es 242-1 has been researched along with dizocilpine maleate in 4 studies
| Studies (es 242-1) | Trials (es 242-1) | Recent Studies (post-2010) (es 242-1) | Studies (dizocilpine maleate) | Trials (dizocilpine maleate) | Recent Studies (post-2010) (dizocilpine maleate) |
|---|---|---|---|---|---|
| 5 | 0 | 0 | 7,741 | 9 | 1,449 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 3 (75.00) | 18.2507 |
| 2000's | 1 (25.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Matsuda, Y; Nonaka, H; Nozawa, M; Toki, S; Tsukuda, E; Yoshida, M | 1 |
| Ando, K; Kawamoto, I; Matsuda, Y; Sano, H; Toki, S; Yoshida, M | 1 |
| Matsuda, Y; Nozawa, M; Toki, S; Tsukuda, E | 1 |
| Goto, H; Hamada, F; Hamada, Y; Noutsuka, H | 1 |
4 other study(ies) available for es 242-1 and dizocilpine maleate
| Article | Year |
|---|---|
The ES-242s, novel N-methyl-D-aspartate antagonists of microbial origin, interact with both the neurotransmitter recognition site and the ion channel domain.
Topics: Animals; Binding, Competitive; Biological Transport; Calcium; Cells, Cultured; Cyclic GMP; Dizocilpine Maleate; Hippocampus; Ion Channels; Kinetics; Mice; N-Methylaspartate; Neurons; Neurotransmitter Agents; Phencyclidine; Pipecolic Acids; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes | 1992 |
ES-242-1, a novel compound from Verticillium sp., binds to a site on N-methyl-D-aspartate receptor that is coupled to the channel domain.
Topics: Animals; Bacteria; Binding, Competitive; Centrifugation; Chromatography, High Pressure Liquid; Chromatography, Thin Layer; Culture Techniques; Dizocilpine Maleate; Dose-Response Relationship, Drug; Fermentation; Kainic Acid; Ketamine; Mitosporic Fungi; Molecular Structure; Phencyclidine; Pyrans; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Soil Microbiology; Solubility; Synaptic Membranes | 1992 |
Effects of a novel N-methyl-D-aspartate (NMDA) receptor antagonist, 3,3'-dimethyl-3,4,3',4'-tetrahydro-6,8,6',8'-tetramethoxy-[10,10' -bi-2- oxanthracene]-4,9,9'-(1H,1'H)-triol 4-acetate (ES-242-1), on NMDA-induced increases of intracellular Ca2+ concentr
Topics: Animals; Calcium; Cells, Cultured; Dizocilpine Maleate; Hippocampus; Mice; N-Methylaspartate; Pyrans; Receptors, N-Methyl-D-Aspartate; Temperature | 1994 |
Comparison of the spinal anti-nociceptive effects of ES-242-1 and MK-801, two different NMDA antagonists, in rats.
Topics: Animals; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pain Threshold; Pyrans; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Time Factors | 2001 |