Page last updated: 2024-09-03

es 242-1 and n-methylaspartate

es 242-1 has been researched along with n-methylaspartate in 2 studies

Compound Research Comparison

Studies (es 242-1)	Trials (es 242-1)	Recent Studies (post-2010) (es 242-1)	Studies (n-methylaspartate)	Trials (n-methylaspartate)	Recent Studies (post-2010) (n-methylaspartate)
5	0	0	10,408	59	1,902

Protein Interaction Comparison

Protein	Taxonomy	n-methylaspartate (IC50)
Glutamate receptor ionotropic, NMDA 1	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 2A	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 2B	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 2C	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 2D	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 3B	Rattus norvegicus (Norway rat)	5.175
Glutamate receptor ionotropic, NMDA 3A	Rattus norvegicus (Norway rat)	5.175

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	2 (100.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	0 (0.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Matsuda, Y; Nonaka, H; Nozawa, M; Toki, S; Tsukuda, E; Yoshida, M	1
Matsuda, Y; Nozawa, M; Toki, S; Tsukuda, E	1

Other Studies

2 other study(ies) available for es 242-1 and n-methylaspartate

Article	Year
The ES-242s, novel N-methyl-D-aspartate antagonists of microbial origin, interact with both the neurotransmitter recognition site and the ion channel domain. The Journal of biological chemistry, 1992, Jul-25, Volume: 267, Issue:21 Topics: Animals; Binding, Competitive; Biological Transport; Calcium; Cells, Cultured; Cyclic GMP; Dizocilpine Maleate; Hippocampus; Ion Channels; Kinetics; Mice; N-Methylaspartate; Neurons; Neurotransmitter Agents; Phencyclidine; Pipecolic Acids; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes	1992
Effects of a novel N-methyl-D-aspartate (NMDA) receptor antagonist, 3,3'-dimethyl-3,4,3',4'-tetrahydro-6,8,6',8'-tetramethoxy-[10,10' -bi-2- oxanthracene]-4,9,9'-(1H,1'H)-triol 4-acetate (ES-242-1), on NMDA-induced increases of intracellular Ca2+ concentr Biochemical pharmacology, 1994, Dec-16, Volume: 48, Issue:12 Topics: Animals; Calcium; Cells, Cultured; Dizocilpine Maleate; Hippocampus; Mice; N-Methylaspartate; Pyrans; Receptors, N-Methyl-D-Aspartate; Temperature	1994

Article

Year

The ES-242s, novel N-methyl-D-aspartate antagonists of microbial origin, interact with both the neurotransmitter recognition site and the ion channel domain.

The Journal of biological chemistry, 1992, Jul-25, Volume: 267, Issue:21

Topics: Animals; Binding, Competitive; Biological Transport; Calcium; Cells, Cultured; Cyclic GMP; Dizocilpine Maleate; Hippocampus; Ion Channels; Kinetics; Mice; N-Methylaspartate; Neurons; Neurotransmitter Agents; Phencyclidine; Pipecolic Acids; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes

1992

Effects of a novel N-methyl-D-aspartate (NMDA) receptor antagonist, 3,3'-dimethyl-3,4,3',4'-tetrahydro-6,8,6',8'-tetramethoxy-[10,10' -bi-2- oxanthracene]-4,9,9'-(1H,1'H)-triol 4-acetate (ES-242-1), on NMDA-induced increases of intracellular Ca2+ concentr

Biochemical pharmacology, 1994, Dec-16, Volume: 48, Issue:12

Topics: Animals; Calcium; Cells, Cultured; Dizocilpine Maleate; Hippocampus; Mice; N-Methylaspartate; Pyrans; Receptors, N-Methyl-D-Aspartate; Temperature

1994