy | eseroline (IC50) | naloxone (IC50) |
---|---|---|---|
Cytochrome P450 2D6 | Homo sapiens (human) | 2 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 0.043 | |
Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0219 | |
Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0019 | |
Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0019 | |
Mu-type opioid receptor | Homo sapiens (human) | 0.0397 | |
Delta-type opioid receptor | Homo sapiens (human) | 0.1896 | |
Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.05 | |
Kappa-type opioid receptor | Homo sapiens (human) | 0.0795 | |
Mu-type opioid receptor | Mus musculus (house mouse) | 0.0154 | |
Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0089 | |
Beta-2 adrenergic receptor | Cavia porcellus (domestic guinea pig) | 0.0055 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (87.50) | 18.7374 |
1990's | 1 (12.50) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Brossi, A; Flippen-Anderson, JL; Gilardi, R; Jacobson, AE; Klee, WA; Schönenberger, B; Streaty, R | 1 |
Bartolini, A; Bartolini, R; Galli, A; Malmberg-Aiello, P; Renzi, G | 1 |
Liu, WF | 1 |
Bartolini, A; Conte, B; Giuliani, S; Maggi, CA; Meli, A; Patacchini, R; Santicioli, P | 1 |
Biella, G; Braga, PC; Fraschini, F; Tiengo, M | 1 |
Biella, G; Braga, PC; Dall'Oglio, G; Fraschini, F; Tiengo, M | 1 |
Aiello-Malmberg, P; Bartolini, A; Bartolini, R; Friedmann, T; Fürst, S; Galli, A; Knoll, J; Somogyi, GT | 1 |
Elliott, J; Jhamandas, K; Sutak, M | 1 |
8 other study(ies) available for eseroline and naloxone
Article | Year |
---|---|
Comparison of (-)-eseroline with (+)-eseroline and dihydroseco analogues in antinociceptive assays: confirmation of rubreserine structure by X-ray analysis.
Topics: Adenylyl Cyclase Inhibitors; Analgesics; Animals; In Vitro Techniques; Indoles; Physostigmine; Rats; Receptors, Opioid; Stereoisomerism; Structure-Activity Relationship; X-Ray Diffraction | 1986 |
Inhibition of [3H]naloxone binding in homogenates of rat brain by eseroline, a drug, with analgesic activity, related to physostigmine.
Topics: Analgesics; Animals; Binding, Competitive; Brain; In Vitro Techniques; Indoles; Kinetics; Naloxone; Physostigmine; Rats; Receptors, Opioid | 1979 |
Effect of eseroline on schedule-controlled behavior in the rat.
Topics: Analgesics; Animals; Atropine; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Indoles; Male; Naloxone; Rats; Rats, Inbred Strains; Reinforcement Schedule; Time Factors | 1991 |
Opioid-like action of eseroline on micturition reflex in rats.
Topics: Acetylcholine; Analgesics, Opioid; Animals; Atropine; Cholinesterase Inhibitors; Electric Stimulation; Indoles; Male; Morphine; Naloxone; Rats; Rats, Inbred Strains; Urinary Bladder; Urination | 1989 |
Eseroline depresses the responses of dorsal horn neurons to C-fiber afferents in the spinal rat.
Topics: Action Potentials; Analgesics, Opioid; Animals; Indoles; Male; Morphine; Naloxone; Nerve Fibers; Rats; Rats, Inbred Strains; Spinal Cord; Spinothalamic Tracts | 1986 |
Inhibitory effect of eseroline, an opiate like drug, on the rat nociceptive thalamic neurons activated by peripheral noxious stimuli.
Topics: Analgesics, Opioid; Animals; Electric Conductivity; Hot Temperature; Indoles; Male; Naloxone; Neurons; Nociceptors; Pain; Physical Stimulation; Rats; Rats, Inbred Strains; Thalamus | 1984 |
Direct evidence that eseroline possesses morphine-like effects.
Topics: Acetylcholine; Animals; Catalepsy; Cats; Female; Guinea Pigs; Humans; In Vitro Techniques; Indoles; Male; Morphine; Muscle Contraction; Muscles; Naloxone; Nociceptors; Rats; Receptors, Opioid; Sleep | 1982 |
Opiatelike actions of eseroline, an eserine derivative.
Topics: Acetylcholine; Analgesics; Animals; Catalepsy; Cerebral Cortex; Guinea Pigs; Humans; Indoles; Male; Muscle Contraction; Naloxone; Narcotics; Rats | 1981 |