erythrosine has been researched along with verapamil in 68 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (4.41) | 18.7374 |
1990's | 19 (27.94) | 18.2507 |
2000's | 30 (44.12) | 29.6817 |
2010's | 15 (22.06) | 24.3611 |
2020's | 1 (1.47) | 2.80 |
Authors | Studies |
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Larsson, R; Nygren, P | 1 |
Allen, CN; Gray, TJ; Harpur, ES; Hirst, BH; Simmons, NL | 1 |
Durán, WN; Paul, J | 1 |
Fleming, JT; Joshua, IG; Miller, FN; Parekh, N | 1 |
Joyner, WL; Mayhan, WG | 1 |
Israeli, D; Senderoff, DM; Urken, ML; Weinberg, H; Zhang, WX | 1 |
Blom-Roosemalen, MC; Breimer, DD; de Boer, AG; Noach, AB; Sakai, M | 1 |
Ichimura, K; Kashiwagura, T; Kawahara, K; Koike, M; Matsui, W; Takeguchi, N | 1 |
Brezden, CB; Hedley, DW; Rauth, AM | 1 |
Holló, M; Homolya, L; Mechetner, EB; Müller, M; Sarkadi, B | 1 |
Loor, F; Tiberghien, F | 1 |
Fujita, T; Fukuzumi, M; Muranishi, S; Nishimaki, A; Yamada, H; Yamamoto, A | 1 |
Ford, PJ; Germann, UA; Harding, MW; Mason, VS; Shlyakhter, D | 1 |
Arttamangkul, S; Poot, M | 1 |
Bakos, E; Klein, I; Müller, M; Sarkadi, B; Szabó, K; Váradi, A; Welker, E | 1 |
Hauser, IA; Jakob, I; Lindemann, B; Thévenod, F | 1 |
Müller, M; Roninson, I; Sarkadi, B; Szabó, K; Váradi, A; Welker, E | 1 |
Hauser, IA; Hopfer, U; Koziolek, M; Thévenod, F | 1 |
Antal, F; Jakab, K; Sarkadi, B; Szakács, G | 1 |
Dagger, F; Essodaïgui, M; Frézard, F; Garnier-Suillerot, A; Moreira, ES | 1 |
Behnam-Motlagh, P; Grankvist, K; Henriksson, R; Jonsson, O; Persson, M | 1 |
Friedmann, JM; Hauser, IA; Katsen, AD; Thévenod, F | 1 |
Serrão, MP; Soares-Da-Silva, P | 1 |
Kamata, K; Maitani, Y; Nagai, T; Nakamura, K; Suenaga, H; Takayama, K | 1 |
Grand-Perret, T; Issandou, M | 1 |
Leitch, GJ; Scanlon, M; Shaw, A; Visvesvara, GS | 1 |
Balboni, G; Bryant, SD; Cooper, PS; Guerrini, R; Hardison, J; Lazarus, LH; Lovekamp, T; Salvadori, S | 1 |
Hamada, A; Nakano, M; Ohmura, T; Oyama, N; Shiraki, N; Tokunaga, J | 1 |
Bebawy, M; Morris, MB; Roufogalis, BD | 1 |
Anagnostopoulos, N; Androutsos, G; Galanopoulos, A; Kalmantis, T; Meletis, J; Paterakis, G; Rombos, Y; Sagriotis, A; Symeonidis, A; Tiniakou, M; Tsimberidou, AM; Yataganas, X; Zoumbos, N | 1 |
Andersson, U; Behnam-Motlagh, P; Bergenheim, AT; Grankvist, K; Hedman, H; Henriksson, R | 1 |
Pajeva, IK; Wiese, M | 1 |
Bartlett, MC; Clarke, DM; Loo, TW | 2 |
Litman, T; Skovsgaard, T; Stein, WD | 1 |
Bacchelli, B; Boraldi, F; Croce, MA; Garcia Fernandez, MI; Gheduzzi, D; Pasquali Ronchetti, I; Quaglino, D; Tiozzo, R | 1 |
Elliott, JI; Higgins, CF; Raguz, S | 1 |
Bailly, C; Cuevas, C; Kluza, J; Lansiaux, A; Otero, G; Tardy, C; Vanhuyse, M | 1 |
Frigieri, A; Huet, H; Huynh-Delerme, C; Kolf-Clauw, M; Noël, L | 1 |
Angelini, A; Baccante, G; Ciofani, G; Cuccurullo, F; Di Febbo, C; Di Ilio, C; Di Nisio, M; Porreca, E | 1 |
Foth, H; Glahn, F; Stehfest, E; Torky, A | 1 |
Ando, M; Bai, J; Dai, J; Hasegawa, T; Hirose, K; Kiuchi, M; Li, M; Nishizawa, S; Oka, S; Sakai, J; Tomida, A; Tsuruo, T | 1 |
Cole, B; Epel, D; Hamdoun, A; Thurber, RV | 1 |
Bubik, M; Fricker, G; Mahringer, A; Ott, M | 1 |
Ando, M; Bai, LM; Furuya, Y; Hasegawa, T; Kakuta, S; Kataoka, T; Li, N; Ogura, H; Sakai, J; Tomida, A; Tsuruo, T; Wang, LY; Wu, JL | 1 |
Baubichon-Cortay, H; Chang, XB; Di Pietro, A; Perrotton, T; Trompier, D | 1 |
Chen, YH; Lan, ZJ; Ning, BT; Qian, BQ; Shen, HQ; Tang, YM | 1 |
Gassner, B; Gekle, M; Kelleher, DK; Thews, O | 1 |
Brennan, NK; Detty, MR; Moore, TM; Raub, TJ; Sawada, GA; Tombline, G; William Higgins, J | 1 |
Abdel-Tawab, M; Fricker, G; Hummel, J; Kanzer, J; Krüger, P; Schubert-Zsilavecz, M | 1 |
Chatterjee, M; Mandal, G; Saha, P; Sarkar, A; Singh, N; Sundar, S | 1 |
Choy, E; Duan, Z; Hornicek, F; Mankin, H; Schwab, J; Susa, M; Yang, C | 1 |
Chattipakorn, N; Chattipakorn, S; Fucharoen, S; Kumfu, S; Settakorn, J; Srichairatanakool, S | 1 |
Chen, HY; Hsu, CY; Huang, FH; Huang, LY; Lai, PS; Shieh, MJ | 1 |
Bertelli, E; Dragoni, S; Franco, G; Frosini, M; Gori, M; Possidente, M; Teodori, E; Valoti, M | 1 |
Kuo, YC; Lu, CH | 1 |
Gabriel, S; Heinemann, U; Kovács, R; Raue, C | 1 |
Baba, K; Hamahata, Y; Iwanaga, K; Kakemi, M; Miyazaki, M; Shibano, M; Taniguchi, M; Yoneda, S | 1 |
Jakob, I; Molinas, A; Sicard, G | 1 |
de Araújo Leite, JC; Marques-Santos, LF; Santi-Gadelha, T; Silva-Neta, HL; Torrezan, E | 1 |
Chiou, MH; Hsieh, YW; Huang, CL; Hung, CC; Lane, HY; Teng, YN | 1 |
Bolzani, Vda S; Efferth, T; Fricker, G; Ishikawa, T; Kadioglu, O; Mitani, Y; Murase, H; Nakagawa, H; Regasini, LO; Satake, K; Tajima, Y; Tamura, A | 1 |
Abele, D; Bickmeyer, U; Dringen, R; Petters, C; Rivera-Ingraham, G; Tietje, K | 1 |
Achilli, TM; McCalla, S; Meyer, J; Morgan, JR; Tripathi, A | 1 |
Fukaki, H; Iida, H; Ishizaki, K; Kadohama, N; Kajiyama, T; Kambara, H; Mimura, T; Ohnishi, M; Shichijo, C; Suzuki, Y | 1 |
Vrzal, R | 1 |
Hung, CC; Lan, YH; Lin, KI; Lin, YC; Teng, YN; Thang, TD | 1 |
Boheim, G; Engelberth, J; Klüsener, B; Liss, H; Weiler, EW | 1 |
1 review(s) available for erythrosine and verapamil
Article | Year |
---|---|
Diagnostics of multidrug resistance in cancer.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport; Diagnosis; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Neoplasms; Neoplastic Stem Cells; Prostaglandins A; RNA, Messenger; RNA, Neoplasm; Verapamil | 1998 |
67 other study(ies) available for erythrosine and verapamil
Article | Year |
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Pharmacological modification of multi-drug resistance (MDR) in vitro detected by a novel fluorometric microculture cytotoxicity assay. Reversal of resistance and selective cytotoxic actions of cyclosporin A and verapamil on MDR leukemia T-cells.
Topics: Benzimidazoles; Cell Division; Cell Line; Cell Survival; Cyclosporins; Cytological Techniques; Dose-Response Relationship, Drug; Drug Resistance; Drug Screening Assays, Antitumor; Fluoresceins; Fluorescent Dyes; Fluorometry; Humans; Precursor Cell Lymphoblastic Leukemia-Lymphoma; T-Lymphocytes; Tumor Cells, Cultured; Verapamil; Vincristine | 1990 |
Efflux of bis-carboxyethyl-carboxyfluorescein (BCECF) by a novel ATP-dependent transport mechanism in epithelial cells.
Topics: Adenocarcinoma; Adenosine Triphosphate; Animals; Cell Line; Epithelium; Fluoresceins; Fluorescent Dyes; Humans; Indomethacin; Kinetics; Nifedipine; Reserpine; Verapamil; Vinblastine | 1990 |
Concentration dependent effects of calcium blockade on vessel diameter and microvascular macromolecular clearance.
Topics: Animals; Arteries; Arterioles; Dextrans; Dose-Response Relationship, Drug; Fluorescein-5-isothiocyanate; Fluoresceins; Macromolecular Substances; Male; Metabolic Clearance Rate; Permeability; Rats; Rats, Inbred WF; Vasodilation; Verapamil | 1989 |
Histamine-induced protein leakage in hypertensive rats: inhibition by verapamil.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Fluorescein-5-isothiocyanate; Fluoresceins; Heart Rate; Histamine; Hypertension, Renal; Male; Proteins; Rats; Rats, Inbred Strains; Serum Albumin; Thiocyanates; Verapamil | 1986 |
The effect of altering the external calcium concentration and a calcium channel blocker, verapamil, on microvascular leaky sites and dextran clearance in the hamster cheek pouch.
Topics: Animals; Calcium; Calcium Channel Blockers; Capillary Permeability; Cheek; Cricetinae; Dextrans; Endothelium; Fluorescein-5-isothiocyanate; Fluoresceins; Histamine; Male; Mesocricetus; Mouth Mucosa; Muscle, Smooth, Vascular; Verapamil | 1984 |
Enhancement of fluorescein perfusion in experimental skin flaps following postischemic washout with iloprost, urokinase, verapamil, and University of Wisconsin solution.
Topics: Adenosine; Allopurinol; Animals; Female; Fluorescein; Fluoresceins; Glutathione; Iloprost; Insulin; Ischemia; Organ Preservation Solutions; Perfusion; Raffinose; Rats; Rats, Sprague-Dawley; Skin; Surgical Flaps; Tissue Preservation; Urokinase-Type Plasminogen Activator; Verapamil | 1993 |
Absorption enhancement of hydrophilic compounds by verapamil in Caco-2 cell monolayers.
Topics: Biological Transport; Cell Line; Dextrans; Electric Impedance; Fluorescein; Fluorescein-5-isothiocyanate; Fluoresceins; Humans; Intestinal Absorption; Stereoisomerism; Trypan Blue; Verapamil | 1994 |
Inhibition of the multidrug efflux pump in isolated hepatocyte couplets by immunosuppressants FK506 and cyclosporine.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile Canaliculi; Cyclosporine; Daunorubicin; Drug Resistance; Fluoresceins; Fluorescent Dyes; Fura-2; Liver; Membrane Glycoproteins; Microscopy, Fluorescence; Progesterone; Rats; Signal Processing, Computer-Assisted; Tacrolimus; Verapamil; Vinblastine | 1993 |
Constitutive expression of P-glycoprotein as a determinant of loading with fluorescent calcium probes.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium; CHO Cells; Cricetinae; Cricetulus; Cyclosporine; Cytosol; Female; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; Indoles; Rhodamine 123; Rhodamines; Verapamil | 1994 |
A new method for a quantitative assessment of P-glycoprotein-related multidrug resistance in tumour cells.
Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Blotting, Western; Cell Membrane; Drug Resistance, Multiple; Flow Cytometry; Fluoresceins; Fluorometry; Humans; KB Cells; Leukemia P388; Leukemia, Erythroblastic, Acute; Mice; Multidrug Resistance-Associated Proteins; Neoplasms, Experimental; Verapamil | 1996 |
Ranking of P-glycoprotein substrates and inhibitors by a calcein-AM fluorometry screening assay.
Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Drug Screening Assays, Antitumor; Fluoresceins; Fluorescent Dyes; Humans; Mice; Peptides, Cyclic; Tumor Cells, Cultured; Verapamil; Vinblastine | 1996 |
Calcein is excreted from the intestinal mucosal cell membrane by the active transport system.
Topics: Animals; Azides; Biological Transport, Active; Caco-2 Cells; Calcium Channel Blockers; Cell Membrane; Cell Membrane Permeability; Daunorubicin; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Humans; In Vitro Techniques; Intestinal Mucosa; Jejunum; Probenecid; Rats; Renal Agents; Sodium Azide; Sodium Fluoride; Verapamil | 1997 |
Chemosensitization and drug accumulation effects of VX-710, verapamil, cyclosporin A, MS-209 and GF120918 in multidrug resistant HL60/ADR cells expressing the multidrug resistance-associated protein MRP.
Topics: Acridines; Affinity Labels; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Cyclosporine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Etoposide; Fluoresceins; HL-60 Cells; Humans; Isoquinolines; Multidrug Resistance-Associated Proteins; Piperidines; Pyridines; Quinolines; Tetrahydroisoquinolines; Tritium; Verapamil; Vincristine | 1997 |
Verapamil inhibition of enzymatic product efflux leads to improved detection of beta-galactosidase activity in lacZ-transfected cells.
Topics: 3T3 Cells; alpha-Galactosidase; Animals; beta-Galactosidase; Cell Line; Chloroquine; Chromatography, High Pressure Liquid; Fibroblasts; Flow Cytometry; Fluoresceins; Galactosides; Gene Expression; Lac Operon; Lysosomes; Mice; Substrate Specificity; Transfection; Verapamil | 1997 |
Characterization of the human multidrug resistance protein containing mutations in the ATP-binding cassette signature region.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Binding Sites; Calcium Channel Blockers; Consensus Sequence; DNA, Complementary; Drug Resistance, Multiple; Fluoresceins; Genetic Vectors; Humans; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Nucleopolyhedroviruses; Recombinant Fusion Proteins; Rhodamine 123; Rhodamines; Spodoptera; Structure-Activity Relationship; Valinomycin; Verapamil | 1997 |
MDR1 in taste buds of rat vallate papilla: functional, immunohistochemical, and biochemical evidence.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Connective Tissue Cells; Cyclosporine; Epithelial Cells; Female; Fluoresceins; Fluorescent Dyes; Immunoglobulin G; In Vitro Techniques; Kinetics; Male; Microscopy, Fluorescence; Rats; Rats, Sprague-Dawley; Tamoxifen; Taste Buds; Tongue; Verapamil | 1998 |
Drug-stimulated nucleotide trapping in the human multidrug transporter MDR1. Cooperation of the nucleotide binding domains.
Topics: Adenine Nucleotides; Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cyclosporine; Enzyme Inhibitors; Ethylmaleimide; Fluoresceins; Fluorouracil; Humans; Protein Binding; Recombinant Proteins; Verapamil | 1998 |
Therapeutic concentrations of cyclosporine A, but not FK506, increase P-glycoprotein expression in endothelial and renal tubule cells.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Line; Cyclosporine; Endothelium, Vascular; Fluoresceins; Fluorescent Dyes; Humans; Immunohistochemistry; Kidney Tubules; Kinetics; Rats; Tacrolimus; Verapamil | 1998 |
Energy-dependent efflux from Leishmania promastigotes of substrates of the mammalian multidrug resistance pumps.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; Biological Transport; Cyclic P-Oxides; Doxorubicin; Drug Resistance, Multiple; Energy Metabolism; Fluoresceins; Fluorescent Dyes; Leishmania; Nicotinic Acids; Phenothiazines; Tumor Cells, Cultured; Verapamil | 1999 |
Increase in doxorubicin cytotoxicity by carvedilol inhibition of P-glycoprotein activity.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Carbazoles; Carvedilol; Cell Division; Doxorubicin; Drug Synergism; Fluoresceins; Fluorescence; Free Radicals; Humans; Propanolamines; Pyrogallol; Tumor Cells, Cultured; Verapamil | 1999 |
Up-regulation of multidrug resistance P-glycoprotein via nuclear factor-kappaB activation protects kidney proximal tubule cells from cadmium- and reactive oxygen species-induced apoptosis.
Topics: Animals; Annexin A5; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cadmium; Cadmium Chloride; Calcium Channel Blockers; Cell Line; Cyclosporine; Cyclosporins; Enzyme Inhibitors; Fluoresceins; Kidney Tubules, Proximal; Kinetics; Necrosis; NF-kappa B; Oxidative Stress; Rats; Rats, Inbred WKY; Reactive Oxygen Species; Time Factors; Up-Regulation; Verapamil | 2000 |
Outward transfer of dopamine precursor L-3,4-dihydroxyphenylalanine (L-dopa) by native and human P-glycoprotein in LLC-PK(1) and LLC-GA5 col300 renal cells.
Topics: Animals; Antibodies, Monoclonal; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cell Line; Dopamine; Fluoresceins; Fluorescent Dyes; Humans; Kidney; Kinetics; Levodopa; LLC-PK1 Cells; Proteins; Rhodamine 123; Swine; Verapamil; Vinblastine | 2000 |
The enhancing effect of soybean-derived sterylglucoside and beta-sitosterol beta-D-glucoside on nasal absorption in rabbits.
Topics: Absorption; Administration, Intranasal; Animals; Area Under Curve; Biological Availability; Calcium; Calcium Channel Blockers; Cholestenes; Drug Carriers; Fluoresceins; Hypoglycemic Agents; Insulin; Liposomes; Male; Nasal Mucosa; Powders; Rabbits; Sitosterols; Verapamil | 2000 |
Multidrug resistance P-glycoprotein is not involved in cholesterol esterification.
Topics: Acridines; Anticholesteremic Agents; Atorvastatin; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cholesterol; Cholesterol Esters; DNA-Binding Proteins; Fluoresceins; Fluorescent Dyes; Heptanoic Acids; Humans; Isoquinolines; Kinetics; Multidrug Resistance-Associated Proteins; MutS Homolog 3 Protein; Probenecid; Progesterone; Pyrroles; Sterol O-Acyltransferase; Tetrahydroisoquinolines; Tumor Cells, Cultured; Verapamil | 2000 |
Role of P glycoprotein in the course and treatment of Encephalitozoon microsporidiosis.
Topics: Acquired Immunodeficiency Syndrome; Albendazole; Animals; Anthelmintics; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Cells, Cultured; Chlorocebus aethiops; Cyclosporine; Encephalitozoon; Encephalitozoonosis; Fluoresceins; Genes, MDR; Immunohistochemistry; Immunosuppressive Agents; Verapamil | 2001 |
Inhibition of human multidrug resistance P-glycoprotein 1 by analogues of a potent delta-opioid antagonist.
Topics: 3T3 Cells; Adamantane; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Dipeptides; Drug Resistance, Multiple; Fibroblasts; Fluoresceins; Humans; Mice; Narcotic Antagonists; Oligopeptides; Peptides, Cyclic; Receptors, Opioid, delta; Structure-Activity Relationship; Tetrahydroisoquinolines; Transfection; Verapamil | 2001 |
Increase in doxorubicin cytotoxicity by inhibition of P-glycoprotein activity with lomerizine.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Doxorubicin; Drug Resistance, Multiple; Fluoresceins; Humans; K562 Cells; Piperazines; Rhodamine 123; Verapamil | 2001 |
Selective modulation of P-glycoprotein-mediated drug resistance.
Topics: Allosteric Regulation; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Calcium Channel Blockers; Cell Division; Cell Membrane; Chlorpromazine; Colchicine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Membrane Lipids; Neoplasm Proteins; Phospholipids; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Temperature; Tumor Cells, Cultured; Verapamil; Vinblastine | 2001 |
Evaluation of the clinical relevance of the expression and function of P-glycoprotein, multidrug resistance protein and lung resistance protein in patients with primary acute myelogenous leukemia.
Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow Transplantation; Calcium Channel Blockers; Carbocyanines; Combined Modality Therapy; Cytarabine; Daunorubicin; Disease-Free Survival; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Female; Fluoresceins; Fluorescent Dyes; Genistein; Humans; Idarubicin; Immunophenotyping; Leukemia, Myeloid; Male; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; Prognosis; Prospective Studies; Rhodamine 123; Survival Analysis; Tumor Cells, Cultured; Vault Ribonucleoprotein Particles; Verapamil | 2002 |
Rapid induction of long-lasting drug efflux activity in brain vascular endothelial cells but not malignant glioma following irradiation.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Sub-Family B Member 4; ATP-Binding Cassette Transporters; Brain Neoplasms; Calcium Channel Blockers; DNA Primers; Drug Resistance, Neoplasm; Endothelium, Vascular; Fluoresceins; Glioma; Humans; Immunoenzyme Techniques; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Verapamil | 2002 |
Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).
Topics: Adenosine Triphosphatases; Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Binding, Competitive; Caco-2 Cells; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship; Radioligand Assay; Rhodamine 123; Stereoisomerism; Verapamil; Vinblastine | 2002 |
Methanethiosulfonate derivatives of rhodamine and verapamil activate human P-glycoprotein at different sites.
Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Calcium Channel Blockers; Cell Line; Colchicine; Cysteine; Disulfides; DNA, Complementary; Dose-Response Relationship, Drug; Fluoresceins; Fluorescent Dyes; Histidine; Humans; Mesylates; Models, Biological; Models, Chemical; Mutation; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary; Rhodamines; Verapamil | 2003 |
Pumping of drugs by P-glycoprotein: a two-step process?
Topics: Algorithms; Animals; Anti-Bacterial Agents; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Calcium Channel Blockers; Carcinoma, Ehrlich Tumor; Cell Line, Tumor; Cyclosporine; Daunorubicin; Fluoresceins; Humans; Immunosuppressive Agents; Kinetics; Models, Biological; Pharmaceutical Preparations; Quinolines; Verapamil; Vinblastine | 2003 |
Multidrug resistance protein-6 (MRP6) in human dermal fibroblasts. Comparison between cells from normal subjects and from Pseudoxanthoma elasticum patients.
Topics: Adult; Benzbromarone; Cell Count; Cell Division; Chlorambucil; Female; Fibroblasts; Fluoresceins; Fluorescent Dyes; Humans; Indomethacin; Lysosomes; Male; Membrane Transport Proteins; Microscopy, Fluorescence; Middle Aged; Multidrug Resistance-Associated Proteins; Propionates; Pseudoxanthoma Elasticum; Quinolines; Skin; Verapamil; Vinblastine | 2003 |
Multidrug transporter activity in lymphocytes.
Topics: Adrenergic alpha-Antagonists; Aniline Compounds; Animals; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; B-Lymphocytes; Calcium Channel Blockers; Fluoresceins; Fluorescent Dyes; Lymphocytes; Mice; Mice, Knockout; Mitoxantrone; Multidrug Resistance-Associated Proteins; Paclitaxel; Prazosin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; T-Lymphocytes; Verapamil; Xanthenes | 2004 |
Lamellarin D: a novel pro-apoptotic agent from marine origin insensitive to P-glycoprotein-mediated drug efflux.
Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cell Cycle; Coumarins; DNA Topoisomerases, Type I; DNA Topoisomerases, Type II; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Fluoresceins; Heterocyclic Compounds, 4 or More Rings; Isoquinolines; Leukemia P388; Membrane Potentials; Mice; Mitochondria; Rhodamine 123; Topoisomerase I Inhibitors; Topoisomerase II Inhibitors; Verapamil | 2005 |
Increased functional expression of P-glycoprotein in Caco-2 TC7 cells exposed long-term to cadmium.
Topics: ATP Binding Cassette Transporter, Subfamily B; Benzimidazoles; Blotting, Western; Caco-2 Cells; Cadmium Poisoning; Calcium Channel Blockers; Cell Survival; DNA; Drug Resistance, Multiple; Electrophoresis, Agar Gel; Fluoresceins; Fluorescent Dyes; Humans; L-Lactate Dehydrogenase; Neutral Red; Tetrazolium Salts; Thiazoles; Verapamil | 2005 |
Inhibition of P-glycoprotein-mediated multidrug resistance by unfractionated heparin: a new potential chemosensitizer for cancer therapy.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Breast Neoplasms; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Fluoresceins; Heparin; Humans; Verapamil | 2005 |
Non-destructive micromethod for MRP1 functional assay in human lung tumor cells.
Topics: Acetylcysteine; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Buthionine Sulfoximine; Cell Culture Techniques; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluoresceins; Fluorescent Dyes; Fluorometry; Glutathione; Humans; Immunohistochemistry; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Propionates; Quinolines; Sensitivity and Specificity; Verapamil | 2006 |
Transmembrane segment 1 of human P-glycoprotein contributes to the drug-binding pocket.
Topics: Adenosine Triphosphatases; Amino Acid Sequence; Amino Acid Substitution; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Cell Line; Colchicine; Cricetinae; Cyclosporine; Demecolcine; Disulfides; Dithiothreitol; Fluoresceins; Flupenthixol; Humans; Mesylates; Point Mutation; Protein Structure, Tertiary; Verapamil; Vinblastine | 2006 |
A new taxoid from a callus culture of Taxus cuspidata as an MDR reversal agent.
Topics: Antineoplastic Agents, Phytogenic; Calcium Channel Blockers; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Fluoresceins; Humans; Taxoids; Taxus; Verapamil | 2006 |
The sea urchin embryo as a model for studying efflux transporters: roles and energy cost.
Topics: Animals; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Cyclosporins; Cytotoxins; Embryo, Nonmammalian; Energy Metabolism; Etoposide; Fluoresceins; Membrane Transport Proteins; Models, Animal; Propionates; Quinolines; Sea Urchins; Verapamil; Vinblastine | 2006 |
Rapid assessment of p-glycoprotein-drug interactions at the blood-brain barrier.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Blotting, Western; Cells, Cultured; Drug Interactions; Endothelium, Vascular; Fluoresceins; Fluorescent Dyes; Pharmaceutical Preparations; Swine; Verapamil | 2006 |
Bioactive polyketides from Peperomia duclouxii.
Topics: Cyclohexanones; Drugs, Chinese Herbal; Female; Fluoresceins; Humans; Inhibitory Concentration 50; Intercellular Adhesion Molecule-1; Interleukin-1alpha; Molecular Structure; Peperomia; Plants, Medicinal; Sesquiterpenes; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Verapamil | 2007 |
(R)- and (S)-verapamil differentially modulate the multidrug-resistant protein MRP1.
Topics: Adenosine Triphosphatases; Animals; Cell Line; Cell Proliferation; Cell Survival; Cricetinae; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Fluoresceins; Fluorescent Dyes; Formazans; Glutathione; Inhibitory Concentration 50; Kidney; Leukotriene C4; Multidrug Resistance-Associated Proteins; Protein Conformation; Sodium Iodide; Spectrometry, Fluorescence; Stereoisomerism; Tetrazolium Salts; Transfection; Tryptophan; Verapamil | 2007 |
[Evaluation of the P-gp pump function on leukemic cell membrane and proper application of its reversal agents with Calcein-AM and flow cytometry].
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Child; Drug Resistance, Multiple; Flow Cytometry; Fluoresceins; Humans; K562 Cells; Tumor Cells, Cultured; Verapamil; Vincristine | 2007 |
Activity of drug efflux transporters in tumor cells under hypoxic conditions.
Topics: Acidosis; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carcinoma; Cell Hypoxia; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Fluorescent Dyes; Isotonic Solutions; Male; Multidrug Resistance-Associated Proteins; Prostatic Neoplasms; Rats; Rhodamine 123; Ringer's Solution; Time Factors; Verapamil | 2008 |
Chalcogenopyrylium dyes as inhibitors/modulators of P-glycoprotein in multidrug-resistant cells.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cell Membrane Permeability; Cell Polarity; Cells, Cultured; Chalcogens; Dogs; Drug Resistance, Multiple; Fluoresceins; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Verapamil | 2008 |
Permeation of Boswellia extract in the Caco-2 model and possible interactions of its constituents KBA and AKBA with OATP1B3 and MRP2.
Topics: Aniline Compounds; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Boswellia; Caco-2 Cells; Cell Line; Dogs; Electric Impedance; Fluoresceins; Fluorescent Dyes; Humans; Intestinal Absorption; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Organic Anion Transporters, Sodium-Independent; Permeability; Plant Extracts; Propionates; Quinolines; Solubility; Solute Carrier Organic Anion Transporter Family Member 1B3; Sulfobromophthalein; Tight Junctions; Transfection; Triterpenes; Verapamil; Xanthenes | 2009 |
Functionality of drug efflux pumps in antimonial resistant Leishmania donovani field isolates.
Topics: Adenosine Triphosphate; Animals; Antimony; Antiprotozoal Agents; ATP-Binding Cassette Transporters; Drug Resistance, Multiple; Fluoresceins; Humans; Leishmania donovani; Leishmaniasis, Visceral; Multidrug Resistance-Associated Proteins; Ofloxacin; Probenecid; Protozoan Proteins; Rhodamine 123; Verapamil | 2009 |
Multidrug resistance reversal agent, NSC77037, identified with a cell-based screening assay.
Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzylisoquinolines; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Fluoresceins; Humans; Paclitaxel; Substrate Specificity; Time Factors; Verapamil | 2010 |
T-type calcium channel as a portal of iron uptake into cardiomyocytes of beta-thalassemic mice.
Topics: Animals; beta-Thalassemia; Calcium Channels, T-Type; Cell Survival; Cells, Cultured; Deferoxamine; Disease Models, Animal; Fluoresceins; Heterozygote; Immunohistochemistry; Iron; Mice; Mice, Inbred C57BL; Myocytes, Cardiac; Verapamil | 2011 |
Reversal of doxorubicin-resistance by multifunctional nanoparticles in MCF-7/ADR cells.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Cell Line, Tumor; Cell Nucleus; Cell Survival; Cytoplasmic Granules; Cytosol; Doxorubicin; Drug Carriers; Drug Combinations; Drug Resistance, Neoplasm; Female; Fluoresceins; Fluorescent Dyes; Humans; Lactic Acid; Light; Molecular Structure; Nanoparticles; Particle Size; Photochemotherapy; Photosensitizing Agents; Polyesters; Polyethylene Glycols; Polymers; Porphyrins; Verapamil; Vitamin E | 2011 |
Rat intestinal precision-cut slices as an in vitro model to study xenobiotic interaction with transporters.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Transporters; Fluoresceins; Fluorescent Dyes; Glyburide; Indomethacin; Intestine, Small; Male; Microtomy; Multidrug Resistance-Associated Proteins; Rats; Rats, Wistar; Verapamil; Xenobiotics | 2011 |
Regulation of endocytosis into human brain-microvascular endothelial cells by inhibition of efflux proteins.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Brain; Cell Death; Cell Survival; Endocytosis; Endothelial Cells; Fluoresceins; Humans; Microvessels; Multidrug Resistance-Associated Proteins; Probenecid; Tight Junctions; Verapamil | 2011 |
Functional test of multidrug transporter activity in hippocampal-neocortical brain slices from epileptic patients.
Topics: Adjuvants, Pharmaceutic; Anticonvulsants; ATP Binding Cassette Transporter, Subfamily B, Member 1; Epilepsy; Fluoresceins; Gene Expression Regulation; Hippocampus; Humans; In Vitro Techniques; Multidrug Resistance-Associated Proteins; Neocortex; Nerve Tissue Proteins; Neurons; Probenecid; Verapamil | 2011 |
Inhibitory effects of furanocoumarin derivatives in Kampo extract medicines on P-glycoprotein at the blood-brain barrier.
Topics: Animals; Apiaceae; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blood-Brain Barrier; Caco-2 Cells; Cattle; Citrus paradisi; Coumarins; Endothelial Cells; Enzyme Inhibitors; Fluoresceins; Furans; Furocoumarins; Herb-Drug Interactions; Humans; Intestinal Absorption; Male; Medicine, Kampo; Permeability; Plant Extracts; Rats; Rats, Wistar; Rutaceae; Verapamil | 2011 |
Functional evidence of multidrug resistance transporters (MDR) in rodent olfactory epithelium.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Sub-Family B Member 4; Biological Transport; Cyclosporine; Female; Fluoresceins; Gene Expression; Male; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Multidrug Resistance-Associated Proteins; Olfactory Mucosa; Olfactory Receptor Neurons; Probenecid; Propionates; Quinolines; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Verapamil | 2012 |
Involvement of ABCB1 and ABCC1 transporters in sea urchin Echinometra lucunter fertilization.
Topics: Acrosome; Acrosome Reaction; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Calcium Channel Blockers; Fertilization; Fluoresceins; Leukotriene Antagonists; Male; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Oligopeptides; Organic Anion Transporters; Propionates; Quinolines; Sea Urchins; Spermatozoa; Verapamil | 2012 |
Functional impact of ABCB1 variants on interactions between P-glycoprotein and methadone.
Topics: Analysis of Variance; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Fluoresceins; Genetic Variation; HEK293 Cells; Humans; Immunoblotting; Inhibitory Concentration 50; Kinetics; Methadone; Mutagenesis, Site-Directed; Real-Time Polymerase Chain Reaction; Rhodamine 123; Verapamil | 2013 |
Nitensidine A, a guanidine alkaloid from Pterogyne nitens, is a novel substrate for human ABC transporter ABCB1.
Topics: Adenosine Triphosphatases; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B; ATP-Binding Cassette Transporters; Cell Line, Tumor; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fabaceae; Fluoresceins; Guanidines; Humans; Leukemia, T-Cell; Molecular Docking Simulation; Monoterpenes; Phytotherapy; Plant Extracts; Structure-Activity Relationship; Verapamil | 2014 |
Reporter dyes demonstrate functional expression of multidrug resistance proteins in the marine flatworm Macrostomum lignano: the sponge-derived dye Ageladine A is not a substrate of these transporters.
Topics: Aniline Compounds; Animals; Astrocytes; Biological Transport; Brain; Cells, Cultured; Coloring Agents; Fluoresceins; Fluorescent Dyes; Fura-2; Glutathione; Multidrug Resistance-Associated Proteins; Platyhelminths; Probenecid; Pyrroles; Rats; Rats, Wistar; Rhodamines; Verapamil; Xanthenes | 2013 |
Multilayer spheroids to quantify drug uptake and diffusion in 3D.
Topics: ATP Binding Cassette Transporter, Subfamily B; Carbenoxolone; Cell Line; Cell Line, Tumor; Cyclosporine; Diffusion; Fluoresceins; HEK293 Cells; Humans; Loperamide; MCF-7 Cells; Pharmaceutical Preparations; Spheroids, Cellular; Verapamil | 2014 |
Involvement of Ca2+ in Vacuole Degradation Caused by a Rapid Temperature Decrease in Saintpaulia Palisade Cells: A Case of Gene Expression Analysis in a Specialized Small Tissue.
Topics: Calcium; Calcium Channel Blockers; Calcium Chelating Agents; Cold Temperature; Egtazic Acid; Fluoresceins; Gene Expression Regulation, Plant; Hydrogen-Ion Concentration; Intracellular Membranes; Ion Channels; Magnoliopsida; Microscopy, Confocal; Nifedipine; Plant Leaves; Reverse Transcriptase Polymerase Chain Reaction; Vacuoles; Verapamil | 2015 |
Anthocyanidins but not anthocyanins inhibit P-glycoprotein-mediated calcein extrusion - possible implication for orally administered drugs.
Topics: Administration, Oral; Animals; Anthocyanins; ATP Binding Cassette Transporter, Subfamily B, Member 1; Dietary Supplements; Dose-Response Relationship, Drug; Fluoresceins; Food-Drug Interactions; Humans; Swine; Verapamil | 2016 |
A novel flavonoid from Fissistigma cupreonitens, 5‑hydroxy‑7,8‑dimethoxyflavanone, competitively inhibited the efflux function of human P-glycoprotein and reversed cancer multi-drug resistance.
Topics: Annonaceae; Apoptosis; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Cycle; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flavonoids; Fluoresceins; Humans; Molecular Docking Simulation; Phytochemicals; Rhodamine 123; Verapamil | 2021 |
Gadolinium-sensitive, voltage-dependent calcium release channels in the endoplasmic reticulum of a higher plant mechanoreceptor organ.
Topics: Calcium; Calcium Channels; Endoplasmic Reticulum; Erythrosine; Gadolinium; Ion Channel Gating; Plant Shoots; Verapamil | 1995 |